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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [[(2R,3S,4R,5S)-5-(2,4-dioxo-1H-pyrimidin-5-yl)-3,4-dihydroxythiolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate —— C9H15N2O14P3S
[[(2R,3S,4R,5S)-5-(2,4-dioxo-1H-pyrimidin-5-yl)-3,4-dihydroxythiolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
—— 3-(2-cyanopropan-2-yl)-N-[5-[2-(ethylamino)-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]benzamide —— C27H31N7O2
3-(2-cyanopropan-2-yl)-N-[5-[2-(ethylamino)-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]benzamide
—— N-[5-(6-ethoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]-2-(trifluoromethyl)pyridine-4-carboxamide —— C23H23F3N6O3
N-[5-(6-ethoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]-2-(trifluoromethyl)pyridine-4-carboxamide
—— 5-Methyl-3-(5-methyl-1,2,4-oxadiazol-3-yl)pyrazin-2-amine —— C8H9N5O
5-Methyl-3-(5-methyl-1,2,4-oxadiazol-3-yl)pyrazin-2-amine
—— Azane;2,5-dipyridin-4-ylpyrimidin-4-amine —— C14H14N6
Azane;2,5-dipyridin-4-ylpyrimidin-4-amine
—— [8-[2-Fluoro-4-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7,8-dihydropurin-9-yl]carbamic acid —— C20H10F10N6O2
[8-[2-Fluoro-4-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7,8-dihydropurin-9-yl]carbamic acid
—— N-[2-methyl-5-[4-(4-oxo-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-2-yl)pyrimidin-2-yl]pyridin-3-yl]prop-2-enamide —— C20H18N6O2
N-[2-methyl-5-[4-(4-oxo-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-2-yl)pyrimidin-2-yl]pyridin-3-yl]prop-2-enamide
—— 3-(1H-tetrazol-1-yl)-6-vinylpyridazine —— C7H6N6
3-(1H-tetrazol-1-yl)-6-vinylpyridazine
—— 2-(2-(1H-imidazol-1-yl)ethyl)-6-(trifluoromethyl)pyrimidine-4,5-diamine —— C10H11F3N6
2-(2-(1H-imidazol-1-yl)ethyl)-6-(trifluoromethyl)pyrimidine-4,5-diamine
—— 3-[(Z)-prop-1-enyl]-6-(tetrazol-1-yl)pyridazine —— C8H8N6
3-[(Z)-prop-1-enyl]-6-(tetrazol-1-yl)pyridazine
—— N-[6-methyl-5-[5-morpholin-4-yl-6-(oxan-4-yloxy)pyridazin-3-yl]pyridin-3-yl]-6-(trifluoromethyl)pyridazine-4-carboxamide —— C25H26F3N7O4
N-[6-methyl-5-[5-morpholin-4-yl-6-(oxan-4-yloxy)pyridazin-3-yl]pyridin-3-yl]-6-(trifluoromethyl)pyridazine-4-carboxamide
—— 2-(1,1-difluoroethyl)-N-[6-methyl-5-(1-methyl-5-morpholin-4-yl-6-oxopyridazin-3-yl)pyridin-3-yl]pyridine-4-carboxamide —— C23H24F2N6O3
2-(1,1-difluoroethyl)-N-[6-methyl-5-(1-methyl-5-morpholin-4-yl-6-oxopyridazin-3-yl)pyridin-3-yl]pyridine-4-carboxamide
—— 6-methyl-7-(1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)ethyl)pyrrolo[1,2-b]pyridazine-5-carboxylic acid —— C18H22F3N3O2
6-methyl-7-(1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)ethyl)pyrrolo[1,2-b]pyridazine-5-carboxylic acid
—— 2-(6-(1H-tetrazol-1-yl)pyridazin-3-yl)propanal —— C8H8N6O
2-(6-(1H-tetrazol-1-yl)pyridazin-3-yl)propanal
—— N-[5-[2-(2-hydroxyethylamino)-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]-3-(trifluoromethyl)benzamide —— C24H25F3N6O3
N-[5-[2-(2-hydroxyethylamino)-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]-3-(trifluoromethyl)benzamide
—— [8-[2-Methoxy-4-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-3-yl]purin-9-yl]carbamic acid —— C21H11F9N6O3
[8-[2-Methoxy-4-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-3-yl]purin-9-yl]carbamic acid
—— 2-(1,1-difluoropropyl)-N-[6-methyl-5-(1-methyl-5-morpholin-4-yl-6-oxopyridazin-3-yl)pyridin-3-yl]pyridine-4-carboxamide —— C24H26F2N6O3
2-(1,1-difluoropropyl)-N-[6-methyl-5-(1-methyl-5-morpholin-4-yl-6-oxopyridazin-3-yl)pyridin-3-yl]pyridine-4-carboxamide
—— 6-(2-cyanopropan-2-yl)pyridazine-4-carboxylic acid —— C9H9N3O2
6-(2-cyanopropan-2-yl)pyridazine-4-carboxylic acid
—— N-[5-[2-[[(2S)-1-hydroxypropan-2-yl]amino]-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]-3-(trifluoromethyl)benzamide —— C25H27F3N6O3
N-[5-[2-[[(2S)-1-hydroxypropan-2-yl]amino]-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]-3-(trifluoromethyl)benzamide
—— N-[5-[2-(1-hydroxypropan-2-ylamino)-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]-3-(trifluoromethyl)benzamide —— C25H27F3N6O3
N-[5-[2-(1-hydroxypropan-2-ylamino)-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]-3-(trifluoromethyl)benzamide
—— 2-(Hexylamino)-4-(3-pyrimidin-2-ylanilino)pyrimidine-5-carboxamide —— C21H25N7O
2-(Hexylamino)-4-(3-pyrimidin-2-ylanilino)pyrimidine-5-carboxamide
—— 2-(difluoromethyl)-N-[6-methyl-5-(1-methyl-5-morpholin-4-yl-6-oxopyridazin-3-yl)pyridin-3-yl]pyridine-4-carboxamide —— C22H22F2N6O3
2-(difluoromethyl)-N-[6-methyl-5-(1-methyl-5-morpholin-4-yl-6-oxopyridazin-3-yl)pyridin-3-yl]pyridine-4-carboxamide
—— 5-(azidomethyl)-1-[2-[[(1S)-1-[2-(4-chlorophenyl)-1,3-thiazol-5-yl]ethyl]amino]-5-fluoropyrimidin-4-yl]pyrrolidin-2-one —— C20H18ClFN8OS
5-(azidomethyl)-1-[2-[[(1S)-1-[2-(4-chlorophenyl)-1,3-thiazol-5-yl]ethyl]amino]-5-fluoropyrimidin-4-yl]pyrrolidin-2-one
—— [(3S)-1-[2-[[(1S)-1-[5-(4-chlorophenyl)-1,2-oxazol-3-yl]ethyl]amino]pyrimidin-4-yl]-5-oxopyrrolidin-3-yl]carbamic acid —— C20H19ClN6O4
[(3S)-1-[2-[[(1S)-1-[5-(4-chlorophenyl)-1,2-oxazol-3-yl]ethyl]amino]pyrimidin-4-yl]-5-oxopyrrolidin-3-yl]carbamic acid
—— (5S)-1-(2,6-dichloropyrimidin-4-yl)-5-methylpyrrolidin-2-one —— C9H9Cl2N3O
(5S)-1-(2,6-dichloropyrimidin-4-yl)-5-methylpyrrolidin-2-one
—— 5-[[Tert-butyl(dimethyl)silyl]oxymethyl]-1-(2,5-difluoropyrimidin-4-yl)pyrrolidin-2-one —— C15H23F2N3O2Si
5-[[Tert-butyl(dimethyl)silyl]oxymethyl]-1-(2,5-difluoropyrimidin-4-yl)pyrrolidin-2-one
—— 1-(2-(((S)-1-(5-chloro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-5-methylpyrrolidin-2-one —— C18H18ClF4N5O2
1-(2-(((S)-1-(5-chloro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-5-methylpyrrolidin-2-one
—— 8-(2-chloro-5-(trifluoromethyl)phenyl)-6-(trifluoromethyl)-2-(6-(trifluoromethyl)pyridin-3-yl)-9H-purin-9-amine —— C19H8ClF9N6
8-(2-chloro-5-(trifluoromethyl)phenyl)-6-(trifluoromethyl)-2-(6-(trifluoromethyl)pyridin-3-yl)-9H-purin-9-amine
—— N-(2-phenyl-2-trimethylsilyloxyethyl)-1-pyrimidin-2-ylmethanimine —— C16H21N3OSi
N-(2-phenyl-2-trimethylsilyloxyethyl)-1-pyrimidin-2-ylmethanimine
—— [1-[2-[[(1S)-1-[5-(4-chlorophenyl)-1,2-oxazol-3-yl]ethyl]amino]pyrimidin-4-yl]-5-oxopyrrolidin-3-yl]carbamic acid —— C20H19ClN6O4
[1-[2-[[(1S)-1-[5-(4-chlorophenyl)-1,2-oxazol-3-yl]ethyl]amino]pyrimidin-4-yl]-5-oxopyrrolidin-3-yl]carbamic acid
—— (R)-1-(2-chloro-5-fluoropyrimidin-4-yl)-4-hydroxypyrrolidin-2-one —— C8H7ClFN3O2
(R)-1-(2-chloro-5-fluoropyrimidin-4-yl)-4-hydroxypyrrolidin-2-one
—— [8-[2-Chloro-5-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-3-yl]purin-9-yl]carbamic acid —— C20H8ClF9N6O2
[8-[2-Chloro-5-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-3-yl]purin-9-yl]carbamic acid
—— 8-(2-chloro-5-(trifluoromethyl)phenyl)-N-methyl-6-(trifluoromethyl)-2-(6-(trifluoromethyl)pyridin-3-yl)-9H-purin-9-amine —— C20H10ClF9N6
8-(2-chloro-5-(trifluoromethyl)phenyl)-N-methyl-6-(trifluoromethyl)-2-(6-(trifluoromethyl)pyridin-3-yl)-9H-purin-9-amine
—— [[5-Amino-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]amino]-methylcarbamic acid —— C13H10F6N6O2
[[5-Amino-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-3-yl]pyrimidin-4-yl]amino]-methylcarbamic acid
—— [8-[2-Methoxy-4-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-3-yl]purin-9-yl]-methylcarbamic acid —— C22H13F9N6O3
[8-[2-Methoxy-4-(trifluoromethyl)phenyl]-6-(trifluoromethyl)-2-[6-(trifluoromethyl)pyridin-3-yl]purin-9-yl]-methylcarbamic acid
—— [1-[2-[[(1S)-1-[2-(4-chlorophenyl)-1,3-thiazol-5-yl]ethyl]amino]pyrimidin-4-yl]-5-oxopyrrolidin-3-yl]carbamic acid —— C20H19ClN6O3S
[1-[2-[[(1S)-1-[2-(4-chlorophenyl)-1,3-thiazol-5-yl]ethyl]amino]pyrimidin-4-yl]-5-oxopyrrolidin-3-yl]carbamic acid
—— 5,5-Dimethyl-1-[2-(1-phenylethylamino)pyrimidin-4-yl]pyrrolidin-2-one —— C18H22N4O
5,5-Dimethyl-1-[2-(1-phenylethylamino)pyrimidin-4-yl]pyrrolidin-2-one
—— 3-(difluoromethyl)-N-[5-(6-ethoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]benzamide —— C24H25F2N5O3
3-(difluoromethyl)-N-[5-(6-ethoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]benzamide
—— methyl 2-chloro-5,6-dimethylpyrimidine-4-carboxylate —— C8H9ClN2O2
methyl 2-chloro-5,6-dimethylpyrimidine-4-carboxylate
—— 8-(2-methoxy-4-(trifluoromethyl)phenyl)-6-(trifluoromethyl)-2-(6-(trifluoromethyl)pyridin-3-yl)-9H-purin-9-amine —— C20H11F9N6O
8-(2-methoxy-4-(trifluoromethyl)phenyl)-6-(trifluoromethyl)-2-(6-(trifluoromethyl)pyridin-3-yl)-9H-purin-9-amine
—— N-[6-methyl-5-[2-(4-methyl-2-oxo-1,3-oxazolidin-3-yl)-6-morpholin-4-ylpyrimidin-4-yl]pyridin-3-yl]-3-(trifluoromethyl)benzamide —— C26H25F3N6O4
N-[6-methyl-5-[2-(4-methyl-2-oxo-1,3-oxazolidin-3-yl)-6-morpholin-4-ylpyrimidin-4-yl]pyridin-3-yl]-3-(trifluoromethyl)benzamide
—— 2-(5-Methylpyridazin-3-yl)acetonitrile —— C7H7N3
2-(5-Methylpyridazin-3-yl)acetonitrile
—— Methyl 6-amino-2-(2-carbonofluoridoylphenyl)-5-methoxypyrimidine-4-carboxylate —— C14H12FN3O4
Methyl 6-amino-2-(2-carbonofluoridoylphenyl)-5-methoxypyrimidine-4-carboxylate
—— 6-Methyl-5-(6-(methylsulfonyl)-5-morpholinopyridazin-3-yl)pyridin-3-amine —— C15H19N5O3S
6-Methyl-5-(6-(methylsulfonyl)-5-morpholinopyridazin-3-yl)pyridin-3-amine
—— 2-(1,1-difluoroethyl)-N-[5-(6-methoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]pyridine-4-carboxamide —— C23H24F2N6O3
2-(1,1-difluoroethyl)-N-[5-(6-methoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]pyridine-4-carboxamide
—— 3-(difluoromethyl)-N-[5-(6-methoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]benzamide —— C23H23F2N5O3
3-(difluoromethyl)-N-[5-(6-methoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]benzamide
—— N-[5-(6-ethoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]-4-(hydroxymethyl)-3-(trifluoromethyl)benzamide —— C25H26F3N5O4
N-[5-(6-ethoxy-5-morpholin-4-ylpyridazin-3-yl)-6-methylpyridin-3-yl]-4-(hydroxymethyl)-3-(trifluoromethyl)benzamide
—— N-[5-[2-[[(2R)-2-hydroxypropyl]amino]-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]-3-(trifluoromethyl)benzamide —— C25H27F3N6O3
N-[5-[2-[[(2R)-2-hydroxypropyl]amino]-6-morpholin-4-ylpyrimidin-4-yl]-6-methylpyridin-3-yl]-3-(trifluoromethyl)benzamide
—— 3-(5-Methoxy-6-morpholin-4-ylpyrazin-2-yl)-4-methylaniline —— C16H20N4O2
3-(5-Methoxy-6-morpholin-4-ylpyrazin-2-yl)-4-methylaniline
—— 2-N-(cyclopropylmethyl)pyrimido[5,4-d]pyrimidine-2,4,6,8-tetramine —— C10H14N8
2-N-(cyclopropylmethyl)pyrimido[5,4-d]pyrimidine-2,4,6,8-tetramine