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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-{[5-(4-fluorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4-methoxyphenyl)propanamide —— C19H19FN4O2S
2-{[5-(4-fluorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4-methoxyphenyl)propanamide
—— 2-{[5-(3-methoxyphenyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}-N-phenylacetamide —— C18H18N4O2S
2-{[5-(3-methoxyphenyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}-N-phenylacetamide
—— N-cyclohexyl-2-{[5-(3-methoxyphenyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide —— C18H24N4O2S
N-cyclohexyl-2-{[5-(3-methoxyphenyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide
—— 2-{[5-(3,4-dimethoxyphenyl)-4-ethyl-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4,5-dimethyl-1,3-thiazol-2-yl)propanamide —— C20H25N5O3S2
2-{[5-(3,4-dimethoxyphenyl)-4-ethyl-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4,5-dimethyl-1,3-thiazol-2-yl)propanamide
—— N-(2,3-dimethylphenyl)-2-{[5-(3-methoxyphenyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide —— C20H22N4O2S
N-(2,3-dimethylphenyl)-2-{[5-(3-methoxyphenyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide
—— 4-(5-Hydroxy-3,4-dimethyl-pyrazol-1-yl)-benzoic acid —— C12H12N2O3
4-(5-Hydroxy-3,4-dimethyl-pyrazol-1-yl)-benzoic acid
—— 2-{[5-(2-methoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(1,3-thiazol-2-yl)acetamide —— C17H17N5O2S2
2-{[5-(2-methoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(1,3-thiazol-2-yl)acetamide
—— N-[(E)-1-(4-bromophenyl)ethylideneamino]-2-[[5-(3-bromophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H17Br2N5OS
N-[(E)-1-(4-bromophenyl)ethylideneamino]-2-[[5-(3-bromophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— N-cyclohexyl-2-{[5-(2-methoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide —— C20H26N4O2S
N-cyclohexyl-2-{[5-(2-methoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide
—— 2-[(4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)propanamide —— C15H16N6OS2
2-[(4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)propanamide
—— 2-{[4-ethyl-5-(3-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(1,3-thiazol-2-yl)acetamide —— C15H14FN5OS2
2-{[4-ethyl-5-(3-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(1,3-thiazol-2-yl)acetamide
—— 2-{[5-(3,4-dimethoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(5-fluoro-2-methylphenyl)acetamide —— C22H23FN4O3S
2-{[5-(3,4-dimethoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(5-fluoro-2-methylphenyl)acetamide
—— 2-{[4-ethyl-5-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(tricyclo[3.3.1.1~3,7~]dec-1-yl)acetamide —— C23H30N4O2S
2-{[4-ethyl-5-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(tricyclo[3.3.1.1~3,7~]dec-1-yl)acetamide
—— N-(1,3-benzodioxol-5-yl)-2-{[4-ethyl-5-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propanamide —— C20H19FN4O3S
N-(1,3-benzodioxol-5-yl)-2-{[4-ethyl-5-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propanamide
—— N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-{[4-ethyl-5-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propanamide —— C18H20FN5OS2
N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-{[4-ethyl-5-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propanamide
—— 2-{[5-(3-fluorophenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(2-methoxyphenyl)acetamide —— C20H19FN4O2S
2-{[5-(3-fluorophenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(2-methoxyphenyl)acetamide
—— 2-{[4-ethyl-5-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(2-fluorophenyl)acetamide —— C18H16F2N4OS
2-{[4-ethyl-5-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(2-fluorophenyl)acetamide
—— N-(2,5-dimethoxyphenyl)-2-{[4-ethyl-5-(3-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide —— C20H21FN4O3S
N-(2,5-dimethoxyphenyl)-2-{[4-ethyl-5-(3-fluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide
—— N-[4-(acetylamino)phenyl]-2-{[5-(4-fluorophenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide —— C21H20FN5O2S
N-[4-(acetylamino)phenyl]-2-{[5-(4-fluorophenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide
—— N-(1,3-benzothiazol-2-yl)-2-{[5-(3-methoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide —— C21H19N5O2S2
N-(1,3-benzothiazol-2-yl)-2-{[5-(3-methoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetamide
—— 1-(4-methylphenyl)-6-[2-[(3R)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C28H24N6O2S2
1-(4-methylphenyl)-6-[2-[(3R)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[2-[(3R)-3-(4-fluorophenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C29H23FN6O3S
6-[2-[(3R)-3-(4-fluorophenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[2-[(3R)-5-(4-methoxyphenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C30H26N6O3S
6-[2-[(3R)-5-(4-methoxyphenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 2-[(4-methyl-5-phenyl-1H-imidazol-2-yl)sulfanyl]-N-(4-sulfamoylphenyl)acetamide —— C18H18N4O3S2
2-[(4-methyl-5-phenyl-1H-imidazol-2-yl)sulfanyl]-N-(4-sulfamoylphenyl)acetamide
—— 2-({5-[(2,5-dimethylphenoxy)methyl]-4-(propan-2-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)-N-(4,5-dimethyl-1,3-thiazol-2-yl)propanamide —— C22H29N5O2S2
2-({5-[(2,5-dimethylphenoxy)methyl]-4-(propan-2-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)-N-(4,5-dimethyl-1,3-thiazol-2-yl)propanamide
—— 2-{[5-(4-fluorophenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)acetamide —— C16H15FN6OS2
2-{[5-(4-fluorophenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)acetamide
—— 2-({5-[(2,6-dimethylphenoxy)methyl]-4-(propan-2-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)-N-(4,5-dimethyl-1,3-thiazol-2-yl)propanamide —— C22H29N5O2S2
2-({5-[(2,6-dimethylphenoxy)methyl]-4-(propan-2-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)-N-(4,5-dimethyl-1,3-thiazol-2-yl)propanamide
—— 6-[2-[(3S)-5-(4-methoxyphenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C30H26N6O3S
6-[2-[(3S)-5-(4-methoxyphenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— (E)-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]-N-[4-[(3S)-3-methylpiperidin-1-yl]sulfonylphenyl]prop-2-enamide —— C30H29FN4O3S
(E)-3-[3-(4-fluorophenyl)-1-phenylpyrazol-4-yl]-N-[4-[(3S)-3-methylpiperidin-1-yl]sulfonylphenyl]prop-2-enamide
—— N-(2-methyl-1H-benzimidazol-5-yl)-2-[(1-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C18H16N6OS
N-(2-methyl-1H-benzimidazol-5-yl)-2-[(1-phenyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— 6-[2-[(3R)-5-(4-bromophenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-fluorophenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C29H22BrFN6O2S
6-[2-[(3R)-5-(4-bromophenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-fluorophenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[2-[(3S)-3-(4-fluorophenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C29H23FN6O3S
6-[2-[(3S)-3-(4-fluorophenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— (3,5-Dimethyl-1-propylpyrazol-4-yl)-(4-propylpiperazin-1-yl)methanone —— C16H28N4O
(3,5-Dimethyl-1-propylpyrazol-4-yl)-(4-propylpiperazin-1-yl)methanone
—— 6-[2-[(3S)-3-(2,3-dimethoxyphenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-fluorophenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C31H27FN6O5S
6-[2-[(3S)-3-(2,3-dimethoxyphenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-fluorophenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 2-[[4-(3,4-dimethylphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1-methylindol-2-yl)methyl]acetamide —— C23H25N5OS
2-[[4-(3,4-dimethylphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-[(1-methylindol-2-yl)methyl]acetamide
—— 1-(4-fluorophenyl)-6-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C27H21FN6O2S2
1-(4-fluorophenyl)-6-[2-[(3S)-3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-fluorophenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C31H27FN6O5S
6-[2-[(3R)-3-(2,3-dimethoxyphenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-fluorophenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 2-{[5-(2-fluorophenyl)-4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4-methyl-1,3-thiazol-2-yl)acetamide —— C17H18FN5OS2
2-{[5-(2-fluorophenyl)-4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4-methyl-1,3-thiazol-2-yl)acetamide
—— 6-[2-[(3S)-5-(4-bromophenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-fluorophenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C29H22BrFN6O2S
6-[2-[(3S)-5-(4-bromophenyl)-3-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-fluorophenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 2-{[5-(4-methoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4-methyl-1,3-thiazol-2-yl)propanamide —— C19H21N5O2S2
2-{[5-(4-methoxyphenyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4-methyl-1,3-thiazol-2-yl)propanamide
—— 2-[1-benzyl-4-(4-fluorophenyl)imidazol-2-yl]sulfanyl-N-(2-methylphenyl)propanamide —— C26H24FN3OS
2-[1-benzyl-4-(4-fluorophenyl)imidazol-2-yl]sulfanyl-N-(2-methylphenyl)propanamide
—— 6-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-methylphenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C27H21FN6O2S2
6-[2-[(3R)-3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]sulfanyl-1-(4-methylphenyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 5-amino-1-(3,5-dimethylphenyl)-N-(oxolan-2-ylmethyl)triazole-4-carboxamide —— C16H21N5O2
5-amino-1-(3,5-dimethylphenyl)-N-(oxolan-2-ylmethyl)triazole-4-carboxamide
—— 5-amino-1-(4-chlorophenyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]triazole-4-carboxamide —— C19H20ClN5O3
5-amino-1-(4-chlorophenyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]triazole-4-carboxamide
—— 2-[(4-ethyl-5-phenyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-(4-methyl-1,3-thiazol-2-yl)propanamide —— C17H19N5OS2
2-[(4-ethyl-5-phenyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-(4-methyl-1,3-thiazol-2-yl)propanamide
—— N-(4-chlorophenyl)-2-[1-[(2-fluorophenyl)methyl]-4-phenylimidazol-2-yl]sulfanylacetamide —— C24H19ClFN3OS
N-(4-chlorophenyl)-2-[1-[(2-fluorophenyl)methyl]-4-phenylimidazol-2-yl]sulfanylacetamide
—— 5-amino-N-benzyl-1-(3-methylsulfanylphenyl)triazole-4-carboxamide —— C17H17N5OS
5-amino-N-benzyl-1-(3-methylsulfanylphenyl)triazole-4-carboxamide
—— [5-Amino-1-(4-chlorophenyl)triazol-4-yl]-piperidin-1-ylmethanone —— C14H16ClN5O
[5-Amino-1-(4-chlorophenyl)triazol-4-yl]-piperidin-1-ylmethanone
—— [5-Amino-1-(3-fluoro-4-methylphenyl)triazol-4-yl]-pyrrolidin-1-ylmethanone —— C14H16FN5O
[5-Amino-1-(3-fluoro-4-methylphenyl)triazol-4-yl]-pyrrolidin-1-ylmethanone
—— 5-amino-N-(1,3-benzodioxol-5-ylmethyl)-1-(3-fluoro-4-methylphenyl)triazole-4-carboxamide —— C18H16FN5O3
5-amino-N-(1,3-benzodioxol-5-ylmethyl)-1-(3-fluoro-4-methylphenyl)triazole-4-carboxamide