中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
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2-[(4R)-3-tert-butyl-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C31H32ClN5O2S |
|
—— |
2-[(4S)-3-tert-butyl-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C31H32FN5O2S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C31H32ClN5O2S |
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—— |
2-[(4S)-1-(2,3-dimethylphenyl)-4-(3-methylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C35H33N5O2S |
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—— |
2-[(4S)-3-tert-butyl-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C31H32FN5O2S |
|
—— |
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C30H29ClFN5O2S |
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—— |
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C31H32FN5O2S |
|
—— |
2-[(4S)-1-(2,4-dimethylphenyl)-4-(2-fluorophenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C34H30FN5O2S |
|
—— |
2-[(4S)-4-(2,4-difluorophenyl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C34H29F2N5O2S |
|
—— |
2-[(4R)-3-tert-butyl-1-(4-fluorophenyl)-4-(3-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C31H32FN5O2S |
|
—— |
2-[(4R)-1-(2-chlorophenyl)-7-oxo-3-phenyl-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C30H24ClN5O2S2 |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C31H32FN5O2S |
|
—— |
2-[(4S)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C30H29ClFN5O2S |
|
—— |
2-[(4R)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C31H32FN5O2S |
|
—— |
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C30H33N5O2S2 |
|
—— |
2-[(4R)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C29H31N5O2S2 |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-fluorophenyl)-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C31H32FN5O2S |
|
—— |
2-[(4R)-3-tert-butyl-1-(2-chlorophenyl)-4-(3-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C30H29ClFN5O2S |
|
—— |
2-[(4S)-3-tert-butyl-4-(3-chlorophenyl)-1-(2-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C31H32ClN5O2S |
|
—— |
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C30H33N5O2S2 |
|
—— |
2-[(4S)-3-tert-butyl-1-(2-methylphenyl)-7-oxo-4-thiophen-3-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C29H31N5O2S2 |
|
—— |
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C30H33N5O2S2 |
|
—— |
2-[(4S)-3-tert-butyl-4-(2-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C30H29F2N5O2S |
|
—— |
2-[(4S)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C30H33N5O2S2 |
|
—— |
2-[(4R)-3-tert-butyl-4-(2-fluorophenyl)-1-(4-fluorophenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-3-ylmethyl)acetamide |
—— |
C30H29F2N5O2S |
|
—— |
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide |
—— |
C30H33N5O2S2 |
|
—— |
3-[(5Z)-5-[[3-[3-[(3R)-3-methylpiperidin-1-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]propanoic acid |
—— |
C28H28N4O5S3 |
|
—— |
N-(4-bromophenyl)-2-[(3E)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]acetamide |
—— |
C28H24BrN7O3S |
|
—— |
2-[(4R)-3-tert-butyl-1-(2,4-dimethylphenyl)-7-oxo-4-thiophen-2-yl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-4-ylmethyl)acetamide |
—— |
C30H33N5O2S2 |
|
—— |
2-[(3E)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-[2-(trifluoromethyl)phenyl]acetamide |
—— |
C29H24F3N7O3S |
|
—— |
2-[(3E)-5-chloro-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-(4-methylphenyl)acetamide |
—— |
C29H26ClN7O3S |
|
—— |
2-[(3E)-5-chloro-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-(4-fluorophenyl)acetamide |
—— |
C28H23ClFN7O3S |
|
—— |
2-[(3E)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-(2-methoxyphenyl)acetamide |
—— |
C29H27N7O4S |
|
—— |
2-[(3E)-5-chloro-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-(2-methoxyphenyl)acetamide |
—— |
C29H26ClN7O4S |
|
—— |
3-[(5Z)-5-[[3-[3-[(3S)-3-methylpiperidin-1-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]propanoic acid |
—— |
C28H28N4O5S3 |
|
—— |
2-[(3E)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-[3-(trifluoromethyl)phenyl]acetamide |
—— |
C29H24F3N7O3S |
|
—— |
2-[(3E)-5-chloro-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-(4-chlorophenyl)acetamide |
—— |
C28H23Cl2N7O3S |
|
—— |
2-[(3E)-5-chloro-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-(2-methylphenyl)acetamide |
—— |
C29H26ClN7O3S |
|
—— |
2-[(3E)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-(4-sulfamoylphenyl)acetamide |
—— |
C28H26N8O5S2 |
|
—— |
2-[(3E)-5-chloro-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-phenylacetamide |
—— |
C28H24ClN7O3S |
|
—— |
2-[(3E)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-phenylacetamide |
—— |
C28H25N7O3S |
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—— |
2-[(3E)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-(4-fluorophenyl)acetamide |
—— |
C28H24FN7O3S |
|
—— |
2-[(3E)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]-N-(4-methylphenyl)acetamide |
—— |
C29H27N7O3S |
|
—— |
N-(4-chlorophenyl)-2-[(3E)-3-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)carbamothioylhydrazinylidene]-2-oxoindol-1-yl]acetamide |
—— |
C28H24ClN7O3S |
|
—— |
(3R)-N-(1,3-benzodioxol-5-ylmethyl)-1-[4-(tetrazol-1-yl)phenyl]sulfonylpiperidine-3-carboxamide |
—— |
C21H22N6O5S |
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—— |
(Z)-2-(1,3-benzothiazol-2-yl)-3-[3-[3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enenitrile |
—— |
C31H27N5O3S2 |
|
—— |
(Z)-2-(1H-benzimidazol-2-yl)-3-[3-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enenitrile |
—— |
C31H28N6O3S |
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—— |
(4S)-6-amino-3-tert-butyl-4-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile |
—— |
C21H21ClN6O |
|
—— |
(Z)-2-(1H-benzimidazol-2-yl)-3-[3-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]prop-2-enenitrile |
—— |
C31H28N6O3S |
|
—— |
2-[(5Z)-5-[[3-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-1-phenylpyrazol-4-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid |
—— |
C27H26N4O6S3 |
|