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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethyl]-2-ethyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H24N6O
5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethyl]-2-ethyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-fluorophenyl)-5-[(2-pyridin-4-yl-1,3-thiazol-4-yl)methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H14FN5OS
3-(4-fluorophenyl)-5-[(2-pyridin-4-yl-1,3-thiazol-4-yl)methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-methoxyphenyl)-3-methyl-5-[(3S)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N4O3
2-(3-methoxyphenyl)-3-methyl-5-[(3S)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethyl-3-methylpyrazol-4-yl)-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
5-(1-ethyl-3-methylpyrazol-4-yl)-2-methyl-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(4-chloro-1-ethylpyrazol-3-yl)-3-(3,4-dimethoxyphenyl)-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H20ClN5O3
5-(4-chloro-1-ethylpyrazol-3-yl)-3-(3,4-dimethoxyphenyl)-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-3-phenyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H18N4O2
2-ethyl-3-phenyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethyl-3-methylpyrazol-4-yl)-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
5-(1-ethyl-3-methylpyrazol-4-yl)-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-methoxyphenyl)-3-methyl-5-(1-propylpyrazol-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O2
2-(3-methoxyphenyl)-3-methyl-5-(1-propylpyrazol-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-fluorophenyl)-5-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H15F4N5O
3-(4-fluorophenyl)-5-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-3-(4-methoxyphenyl)-5-(1H-pyrazol-5-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H17N5O3
2-(methoxymethyl)-3-(4-methoxyphenyl)-5-(1H-pyrazol-5-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H17N5O
5-(1-ethylpyrazol-3-yl)-3-methyl-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3,4-dimethoxyphenyl)-5-(1-ethylpyrazol-3-yl)-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O3
3-(3,4-dimethoxyphenyl)-5-(1-ethylpyrazol-3-yl)-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethyl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H22N6O
5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethyl]-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-chlorophenyl)-2-methyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H15ClN4O2
3-(4-chlorophenyl)-2-methyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-2-(3-methylphenyl)-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H18N4O2
3-methyl-2-(3-methylphenyl)-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(2R)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H25N5O3
3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(2R)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(2-methoxyphenyl)-3-methyl-5-(1-propylpyrazol-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O2
2-(2-methoxyphenyl)-3-methyl-5-(1-propylpyrazol-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(2S)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H25N5O3
3-(3,4-dimethoxyphenyl)-2-ethyl-5-[(2S)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(4-chloro-1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H20ClN5O3
5-(4-chloro-1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H14FN5O
5-(1-ethylpyrazol-3-yl)-3-(4-fluorophenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O3
5-(1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methoxyphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O2
5-(1-ethylpyrazol-3-yl)-2-(methoxymethyl)-3-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-methylphenyl)-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H16N4O2
3-(4-methylphenyl)-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-2-phenyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H16N4O2
3-methyl-2-phenyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethylpyrazol-3-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H15N5O
5-(1-ethylpyrazol-3-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-3-(4-methoxyphenyl)-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H20N4O4
2-(methoxymethyl)-3-(4-methoxyphenyl)-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-5-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H18F3N5O
3-methyl-5-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethyl-3-methylpyrazol-4-yl)-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O2
5-(1-ethyl-3-methylpyrazol-4-yl)-2-(4-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethyl-3-methylpyrazol-4-yl)-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
5-(1-ethyl-3-methylpyrazol-4-yl)-3-methyl-2-(3-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-5-(1-ethylpyrazol-3-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
2-ethyl-5-(1-ethylpyrazol-3-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-methyl-2-phenyl-5-(1-propylpyrazol-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H19N5O
3-methyl-2-phenyl-5-(1-propylpyrazol-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(1-ethyl-3-methylpyrazol-4-yl)-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O2
5-(1-ethyl-3-methylpyrazol-4-yl)-2-(2-methoxyphenyl)-3-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-5-(1-ethyl-3-methylpyrazol-4-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O
2-ethyl-5-(1-ethyl-3-methylpyrazol-4-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H16F3N5O
5-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-methyl-3-phenyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H16N4O2
2-methyl-3-phenyl-5-(pyridin-2-yloxymethyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3,4-dimethoxyphenyl)-2-ethyl-5-(1-ethyl-3-methylpyrazol-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H25N5O3
3-(3,4-dimethoxyphenyl)-2-ethyl-5-(1-ethyl-3-methylpyrazol-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-3-(4-methylphenyl)-5-[(3R)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H28N4O3
2-(methoxymethyl)-3-(4-methylphenyl)-5-[(3R)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(methoxymethyl)-3-(4-methylphenyl)-5-[(3S)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C23H28N4O3
2-(methoxymethyl)-3-(4-methylphenyl)-5-[(3S)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(2-methoxyphenyl)-3-methyl-5-[(2S)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O2
2-(2-methoxyphenyl)-3-methyl-5-[(2S)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-ethyl-5-[3-(2-methylimidazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H23N5O
2-ethyl-5-[3-(2-methylimidazol-1-yl)propyl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(2-methoxyphenyl)-3-methyl-5-[(2R)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H21N5O2
2-(2-methoxyphenyl)-3-methyl-5-[(2R)-2-pyrazol-1-ylpropyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(3-methoxyphenyl)-1-[(1R,8R)-5-(4-methoxyphenyl)-4,5,11-triazatricyclo[6.2.1.02,6]undeca-2(6),3-dien-11-yl]propan-1-one —— C25H27N3O3
3-(3-methoxyphenyl)-1-[(1R,8R)-5-(4-methoxyphenyl)-4,5,11-triazatricyclo[6.2.1.02,6]undeca-2(6),3-dien-11-yl]propan-1-one
—— 5-[(1R,3S,4R)-2-(benzenesulfonyl)-2-azabicyclo[2.2.1]heptan-3-yl]-3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazole —— C22H23N3O5S
5-[(1R,3S,4R)-2-(benzenesulfonyl)-2-azabicyclo[2.2.1]heptan-3-yl]-3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazole
—— (1S,2R,4R)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C16H20N2O2
(1S,2R,4R)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— (1S,2R,4R)-N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C17H23N3O
(1S,2R,4R)-N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide
—— 2-(methoxymethyl)-5-[(3S)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N4O3
2-(methoxymethyl)-5-[(3S)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(3-methoxyphenyl)-3-methyl-5-[(3R)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H26N4O3
2-(3-methoxyphenyl)-3-methyl-5-[(3R)-1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 3-(4-fluorophenyl)-5-[2-(3-methoxy-1,2-oxazol-5-yl)ethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H15FN4O3
3-(4-fluorophenyl)-5-[2-(3-methoxy-1,2-oxazol-5-yl)ethyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 1-(azetidin-1-yl)-2-[(1S,3S,4S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-azabicyclo[2.2.1]heptan-2-yl]ethanone —— C19H22N4O2
1-(azetidin-1-yl)-2-[(1S,3S,4S)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-azabicyclo[2.2.1]heptan-2-yl]ethanone
—— (1S,2S,4R)-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide —— C18H25N3O
(1S,2S,4R)-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-carboxamide