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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[[(2S)-1-amino-3-oxopropan-2-yl]amino]-2-(4-cyclopentyloxyphenyl)pyrimidine-4-carboxamide —— C19H23N5O3
6-[[(2S)-1-amino-3-oxopropan-2-yl]amino]-2-(4-cyclopentyloxyphenyl)pyrimidine-4-carboxamide
—— 2-Chloro-6-[2-(2,2-dimethyl-1,3-dioxolan-4-yl)ethylsulfonylamino]pyrimidine-4-carboxamide —— C12H17ClN4O5S
2-Chloro-6-[2-(2,2-dimethyl-1,3-dioxolan-4-yl)ethylsulfonylamino]pyrimidine-4-carboxamide
—— 6-(2-Oxopyrrolidin-3-yl)oxy-2-[4-[5-(trifluoromethyl)pyridin-2-yl]oxycyclohexyl]pyrimidine-4-carboxamide —— C21H22F3N5O4
6-(2-Oxopyrrolidin-3-yl)oxy-2-[4-[5-(trifluoromethyl)pyridin-2-yl]oxycyclohexyl]pyrimidine-4-carboxamide
—— 5-(oxazol-4-ylmethoxy)pyrazine-2-carboxylic acid —— C9H7N3O4
5-(oxazol-4-ylmethoxy)pyrazine-2-carboxylic acid
—— 2-Methyl-3-propylimidazo[1,2-b]pyridazin-6-amine —— C10H14N4
2-Methyl-3-propylimidazo[1,2-b]pyridazin-6-amine
—— 4-methyl-N-[3-(1-methylpiperidin-4-yl)propyl]pyrimidin-2-amine —— C14H24N4
4-methyl-N-[3-(1-methylpiperidin-4-yl)propyl]pyrimidin-2-amine
—— 5-(thiazol-2-ylmethoxy)pyrazine-2-carboxylic acid —— C9H7N3O3S
5-(thiazol-2-ylmethoxy)pyrazine-2-carboxylic acid
—— N-methylpropan-1-amine;N-propylimidazo[1,2-b]pyridazin-6-amine —— C13H23N5
N-methylpropan-1-amine;N-propylimidazo[1,2-b]pyridazin-6-amine
—— 2-Chloro-4-ethyl-6-fluoropyrimidine —— C6H6ClFN2
2-Chloro-4-ethyl-6-fluoropyrimidine
—— 3-[7-(3,5-dimethyl-1,2-oxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl]aniline —— C23H21N5O2
3-[7-(3,5-dimethyl-1,2-oxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl]aniline
—— 3-(1H-indol-5-yl)-6-(3,4,5-trimethoxyphenyl)imidazo[1,2-b]pyridazine —— C23H20N4O3
3-(1H-indol-5-yl)-6-(3,4,5-trimethoxyphenyl)imidazo[1,2-b]pyridazine
—— 6-Chloro-2-methyl-3-pentylimidazo[1,2-b]pyridazine —— C12H16ClN3
6-Chloro-2-methyl-3-pentylimidazo[1,2-b]pyridazine
—— N,N-dihydroxypyrazine-2-carboxamide —— C5H5N3O3
N,N-dihydroxypyrazine-2-carboxamide
—— 8-(3,4-Dimethoxyphenyl)-2-methylimidazo[1,2-b]pyridazin-6-amine —— C15H16N4O2
8-(3,4-Dimethoxyphenyl)-2-methylimidazo[1,2-b]pyridazin-6-amine
—— 2-(3-(7-(3,5-dimethylisoxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl)phenyl)-2-methyl-1-(4-morpholinopiperidine-1-yl)propan-1-one —— C36H42N6O4
2-(3-(7-(3,5-dimethylisoxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl)phenyl)-2-methyl-1-(4-morpholinopiperidine-1-yl)propan-1-one
—— 7,8-dimethyl-N-propylimidazo[1,2-b]pyridazin-6-amine —— C11H16N4
7,8-dimethyl-N-propylimidazo[1,2-b]pyridazin-6-amine
—— 2-[7-(3,5-dimethyl-1,2-oxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl]-N,N-dimethylaniline —— C25H25N5O2
2-[7-(3,5-dimethyl-1,2-oxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl]-N,N-dimethylaniline
—— 3-(5,6-dimethoxybenzo[b]thiophen-2-yl)-6-(3-((4-methylpiperazin-1-yl)methyl)phenyl)imidazo[1,2-b]pyridazine —— C28H29N5O2S
3-(5,6-dimethoxybenzo[b]thiophen-2-yl)-6-(3-((4-methylpiperazin-1-yl)methyl)phenyl)imidazo[1,2-b]pyridazine
—— 2,3-dimethyl-N-propylimidazo[1,2-b]pyridazin-6-amine —— C11H16N4
2,3-dimethyl-N-propylimidazo[1,2-b]pyridazin-6-amine
—— 2-(5-(7-(3,5-Dimethylisoxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl)-2-methoxyphenyl)propan-2-ol —— C27H28N4O4
2-(5-(7-(3,5-Dimethylisoxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl)-2-methoxyphenyl)propan-2-ol
—— 3-(2-cyanopropan-2-yl)-5-(7-(3,5-dimethylisoxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl)-N-(1-(oxetan-3-yl)piperidin-4-yl)benzamide —— C36H39N7O4
3-(2-cyanopropan-2-yl)-5-(7-(3,5-dimethylisoxazol-4-yl)-6-methoxy-2-methyl-9H-pyrimido[4,5-b]indol-4-yl)-N-(1-(oxetan-3-yl)piperidin-4-yl)benzamide
—— 1-Azabicyclo[2.2.2]octan-3-yl-[2-(4-fluoro-3-pyrimidin-5-ylphenyl)propan-2-yl]carbamic acid —— C21H25FN4O2
1-Azabicyclo[2.2.2]octan-3-yl-[2-(4-fluoro-3-pyrimidin-5-ylphenyl)propan-2-yl]carbamic acid
—— 3-[2-Methyl-5-[2-methylsulfonyl-4-(trifluoromethyl)phenyl]-3-oxopyridazin-4-yl]propane-1-sulfonic acid —— C16H17F3N2O6S2
3-[2-Methyl-5-[2-methylsulfonyl-4-(trifluoromethyl)phenyl]-3-oxopyridazin-4-yl]propane-1-sulfonic acid
—— (S)-N-(1-(5-(3-amino-1-methyl-1H-indazol-7-yl)-2-(methylthio)pyrimidin-4-yl)-2-(3,5-difluorophenyl)ethyl)-2-(3-(difluoromethyl)-4,4,7,7-tetrafluoro-4,5,6,7-tetrahydro-1H-indazol-1-yl)acetamide —— C31H26F8N8OS
(S)-N-(1-(5-(3-amino-1-methyl-1H-indazol-7-yl)-2-(methylthio)pyrimidin-4-yl)-2-(3,5-difluorophenyl)ethyl)-2-(3-(difluoromethyl)-4,4,7,7-tetrafluoro-4,5,6,7-tetrahydro-1H-indazol-1-yl)acetamide
—— N-(tert-butyl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine-2-sulfonamide —— C14H24BN3O4S
N-(tert-butyl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine-2-sulfonamide
—— 2-((3bS,4aR)-5,5-difluoro-3-(trifluoromethyl)-3b,4,4a,5-tetrahydro-1H-cyclopropa[3,4] cyclopenta[1,2-c]pyrazol-1-yl)-N-((S)-2-(3,5-difluorophenyl)-1-(2-(3-hydroxy-3-methylbut-1-yn-1-yl)-5-(3-oxoisoindolin-5-yl)pyrimidin-4-yl)ethyl)acetamide —— C35H27F7N6O3
2-((3bS,4aR)-5,5-difluoro-3-(trifluoromethyl)-3b,4,4a,5-tetrahydro-1H-cyclopropa[3,4] cyclopenta[1,2-c]pyrazol-1-yl)-N-((S)-2-(3,5-difluorophenyl)-1-(2-(3-hydroxy-3-methylbut-1-yn-1-yl)-5-(3-oxoisoindolin-5-yl)pyrimidin-4-yl)ethyl)acetamide
—— 5-[[3-(dimethylamino)propylamino]methylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C12H20N4O2S
5-[[3-(dimethylamino)propylamino]methylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5E)-1-methyl-5-[(2-piperazin-1-ylethylamino)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C12H19N5O2S
(5E)-1-methyl-5-[(2-piperazin-1-ylethylamino)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-(4-((S)-1-(2-((3bS,4aR)-5,5-difluoro-3-(trifluoromethyl)-3b,4,4a,5-tetrahydro-1H-cycloprop[3,4]cyclopenta[1,2-c]pyrazol-1-yl)acetamido)-2-(3,5-difluorophenyl)ethyl)-2-(3-hydroxy-3-methylbut-1-yn-1-yl)pyrimidin-5-yl)-2-fluorobenzamide —— C34H26F8N6O3
5-(4-((S)-1-(2-((3bS,4aR)-5,5-difluoro-3-(trifluoromethyl)-3b,4,4a,5-tetrahydro-1H-cycloprop[3,4]cyclopenta[1,2-c]pyrazol-1-yl)acetamido)-2-(3,5-difluorophenyl)ethyl)-2-(3-hydroxy-3-methylbut-1-yn-1-yl)pyrimidin-5-yl)-2-fluorobenzamide
—— 2-[2-[2-amino-6-[5-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-4-yl]anilino]ethanol —— C23H22N8O
2-[2-[2-amino-6-[5-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-4-yl]anilino]ethanol
—— 5,10-Dimethyl-11,12-diazatricyclo[7.4.0.04,6]trideca-1(13),9,11-triene —— C13H18N2
5,10-Dimethyl-11,12-diazatricyclo[7.4.0.04,6]trideca-1(13),9,11-triene
—— 2-methyl-4-[[(6-oxo-2-pyrazol-1-yl-1H-pyrimidine-5-carbonyl)amino]methyl]benzoic acid —— C17H15N5O4
2-methyl-4-[[(6-oxo-2-pyrazol-1-yl-1H-pyrimidine-5-carbonyl)amino]methyl]benzoic acid
—— 5-Ethanimidoylpyrimidine-4,6-diamine —— C6H9N5
5-Ethanimidoylpyrimidine-4,6-diamine
—— N-hydroxy-N-(2-phenylpropan-2-yl)-2-pyrazol-1-ylpyrimidine-5-carboxamide —— C17H17N5O2
N-hydroxy-N-(2-phenylpropan-2-yl)-2-pyrazol-1-ylpyrimidine-5-carboxamide
—— 3-[2-[2-amino-6-[5-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-4-yl]anilino]propanamide —— C24H23N9O
3-[2-[2-amino-6-[5-(1-methylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-4-yl]anilino]propanamide
—— 5-amino-2-[(E)-[(2Z,4Z)-hexa-2,4-dienylidene]amino]pyrimidine-4-carboxylic acid —— C11H12N4O2
5-amino-2-[(E)-[(2Z,4Z)-hexa-2,4-dienylidene]amino]pyrimidine-4-carboxylic acid
—— Methyl 4-(3-methoxypyrazin-2-yl)-2-methylpyrazole-3-carboxylate —— C11H12N4O3
Methyl 4-(3-methoxypyrazin-2-yl)-2-methylpyrazole-3-carboxylate
—— 1-(3-Cyclohexyloxy-8-thia-4,6,12-triazatricyclo[7.4.0.02,7]tridec-5-en-12-yl)ethanol —— C17H29N3O2S
1-(3-Cyclohexyloxy-8-thia-4,6,12-triazatricyclo[7.4.0.02,7]tridec-5-en-12-yl)ethanol
—— N-hydroxy-2-[4-[[(3S)-3-methyl-4-[1-(oxan-4-yl)-4-oxo-2H-pyrazolo[3,4-d]pyrimidin-6-yl]pyrrolidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide —— C26H35N9O4
N-hydroxy-2-[4-[[(3S)-3-methyl-4-[1-(oxan-4-yl)-4-oxo-2H-pyrazolo[3,4-d]pyrimidin-6-yl]pyrrolidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide
—— [(1S,3S)-3-[4-(cyclohexylamino)-6-methyl-1,4,5,6-tetrahydropyrimidin-5-yl]-4-sulfanylcyclohexyl]methanol —— C18H33N3OS
[(1S,3S)-3-[4-(cyclohexylamino)-6-methyl-1,4,5,6-tetrahydropyrimidin-5-yl]-4-sulfanylcyclohexyl]methanol
—— N-cyclopropyl-4-pyrimidin-5-yl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)benzamide —— C21H21N5O
N-cyclopropyl-4-pyrimidin-5-yl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)benzamide
—— (1S)-2-[2-cyclopropyl-6-(3,5-dimethyl-1,2,4-triazol-1-yl)pyrimidin-4-yl]cyclopropane-1-carbaldehyde —— C15H17N5O
(1S)-2-[2-cyclopropyl-6-(3,5-dimethyl-1,2,4-triazol-1-yl)pyrimidin-4-yl]cyclopropane-1-carbaldehyde
—— ethyl (1S)-2-[6-(3,5-dimethyl-1,2,4-triazol-1-yl)-2-ethylpyrimidin-4-yl]cyclopropane-1-carboxylate —— C16H21N5O2
ethyl (1S)-2-[6-(3,5-dimethyl-1,2,4-triazol-1-yl)-2-ethylpyrimidin-4-yl]cyclopropane-1-carboxylate
—— 3-(6-Dimethylboranylquinazolin-4-yl)benzamide —— C17H16BN3O
3-(6-Dimethylboranylquinazolin-4-yl)benzamide
—— (1S)-2-[6-(3,5-dimethyl-1,2,4-triazol-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]cyclopropane-1-carbaldehyde —— C13H12F3N5O
(1S)-2-[6-(3,5-dimethyl-1,2,4-triazol-1-yl)-2-(trifluoromethyl)pyrimidin-4-yl]cyclopropane-1-carbaldehyde
—— 1-[(1S)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(cyclopentylamino)pyrimidin-4-yl]pyridin-2-one —— C22H22ClFN4O2
1-[(1S)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(cyclopentylamino)pyrimidin-4-yl]pyridin-2-one
—— 1-[5-Cyclopropyl-3-[[2-[5-[3-(dimethylamino)propylsulfonyl]thiophen-2-yl]-5-ethynylpyrimidin-4-yl]amino]pyrazol-1-yl]ethanone —— C23H26N6O3S2
1-[5-Cyclopropyl-3-[[2-[5-[3-(dimethylamino)propylsulfonyl]thiophen-2-yl]-5-ethynylpyrimidin-4-yl]amino]pyrazol-1-yl]ethanone
—— (2R)-12-cyclohexyloxy-7-thia-4,9,11-triazatricyclo[6.4.0.02,6]dodec-9-ene —— C14H23N3OS
(2R)-12-cyclohexyloxy-7-thia-4,9,11-triazatricyclo[6.4.0.02,6]dodec-9-ene
—— (1S)-2-[6-(3,5-dimethyl-1,2,4-triazol-1-yl)pyridazin-4-yl]cyclopropane-1-carbaldehyde —— C12H13N5O
(1S)-2-[6-(3,5-dimethyl-1,2,4-triazol-1-yl)pyridazin-4-yl]cyclopropane-1-carbaldehyde
—— (1S,4S)-(2,5-diazabicyclo[2.2.1]hept-2-yl)-{3-[6-(4-methoxy-3-trifluoromethylphenyl)quinazolin-4-yl]phenyl}methanone 1431541-37-5 C28H23F3N4O2
(1S,4S)-(2,5-diazabicyclo[2.2.1]hept-2-yl)-{3-[6-(4-methoxy-3-trifluoromethylphenyl)quinazolin-4-yl]phenyl}methanone