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中文名称 英文名称 CAS号 化学式 结构式图片
—— (Z)-2-(1,3-benzothiazol-2-yl)-3-[3-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enenitrile —— C31H27N5O3S2
(Z)-2-(1,3-benzothiazol-2-yl)-3-[3-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enenitrile
—— (Z)-2-(1,3-benzothiazol-2-yl)-3-[3-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enenitrile —— C31H27N5O3S2
(Z)-2-(1,3-benzothiazol-2-yl)-3-[3-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enenitrile
—— (Z)-2-(1H-benzimidazol-2-yl)-3-[3-[3-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enenitrile —— C31H28N6O3S
(Z)-2-(1H-benzimidazol-2-yl)-3-[3-[3-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enenitrile
—— 2-[(5Z)-5-[[3-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid —— C27H26N4O6S3
2-[(5Z)-5-[[3-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid
—— 2-[(5Z)-5-[[3-[3-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid —— C27H26N4O6S3
2-[(5Z)-5-[[3-[3-[(2S,6R)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid
—— (5Z)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[3-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]-1-phenylpyrazol-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H23N3O4S3
(5Z)-3-[(3S)-1,1-dioxothiolan-3-yl]-5-[[3-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]-1-phenylpyrazol-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (1S,2R,5R)-2-[3-(4-chlorophenyl)-4-phenyl-5-sulfanylidene-1,2,4-triazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one —— C20H16ClN3O3S
(1S,2R,5R)-2-[3-(4-chlorophenyl)-4-phenyl-5-sulfanylidene-1,2,4-triazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one
—— (5Z)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[3-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]-1-phenylpyrazol-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H23N3O4S3
(5Z)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[3-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]-1-phenylpyrazol-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (1S,2R,5R)-2-[3-(3,4-dimethoxyphenyl)-4-methyl-5-sulfanylidene-1,2,4-triazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one —— C17H19N3O5S
(1S,2R,5R)-2-[3-(3,4-dimethoxyphenyl)-4-methyl-5-sulfanylidene-1,2,4-triazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one
—— methyl (6R)-6-tert-butyl-2-[[2-(1-methylimidazol-2-yl)sulfanylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C20H27N3O3S2
methyl (6R)-6-tert-butyl-2-[[2-(1-methylimidazol-2-yl)sulfanylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— N-[(1S,2R,4R)-2-bicyclo[2.2.1]heptanyl]-2-[[5-(4-chlorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C17H19ClN4OS
N-[(1S,2R,4R)-2-bicyclo[2.2.1]heptanyl]-2-[[5-(4-chlorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (1S,2R,5R)-2-[5-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]tetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one —— C14H11F3N4O4S
(1S,2R,5R)-2-[5-sulfanylidene-4-[4-(trifluoromethoxy)phenyl]tetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one
—— (5Z)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[3-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]-1-phenylpyrazol-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H23N3O4S3
(5Z)-3-[(3R)-1,1-dioxothiolan-3-yl]-5-[[3-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]-1-phenylpyrazol-4-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— N-[(2-fluorophenyl)methyl]-3-methyl-N-[(1R,2R)-2-methylcyclohexyl]-4-(tetrazol-1-yl)benzenesulfonamide —— C22H26FN5O2S
N-[(2-fluorophenyl)methyl]-3-methyl-N-[(1R,2R)-2-methylcyclohexyl]-4-(tetrazol-1-yl)benzenesulfonamide
—— (2S)-N-cyclopentyl-2-(N-[2-[5-(4-methylphenyl)tetrazol-2-yl]acetyl]anilino)butanamide —— C25H30N6O2
(2S)-N-cyclopentyl-2-(N-[2-[5-(4-methylphenyl)tetrazol-2-yl]acetyl]anilino)butanamide
—— 4-[4-[(Z)-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxo-1,3-thiazol-5-ylidene]methyl]-1-phenylpyrazol-3-yl]-N,N-dimethylbenzenesulfonamide —— C27H29N5O4S2
4-[4-[(Z)-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-4-oxo-1,3-thiazol-5-ylidene]methyl]-1-phenylpyrazol-3-yl]-N,N-dimethylbenzenesulfonamide
—— 4-[4-[(Z)-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxo-1,3-thiazol-5-ylidene]methyl]-1-phenylpyrazol-3-yl]-N,N-dimethylbenzenesulfonamide —— C27H29N5O4S2
4-[4-[(Z)-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-4-oxo-1,3-thiazol-5-ylidene]methyl]-1-phenylpyrazol-3-yl]-N,N-dimethylbenzenesulfonamide
—— 2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C24H30N6O2S2
2-[[5-[(4,6-dimethylpyrimidin-2-yl)sulfanylmethyl]-4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 1-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]urea —— C19H23ClN4O2
1-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]urea
—— (1R,2S,3S)-4-amino-1-(2-phenyltriazol-4-yl)butane-1,2,3-triol —— C12H16N4O3
(1R,2S,3S)-4-amino-1-(2-phenyltriazol-4-yl)butane-1,2,3-triol
—— (1S,2R,5R)-2-[4-(4-chloro-2,5-dimethoxyphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one —— C15H15ClN4O5S
(1S,2R,5R)-2-[4-(4-chloro-2,5-dimethoxyphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one
—— N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]hexanamide —— C26H30N4O4
N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-[(1R,2S,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]hexanamide
—— 1-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]urea —— C19H23ClN4O2
1-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]urea
—— (1R,2R,3S)-4-amino-1-(2-phenyltriazol-4-yl)butane-1,2,3-triol —— C12H16N4O3
(1R,2R,3S)-4-amino-1-(2-phenyltriazol-4-yl)butane-1,2,3-triol
—— N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-[(1R,2S,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]hexanamide —— C26H30N4O4
N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-[(1R,2S,6R,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]hexanamide
—— 2-(4-chlorophenyl)-5-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-1,3-oxazole-4-carbonitrile —— C16H16ClN3O2
2-(4-chlorophenyl)-5-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-1,3-oxazole-4-carbonitrile
—— 1-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]urea —— C19H23ClN4O2
1-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-[[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]urea
—— N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[(7R)-7-methyl-4-oxo-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetamide —— C30H29N5O3S2
N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[(7R)-7-methyl-4-oxo-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetamide
—— N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[(7S)-7-methyl-4-oxo-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetamide —— C30H29N5O3S2
N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[(7S)-7-methyl-4-oxo-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetamide
—— 4-{3-[(1R,2R)-2-phenylcyclopropyl]-5-thioxo-1,5-dihydro-4H-1,2,4-triazol-4-yl}benzoic acid —— C18H15N3O2S
4-{3-[(1R,2R)-2-phenylcyclopropyl]-5-thioxo-1,5-dihydro-4H-1,2,4-triazol-4-yl}benzoic acid
—— (5Z)-5-[[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one —— C32H29ClN4O3S
(5Z)-5-[[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one
—— (Z)-3-[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]-2-cyano-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C31H27ClN4O3
(Z)-3-[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]-2-cyano-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (4R)-6-amino-4-[(1R)-cyclohex-2-en-1-yl]-3-(methoxymethyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C15H18N4O2
(4R)-6-amino-4-[(1R)-cyclohex-2-en-1-yl]-3-(methoxymethyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (5Z)-5-[[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one —— C32H29ClN4O3S
(5Z)-5-[[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one
—— (Z)-3-[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]-2-cyano-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C31H27ClN4O3
(Z)-3-[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]-2-cyano-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (Z)-3-[3-[4-[(4-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]-2-cyano-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C31H27ClN4O3
(Z)-3-[3-[4-[(4-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]-2-cyano-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— (5Z)-5-[[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one —— C32H29ClN4O3S
(5Z)-5-[[3-[4-[(2-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]methylidene]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one
—— (Z)-3-[3-[4-[(4-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]-2-cyano-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C31H27ClN4O3
(Z)-3-[3-[4-[(4-chlorophenyl)methoxy]phenyl]-1-phenylpyrazol-4-yl]-2-cyano-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (NE)-N-[(6S)-3-ethyl-6-[(2R)-2-ethylsulfanylpropyl]-6,7-dihydro-5H-1,2-benzoxazol-4-ylidene]hydroxylamine —— C14H22N2O2S
(NE)-N-[(6S)-3-ethyl-6-[(2R)-2-ethylsulfanylpropyl]-6,7-dihydro-5H-1,2-benzoxazol-4-ylidene]hydroxylamine
—— (1S)-1-(5-chloro-1-methylimidazol-2-yl)ethanol —— C6H9ClN2O
(1S)-1-(5-chloro-1-methylimidazol-2-yl)ethanol
—— (1S,2R,5R)-2-(5-phenyltetrazol-1-yl)-6,8-dioxabicyclo[3.2.1]octan-4-one —— C13H12N4O3
(1S,2R,5R)-2-(5-phenyltetrazol-1-yl)-6,8-dioxabicyclo[3.2.1]octan-4-one
—— (1S,2R,5R)-2-[4-(2,6-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one —— C15H16N4O3S
(1S,2R,5R)-2-[4-(2,6-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one
—— (1S,2R,5R)-2-[4-(3,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one —— C15H16N4O3S
(1S,2R,5R)-2-[4-(3,5-dimethylphenyl)-5-sulfanylidenetetrazol-1-yl]-6,8-dioxabicyclo[3.2.1]octan-4-one
—— Pyrazolo[3,4-d]pyrimidine 9 —— C29H37N9O3S
Pyrazolo[3,4-d]pyrimidine 9
—— trans-3-{4-[(1H-2-indolylmethyl)amino]phenyl}-[4-(4-methylpiperazino)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine —— C31H37N9
trans-3-{4-[(1H-2-indolylmethyl)amino]phenyl}-[4-(4-methylpiperazino)-cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
—— trans-N1-(4-{4-amino-1-[4-(4-methylpiperazino)cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-3-methyl-3-phenylbutanamide —— C34H44N8O2
trans-N1-(4-{4-amino-1-[4-(4-methylpiperazino)cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-3-methyl-3-phenylbutanamide
—— (4Z)-4-[[2-(6-chloro-1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)hydrazinyl]methylidene]-2-methoxycyclohexa-2,5-dien-1-one —— C19H15ClN6O2
(4Z)-4-[[2-(6-chloro-1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)hydrazinyl]methylidene]-2-methoxycyclohexa-2,5-dien-1-one
—— (4Z)-4-[[2-(1,6-diphenylpyrazolo[3,4-d]pyrimidin-4-yl)hydrazinyl]methylidene]-2-methoxycyclohexa-2,5-dien-1-one —— C25H20N6O2
(4Z)-4-[[2-(1,6-diphenylpyrazolo[3,4-d]pyrimidin-4-yl)hydrazinyl]methylidene]-2-methoxycyclohexa-2,5-dien-1-one
—— (6Z)-6-[[[2-(4-methylphenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C21H16N2O2
(6Z)-6-[[[2-(4-methylphenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— 4-[(5S,7S)-3-(4-methylphenyl)-1-adamantyl]-1,3-thiazol-2-amine —— C20H24N2S
4-[(5S,7S)-3-(4-methylphenyl)-1-adamantyl]-1,3-thiazol-2-amine