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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1,5-anhydro-2,4-dideoxy-4-{[(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)carbonyl]amino}-3-O-(1,3-thiazol-4-ylmethyl)-D-erythro-pentitol —— C14H18N4O4S
1,5-anhydro-2,4-dideoxy-4-{[(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)carbonyl]amino}-3-O-(1,3-thiazol-4-ylmethyl)-D-erythro-pentitol
—— 3-methyl-N-[(3R,4S)-4-(3-methylbut-2-enoxy)oxan-3-yl]pyrazin-2-amine —— C15H23N3O2
3-methyl-N-[(3R,4S)-4-(3-methylbut-2-enoxy)oxan-3-yl]pyrazin-2-amine
—— {5-[(5-chloro-2-methylpyrimidin-4-yl)carbonyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol —— C14H16ClN5O2
{5-[(5-chloro-2-methylpyrimidin-4-yl)carbonyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol
—— 3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}propanamide —— C16H20F3N5O2
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}propanamide
—— 1,5-anhydro-2,3-dideoxy-4-O-[2-(dimethylamino)ethyl]-3-{[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]amino}-D-threo-pentitol —— C16H28N4O4
1,5-anhydro-2,3-dideoxy-4-O-[2-(dimethylamino)ethyl]-3-{[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]amino}-D-threo-pentitol
—— 5-Hydroxy-N-[1-(4-methyl-1H-imidazol-2-YL)ethyl]pyrazine-2-carboxamide —— C11H13N5O2
5-Hydroxy-N-[1-(4-methyl-1H-imidazol-2-YL)ethyl]pyrazine-2-carboxamide
—— N-Ethyl-5-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-YL)methyl]pyrazine-2-carboxamide —— C12H15N5O2
N-Ethyl-5-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-YL)methyl]pyrazine-2-carboxamide
—— 1,5-anhydro-2,3-dideoxy-3-{[(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)acetyl]amino}-4-O-(1,3-thiazol-4-ylmethyl)-D-threo-pentitol —— C16H20N4O5S
1,5-anhydro-2,3-dideoxy-3-{[(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)acetyl]amino}-4-O-(1,3-thiazol-4-ylmethyl)-D-threo-pentitol
—— 2-Amino-N-ethyl-6-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-YL)methyl]pyrimidine-4-carboxamide —— C12H16N6O2
2-Amino-N-ethyl-6-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-YL)methyl]pyrimidine-4-carboxamide
—— 1,5-anhydro-2-O-(cyclopropylmethyl)-3,4-dideoxy-3-{[(4,6-dimethyl-2-oxopyrimidin-1(2H)-yl)acetyl]amino}-D-threo-pentitol —— C17H25N3O4
1,5-anhydro-2-O-(cyclopropylmethyl)-3,4-dideoxy-3-{[(4,6-dimethyl-2-oxopyrimidin-1(2H)-yl)acetyl]amino}-D-threo-pentitol
—— 2-Isopropyl-4-[(3-propoxypiperidin-1-yl)carbonyl]pyrimidine —— C16H25N3O2
2-Isopropyl-4-[(3-propoxypiperidin-1-yl)carbonyl]pyrimidine
—— N-{2-[3-(Methoxymethyl)-1,2,4-oxadiazol-5-YL]ethyl}pyrazine-2-carboxamide —— C11H13N5O3
N-{2-[3-(Methoxymethyl)-1,2,4-oxadiazol-5-YL]ethyl}pyrazine-2-carboxamide
—— 1,5-anhydro-2,3-dideoxy-3-{[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]amino}-4-O-pyridin-2-yl-D-threo-pentitol —— C17H20N4O4
1,5-anhydro-2,3-dideoxy-3-{[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]amino}-4-O-pyridin-2-yl-D-threo-pentitol
—— 1,5-anhydro-2,3-dideoxy-3-[(2,6-dimethoxypyrimidin-4-yl)amino]-4-O-[2-(dimethylamino)ethyl]-D-threo-pentitol —— C15H26N4O4
1,5-anhydro-2,3-dideoxy-3-[(2,6-dimethoxypyrimidin-4-yl)amino]-4-O-[2-(dimethylamino)ethyl]-D-threo-pentitol
—— 6-(3-aminocyclobutyl)-N~4~-(1H-tetrazol-5-ylmethyl)pyrimidine-2,4-diamine —— C10H15N9
6-(3-aminocyclobutyl)-N~4~-(1H-tetrazol-5-ylmethyl)pyrimidine-2,4-diamine
—— 2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]acetamide —— C15H21N5O3
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]acetamide
—— 2-cyclopropyl-6-{cis-3-[(2,6-dimethoxypyrimidin-4-yl)amino]cyclobutyl}pyrimidin-4(3H)-one —— C17H21N5O3
2-cyclopropyl-6-{cis-3-[(2,6-dimethoxypyrimidin-4-yl)amino]cyclobutyl}pyrimidin-4(3H)-one
—— 5-hydroxy-N-(2-{2-[(methylthio)methyl]-1,3-thiazol-4-yl}ethyl)pyrazine-2-carboxamide —— C12H14N4O2S2
5-hydroxy-N-(2-{2-[(methylthio)methyl]-1,3-thiazol-4-yl}ethyl)pyrazine-2-carboxamide
—— Methyl 2-({[2-(4-phenylpyrimidin-2-yl)ethyl]amino}carbonyl)piperidine-1-carboxylate —— C20H24N4O3
Methyl 2-({[2-(4-phenylpyrimidin-2-yl)ethyl]amino}carbonyl)piperidine-1-carboxylate
—— 2-cyclopropyl-6-[trans-3-(1,4-dithiepan-6-ylamino)cyclobutyl]pyrimidin-4(3H)-one —— C16H23N3OS2
2-cyclopropyl-6-[trans-3-(1,4-dithiepan-6-ylamino)cyclobutyl]pyrimidin-4(3H)-one
—— 6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-(3-morpholin-4-ylpropyl)pyrimidin-4-amine —— C17H29N5O2
6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-(3-morpholin-4-ylpropyl)pyrimidin-4-amine
—— 1-(2-{[6-(cis-3-Aminocyclobutyl)pyrimidin-4-yl]amino}ethyl)piperidin-2-one —— C15H23N5O
1-(2-{[6-(cis-3-Aminocyclobutyl)pyrimidin-4-yl]amino}ethyl)piperidin-2-one
—— 6-(cis-3-aminocyclobutyl)-N-[3-(3,5-dimethylisoxazol-4-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine —— C18H27N5O2
6-(cis-3-aminocyclobutyl)-N-[3-(3,5-dimethylisoxazol-4-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 2-Amino-6-methyl-N-[1-(6-methylpyridin-2-YL)ethyl]pyrimidine-4-carboxamide —— C14H17N5O
2-Amino-6-methyl-N-[1-(6-methylpyridin-2-YL)ethyl]pyrimidine-4-carboxamide
—— 2-(2,4-dioxo-1H-pyrimidin-5-yl)-N-[(3R,4R)-3-(6-methylpyridin-3-yl)oxyoxan-4-yl]acetamide —— C17H20N4O5
2-(2,4-dioxo-1H-pyrimidin-5-yl)-N-[(3R,4R)-3-(6-methylpyridin-3-yl)oxyoxan-4-yl]acetamide
—— [2-({4-[(2-Amino-6-isopropylpyrimidin-4-yl)carbonyl]piperazin-1-yl}methyl)phenyl]methanol —— C20H27N5O2
[2-({4-[(2-Amino-6-isopropylpyrimidin-4-yl)carbonyl]piperazin-1-yl}methyl)phenyl]methanol
—— 6-(cis-3-aminocyclobutyl)-N-[3-(2-fluorophenyl)propyl]-2-(methoxymethyl)pyrimidin-4-amine —— C19H25FN4O
6-(cis-3-aminocyclobutyl)-N-[3-(2-fluorophenyl)propyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-[(2-pyrazin-2-yl-1,3-thiazol-4-yl)methyl]pyrimidin-4-amine —— C16H17N7S
6-(trans-3-aminocyclobutyl)-N-[(2-pyrazin-2-yl-1,3-thiazol-4-yl)methyl]pyrimidin-4-amine
—— 1,5-anhydro-2-{[(5-chloro-2-methylpyrimidin-4-yl)carbonyl]amino}-2,4-dideoxy-D-threo-pentitol —— C11H14ClN3O3
1,5-anhydro-2-{[(5-chloro-2-methylpyrimidin-4-yl)carbonyl]amino}-2,4-dideoxy-D-threo-pentitol
—— 1-{5-[(2-Amino-6-methylpyrimidin-4-yl)carbonyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}-2-(methylsulfonyl)ethanol —— C15H20N6O4S
1-{5-[(2-Amino-6-methylpyrimidin-4-yl)carbonyl]-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl}-2-(methylsulfonyl)ethanol
—— {5-[(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol —— C16H22N6O2
{5-[(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-5,6,7,8-tetrahydro-4H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methanol
—— 6-(3-aminocyclobutyl)-N~4~-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyrimidine-2,4-diamine —— C14H20N6S
6-(3-aminocyclobutyl)-N~4~-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyrimidine-2,4-diamine
—— 1,5-anhydro-2,4-dideoxy-3-O-[(3,5-dimethylisoxazol-4-yl)methyl]-4-({[2-(methylamino)pyrimidin-5-yl]carbonyl}amino)-D-erythro-pentitol —— C17H23N5O4
1,5-anhydro-2,4-dideoxy-3-O-[(3,5-dimethylisoxazol-4-yl)methyl]-4-({[2-(methylamino)pyrimidin-5-yl]carbonyl}amino)-D-erythro-pentitol
—— 1,5-anhydro-2-O-benzyl-3,4-dideoxy-3-{[(2-isopropylpyrimidin-4-yl)carbonyl]amino}-D-threo-pentitol —— C20H25N3O3
1,5-anhydro-2-O-benzyl-3,4-dideoxy-3-{[(2-isopropylpyrimidin-4-yl)carbonyl]amino}-D-threo-pentitol
—— N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(pyridin-3-yloxy)acetamide —— C14H16N4O3
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(pyridin-3-yloxy)acetamide
—— 4,6-dimethyl-1-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)pyrimidin-2(1H)-one —— C17H24N6O2
4,6-dimethyl-1-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)pyrimidin-2(1H)-one
—— 1,5-anhydro-2,3-dideoxy-4-O-[(3,5-dimethylisoxazol-4-yl)methyl]-3-{[(3-hydroxypyrazin-2-yl)carbonyl]amino}-D-threo-pentitol —— C16H20N4O5
1,5-anhydro-2,3-dideoxy-4-O-[(3,5-dimethylisoxazol-4-yl)methyl]-3-{[(3-hydroxypyrazin-2-yl)carbonyl]amino}-D-threo-pentitol
—— 2-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-2,5,6,7-tetrahydro-1H-cyclopenta[b]pyridine-3-carboxamide —— C21H20N4O2
2-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-2,5,6,7-tetrahydro-1H-cyclopenta[b]pyridine-3-carboxamide
—— 2-amino-N-(2-azepan-1-ylethyl)-N-ethyl-6-isopropylpyrimidine-4-carboxamide —— C18H31N5O
2-amino-N-(2-azepan-1-ylethyl)-N-ethyl-6-isopropylpyrimidine-4-carboxamide
—— 2-(5-methyl-2,4-dioxopyrimidin-1-yl)-N-[(3R,4R)-4-pyrrolidin-1-yloxolan-3-yl]acetamide —— C15H22N4O4
2-(5-methyl-2,4-dioxopyrimidin-1-yl)-N-[(3R,4R)-4-pyrrolidin-1-yloxolan-3-yl]acetamide
—— 6-(trans-3-aminocyclobutyl)-N~4~-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrimidine-2,4-diamine —— C16H20F3N7
6-(trans-3-aminocyclobutyl)-N~4~-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrimidine-2,4-diamine
—— N-{trans-3-[4-ethyl-5-(hydroxymethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide —— C16H22N6O4
N-{trans-3-[4-ethyl-5-(hydroxymethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
—— N-{trans-3-[4-cyclopropyl-5-(hydroxymethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide —— C17H24N6O3
N-{trans-3-[4-cyclopropyl-5-(hydroxymethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
—— N-[(3R,4R)-3-(6-methylpyridin-3-yl)oxyoxan-4-yl]-4-propylpyrimidine-5-carboxamide —— C19H24N4O3
N-[(3R,4R)-3-(6-methylpyridin-3-yl)oxyoxan-4-yl]-4-propylpyrimidine-5-carboxamide
—— 1-(2-{[6-(3-Aminocyclobutyl)-2-(methoxymethyl)pyrimidin-4-YL]amino}ethyl)piperidin-4-OL —— C17H29N5O2
1-(2-{[6-(3-Aminocyclobutyl)-2-(methoxymethyl)pyrimidin-4-YL]amino}ethyl)piperidin-4-OL
—— N'-[(E)-[2,4,6-trioxo-1-(2-phenylethyl)-1,3-diazinan-5-ylidene]methyl]pentanehydrazide —— C18H22N4O4
N'-[(E)-[2,4,6-trioxo-1-(2-phenylethyl)-1,3-diazinan-5-ylidene]methyl]pentanehydrazide
—— dichlorocopper;[dimethylamino(sulfoniumylidene)methyl]-[(Z)-pyrazin-2-ylmethylideneamino]azanide —— C8H11Cl2CuN5S
dichlorocopper;[dimethylamino(sulfoniumylidene)methyl]-[(Z)-pyrazin-2-ylmethylideneamino]azanide
—— 6-(3-aminocyclobutyl)-N-{2-[(3-chlorobenzyl)thio]ethyl}pyrimidin-4-amine —— C17H21ClN4S
6-(3-aminocyclobutyl)-N-{2-[(3-chlorobenzyl)thio]ethyl}pyrimidin-4-amine
—— (NZ)-N-[5-(4-chlorophenyl)dithiol-3-ylidene]-2-(4-ethoxy-2-oxopyrimidin-1-yl)acetamide —— C17H14ClN3O3S2
(NZ)-N-[5-(4-chlorophenyl)dithiol-3-ylidene]-2-(4-ethoxy-2-oxopyrimidin-1-yl)acetamide
—— N-[(3R,4R)-3-(6-methylpyridin-3-yl)oxyoxan-4-yl]-6-oxo-4,5-dihydro-1H-pyridazine-3-carboxamide —— C16H20N4O4
N-[(3R,4R)-3-(6-methylpyridin-3-yl)oxyoxan-4-yl]-6-oxo-4,5-dihydro-1H-pyridazine-3-carboxamide