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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
2-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N4O2
2-ethyl-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-fluorophenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18FN5O
3-(4-fluorophenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
2-(methoxymethyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19ClN6O
2-(3-chlorophenyl)-5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2S)-2-(benzotriazol-1-yl)propyl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H22N6O2
5-[(2S)-2-(benzotriazol-1-yl)propyl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H27N5O3
3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(4-fluorophenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19FN4O3
2-(4-fluorophenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-chlorophenyl)-2-methyl-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H17ClN4O2
3-(4-chlorophenyl)-2-methyl-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(benzotriazol-1-yl)propyl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H20N6O
5-[(2R)-2-(benzotriazol-1-yl)propyl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-3-(4-methoxyphenyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O4
2-(methoxymethyl)-3-(4-methoxyphenyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N6O
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N6O
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-fluorophenyl)-5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19FN4O3
3-(4-fluorophenyl)-5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18ClN5O
2-(3-chlorophenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(2,4-dimethoxyphenyl)-4-methyl-1H-pyrazole-5-carboxamide —— C22H29N3O3
N-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(2,4-dimethoxyphenyl)-4-methyl-1H-pyrazole-5-carboxamide
—— 3-(4-fluorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19FN4O3
3-(4-fluorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O3
2-ethyl-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19ClN4O2
5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-3-methyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H17ClN4O2
2-(3-chlorophenyl)-3-methyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-[(5S,7S)-3-(5-phenyltetrazol-2-yl)-1-adamantyl]acetic acid —— C19H22N4O2
2-[(5S,7S)-3-(5-phenyltetrazol-2-yl)-1-adamantyl]acetic acid
—— 2-(3-chlorophenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18ClN5O
2-(3-chlorophenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19ClN4O3
2-(3-chlorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H18N4O2
5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(4-methoxyphenyl)-3-methyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N4O3
2-(4-methoxyphenyl)-3-methyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-fluorophenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18FN5O
3-(4-fluorophenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-3-methyl-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H17ClN4O2
2-(3-chlorophenyl)-3-methyl-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(2-methoxyphenyl)-3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O2
2-(2-methoxyphenyl)-3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(benzotriazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H17FN6O
5-[(2R)-2-(benzotriazol-1-yl)propyl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-chlorophenyl)-2-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H20ClN5O
3-(4-chlorophenyl)-2-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N4O2
3-methyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2S)-2-(benzotriazol-1-yl)propyl]-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H17FN6O
5-[(2S)-2-(benzotriazol-1-yl)propyl]-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-fluorophenyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H15FN4O2
3-(4-fluorophenyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(2,4-dichlorophenyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H14Cl2N4O2
2-(2,4-dichlorophenyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N4O4
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H20N4O2
5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N4O2
2-ethyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-3-(4-methylphenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H25N5O2
2-(methoxymethyl)-3-(4-methylphenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N4O4
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H16N4O2
5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-chlorophenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19ClN4O3
3-(4-chlorophenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H24N4O2
5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
2-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H20ClN5O
2-(3-chlorophenyl)-3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one