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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(4-methoxyphenyl)methyl]-2-methyl-4-[(2S)-1-[(3-methylphenyl)methyl]pyrrolidin-2-yl]pyrimidine-5-carboxamide —— C26H30N4O2
N-[(4-methoxyphenyl)methyl]-2-methyl-4-[(2S)-1-[(3-methylphenyl)methyl]pyrrolidin-2-yl]pyrimidine-5-carboxamide
—— 5-methyl-N-[(4S)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]azepan-4-yl]pyrazine-2-carboxamide —— C18H23N5O2S
5-methyl-N-[(4S)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]azepan-4-yl]pyrazine-2-carboxamide
—— 2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-N-[(1S)-1-phenylethyl]acetamide —— C22H28N4O2
2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-N-[(1S)-1-phenylethyl]acetamide
—— N-[(4S)-1-[3-(4-methoxy-3-methylphenyl)propanoyl]azepan-4-yl]-5-methylpyrazine-2-carboxamide —— C23H30N4O3
N-[(4S)-1-[3-(4-methoxy-3-methylphenyl)propanoyl]azepan-4-yl]-5-methylpyrazine-2-carboxamide
—— N-methyl-N-[(4S)-1-[2-(methylamino)pyrimidine-5-carbonyl]azepan-4-yl]-1-phenylmethanesulfonamide —— C20H27N5O3S
N-methyl-N-[(4S)-1-[2-(methylamino)pyrimidine-5-carbonyl]azepan-4-yl]-1-phenylmethanesulfonamide
—— 5-methyl-N-[(4R)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]azepan-4-yl]pyrazine-2-carboxamide —— C18H23N5O2S
5-methyl-N-[(4R)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]azepan-4-yl]pyrazine-2-carboxamide
—— 4-methyl-N-[(4S)-1-[2-(methylamino)pyrimidine-5-carbonyl]azepan-4-yl]-1,3-thiazole-5-carboxamide —— C17H22N6O2S
4-methyl-N-[(4S)-1-[2-(methylamino)pyrimidine-5-carbonyl]azepan-4-yl]-1,3-thiazole-5-carboxamide
—— N-[(4R)-1-(2,4-dimethylpyrimidine-5-carbonyl)azepan-4-yl]-3-methoxy-N-methylbenzamide —— C22H28N4O3
N-[(4R)-1-(2,4-dimethylpyrimidine-5-carbonyl)azepan-4-yl]-3-methoxy-N-methylbenzamide
—— N-methyl-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]-N-(2-pyridin-2-ylethyl)azetidine-3-carboxamide —— C19H23N5O3
N-methyl-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]-N-(2-pyridin-2-ylethyl)azetidine-3-carboxamide
—— 2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-N-[2-(2-fluorophenyl)ethyl]acetamide —— C22H27FN4O2
2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-N-[2-(2-fluorophenyl)ethyl]acetamide
—— 5-methyl-N-[(4S)-1-(1-methyl-6-oxopyridine-3-carbonyl)azepan-4-yl]pyrazine-2-carboxamide —— C19H23N5O3
5-methyl-N-[(4S)-1-(1-methyl-6-oxopyridine-3-carbonyl)azepan-4-yl]pyrazine-2-carboxamide
—— 2-[1-(2-amino-4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-N-[(1S)-1-phenylethyl]acetamide —— C21H27N5O2
2-[1-(2-amino-4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-N-[(1S)-1-phenylethyl]acetamide
—— 5-methyl-N-[(4R)-1-(2-propan-2-yloxyacetyl)azepan-4-yl]pyrazine-2-carboxamide —— C17H26N4O3
5-methyl-N-[(4R)-1-(2-propan-2-yloxyacetyl)azepan-4-yl]pyrazine-2-carboxamide
—— (3S)-N-[2-(4-chlorophenyl)ethyl]-1-[2-(methylamino)pyrimidine-5-carbonyl]pyrrolidine-3-carboxamide —— C19H22ClN5O2
(3S)-N-[2-(4-chlorophenyl)ethyl]-1-[2-(methylamino)pyrimidine-5-carbonyl]pyrrolidine-3-carboxamide
—— 5-methyl-N-[(4R)-1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]azepan-4-yl]pyrazine-2-carboxamide —— C18H24N6O3
5-methyl-N-[(4R)-1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]azepan-4-yl]pyrazine-2-carboxamide
—— 1-[4-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]-2-propan-2-yloxyethanone —— C21H32N4O3
1-[4-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]-2-propan-2-yloxyethanone
—— (3R)-N-cyclopentyl-1-(2,4-dimethylpyrimidine-5-carbonyl)pyrrolidine-3-carboxamide —— C17H24N4O2
(3R)-N-cyclopentyl-1-(2,4-dimethylpyrimidine-5-carbonyl)pyrrolidine-3-carboxamide
—— (6-methoxypyridin-3-yl)-[4-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]methanone —— C23H29N5O3
(6-methoxypyridin-3-yl)-[4-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]methanone
—— [(2S)-2-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C23H31N5O3
[(2S)-2-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— 3-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[4-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]propan-1-one —— C23H32N6O3
3-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[4-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]propan-1-one
—— [4-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]-(4-methylpyrimidin-5-yl)methanone —— C22H28N6O2
[4-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]-(4-methylpyrimidin-5-yl)methanone
—— (4-methylpyrimidin-5-yl)-[4-[(2S)-1-methylsulfonylpiperidin-2-yl]piperidin-1-yl]methanone —— C17H26N4O3S
(4-methylpyrimidin-5-yl)-[4-[(2S)-1-methylsulfonylpiperidin-2-yl]piperidin-1-yl]methanone
—— 1-[4-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]-2-propan-2-yloxyethanone —— C21H32N4O3
1-[4-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]-2-propan-2-yloxyethanone
—— Azepan-1-yl-[1-(2,4-dimethylpyrimidine-5-carbonyl)azetidin-3-yl]methanone —— C17H24N4O2
Azepan-1-yl-[1-(2,4-dimethylpyrimidine-5-carbonyl)azetidin-3-yl]methanone
—— (4-methylpyrimidin-5-yl)-[4-[(2R)-1-methylsulfonylpiperidin-2-yl]piperidin-1-yl]methanone —— C17H26N4O3S
(4-methylpyrimidin-5-yl)-[4-[(2R)-1-methylsulfonylpiperidin-2-yl]piperidin-1-yl]methanone
—— (3S)-N-cyclopentyl-1-(2,4-dimethylpyrimidine-5-carbonyl)pyrrolidine-3-carboxamide —— C17H24N4O2
(3S)-N-cyclopentyl-1-(2,4-dimethylpyrimidine-5-carbonyl)pyrrolidine-3-carboxamide
—— (5-methylpyrazin-2-yl)-[(2R)-2-[1-(4-methylthiadiazole-5-carbonyl)piperidin-4-yl]piperidin-1-yl]methanone —— C20H26N6O2S
(5-methylpyrazin-2-yl)-[(2R)-2-[1-(4-methylthiadiazole-5-carbonyl)piperidin-4-yl]piperidin-1-yl]methanone
—— [2-(methylamino)pyrimidin-5-yl]-[4-[(2R)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]piperidin-1-yl]methanone —— C21H28N6O2S
[2-(methylamino)pyrimidin-5-yl]-[4-[(2R)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]piperidin-1-yl]methanone
—— (3S)-N,3-dimethyl-1-(4-methylpyrimidine-5-carbonyl)piperidine-3-carboxamide —— C14H20N4O2
(3S)-N,3-dimethyl-1-(4-methylpyrimidine-5-carbonyl)piperidine-3-carboxamide
—— N-[2-[(2S)-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-2-yl]ethyl]methanesulfonamide —— C14H23N5O3S
N-[2-[(2S)-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-2-yl]ethyl]methanesulfonamide
—— 2-[1-(2-Propan-2-ylpyrimidine-5-carbonyl)piperidin-4-yl]acetic acid —— C15H21N3O3
2-[1-(2-Propan-2-ylpyrimidine-5-carbonyl)piperidin-4-yl]acetic acid
—— 2-(3,5-dimethylpyrazol-1-yl)-1-[4-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]ethanone —— C23H32N6O2
2-(3,5-dimethylpyrazol-1-yl)-1-[4-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]piperidin-1-yl]ethanone
—— (3R)-3-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-3-methyl-1-(2-phenylethyl)azepan-2-one —— C27H36N4O2
(3R)-3-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-3-methyl-1-(2-phenylethyl)azepan-2-one
—— 2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-N,N-dimethylacetamide —— C16H24N4O2
2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-N,N-dimethylacetamide
—— 2-methoxy-N-[2-[(2R)-1-(4-methylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl]acetamide —— C16H24N4O3
2-methoxy-N-[2-[(2R)-1-(4-methylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl]acetamide
—— (3S)-3-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]-1-(2-phenylethyl)azepan-2-one —— C25H32N4O2
(3S)-3-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]-1-(2-phenylethyl)azepan-2-one
—— (3R)-1-[2-(methylamino)pyrimidine-5-carbonyl]-N-propylpyrrolidine-3-carboxamide —— C14H21N5O2
(3R)-1-[2-(methylamino)pyrimidine-5-carbonyl]-N-propylpyrrolidine-3-carboxamide
—— (3R)-3-[1-(2-amino-4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-1-benzyl-3-methylazepan-2-one —— C25H33N5O2
(3R)-3-[1-(2-amino-4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-1-benzyl-3-methylazepan-2-one
—— (3S)-3-methyl-1-(2-phenylethyl)-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]azepan-2-one —— C25H32N4O2
(3S)-3-methyl-1-(2-phenylethyl)-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]azepan-2-one
—— (3S)-3-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-3-methyl-1-(2-phenylethyl)azepan-2-one —— C27H36N4O2
(3S)-3-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-3-methyl-1-(2-phenylethyl)azepan-2-one
—— [2-(3-fluorophenyl)-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl]-(5-methylpyrazin-2-yl)methanone —— C18H15FN4OS
[2-(3-fluorophenyl)-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridin-5-yl]-(5-methylpyrazin-2-yl)methanone
—— [(3R)-3-(imidazol-1-ylmethyl)piperidin-1-yl]-[7-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]methanone —— C23H24N6O2
[(3R)-3-(imidazol-1-ylmethyl)piperidin-1-yl]-[7-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]methanone
—— 2-morpholin-4-yl-N-[(2R)-2-morpholin-4-ylpropyl]pyrimidine-5-carboxamide —— C16H25N5O3
2-morpholin-4-yl-N-[(2R)-2-morpholin-4-ylpropyl]pyrimidine-5-carboxamide
—— 6-methyl-N-[5-[(1R)-1-phenoxyethyl]-1,3,4-thiadiazol-2-yl]-2-piperidin-1-ylpyrimidine-4-carboxamide —— C21H24N6O2S
6-methyl-N-[5-[(1R)-1-phenoxyethyl]-1,3,4-thiadiazol-2-yl]-2-piperidin-1-ylpyrimidine-4-carboxamide
—— 1-[2-[[2-methyl-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-yl]amino]ethyl]pyrrolidin-2-one —— C20H30N6O
1-[2-[[2-methyl-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-yl]amino]ethyl]pyrrolidin-2-one
—— 4-N-[(2R)-2-(4-fluorophenyl)-2-pyrrolidin-1-ylethyl]-6-(1-methylpyrazol-4-yl)pyrimidine-2,4-diamine —— C20H24FN7
4-N-[(2R)-2-(4-fluorophenyl)-2-pyrrolidin-1-ylethyl]-6-(1-methylpyrazol-4-yl)pyrimidine-2,4-diamine
—— 2-(methylamino)-N-[(2S)-2-(4-methylphenyl)-2-morpholin-4-ylethyl]pyrimidine-5-carboxamide —— C19H25N5O2
2-(methylamino)-N-[(2S)-2-(4-methylphenyl)-2-morpholin-4-ylethyl]pyrimidine-5-carboxamide
—— 1-[3-[[2-methyl-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-yl]amino]propyl]pyrrolidin-2-one —— C21H32N6O
1-[3-[[2-methyl-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-yl]amino]propyl]pyrrolidin-2-one
—— 2-(methylamino)-N-[5-[(1R)-1-phenoxyethyl]-1,3,4-thiadiazol-2-yl]pyrimidine-5-carboxamide —— C16H16N6O2S
2-(methylamino)-N-[5-[(1R)-1-phenoxyethyl]-1,3,4-thiadiazol-2-yl]pyrimidine-5-carboxamide
—— N-[(2R)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-2-(methylamino)pyrimidine-5-carboxamide —— C18H22ClN5O2
N-[(2R)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-2-(methylamino)pyrimidine-5-carboxamide