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中文名称 英文名称 CAS号 化学式 结构式图片
—— (1S,2R,4R)-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C18H25N3O
(1S,2R,4R)-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— 2-(methoxymethyl)-5-[3-(2-oxopyrrolidin-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O3
2-(methoxymethyl)-5-[3-(2-oxopyrrolidin-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (1S,2S,4R)-N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C17H23N3O
(1S,2S,4R)-N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— (1S,2S,4R)-N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C17H23N3O
(1S,2S,4R)-N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— 5-[(1S,3S,4S)-2-(benzenesulfonyl)-2-azabicyclo[2.2.1]heptan-3-yl]-3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazole —— C22H23N3O5S
5-[(1S,3S,4S)-2-(benzenesulfonyl)-2-azabicyclo[2.2.1]heptan-3-yl]-3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazole
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O3
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2S)-2-(benzotriazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H18N6O
5-[(2S)-2-(benzotriazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-3-(4-methylphenyl)-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H20N4O3
2-(methoxymethyl)-3-(4-methylphenyl)-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O2
5-(1-ethylpyrazol-3-yl)-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(4-methoxyphenyl)-3-methyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H18N4O3
2-(4-methoxyphenyl)-3-methyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (1S,2S,4R)-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C18H25N3O
(1S,2S,4R)-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— 2-(3-methoxyphenyl)-3-methyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H18N4O3
2-(3-methoxyphenyl)-3-methyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (1S,2S,4R)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C14H17N3O2
(1S,2S,4R)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— 2-(methoxymethyl)-5-[(3R)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N4O3
2-(methoxymethyl)-5-[(3R)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3-methoxyphenyl)-1-[(1S,8S)-5-(4-methoxyphenyl)-4,5,11-triazatricyclo[6.2.1.02,6]undeca-2(6),3-dien-11-yl]propan-1-one —— C25H27N3O3
3-(3-methoxyphenyl)-1-[(1S,8S)-5-(4-methoxyphenyl)-4,5,11-triazatricyclo[6.2.1.02,6]undeca-2(6),3-dien-11-yl]propan-1-one
—— 5-(1-ethylpyrazol-3-yl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H17N5O
5-(1-ethylpyrazol-3-yl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethyl-3-methylpyrazol-4-yl)-2-(3-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O2
5-(1-ethyl-3-methylpyrazol-4-yl)-2-(3-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1R,3S,4R)-2-(3-methyl-1-propan-2-ylpyrazol-4-yl)sulfonyl-2-azabicyclo[2.2.1]heptan-3-yl]-3-phenyl-1,2,4-oxadiazole —— C21H25N5O3S
5-[(1R,3S,4R)-2-(3-methyl-1-propan-2-ylpyrazol-4-yl)sulfonyl-2-azabicyclo[2.2.1]heptan-3-yl]-3-phenyl-1,2,4-oxadiazole
—— 2-(3-chlorophenyl)-3-methyl-5-[(3R)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23ClN4O2
2-(3-chlorophenyl)-3-methyl-5-[(3R)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-2-(3-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O2
5-(1-ethylpyrazol-3-yl)-2-(3-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (1S,2R,4R)-N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C17H23N3O
(1S,2R,4R)-N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— 5-[(1R,3S,4R)-2-(1-ethylpyrazol-4-yl)sulfonyl-2-azabicyclo[2.2.1]heptan-3-yl]-3-phenyl-1,2,4-oxadiazole —— C19H21N5O3S
5-[(1R,3S,4R)-2-(1-ethylpyrazol-4-yl)sulfonyl-2-azabicyclo[2.2.1]heptan-3-yl]-3-phenyl-1,2,4-oxadiazole
—— (1S,2S,4R)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C16H20N2O2
(1S,2S,4R)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— (1S,2R,4R)-N-methyl-N-[2-(2-methylimidazol-1-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C17H23N3O
(1S,2R,4R)-N-methyl-N-[2-(2-methylimidazol-1-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— (1S,2R,4R)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C14H17N3O2
(1S,2R,4R)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[(5R,7R)-3-(1,2,4-triazol-1-yl)-1-adamantyl]acetamide —— C20H27N5O2
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[(5R,7R)-3-(1,2,4-triazol-1-yl)-1-adamantyl]acetamide
—— (1S,2S,4R)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C15H19N3O2
(1S,2S,4R)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— (1S,2S,4R)-N-methyl-N-[2-(2-methylimidazol-1-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C17H23N3O
(1S,2S,4R)-N-methyl-N-[2-(2-methylimidazol-1-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— (1S,2R,4R)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C15H19N3O2
(1S,2R,4R)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[(5S,7S)-3-(1,2,4-triazol-1-yl)-1-adamantyl]acetamide —— C20H27N5O2
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[(5S,7S)-3-(1,2,4-triazol-1-yl)-1-adamantyl]acetamide
—— (+/-)-4-(2-(5,5-Dimethylhex-1-ynyl)cyclopropyl)imidazole —— C14H20N2
(+/-)-4-(2-(5,5-Dimethylhex-1-ynyl)cyclopropyl)imidazole
—— ethyl (4S)-4-[(4R)-3-ethoxycarbonyl-5-oxo-1-phenyl-4H-pyrazol-4-yl]-5-oxo-1-phenyl-4H-pyrazole-3-carboxylate —— C24H22N4O6
ethyl (4S)-4-[(4R)-3-ethoxycarbonyl-5-oxo-1-phenyl-4H-pyrazol-4-yl]-5-oxo-1-phenyl-4H-pyrazole-3-carboxylate
—— 1-[(1R,12R)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one —— C21H22N4O2
1-[(1R,12R)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one
—— 1-[(1S,12S)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one —— C22H24N4O2
1-[(1S,12S)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one
—— 1-[(1R,12R)-7-(3-fluorophenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one —— C21H21FN4O
1-[(1R,12R)-7-(3-fluorophenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one
—— 2-methoxy-1-[(1R,12R)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone —— C21H22N4O3
2-methoxy-1-[(1R,12R)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone
—— (1S,5R,6S,7S)-3-methyl-N-[(2S)-1-(4-methyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)propan-2-yl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide —— C24H25N5O4
(1S,5R,6S,7S)-3-methyl-N-[(2S)-1-(4-methyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)propan-2-yl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
—— 2-[(1S,2S,6S,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-[2-(4-methyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)ethyl]acetamide —— C24H25N5O4
2-[(1S,2S,6S,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-[2-(4-methyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)ethyl]acetamide
—— (1S,5R,6R,7S)-3-methyl-N-[(2R)-1-(4-methyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)propan-2-yl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide —— C24H25N5O4
(1S,5R,6R,7S)-3-methyl-N-[(2R)-1-(4-methyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)propan-2-yl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
—— (1R,12R)-7-(4-methoxyphenyl)-15-[(2-methylpyrazol-3-yl)methyl]-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraene —— C23H24N6O
(1R,12R)-7-(4-methoxyphenyl)-15-[(2-methylpyrazol-3-yl)methyl]-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraene
—— 2-methoxy-1-[(1S,12S)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone —— C21H22N4O3
2-methoxy-1-[(1S,12S)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]ethanone
—— 1-[(1S,12S)-7-(4-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one —— C22H24N4O2
1-[(1S,12S)-7-(4-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one
—— (1S,5R,6S,7S)-N-[2-(4,8-dimethyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)ethyl]-3-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide —— C24H25N5O4
(1S,5R,6S,7S)-N-[2-(4,8-dimethyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)ethyl]-3-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
—— 1-[(1S,12S)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one —— C21H22N4O2
1-[(1S,12S)-7-(2-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one
—— 1-[(1R,12R)-7-(4-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one —— C22H24N4O2
1-[(1R,12R)-7-(4-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]butan-1-one
—— (1R,12R)-7-(3-fluorophenyl)-15-[(2-methylpyrazol-3-yl)methyl]-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraene —— C22H21FN6
(1R,12R)-7-(3-fluorophenyl)-15-[(2-methylpyrazol-3-yl)methyl]-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraene
—— 1-[(1R,12R)-7-(4-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one —— C21H22N4O2
1-[(1R,12R)-7-(4-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one
—— 1-[(1S,12S)-7-(4-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one —— C21H22N4O2
1-[(1S,12S)-7-(4-methoxyphenyl)-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]propan-1-one
—— 5-Methyl-2-propylthiazole —— C7H11NS
5-Methyl-2-propylthiazole
—— 2-[(1S,2R,6S,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-[2-(4-methyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)ethyl]acetamide —— C24H25N5O4
2-[(1S,2R,6S,7S)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-[2-(4-methyl-1-oxo-[1,2,4]triazolo[4,3-a]quinolin-2-yl)ethyl]acetamide