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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (1R)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-3,4-dihydro-1H-isochromene-1-carboxamide —— C24H23N5O3
(1R)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-3,4-dihydro-1H-isochromene-1-carboxamide
—— N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(3-methylphenyl)acetamide —— C23H23N5O2
N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(3-methylphenyl)acetamide
—— N-[(1S)-1-[7-(4-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(4-methoxyphenoxy)acetamide —— C22H20FN5O3
N-[(1S)-1-[7-(4-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(4-methoxyphenoxy)acetamide
—— 2-(3-fluorophenoxy)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide —— C22H20FN5O3
2-(3-fluorophenoxy)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide
—— (2R)-2-(2-fluorophenoxy)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]butanamide —— C24H24FN5O3
(2R)-2-(2-fluorophenoxy)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]butanamide
—— (2S)-2-(4-fluorophenoxy)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]propanamide —— C23H22FN5O3
(2S)-2-(4-fluorophenoxy)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]propanamide
—— (4R)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide —— C23H25N5O4
(4R)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
—— (2R)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(4-methylphenoxy)propanamide —— C24H25N5O3
(2R)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(4-methylphenoxy)propanamide
—— N-[(3R)-1-cycloheptylpiperidin-3-yl]pyrazine-2-carboxamide —— C17H26N4O
N-[(3R)-1-cycloheptylpiperidin-3-yl]pyrazine-2-carboxamide
—— N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-1,3-benzodioxole-5-carboxamide —— C22H19N5O4
N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-1,3-benzodioxole-5-carboxamide
—— N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-6-methoxy-2H-chromene-3-carboxamide —— C24H20FN5O3
N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-6-methoxy-2H-chromene-3-carboxamide
—— N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2,2-dimethylpropanamide —— C19H23N5O2
N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2,2-dimethylpropanamide
—— (3R)-3-[2-[(3S)-3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl]-2-oxoethyl]-6-methoxy-1,3-dihydroindol-2-one —— C27H27FN4O3
(3R)-3-[2-[(3S)-3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl]-2-oxoethyl]-6-methoxy-1,3-dihydroindol-2-one
—— 6-[(3S)-3-(4-methoxyanilino)piperidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C19H24N4O4
6-[(3S)-3-(4-methoxyanilino)piperidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[(3R)-3-(4-methoxyanilino)piperidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C19H24N4O4
6-[(3R)-3-(4-methoxyanilino)piperidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— N-ethyl-N-[[(3S)-1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl]methyl]-1,3-dimethyl-2,6-dioxopyrimidine-4-carboxamide —— C23H31FN4O3
N-ethyl-N-[[(3S)-1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl]methyl]-1,3-dimethyl-2,6-dioxopyrimidine-4-carboxamide
—— 6-chloro-2-[(3S)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline —— C29H23ClN4O2S
6-chloro-2-[(3S)-3-(2,3-dimethoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline
—— (5E)-5-[[2-(dimethylamino)ethylamino]methylidene]-1-[(4-fluorophenyl)methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C16H19FN4O2S
(5E)-5-[[2-(dimethylamino)ethylamino]methylidene]-1-[(4-fluorophenyl)methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— ethyl (4R)-4-(4-chlorophenyl)-6-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H20ClN5O3S
ethyl (4R)-4-(4-chlorophenyl)-6-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(4-chlorophenyl)-6-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H18ClN5O3S
ethyl (4S)-4-(4-chlorophenyl)-6-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(4-chlorophenyl)-6-[[1-(furan-2-ylmethyl)tetrazol-5-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H19ClN6O4S
ethyl (4R)-4-(4-chlorophenyl)-6-[[1-(furan-2-ylmethyl)tetrazol-5-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(4-chlorophenyl)-6-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H18ClN5O3S2
ethyl (4S)-4-(4-chlorophenyl)-6-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(2-ethoxypyridine-3-carbonyl)oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H25N3O7
ethyl (4R)-6-[(2-ethoxypyridine-3-carbonyl)oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[1-(4-chlorophenyl)cyclopropanecarbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H23ClN2O5
ethyl (4S)-6-[[1-(4-chlorophenyl)cyclopropanecarbonyl]oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(4-chlorophenyl)-2-oxo-6-[(5-propan-2-yl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H22ClN5O3S
ethyl (4R)-4-(4-chlorophenyl)-2-oxo-6-[(5-propan-2-yl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-[(2Z)-2-[(4-butoxyphenyl)methylidene]hydrazinyl]-4-phenyl-1H-pyrimidin-6-one —— C21H22N4O2
2-[(2Z)-2-[(4-butoxyphenyl)methylidene]hydrazinyl]-4-phenyl-1H-pyrimidin-6-one
—— 1,3-dimethyl-6-[[[(2S)-3-methylbutan-2-yl]amino]methyl]pyrimidine-2,4-dione —— C12H21N3O2
1,3-dimethyl-6-[[[(2S)-3-methylbutan-2-yl]amino]methyl]pyrimidine-2,4-dione
—— ethyl (4S)-4-(4-chlorophenyl)-2-oxo-6-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H24ClN5O3S
ethyl (4S)-4-(4-chlorophenyl)-2-oxo-6-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (6E)-2-benzyl-6-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H15ClN4O2S
(6E)-2-benzyl-6-[[5-(3-chlorophenyl)furan-2-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— ethyl (4R)-4-(4-chlorophenyl)-2-oxo-6-[[5-(propan-2-ylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H22ClN5O3S2
ethyl (4R)-4-(4-chlorophenyl)-2-oxo-6-[[5-(propan-2-ylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[(3,4-difluorophenyl)sulfanylmethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H16F2N2O3S2
ethyl (4R)-6-[(3,4-difluorophenyl)sulfanylmethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 6-chloro-2-[(3R)-3-[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]-5-phenyl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline —— C39H29ClN6
6-chloro-2-[(3R)-3-[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]-5-phenyl-3,4-dihydropyrazol-2-yl]-4-phenylquinazoline
—— ethyl (4S)-4-(4-chlorophenyl)-6-[[5-(3,4-dimethylphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H23ClN4O4S
ethyl (4S)-4-(4-chlorophenyl)-6-[[5-(3,4-dimethylphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(5-benzyl-4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-4-(4-chlorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H24ClN5O3S
ethyl (4S)-6-[(5-benzyl-4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-4-(4-chlorophenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H26N4O4S2
ethyl (4R)-6-[[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H26N4O4S2
ethyl (4S)-6-[[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-(4-chlorophenyl)-2-oxo-6-[(1,3,5-trimethylpyrazole-4-carbonyl)oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H23ClN4O5
ethyl (4S)-4-(4-chlorophenyl)-2-oxo-6-[(1,3,5-trimethylpyrazole-4-carbonyl)oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 4-chloro-5-[[(1R)-1-(2-methylphenyl)ethyl]amino]-2-[5-(trifluoromethyl)pyridin-2-yl]pyridazin-3-one —— C19H16ClF3N4O
4-chloro-5-[[(1R)-1-(2-methylphenyl)ethyl]amino]-2-[5-(trifluoromethyl)pyridin-2-yl]pyridazin-3-one
—— ethyl (E)-3-[1-[6-(hydroxymethyl)spiro[3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxole-2,1'-cyclohexane]-4-yl]-2,4-dioxopyrimidin-5-yl]prop-2-enoate —— C20H26N2O8
ethyl (E)-3-[1-[6-(hydroxymethyl)spiro[3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxole-2,1'-cyclohexane]-4-yl]-2,4-dioxopyrimidin-5-yl]prop-2-enoate
—— ethyl (4R)-6-[(2-chlorocyclohexene-1-carbonyl)oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H25ClN2O6
ethyl (4R)-6-[(2-chlorocyclohexene-1-carbonyl)oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(Z)-(2-methoxyphenyl)methylideneamino]-6-methyl-4-phenylquinazolin-2-amine —— C23H20N4O
N-[(Z)-(2-methoxyphenyl)methylideneamino]-6-methyl-4-phenylquinazolin-2-amine
—— ethyl (4S)-4-(4-chlorophenyl)-6-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H18ClFN4O4S
ethyl (4S)-4-(4-chlorophenyl)-6-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 4-amino-2-[(2R)-1-(4-fluoroanilino)-1-oxobutan-2-yl]sulfanylpyrimidine-5-carboxylate —— C17H19FN4O3S
ethyl 4-amino-2-[(2R)-1-(4-fluoroanilino)-1-oxobutan-2-yl]sulfanylpyrimidine-5-carboxylate
—— 6-[ethyl-[(Z)-(4-ethylphenyl)methylideneamino]amino]-3-methyl-1H-pyrimidine-2,4-dione —— C16H20N4O2
6-[ethyl-[(Z)-(4-ethylphenyl)methylideneamino]amino]-3-methyl-1H-pyrimidine-2,4-dione
—— 1-[(1S)-1-(2-bromophenyl)ethyl]-3-(pyrazine-2-carbonylamino)urea —— C14H14BrN5O2
1-[(1S)-1-(2-bromophenyl)ethyl]-3-(pyrazine-2-carbonylamino)urea
—— ethyl (4R)-6-[(5-chlorothiophene-2-carbonyl)oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H17ClN2O5S
ethyl (4R)-6-[(5-chlorothiophene-2-carbonyl)oxymethyl]-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1-[[(E)-(1-cyclohexyl-4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]amino]-3-phenylthiourea —— C18H21N5O2S2
1-[[(E)-(1-cyclohexyl-4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]amino]-3-phenylthiourea
—— (8R)-8-phenyl-10-thiophen-2-yl-2,4,5,6,7,11,12-heptazatricyclo[7.4.0.03,7]trideca-1,3,9,11-tetraen-13-one —— C16H11N7OS
(8R)-8-phenyl-10-thiophen-2-yl-2,4,5,6,7,11,12-heptazatricyclo[7.4.0.03,7]trideca-1,3,9,11-tetraen-13-one
—— 4-methyl-2-[(2E)-2-(3,5,5-trimethylcyclohex-2-en-1-ylidene)hydrazinyl]-1H-pyrimidin-6-one —— C14H20N4O
4-methyl-2-[(2E)-2-(3,5,5-trimethylcyclohex-2-en-1-ylidene)hydrazinyl]-1H-pyrimidin-6-one
—— (6E)-2-bromo-6-[[2-(4,6-diphenylpyrimidin-2-yl)hydrazinyl]methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C23H16BrN5O3
(6E)-2-bromo-6-[[2-(4,6-diphenylpyrimidin-2-yl)hydrazinyl]methylidene]-4-nitrocyclohexa-2,4-dien-1-one