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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (4R)-6-(benzenesulfonylmethyl)-4-(3,4-difluorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H18F2N2O5S
ethyl (4R)-6-(benzenesulfonylmethyl)-4-(3,4-difluorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(4-fluorophenyl)sulfonylmethyl]-4-(4-methylsulfanylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H21FN2O5S2
ethyl (4R)-6-[(4-fluorophenyl)sulfonylmethyl]-4-(4-methylsulfanylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(3,4-dimethylphenyl)sulfonylmethyl]-4-(2-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H26N2O5S
ethyl (4R)-6-[(3,4-dimethylphenyl)sulfonylmethyl]-4-(2-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(4-fluorophenyl)sulfonylmethyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H21FN2O5S
ethyl (4S)-6-[(4-fluorophenyl)sulfonylmethyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 3-(4-chlorophenyl)-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine —— C19H22ClN5O
3-(4-chlorophenyl)-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
—— ethyl (4S)-4-(3-bromophenyl)-6-[(4-fluorophenyl)sulfonylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H18BrFN2O5S
ethyl (4S)-4-(3-bromophenyl)-6-[(4-fluorophenyl)sulfonylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(4-chlorophenyl)sulfonylmethyl]-4-(2-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H21ClN2O6S
ethyl (4R)-6-[(4-chlorophenyl)sulfonylmethyl]-4-(2-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 3-(4-chlorophenyl)-N-[3-[(2S,6S)-2,6-dimethylpiperidin-1-yl]propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine —— C21H26ClN5O
3-(4-chlorophenyl)-N-[3-[(2S,6S)-2,6-dimethylpiperidin-1-yl]propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
—— ethyl (4S)-6-[(3-chloro-4-fluorophenyl)sulfonylmethyl]-4-(4-ethoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H22ClFN2O6S
ethyl (4S)-6-[(3-chloro-4-fluorophenyl)sulfonylmethyl]-4-(4-ethoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(3-chloro-4-fluorophenyl)sulfonylmethyl]-4-(3,4-difluorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H16ClF3N2O5S
ethyl (4S)-6-[(3-chloro-4-fluorophenyl)sulfonylmethyl]-4-(3,4-difluorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(4-chlorophenyl)sulfonylmethyl]-4-(2-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H21ClN2O5S
ethyl (4S)-6-[(4-chlorophenyl)sulfonylmethyl]-4-(2-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(3,4-dimethylphenyl)sulfonylmethyl]-4-(4-methylsulfanylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H26N2O5S2
ethyl (4S)-6-[(3,4-dimethylphenyl)sulfonylmethyl]-4-(4-methylsulfanylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[(2-methoxyphenyl)methylamino]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H25N3O4
ethyl (4S)-6-[[(2-methoxyphenyl)methylamino]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[4-[(2S)-butan-2-yl]piperazin-1-yl]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H32N4O3
ethyl (4R)-6-[[4-[(2S)-butan-2-yl]piperazin-1-yl]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[(3-methoxyphenyl)methylamino]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H25N3O4
ethyl (4R)-6-[[(3-methoxyphenyl)methylamino]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[cyclohexyl(furan-2-ylmethyl)amino]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H31N3O4
ethyl (4R)-6-[[cyclohexyl(furan-2-ylmethyl)amino]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-2-oxo-4-phenyl-6-[(thiophen-2-ylmethylamino)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H21N3O3S
ethyl (4S)-2-oxo-4-phenyl-6-[(thiophen-2-ylmethylamino)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[(3-methoxyphenyl)methylamino]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H25N3O4
ethyl (4S)-6-[[(3-methoxyphenyl)methylamino]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(2-methoxyethylamino)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H23N3O4
ethyl (4R)-6-[(2-methoxyethylamino)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-2-oxo-4-phenyl-6-[(pyridin-3-ylamino)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H20N4O3
ethyl (4R)-2-oxo-4-phenyl-6-[(pyridin-3-ylamino)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(4-cyclohexylpiperazin-1-yl)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H34N4O3
ethyl (4R)-6-[(4-cyclohexylpiperazin-1-yl)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[4-[(2R)-butan-2-yl]piperazin-1-yl]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H32N4O3
ethyl (4R)-6-[[4-[(2R)-butan-2-yl]piperazin-1-yl]methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(4-methylanilino)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H23N3O3
ethyl (4R)-6-[(4-methylanilino)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(3,4-dimethylanilino)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H25N3O3
ethyl (4R)-6-[(3,4-dimethylanilino)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(2-methoxyethylamino)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H23N3O4
ethyl (4S)-6-[(2-methoxyethylamino)methyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-(6-amino-1-benzyl-2,4-dioxopyrimidin-5-yl)-N-(2-methylpropyl)-3-thiophen-2-ylprop-2-enamide —— C22H24N4O3S
(E)-N-(6-amino-1-benzyl-2,4-dioxopyrimidin-5-yl)-N-(2-methylpropyl)-3-thiophen-2-ylprop-2-enamide
—— ethyl (4S)-6-[(4-cyclohexylpiperazin-1-yl)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H40N4O4
ethyl (4S)-6-[(4-cyclohexylpiperazin-1-yl)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-(6-amino-1-benzyl-2,4-dioxopyrimidin-5-yl)-N-methyl-3-thiophen-2-ylprop-2-enamide —— C19H18N4O3S
(E)-N-(6-amino-1-benzyl-2,4-dioxopyrimidin-5-yl)-N-methyl-3-thiophen-2-ylprop-2-enamide
—— ethyl (4R)-6-(morpholin-4-ylmethyl)-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H29N3O5
ethyl (4R)-6-(morpholin-4-ylmethyl)-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-(azepan-1-ylmethyl)-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H33N3O4
ethyl (4R)-6-(azepan-1-ylmethyl)-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(4-chlorophenyl)-6-[[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H25ClN4O3
ethyl (4R)-4-(4-chlorophenyl)-6-[[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(4-fluoro-N-methylanilino)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H28FN3O4
ethyl (4R)-6-[(4-fluoro-N-methylanilino)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[cyclopentyl(furan-2-ylmethyl)amino]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H35N3O5
ethyl (4S)-6-[[cyclopentyl(furan-2-ylmethyl)amino]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[4-[(2R)-butan-2-yl]piperazin-1-yl]methyl]-4-(4-fluorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H31FN4O3
ethyl (4S)-6-[[4-[(2R)-butan-2-yl]piperazin-1-yl]methyl]-4-(4-fluorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]-4-(4-fluorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H28FN3O3
ethyl (4R)-6-[[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]-4-(4-fluorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(4-benzylpiperazin-1-yl)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C28H36N4O4
ethyl (4R)-6-[(4-benzylpiperazin-1-yl)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(N-methylanilino)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H29N3O4
ethyl (4R)-6-[(N-methylanilino)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(N-ethylanilino)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H31N3O4
ethyl (4R)-6-[(N-ethylanilino)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(4-carbamoylpiperidin-1-yl)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H32N4O5
ethyl (4R)-6-[(4-carbamoylpiperidin-1-yl)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(4-chlorophenyl)-2-oxo-6-[(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H26ClN3O3
ethyl (4R)-4-(4-chlorophenyl)-2-oxo-6-[(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[furan-2-ylmethyl(2-methoxyethyl)amino]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H33N3O6
ethyl (4S)-6-[[furan-2-ylmethyl(2-methoxyethyl)amino]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(4-chlorophenyl)-6-[(N-ethylanilino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H24ClN3O3
ethyl (4R)-4-(4-chlorophenyl)-6-[(N-ethylanilino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(4-chlorophenyl)-6-[(4-fluoro-N-methylanilino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H21ClFN3O3
ethyl (4S)-4-(4-chlorophenyl)-6-[(4-fluoro-N-methylanilino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(4-chlorophenyl)-6-[[2-methoxyethyl(thiophen-2-ylmethyl)amino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H26ClN3O4S
ethyl (4R)-4-(4-chlorophenyl)-6-[[2-methoxyethyl(thiophen-2-ylmethyl)amino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(4-cyclohexylpiperazin-1-yl)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H40N4O4
ethyl (4R)-6-[(4-cyclohexylpiperazin-1-yl)methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[4-[(2S)-butan-2-yl]piperazin-1-yl]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H38N4O4
ethyl (4S)-6-[[4-[(2S)-butan-2-yl]piperazin-1-yl]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-2-oxo-6-(piperidin-1-ylmethyl)-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H31N3O4
ethyl (4S)-2-oxo-6-(piperidin-1-ylmethyl)-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(4-chlorophenyl)-6-[[cyclohexyl(furan-2-ylmethyl)amino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H30ClN3O4
ethyl (4R)-4-(4-chlorophenyl)-6-[[cyclohexyl(furan-2-ylmethyl)amino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C25H32N4O4
ethyl (4R)-6-[[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(3-methoxypropylamino)methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H27N3O4
ethyl (4R)-6-[(3-methoxypropylamino)methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate