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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(4-fluorophenyl)methyl]-4-methyl-2-[1-(1-methylimidazole-2-carbonyl)piperidin-4-yl]pyrimidine-5-carboxamide —— C23H25FN6O2
N-[(4-fluorophenyl)methyl]-4-methyl-2-[1-(1-methylimidazole-2-carbonyl)piperidin-4-yl]pyrimidine-5-carboxamide
—— N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]pyrimidine-5-carboxamide —— C24H32N4O3
N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]pyrimidine-5-carboxamide
—— cyclopentyl-[(2S)-2-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]methanone —— C22H32N4O2
cyclopentyl-[(2S)-2-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]methanone
—— N-benzyl-4-methyl-2-[(2S)-1-(1-methylimidazole-2-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide —— C23H26N6O2
N-benzyl-4-methyl-2-[(2S)-1-(1-methylimidazole-2-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide
—— [2-[(2S)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl]-4-methylpyrimidin-5-yl]-piperidin-1-ylmethanone —— C21H30N6O3S
[2-[(2S)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl]-4-methylpyrimidin-5-yl]-piperidin-1-ylmethanone
—— N-[(4-fluorophenyl)methyl]-2-[1-(2-methoxyacetyl)piperidin-4-yl]-4-methylpyrimidine-5-carboxamide —— C21H25FN4O3
N-[(4-fluorophenyl)methyl]-2-[1-(2-methoxyacetyl)piperidin-4-yl]-4-methylpyrimidine-5-carboxamide
—— 2-(4-fluorophenoxy)-1-[(2R)-2-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]ethanone —— C24H29FN4O3
2-(4-fluorophenoxy)-1-[(2R)-2-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]ethanone
—— N-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropyl)piperidin-2-yl]pyrimidine-5-carboxamide —— C22H29FN4O
N-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropyl)piperidin-2-yl]pyrimidine-5-carboxamide
—— 3-(4-fluorophenyl)-1-[(2S)-2-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]propan-1-one —— C25H31FN4O2
3-(4-fluorophenyl)-1-[(2S)-2-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]propan-1-one
—— N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide —— C24H26N6O3
N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(pyrazine-2-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide
—— N-benzyl-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide —— C24H25N5O2
N-benzyl-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide
—— 1-[(2R)-2-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]-3-phenylpropan-1-one —— C25H32N4O2
1-[(2R)-2-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]-3-phenylpropan-1-one
—— 2-[(3S)-1-[3-(4-fluorophenyl)sulfonylpropanoyl]piperidin-3-yl]-N,4-dimethylpyrimidine-5-carboxamide —— C21H25FN4O4S
2-[(3S)-1-[3-(4-fluorophenyl)sulfonylpropanoyl]piperidin-3-yl]-N,4-dimethylpyrimidine-5-carboxamide
—— [4-methyl-2-[(3S)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]pyrimidin-5-yl]-piperidin-1-ylmethanone —— C21H27N5O2S
[4-methyl-2-[(3S)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]pyrimidin-5-yl]-piperidin-1-ylmethanone
—— 2-[(3S)-1-[3-(4,6-dimethyl-2-oxopyrimidin-1-yl)propanoyl]piperidin-3-yl]-N,4-dimethylpyrimidine-5-carboxamide —— C21H28N6O3
2-[(3S)-1-[3-(4,6-dimethyl-2-oxopyrimidin-1-yl)propanoyl]piperidin-3-yl]-N,4-dimethylpyrimidine-5-carboxamide
—— N-benzyl-2-[(2R)-1-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methylpyrimidine-5-carboxamide —— C26H34N6O
N-benzyl-2-[(2R)-1-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]piperidin-2-yl]-4-methylpyrimidine-5-carboxamide
—— N-benzyl-2-[(3S)-1-[2-(4-fluorophenoxy)ethyl]piperidin-3-yl]-4-methylpyrimidine-5-carboxamide —— C26H29FN4O2
N-benzyl-2-[(3S)-1-[2-(4-fluorophenoxy)ethyl]piperidin-3-yl]-4-methylpyrimidine-5-carboxamide
—— 2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide —— C22H28N4O4
2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide
—— 2-[(3R)-1-[2-(4-fluorophenoxy)ethyl]piperidin-3-yl]-N,N,4-trimethylpyrimidine-5-carboxamide —— C21H27FN4O2
2-[(3R)-1-[2-(4-fluorophenoxy)ethyl]piperidin-3-yl]-N,N,4-trimethylpyrimidine-5-carboxamide
—— 2-[(3S)-1-(cyclopentanecarbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide —— C25H32N4O3
2-[(3S)-1-(cyclopentanecarbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide
—— [2-[(2S)-1-(1,5-dimethylpyrazol-4-yl)sulfonylpiperidin-2-yl]-4-methylpyrimidin-5-yl]-piperidin-1-ylmethanone —— C21H30N6O3S
[2-[(2S)-1-(1,5-dimethylpyrazol-4-yl)sulfonylpiperidin-2-yl]-4-methylpyrimidin-5-yl]-piperidin-1-ylmethanone
—— 2-[(3S)-1-(2-cyclopentylacetyl)piperidin-3-yl]-N-[(4-fluorophenyl)methyl]-4-methylpyrimidine-5-carboxamide —— C25H31FN4O2
2-[(3S)-1-(2-cyclopentylacetyl)piperidin-3-yl]-N-[(4-fluorophenyl)methyl]-4-methylpyrimidine-5-carboxamide
—— 2-[(2R)-1-(2-cyclopentylacetyl)piperidin-2-yl]-N-[(4-fluorophenyl)methyl]-4-methylpyrimidine-5-carboxamide —— C25H31FN4O2
2-[(2R)-1-(2-cyclopentylacetyl)piperidin-2-yl]-N-[(4-fluorophenyl)methyl]-4-methylpyrimidine-5-carboxamide
—— 2-amino-N-cyclopentyl-6-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]pyridine-3-carboxamide —— C23H30N6O2
2-amino-N-cyclopentyl-6-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]pyridine-3-carboxamide
—— N-benzyl-4-methyl-2-[(3R)-1-(1H-pyrazole-5-carbonyl)piperidin-3-yl]pyrimidine-5-carboxamide —— C22H24N6O2
N-benzyl-4-methyl-2-[(3R)-1-(1H-pyrazole-5-carbonyl)piperidin-3-yl]pyrimidine-5-carboxamide
—— 2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide —— C22H28N4O4
2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide
—— [(3R)-3-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone —— C22H27N5O2
[(3R)-3-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]-pyridin-3-ylmethanone
—— N,N,4-trimethyl-2-[(3S)-1-[4-(2-methylphenoxy)butanoyl]piperidin-3-yl]pyrimidine-5-carboxamide —— C24H32N4O3
N,N,4-trimethyl-2-[(3S)-1-[4-(2-methylphenoxy)butanoyl]piperidin-3-yl]pyrimidine-5-carboxamide
—— N-benzyl-2-[(2S)-1-(2-cyclopentylacetyl)piperidin-2-yl]-4-methylpyrimidine-5-carboxamide —— C25H32N4O2
N-benzyl-2-[(2S)-1-(2-cyclopentylacetyl)piperidin-2-yl]-4-methylpyrimidine-5-carboxamide
—— 2-[(3R)-1-(cyclopentanecarbonyl)piperidin-3-yl]-N-[(4-fluorophenyl)methyl]-4-methylpyrimidine-5-carboxamide —— C24H29FN4O2
2-[(3R)-1-(cyclopentanecarbonyl)piperidin-3-yl]-N-[(4-fluorophenyl)methyl]-4-methylpyrimidine-5-carboxamide
—— 2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide —— C22H28N4O4
2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide
—— 2-methoxy-1-[(3R)-3-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]ethanone —— C19H28N4O3
2-methoxy-1-[(3R)-3-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]ethanone
—— 2-methoxy-1-[(3S)-3-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]ethanone —— C19H28N4O3
2-methoxy-1-[(3S)-3-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]ethanone
—— 2-[(3S)-1-[4-(benzenesulfonyl)butanoyl]piperidin-3-yl]-N,4-dimethylpyrimidine-5-carboxamide —— C22H28N4O4S
2-[(3S)-1-[4-(benzenesulfonyl)butanoyl]piperidin-3-yl]-N,4-dimethylpyrimidine-5-carboxamide
—— 2-[(3R)-1-[3-(4,6-dimethyl-2-oxopyrimidin-1-yl)propanoyl]piperidin-3-yl]-N,4-dimethylpyrimidine-5-carboxamide —— C21H28N6O3
2-[(3R)-1-[3-(4,6-dimethyl-2-oxopyrimidin-1-yl)propanoyl]piperidin-3-yl]-N,4-dimethylpyrimidine-5-carboxamide
—— N-benzyl-4-methyl-2-[(2R)-1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-2-yl]pyrimidine-5-carboxamide —— C24H28N6O3
N-benzyl-4-methyl-2-[(2R)-1-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propanoyl]piperidin-2-yl]pyrimidine-5-carboxamide
—— N,N-diethyl-2-[(2S)-1-(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)piperidin-2-yl]-4-methylpyrimidine-5-carboxamide —— C22H28N6O2S
N,N-diethyl-2-[(2S)-1-(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)piperidin-2-yl]-4-methylpyrimidine-5-carboxamide
—— [4-methyl-2-[(3R)-1-morpholin-4-ylsulfonylpiperidin-3-yl]pyrimidin-5-yl]-piperidin-1-ylmethanone —— C20H31N5O4S
[4-methyl-2-[(3R)-1-morpholin-4-ylsulfonylpiperidin-3-yl]pyrimidin-5-yl]-piperidin-1-ylmethanone
—— 3-(2-methoxyphenyl)-1-[(3R)-3-[4-methyl-5-(pyrrolidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]propan-1-one —— C25H32N4O3
3-(2-methoxyphenyl)-1-[(3R)-3-[4-methyl-5-(pyrrolidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]propan-1-one
—— N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(3-methylbutanoyl)piperidin-3-yl]pyrimidine-5-carboxamide —— C24H32N4O3
N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(3-methylbutanoyl)piperidin-3-yl]pyrimidine-5-carboxamide
—— [4-methyl-2-[(3R)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]pyrimidin-5-yl]-piperidin-1-ylmethanone —— C21H27N5O2S
[4-methyl-2-[(3R)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]pyrimidin-5-yl]-piperidin-1-ylmethanone
—— 2-[(2S)-1-(cyclopentanecarbonyl)piperidin-2-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide —— C25H32N4O3
2-[(2S)-1-(cyclopentanecarbonyl)piperidin-2-yl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide
—— [2-[(3R)-1-[2-(4-fluorophenoxy)ethyl]piperidin-3-yl]-4-methylpyrimidin-5-yl]-piperidin-1-ylmethanone —— C24H31FN4O2
[2-[(3R)-1-[2-(4-fluorophenoxy)ethyl]piperidin-3-yl]-4-methylpyrimidin-5-yl]-piperidin-1-ylmethanone
—— 1-[(3S)-3-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]-4-morpholin-4-ylbutan-1-one —— C24H37N5O3
1-[(3S)-3-[4-methyl-5-(piperidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]-4-morpholin-4-ylbutan-1-one
—— [2-[(2R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl]-4-methylpyrimidin-5-yl]-piperidin-1-ylmethanone —— C21H30N6O3S
[2-[(2R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl]-4-methylpyrimidin-5-yl]-piperidin-1-ylmethanone
—— 3-[4-(dimethylamino)phenyl]-1-[(3S)-3-[4-methyl-5-(pyrrolidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]propan-1-one —— C26H35N5O2
3-[4-(dimethylamino)phenyl]-1-[(3S)-3-[4-methyl-5-(pyrrolidine-1-carbonyl)pyrimidin-2-yl]piperidin-1-yl]propan-1-one
—— N-benzyl-4-methyl-2-[(3S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]pyrimidine-5-carboxamide —— C25H30N6O2
N-benzyl-4-methyl-2-[(3S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-3-yl]pyrimidine-5-carboxamide
—— N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidine-5-carboxamide —— C25H29N5O2
N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidine-5-carboxamide
—— N-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methylpyrimidine-5-carboxamide —— C21H25FN4O3
N-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methylpyrimidine-5-carboxamide
—— [4-methyl-2-[(3R)-1-(1-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]pyrimidin-5-yl]-piperidin-1-ylmethanone —— C20H28N6O3S
[4-methyl-2-[(3R)-1-(1-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]pyrimidin-5-yl]-piperidin-1-ylmethanone