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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(2R)-2-(benzotriazol-1-yl)propyl]-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H17FN6O
5-[(2R)-2-(benzotriazol-1-yl)propyl]-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N4O3
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-fluorophenyl)-5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19FN4O3
3-(4-fluorophenyl)-5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(4-methoxyphenyl)-3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O2
2-(4-methoxyphenyl)-3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-2-(3-methylphenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O
3-methyl-2-(3-methylphenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-methylphenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
3-(4-methylphenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(2,4-dichlorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18Cl2N4O3
2-(2,4-dichlorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19FN4O2
5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3,4-dimethoxyphenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O5
2-(3,4-dimethoxyphenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-methyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H18N4O2
2-methyl-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-chlorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21ClN4O3
3-(4-chlorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21ClN6O
2-(3-chlorophenyl)-5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-chlorophenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18ClN5O
3-(4-chlorophenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(4-methoxyphenyl)-3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O2
2-(4-methoxyphenyl)-3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2S)-2-(benzotriazol-1-yl)propyl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H20N6O
5-[(2S)-2-(benzotriazol-1-yl)propyl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H27N5O3
3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(4-fluorophenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18FN5O
2-(4-fluorophenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N4O3
2-(methoxymethyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-methylphenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
2-(3-methylphenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3,4-dimethoxyphenyl)-2-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H25N5O3
3-(3,4-dimethoxyphenyl)-2-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O3
2-ethyl-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19FN4O2
5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O
2-ethyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(2-methoxyphenyl)-3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O2
2-(2-methoxyphenyl)-3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H15ClN4O2
2-(3-chlorophenyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N4O3
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-chlorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19ClN4O3
3-(4-chlorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3,4-dimethoxyphenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O5
2-(3,4-dimethoxyphenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(benzotriazol-1-yl)propyl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H22N6O2
5-[(2R)-2-(benzotriazol-1-yl)propyl]-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-[(5R,7R)-3-(5-phenyltetrazol-2-yl)-1-adamantyl]acetic acid —— C19H22N4O2
2-[(5R,7R)-3-(5-phenyltetrazol-2-yl)-1-adamantyl]acetic acid
—— 5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19ClN4O2
5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H20ClN5O
2-(3-chlorophenyl)-3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-methoxyphenyl)-3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O2
2-(3-methoxyphenyl)-3-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(2,4-dimethoxyphenyl)-4-methyl-1H-pyrazole-5-carboxamide —— C22H29N3O3
N-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(2,4-dimethoxyphenyl)-4-methyl-1H-pyrazole-5-carboxamide
—— 2-(3-chlorophenyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H15ClN4O2
2-(3-chlorophenyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (1S,2S,4R)-N-[5-(2-methoxyphenyl)-2-methylpyrazol-3-yl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C21H23N3O2
(1S,2S,4R)-N-[5-(2-methoxyphenyl)-2-methylpyrazol-3-yl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(2,4-dichlorophenyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H14Cl2N4O2
2-(2,4-dichlorophenyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(2,4-dimethoxyphenyl)-4-methyl-1H-pyrazole-5-carboxamide —— C22H29N3O3
N-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(2,4-dimethoxyphenyl)-4-methyl-1H-pyrazole-5-carboxamide
—— 5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H16N4O2
5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(benzotriazol-1-yl)propyl]-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H22N6O2
5-[(2R)-2-(benzotriazol-1-yl)propyl]-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (E)-1-(2,3-dimethylimidazo[2,1-b]thiazol-5-yl)-3-(2-furyl)prop-2-en-1-ol —— C14H14N2O2S
(E)-1-(2,3-dimethylimidazo[2,1-b]thiazol-5-yl)-3-(2-furyl)prop-2-en-1-ol
—— N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(2,4-dimethoxyphenyl)-4-methyl-1H-pyrazole-5-carboxamide —— C22H29N3O3
N-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-3-(2,4-dimethoxyphenyl)-4-methyl-1H-pyrazole-5-carboxamide