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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-pyridin-4-ylmethanone —— C21H22N6O
[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-pyridin-4-ylmethanone
—— N-methyl-2-pyridin-4-yl-6-[(3R)-1-(quinolin-5-ylmethyl)piperidin-3-yl]pyrimidin-4-amine —— C25H26N6
N-methyl-2-pyridin-4-yl-6-[(3R)-1-(quinolin-5-ylmethyl)piperidin-3-yl]pyrimidin-4-amine
—— 4-[(2R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C21H24N6O
4-[(2R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]-2-pyridin-3-yl-1H-pyrimidin-6-one
—— 4-(methoxymethyl)-N-[[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]methyl]benzamide —— C20H21N5O2
4-(methoxymethyl)-N-[[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]methyl]benzamide
—— 6-[(3S)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C22H25N5O3S
6-[(3S)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[1-(4-chlorophenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C21H22ClN5O2S
6-[1-(4-chlorophenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— [2-(Dimethylamino)pyridin-4-yl]-[4-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C23H27N7O
[2-(Dimethylamino)pyridin-4-yl]-[4-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]methanone
—— 2-(4-Fluorophenoxy)-1-[4-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]ethanone —— C23H24FN5O2
2-(4-Fluorophenoxy)-1-[4-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]ethanone
—— 2-methoxy-1-[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]ethanone —— C18H23N5O2
2-methoxy-1-[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]ethanone
—— 7-[(1-methyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O
7-[(1-methyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— N-[3-(4-methylpiperazin-1-yl)propyl]-4-(1,3-thiazol-2-yl)-5-thiophen-2-ylpyrimidin-2-amine —— C19H24N6S2
N-[3-(4-methylpiperazin-1-yl)propyl]-4-(1,3-thiazol-2-yl)-5-thiophen-2-ylpyrimidin-2-amine
—— 1-[(3S)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-fluoro-4-methoxyphenyl)ethanone —— C25H28FN5O2
1-[(3S)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-fluoro-4-methoxyphenyl)ethanone
—— (3S)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-1-methyl-5-oxopyrrolidine-3-carboxamide —— C18H22N6O2
(3S)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-1-methyl-5-oxopyrrolidine-3-carboxamide
—— (3R)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-1-methyl-5-oxopyrrolidine-3-carboxamide —— C18H22N6O2
(3R)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-1-methyl-5-oxopyrrolidine-3-carboxamide
—— N-methyl-N-[[5-[(4-oxo-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-7-yl)methyl]furan-2-yl]methyl]methanesulfonamide —— C21H25N5O4S
N-methyl-N-[[5-[(4-oxo-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-7-yl)methyl]furan-2-yl]methyl]methanesulfonamide
—— 2-(dimethylamino)-N,N-dimethyl-4-[4-[[[2-(2-oxopyrrolidin-1-yl)acetyl]amino]methyl]phenyl]pyrimidine-5-carboxamide —— C22H28N6O3
2-(dimethylamino)-N,N-dimethyl-4-[4-[[[2-(2-oxopyrrolidin-1-yl)acetyl]amino]methyl]phenyl]pyrimidine-5-carboxamide
—— 2-(2,5-dimethoxyphenyl)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]acetamide —— C22H25N5O3
2-(2,5-dimethoxyphenyl)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]acetamide
—— 4-[(2R)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-2-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C22H26N6O
4-[(2R)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-2-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— Cyclopropyl-[4-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C20H25N5O
Cyclopropyl-[4-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methanone
—— 4-[(2R)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-2-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C22H26N6O
4-[(2R)-1-[[2-(dimethylamino)pyridin-3-yl]methyl]piperidin-2-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— N,N-dimethyl-6-piperidin-4-yl-2-pyridin-3-ylpyrimidin-4-amine —— C16H21N5
N,N-dimethyl-6-piperidin-4-yl-2-pyridin-3-ylpyrimidin-4-amine
—— N-[(1R)-2-[2-cyclopropyl-6-(dimethylamino)pyrimidin-4-yl]-1-phenylethyl]pyrazine-2-carboxamide —— C22H24N6O
N-[(1R)-2-[2-cyclopropyl-6-(dimethylamino)pyrimidin-4-yl]-1-phenylethyl]pyrazine-2-carboxamide
—— N-[(1S)-1-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]-2-phenylethyl]-2-pyridin-2-ylacetamide —— C26H26N6O
N-[(1S)-1-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]-2-phenylethyl]-2-pyridin-2-ylacetamide
—— 5-[(3R)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H24N6O2
5-[(3R)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— 1-[(3S)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-2-(2-fluorophenyl)ethanone —— C24H26FN5O
1-[(3S)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-2-(2-fluorophenyl)ethanone
—— 1-[(3S)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-methoxyphenyl)ethanone —— C25H29N5O2
1-[(3S)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-methoxyphenyl)ethanone
—— 1-[(3R)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-methoxyphenyl)ethanone —— C25H29N5O2
1-[(3R)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-methoxyphenyl)ethanone
—— N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-2-(2-methoxyphenyl)acetamide —— C21H23N5O2
N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-2-(2-methoxyphenyl)acetamide
—— (1S)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]cyclohex-3-ene-1-carboxamide —— C19H23N5O
(1S)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]cyclohex-3-ene-1-carboxamide
—— [(3S)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-pyridin-2-ylmethanone —— C22H24N6O
[(3S)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-pyridin-2-ylmethanone
—— 2-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methoxy]-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]acetamide —— C23H25N5O4
2-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methoxy]-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]acetamide
—— 2-cyclohexyl-1-[(3S)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]ethanone —— C24H33N5O
2-cyclohexyl-1-[(3S)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]ethanone
—— 1-[2-[(3R)-3-[2-(dimethylamino)-6-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-oxoethyl]pyrrolidin-2-one —— C23H29N5O3
1-[2-[(3R)-3-[2-(dimethylamino)-6-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-oxoethyl]pyrrolidin-2-one
—— N-[(1R)-1-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]-2-phenylethyl]-2-methoxyacetamide —— C22H25N5O2
N-[(1R)-1-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]-2-phenylethyl]-2-methoxyacetamide
—— 6-[(3R)-1-[(7-methoxy-1-benzofuran-2-yl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine —— C26H29N5O2
6-[(3R)-1-[(7-methoxy-1-benzofuran-2-yl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine
—— 4-[4-(4-fluorophenyl)-5-(1H-imidazol-2-yl)pyrimidin-2-yl]-N,N-dimethylpiperazine-1-sulfonamide —— C19H22FN7O2S
4-[4-(4-fluorophenyl)-5-(1H-imidazol-2-yl)pyrimidin-2-yl]-N,N-dimethylpiperazine-1-sulfonamide
—— 4-(2-methylfuran-3-yl)-N-[3-(4-methylpiperazin-1-yl)propyl]-5-pyridin-4-ylpyrimidin-2-amine —— C22H28N6O
4-(2-methylfuran-3-yl)-N-[3-(4-methylpiperazin-1-yl)propyl]-5-pyridin-4-ylpyrimidin-2-amine
—— N,N-dimethyl-2-pyridin-3-yl-6-(1-pyridin-3-ylsulfonylpiperidin-4-yl)pyrimidin-4-amine —— C21H24N6O2S
N,N-dimethyl-2-pyridin-3-yl-6-(1-pyridin-3-ylsulfonylpiperidin-4-yl)pyrimidin-4-amine
—— N-[(1R)-1-(4-fluorophenyl)-2-(6-oxo-2-pyridin-4-yl-1H-pyrimidin-4-yl)ethyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide —— C23H20FN5O3
N-[(1R)-1-(4-fluorophenyl)-2-(6-oxo-2-pyridin-4-yl-1H-pyrimidin-4-yl)ethyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
—— 2-(dimethylamino)-1-[(2S)-2-[4-(3-fluoroanilino)-6-pyridin-3-ylpyrimidin-2-yl]piperidin-1-yl]ethanone —— C24H27FN6O
2-(dimethylamino)-1-[(2S)-2-[4-(3-fluoroanilino)-6-pyridin-3-ylpyrimidin-2-yl]piperidin-1-yl]ethanone
—— 1,2-dimethyl-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]indole-3-carboxamide —— C24H25N5O2S
1,2-dimethyl-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]indole-3-carboxamide
—— 3,5-dimethyl-N-[(1R)-2-(6-oxo-2-propan-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]-1,2-oxazole-4-carboxamide —— C21H24N4O3
3,5-dimethyl-N-[(1R)-2-(6-oxo-2-propan-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]-1,2-oxazole-4-carboxamide
—— 3,5-dimethyl-N-[(1S)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]-1,2-oxazole-4-carboxamide —— C23H21N5O3
3,5-dimethyl-N-[(1S)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]-1,2-oxazole-4-carboxamide
—— 1,3,6-trimethyl-5-[[[(1S,6R,7S,8R)-8-phenyl-7-bicyclo[4.2.0]octanyl]amino]methyl]pyrimidine-2,4-dione —— C22H29N3O2
1,3,6-trimethyl-5-[[[(1S,6R,7S,8R)-8-phenyl-7-bicyclo[4.2.0]octanyl]amino]methyl]pyrimidine-2,4-dione
—— 2-tert-butyl-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide —— C15H21N5O
2-tert-butyl-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
—— 1,3,6-trimethyl-5-[[(3S)-3-(4-oxo-6-thiophen-2-yl-1H-pyrimidin-2-yl)piperidin-1-yl]methyl]pyrimidine-2,4-dione —— C21H25N5O3S
1,3,6-trimethyl-5-[[(3S)-3-(4-oxo-6-thiophen-2-yl-1H-pyrimidin-2-yl)piperidin-1-yl]methyl]pyrimidine-2,4-dione
—— N,N-dimethyl-4-[4-[[[(2R)-oxolane-2-carbonyl]amino]methyl]phenyl]pyrimidine-5-carboxamide —— C19H22N4O3
N,N-dimethyl-4-[4-[[[(2R)-oxolane-2-carbonyl]amino]methyl]phenyl]pyrimidine-5-carboxamide
—— N-[(1R)-2-(2-cyclopropyl-6-oxo-1H-pyrimidin-4-yl)-1-(4-fluorophenyl)ethyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide —— C21H21FN4O3
N-[(1R)-2-(2-cyclopropyl-6-oxo-1H-pyrimidin-4-yl)-1-(4-fluorophenyl)ethyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
—— 2-[1-[1-(Difluoromethyl)-3,5-dimethylpyrazol-4-yl]sulfonylazetidin-3-yl]-6-phenylpyridazin-3-one —— C19H19F2N5O3S
2-[1-[1-(Difluoromethyl)-3,5-dimethylpyrazol-4-yl]sulfonylazetidin-3-yl]-6-phenylpyridazin-3-one
—— [(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-(3,5-dimethyl-1,2-oxazol-4-yl)methanone —— C25H24N6O2
[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-(3,5-dimethyl-1,2-oxazol-4-yl)methanone