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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-methyl-2-(3-methylphenyl)-5-[(2S)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
3-methyl-2-(3-methylphenyl)-5-[(2S)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-3-(4-methoxyphenyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O4
2-(methoxymethyl)-3-(4-methoxyphenyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-methylphenyl)-5-[(2R)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
3-(4-methylphenyl)-5-[(2R)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-methoxyphenyl)-3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O2
2-(3-methoxyphenyl)-3-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19ClN4O2
5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-methyl-7-oxo-3-phenyl-N-[(2S)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidine-5-carboxamide —— C23H26N6O2
2-methyl-7-oxo-3-phenyl-N-[(2S)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidine-5-carboxamide
—— 4-[2-[(3S)-3-hydroxy-3-(4-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl]-5-methyl-2-(4-methylphenyl)-1H-pyrazol-3-one —— C24H27N3O3
4-[2-[(3S)-3-hydroxy-3-(4-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl]-5-methyl-2-(4-methylphenyl)-1H-pyrazol-3-one
—— 5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H20N4O3
5-[(3R)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H20N4O3
5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[(1R)-1-(1,5-dimethylpyrazol-4-yl)ethyl]-3-[3-oxo-5-(trifluoromethyl)-1H-pyrazol-2-yl]benzamide —— C18H18F3N5O2
N-[(1R)-1-(1,5-dimethylpyrazol-4-yl)ethyl]-3-[3-oxo-5-(trifluoromethyl)-1H-pyrazol-2-yl]benzamide
—— 5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N6O3
5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1S)-1-(2-methoxyphenoxy)ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H19N3O3
5-[(1S)-1-(2-methoxyphenoxy)ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-[(5R,7R)-3-(5-methyltetrazol-2-yl)-1-adamantyl]acetyl chloride —— C14H19ClN4O
2-[(5R,7R)-3-(5-methyltetrazol-2-yl)-1-adamantyl]acetyl chloride
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N4O4
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(methoxymethyl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C25H24N4O2
5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1R)-1-(2-methoxyphenoxy)ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H19N3O3
5-[(1R)-1-(2-methoxyphenoxy)ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-2-(3-methylphenyl)-5-[(3S)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H23N5O2
3-methyl-2-(3-methylphenyl)-5-[(3S)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H19ClN4O2
5-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-3-(4-chlorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[[3-(4-fluorophenyl)-1-methylpyrazol-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H16FN5O
5-[[3-(4-fluorophenyl)-1-methylpyrazol-4-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N4O3
2-(methoxymethyl)-5-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(2,4-dichlorophenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18Cl2N4O3
2-(2,4-dichlorophenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-methyl-7-oxo-3-phenyl-N-[(2R)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidine-5-carboxamide —— C23H26N6O2
2-methyl-7-oxo-3-phenyl-N-[(2R)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidine-5-carboxamide
—— 2-tert-butyl-5-[[3-(4-fluorophenyl)-1-methylpyrazol-4-yl]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H22FN5O
2-tert-butyl-5-[[3-(4-fluorophenyl)-1-methylpyrazol-4-yl]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H24N6O
5-[(2R)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 1-[(2S)-butan-2-yl]-5-methylpyrazole-4-sulfonyl chloride —— C8H13ClN2O2S
1-[(2S)-butan-2-yl]-5-methylpyrazole-4-sulfonyl chloride
—— 3-(4-methylphenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
3-(4-methylphenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5Z)-5-benzylidene-3-[2-(2-methyl-5-nitro-imidazol-1-yl)ethyl]thiazolidine-2,4-dione —— C16H14N4O4S
(5Z)-5-benzylidene-3-[2-(2-methyl-5-nitro-imidazol-1-yl)ethyl]thiazolidine-2,4-dione
—— N-[5-(3,4-dimethylphenyl)-1-methylimidazol-2-yl]-3-[(3R)-2-oxo-1,3-dihydroindol-3-yl]propanamide —— C23H24N4O2
N-[5-(3,4-dimethylphenyl)-1-methylimidazol-2-yl]-3-[(3R)-2-oxo-1,3-dihydroindol-3-yl]propanamide
—— 3-(4-chlorophenyl)-5-[(3S)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H18ClN5O2
3-(4-chlorophenyl)-5-[(3S)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1S)-1-(2-methoxyphenoxy)ethyl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H21N3O3
5-[(1S)-1-(2-methoxyphenoxy)ethyl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-chlorophenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19ClN4O3
2-(3-chlorophenyl)-5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— N-[5-(4-fluorophenyl)-1-methylimidazol-2-yl]-3-[(3R)-2-oxo-1,3-dihydroindol-3-yl]propanamide —— C21H19FN4O2
N-[5-(4-fluorophenyl)-1-methylimidazol-2-yl]-3-[(3R)-2-oxo-1,3-dihydroindol-3-yl]propanamide
—— 3-(4-methylphenyl)-5-[(3R)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H21N5O2
3-(4-methylphenyl)-5-[(3R)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(1R)-1-(2-methoxyphenoxy)ethyl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H21N3O3
5-[(1R)-1-(2-methoxyphenoxy)ethyl]-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H22N4O3
5-[(3S)-1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H20N6O
5-[(2S)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-chlorophenyl)-2-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H20ClN5O
3-(4-chlorophenyl)-2-methyl-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-methylphenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
2-(3-methylphenyl)-5-[(2S)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
2-(methoxymethyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(4-fluorophenyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H15FN4O2
2-(4-fluorophenyl)-5-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-chlorophenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H18ClN5O
3-(4-chlorophenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3,4-dimethoxyphenyl)-2-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H25N5O3
3-(3,4-dimethoxyphenyl)-2-methyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H22N4O3
5-[(3R)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O
2-ethyl-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-2-(3-methylphenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O
3-methyl-2-(3-methylphenyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(4-fluorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19FN4O3
2-(4-fluorophenyl)-5-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O2
2-(methoxymethyl)-5-[(2R)-1-(5-methylpyrazol-1-yl)propan-2-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H22N4O2
5-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one