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中文名称 英文名称 CAS号 化学式 结构式图片
—— (1S)-N-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)cyclohex-3-ene-1-carboxamide —— C21H21N3O
(1S)-N-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)cyclohex-3-ene-1-carboxamide
—— [(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-(3-phenylimidazol-4-yl)methanone —— C22H20N4OS
[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-(3-phenylimidazol-4-yl)methanone
—— 5-chloro-N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide —— C21H25ClN4OS
5-chloro-N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide
—— 5-chloro-N-[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide —— C21H25ClN4OS
5-chloro-N-[(2S)-2-(dimethylamino)-2-thiophen-2-ylethyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide
—— 2-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]acetamide —— C20H23N5O2
2-(3,5-dimethyl-1,2-oxazol-4-yl)-N-[4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]acetamide
—— (4-Benzylsulfonylpiperazin-1-yl)-(3-phenylimidazol-4-yl)methanone —— C21H22N4O3S
(4-Benzylsulfonylpiperazin-1-yl)-(3-phenylimidazol-4-yl)methanone
—— [(1R)-2-[[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carbonyl]amino]-1-thiophen-2-ylethyl]-dimethylazanium —— C21H26ClN4OS+
[(1R)-2-[[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carbonyl]amino]-1-thiophen-2-ylethyl]-dimethylazanium
—— N-[(4-methylphenyl)methyl]-3-(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)propanamide —— C22H21N5O2
N-[(4-methylphenyl)methyl]-3-(4-oxo-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)propanamide
—— N-[2-[(2R)-1-cyanopropan-2-yl]sulfanylphenyl]-2-(5-phenyltetrazol-2-yl)acetamide —— C19H18N6OS
N-[2-[(2R)-1-cyanopropan-2-yl]sulfanylphenyl]-2-(5-phenyltetrazol-2-yl)acetamide
—— (3R)-N-[2-methyl-6-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)phenyl]oxolane-3-carboxamide —— C17H21N3O3
(3R)-N-[2-methyl-6-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)phenyl]oxolane-3-carboxamide
—— 1-[3-[ethylsulfonyl(methyl)amino]propyl]-3-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C13H24N4O3S2
1-[3-[ethylsulfonyl(methyl)amino]propyl]-3-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C22H17F3N4O2S
N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C22H17F3N4O2S
N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— tert-butyl N-[(3R)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl]-N-methylcarbamate —— C14H19N3O3S
tert-butyl N-[(3R)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl]-N-methylcarbamate
—— 1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-[(2S)-1-thiophen-2-ylpropan-2-yl]urea —— C14H19N3OS2
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-[(2S)-1-thiophen-2-ylpropan-2-yl]urea
—— 2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanyl-N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]acetamide —— C22H22F3N3O2S
2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanyl-N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]acetamide
—— N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]acetamide —— C20H19F3N4O3S
N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]acetamide
—— 2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanyl-N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]acetamide —— C22H22F3N3O2S
2-[1-(2,5-dimethylphenyl)imidazol-2-yl]sulfanyl-N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]acetamide
—— N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C21H17F6N3O2
N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— tert-butyl N-[(3S)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl]-N-methylcarbamate —— C14H19N3O3S
tert-butyl N-[(3S)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl]-N-methylcarbamate
—— N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide —— C21H17F6N3O2
N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carboxamide
—— N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-3-(2-methoxyphenyl)-1-phenylpyrazole-4-carboxamide —— C26H22F3N3O3
N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-3-(2-methoxyphenyl)-1-phenylpyrazole-4-carboxamide
—— N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-3-(3-methoxyphenyl)-1-phenylpyrazole-4-carboxamide —— C26H22F3N3O3
N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-3-(3-methoxyphenyl)-1-phenylpyrazole-4-carboxamide
—— N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]acetamide —— C20H19F3N4O3S
N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-2-[3-(4-methoxyphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]acetamide
—— N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1-(4-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide —— C21H17F6N3O2
N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1-(4-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
—— 4-cyclohexyl-3-(3,4-dimethoxyphenyl)-5-[[(2R)-oxan-2-yl]methylsulfanyl]-1,2,4-triazole —— C22H31N3O3S
4-cyclohexyl-3-(3,4-dimethoxyphenyl)-5-[[(2R)-oxan-2-yl]methylsulfanyl]-1,2,4-triazole
—— N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-3-(2-methoxyphenyl)-1-phenylpyrazole-4-carboxamide —— C26H22F3N3O3
N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-3-(2-methoxyphenyl)-1-phenylpyrazole-4-carboxamide
—— N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-3-(3-methoxyphenyl)-1-phenylpyrazole-4-carboxamide —— C26H22F3N3O3
N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-3-(3-methoxyphenyl)-1-phenylpyrazole-4-carboxamide
—— 2-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(7-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)acetamide —— C24H21N3O3
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(7-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)acetamide
—— N-(3-acetamidophenyl)-2-[1-(2-methylpropyl)-5-phenylimidazol-2-yl]sulfanylacetamide —— C23H26N4O2S
N-(3-acetamidophenyl)-2-[1-(2-methylpropyl)-5-phenylimidazol-2-yl]sulfanylacetamide
—— 1-(4-chlorophenyl)-N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-5-propan-2-ylpyrazole-4-carboxamide —— C22H21ClF3N3O2
1-(4-chlorophenyl)-N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-5-propan-2-ylpyrazole-4-carboxamide
—— (2S)-2-(4-methoxyphenyl)-N-[(5-phenyl-1H-imidazol-2-yl)methyl]propanamide —— C20H21N3O2
(2S)-2-(4-methoxyphenyl)-N-[(5-phenyl-1H-imidazol-2-yl)methyl]propanamide
—— N-[4-(1,3-benzodioxol-5-yl)-1,3-thiazol-2-yl]-3-(4-fluorophenyl)imidazole-4-carboxamide —— C20H13FN4O3S
N-[4-(1,3-benzodioxol-5-yl)-1,3-thiazol-2-yl]-3-(4-fluorophenyl)imidazole-4-carboxamide
—— N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-[1]benzofuro[3,2-d]pyrimidin-4-amine —— C20H16N6O
N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-[1]benzofuro[3,2-d]pyrimidin-4-amine
—— 1-[(1S)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-[(1R,3S)-3-(trifluoromethyl)cyclohexyl]urea —— C14H20F3N3OS
1-[(1S)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-[(1R,3S)-3-(trifluoromethyl)cyclohexyl]urea
—— 1-[(6-chloropyridin-3-yl)methyl]-3-[(1S)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C13H15ClN4OS
1-[(6-chloropyridin-3-yl)methyl]-3-[(1S)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— 1-[(1S)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-3-[(2-methyl-1,3-thiazol-5-yl)methyl]urea —— C15H22N6OS
1-[(1S)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-3-[(2-methyl-1,3-thiazol-5-yl)methyl]urea
—— N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide —— C22H22F3N3O4
N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
—— N-[(1S)-1-(1H-benzimidazol-2-yl)-2-methylpropyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanamide —— C25H29N5O
N-[(1S)-1-(1H-benzimidazol-2-yl)-2-methylpropyl]-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanamide
—— 1-[(2R)-1-(2-methylpropoxy)propan-2-yl]-3-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C14H25N3O2S
1-[(2R)-1-(2-methylpropoxy)propan-2-yl]-3-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— 1-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-[(1R,3S)-3-(trifluoromethyl)cyclohexyl]urea —— C14H20F3N3OS
1-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-[(1R,3S)-3-(trifluoromethyl)cyclohexyl]urea
—— N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1-(4-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide —— C21H17F6N3O2
N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1-(4-methylphenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
—— (3-methyl-1-phenylthieno[2,3-c]pyrazol-5-yl)-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)methanone —— C24H21N3OS
(3-methyl-1-phenylthieno[2,3-c]pyrazol-5-yl)-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)methanone
—— 1-(4-imidazol-1-ylbutyl)-3-[(1S)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C14H21N5OS
1-(4-imidazol-1-ylbutyl)-3-[(1S)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— [(3R)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl] 2-(4-chlorophenyl)acetate —— C16H13ClN2O3S
[(3R)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl] 2-(4-chlorophenyl)acetate
—— 1-[(6-chloropyridin-3-yl)methyl]-3-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea —— C13H15ClN4OS
1-[(6-chloropyridin-3-yl)methyl]-3-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]urea
—— 1-[(1R)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-3-[(2-methyl-1,3-thiazol-5-yl)methyl]urea —— C15H22N6OS
1-[(1R)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-3-[(2-methyl-1,3-thiazol-5-yl)methyl]urea
—— 1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-[(2R)-1-thiophen-2-ylpropan-2-yl]urea —— C14H19N3OS2
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-[(2R)-1-thiophen-2-ylpropan-2-yl]urea
—— 2-[(1S)-3-oxo-1H-2-benzofuran-1-yl]-N-[4-(tetrazol-1-yl)phenyl]acetamide —— C17H13N5O3
2-[(1S)-3-oxo-1H-2-benzofuran-1-yl]-N-[4-(tetrazol-1-yl)phenyl]acetamide
—— 1-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-[(1S,3S)-3-(trifluoromethyl)cyclohexyl]urea —— C14H20F3N3OS
1-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]-3-[(1S,3S)-3-(trifluoromethyl)cyclohexyl]urea