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中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-1-[(4-fluorophenyl)methyl]-6,6-dimethyl-3-(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-3-(trifluoromethyl)-5,7-dihydroindole-2,4-dione —— C28H25F4N3O3
(3S)-1-[(4-fluorophenyl)methyl]-6,6-dimethyl-3-(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-3-(trifluoromethyl)-5,7-dihydroindole-2,4-dione
—— (3S,5S,8R)-8-(butoxymethyl)-3-[2-[[5-(2-chlorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetyl]-3-methyl-2,7-dioxaspiro[4.4]nonane-1,6-dione —— C23H26ClN3O6S
(3S,5S,8R)-8-(butoxymethyl)-3-[2-[[5-(2-chlorophenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]acetyl]-3-methyl-2,7-dioxaspiro[4.4]nonane-1,6-dione
—— (5R)-1-(4-fluorophenyl)-5-(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-5-(trifluoromethyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4,6-trione —— C23H15F4N5O4
(5R)-1-(4-fluorophenyl)-5-(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-5-(trifluoromethyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4,6-trione
—— (5S)-1-(4-fluorophenyl)-5-(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-5-(trifluoromethyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4,6-trione —— C23H15F4N5O4
(5S)-1-(4-fluorophenyl)-5-(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-5-(trifluoromethyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4,6-trione
—— N-[(Z)-[(3R)-5-bromo-2-oxo-1,3-dihydroindol-3-yl]methylideneamino]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C20H16BrN5O3
N-[(Z)-[(3R)-5-bromo-2-oxo-1,3-dihydroindol-3-yl]methylideneamino]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— (NZ)-N-[(1S,3R,4S)-3-(2,4-dimethyl-5-phenylimidazol-1-yl)-2-bicyclo[2.2.1]heptanylidene]hydroxylamine —— C18H21N3O
(NZ)-N-[(1S,3R,4S)-3-(2,4-dimethyl-5-phenylimidazol-1-yl)-2-bicyclo[2.2.1]heptanylidene]hydroxylamine
—— (NZ)-N-[(1S,3S,4S)-3-(2,4-dimethyl-5-phenylimidazol-1-yl)-2-bicyclo[2.2.1]heptanylidene]hydroxylamine —— C18H21N3O
(NZ)-N-[(1S,3S,4S)-3-(2,4-dimethyl-5-phenylimidazol-1-yl)-2-bicyclo[2.2.1]heptanylidene]hydroxylamine
—— (3aS)-3a-[(E)-2-[3-(4-ethoxyphenyl)-1-phenylpyrazol-4-yl]ethenyl]-4,4,6-trimethyl-1,3-dihydroimidazo[1,2-a]indol-2-one —— C32H32N4O2
(3aS)-3a-[(E)-2-[3-(4-ethoxyphenyl)-1-phenylpyrazol-4-yl]ethenyl]-4,4,6-trimethyl-1,3-dihydroimidazo[1,2-a]indol-2-one
—— (1R,2S,3S,4R)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C19H21N3O3
(1R,2S,3S,4R)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— (1R,3S,4R)-4,7,7-trimethyl-3-(1-phenyltetrazol-5-yl)sulfanylbicyclo[2.2.1]heptan-2-one —— C17H20N4OS
(1R,3S,4R)-4,7,7-trimethyl-3-(1-phenyltetrazol-5-yl)sulfanylbicyclo[2.2.1]heptan-2-one
—— (NE)-N-[(1S,3R,4S)-3-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-2-bicyclo[2.2.1]heptanylidene]hydroxylamine —— C22H20N2O2S
(NE)-N-[(1S,3R,4S)-3-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-2-bicyclo[2.2.1]heptanylidene]hydroxylamine
—— (1R,3S,4R)-3-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-4,7,7-trimethylbicyclo[2.2.1]heptan-2-one —— C25H25NO2S
(1R,3S,4R)-3-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-4,7,7-trimethylbicyclo[2.2.1]heptan-2-one
—— (1S,3S,4S)-3-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-4,7,7-trimethylbicyclo[2.2.1]heptan-2-one —— C25H25NO2S
(1S,3S,4S)-3-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-4,7,7-trimethylbicyclo[2.2.1]heptan-2-one
—— (NE)-N-[(1S,3S,4S)-3-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-2-bicyclo[2.2.1]heptanylidene]hydroxylamine —— C22H20N2O2S
(NE)-N-[(1S,3S,4S)-3-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]-2-bicyclo[2.2.1]heptanylidene]hydroxylamine
—— (1S,3S,4S)-4,7,7-trimethyl-3-(1-phenyltetrazol-5-yl)sulfanylbicyclo[2.2.1]heptan-2-one —— C17H20N4OS
(1S,3S,4S)-4,7,7-trimethyl-3-(1-phenyltetrazol-5-yl)sulfanylbicyclo[2.2.1]heptan-2-one
—— (1R,2S,3R,4R)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid —— C19H21N3O3
(1R,2S,3R,4R)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid
—— 5-methyl-4-[(Z)-2-[(4S)-3-methyl-5-oxo-1,4-dihydropyrazol-4-yl]ethenyl]-2-phenyl-1H-pyrazol-3-one —— C16H16N4O2
5-methyl-4-[(Z)-2-[(4S)-3-methyl-5-oxo-1,4-dihydropyrazol-4-yl]ethenyl]-2-phenyl-1H-pyrazol-3-one
—— 5-methyl-4-[(Z)-2-[(4R)-3-methyl-5-oxo-1,4-dihydropyrazol-4-yl]ethenyl]-2-phenyl-1H-pyrazol-3-one —— C16H16N4O2
5-methyl-4-[(Z)-2-[(4R)-3-methyl-5-oxo-1,4-dihydropyrazol-4-yl]ethenyl]-2-phenyl-1H-pyrazol-3-one
—— (3S,5S,8R)-3-(2-amino-1,3-thiazol-4-yl)-3-methyl-8-(2-methylpropoxymethyl)-2,7-dioxaspiro[4.4]nonane-1,6-dione —— C16H22N2O5S
(3S,5S,8R)-3-(2-amino-1,3-thiazol-4-yl)-3-methyl-8-(2-methylpropoxymethyl)-2,7-dioxaspiro[4.4]nonane-1,6-dione
—— methyl (4R)-2-methyl-4-(3-nitrophenyl)-6-[(1-phenylimidazol-2-yl)sulfanylmethyl]-1,4-dihydropyridine-3-carboxylate —— C24H22N4O4S
methyl (4R)-2-methyl-4-(3-nitrophenyl)-6-[(1-phenylimidazol-2-yl)sulfanylmethyl]-1,4-dihydropyridine-3-carboxylate
—— methyl (4S)-2-methyl-4-(3-nitrophenyl)-6-[(1-phenylimidazol-2-yl)sulfanylmethyl]-1,4-dihydropyridine-3-carboxylate —— C24H22N4O4S
methyl (4S)-2-methyl-4-(3-nitrophenyl)-6-[(1-phenylimidazol-2-yl)sulfanylmethyl]-1,4-dihydropyridine-3-carboxylate
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C32H34FN5O2S
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— (1R,7R)-1,10,10-trimethyl-3-phenyl-3,4-diazatricyclo[5.2.1.02,6]deca-2(6),4-diene-5-carboxylic acid —— C18H20N2O2
(1R,7R)-1,10,10-trimethyl-3-phenyl-3,4-diazatricyclo[5.2.1.02,6]deca-2(6),4-diene-5-carboxylic acid
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H37N5O2S
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-4-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H30FN5O2S
2-[(4R)-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C29H31N5O2S2
2-[(4R)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-4-(2-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C32H25ClFN5O2S
2-[(4R)-4-(2-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C31H32ClN5O2S
2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4R)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H30FN5O2S
2-[(4R)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C29H31N5O2S2
2-[(4R)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-4-(2-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C32H25ClFN5O2S
2-[(4S)-4-(2-chlorophenyl)-1-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C30H29F2N5O2S
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H30FN5O2S
2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C31H31F2N5O2S
2-[(4S)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4R)-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C34H30FN5O2S
2-[(4R)-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C30H29F2N5O2S
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-4-(3-fluorophenyl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C33H28FN5O2S
2-[(4R)-4-(3-fluorophenyl)-1-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H29F2N5O2S
2-[(4R)-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C31H31F2N5O2S
2-[(4R)-3-tert-butyl-4-(2,4-difluorophenyl)-1-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C30H29F2N5O2S
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C29H31N5O2S2
2-[(4S)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C34H29F2N5O2S
2-[(4S)-4-(2,4-difluorophenyl)-1-(2,3-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-4-(2-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C30H29F2N5O2S
2-[(4R)-3-tert-butyl-4-(2-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C35H33N5O2S
2-[(4R)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C29H31N5O2S2
2-[(4R)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide —— C31H32FN5O2S
2-[(4S)-3-tert-butyl-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide
—— 2-[(4S)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C34H30FN5O2S
2-[(4S)-1-(2,3-dimethylphenyl)-4-(4-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-1-(2,3-dimethylphenyl)-4-(3-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide —— C34H30FN5O2S
2-[(4R)-1-(2,3-dimethylphenyl)-4-(3-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C30H29ClFN5O2S
2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C30H33N5O2S2
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide