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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(1S)-1-[7-(4-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide —— C23H22FN5O2
N-[(1S)-1-[7-(4-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
—— N-[[4-[2-cyclopropyl-5-(dimethylcarbamoyl)pyrimidin-4-yl]phenyl]methyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide —— C23H25N5O3
N-[[4-[2-cyclopropyl-5-(dimethylcarbamoyl)pyrimidin-4-yl]phenyl]methyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
—— 4-[(3S)-1-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-6-one —— C22H29N5OS
4-[(3S)-1-[(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-6-one
—— 2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)-N-[(1-methylimidazol-2-yl)methyl]acetamide —— C13H17N5O2
2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)-N-[(1-methylimidazol-2-yl)methyl]acetamide
—— 2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(1R)-2-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]acetamide —— C24H24N6O2
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(1R)-2-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]acetamide
—— 2,3-dimethyl-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-7-carboxamide —— C24H25N5O2S
2,3-dimethyl-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-7-carboxamide
—— (3-ethylimidazol-4-yl)-[4-(2-fluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone —— C24H22FN7O
(3-ethylimidazol-4-yl)-[4-(2-fluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone
—— [(2R)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-(3,5-dimethyl-1,2-oxazol-4-yl)methanone —— C25H24N6O2
[(2R)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-(3,5-dimethyl-1,2-oxazol-4-yl)methanone
—— (3-ethylimidazol-4-yl)-[4-(3-fluoroanilino)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone —— C24H22FN7O
(3-ethylimidazol-4-yl)-[4-(3-fluoroanilino)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone
—— (2R)-N-cyclooctyl-2-[6-oxo-3-(1,3,5-trimethylpyrazol-4-yl)pyridazin-1-yl]propanamide —— C21H31N5O2
(2R)-N-cyclooctyl-2-[6-oxo-3-(1,3,5-trimethylpyrazol-4-yl)pyridazin-1-yl]propanamide
—— 4-fluoro-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-2-carboxamide —— C22H20FN5O2S
4-fluoro-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-2-carboxamide
—— N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]cyclopentanecarboxamide —— C19H24N4O2S
N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]cyclopentanecarboxamide
—— N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]pyridine-3-carboxamide —— C19H19N5O2S
N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]pyridine-3-carboxamide
—— (3S)-N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-1,1-dioxothiolane-3-carboxamide —— C18H18FN5O3S
(3S)-N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-1,1-dioxothiolane-3-carboxamide
—— N-[(1R)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-3-methoxypropanamide —— C17H18FN5O2
N-[(1R)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-3-methoxypropanamide
—— 2-(4-methoxyphenoxy)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide —— C23H23N5O4
2-(4-methoxyphenoxy)-N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide
—— N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]cyclopentanecarboxamide —— C19H24N4O2S
N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]cyclopentanecarboxamide
—— 2-[(2R)-1-[3-(3,5-dimethylpyrazol-1-yl)propanoyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C21H24N6O2
2-[(2R)-1-[3-(3,5-dimethylpyrazol-1-yl)propanoyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— N-[(1R)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(4-methoxyphenyl)acetamide —— C22H20FN5O2
N-[(1R)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(4-methoxyphenyl)acetamide
—— N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]-1,3-benzodioxole-5-carboxamide —— C21H20N4O4S
N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]-1,3-benzodioxole-5-carboxamide
—— 2-(2-fluorophenyl)-N-[(1S)-1-[7-(4-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide —— C21H17F2N5O
2-(2-fluorophenyl)-N-[(1S)-1-[7-(4-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide
—— N-[(1S)-1-[7-(4-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(3-methoxyphenyl)acetamide —— C22H20FN5O2
N-[(1S)-1-[7-(4-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(3-methoxyphenyl)acetamide
—— N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]pyridine-4-carboxamide —— C19H19N5O2S
N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]pyridine-4-carboxamide
—— N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]pyridine-2-carboxamide —— C19H19N5O2S
N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]pyridine-2-carboxamide
—— 2-(4-fluorophenyl)-N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide —— C21H17F2N5O
2-(4-fluorophenyl)-N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide
—— N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-5-methoxythiophene-2-carboxamide —— C19H16FN5O2S
N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-5-methoxythiophene-2-carboxamide
—— N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C22H24N4O2S2
N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]pyridine-4-carboxamide —— C19H19N5O2S
N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]pyridine-4-carboxamide
—— 2-(4-methoxy-3-methylphenyl)-N-[(1R)-2-methyl-1-(6-oxo-2-pyridin-4-yl-1H-pyrimidin-4-yl)propyl]acetamide —— C23H26N4O3
2-(4-methoxy-3-methylphenyl)-N-[(1R)-2-methyl-1-(6-oxo-2-pyridin-4-yl-1H-pyrimidin-4-yl)propyl]acetamide
—— 3-(4,6-dimethyl-2-oxopyrimidin-1-yl)-N-[(1R)-1-pyridin-3-yl-2-thiophen-3-ylethyl]propanamide —— C20H22N4O2S
3-(4,6-dimethyl-2-oxopyrimidin-1-yl)-N-[(1R)-1-pyridin-3-yl-2-thiophen-3-ylethyl]propanamide
—— 2-[(3S)-1-(2-methoxypyrimidine-5-carbonyl)pyrrolidin-3-yl]-4-pyridin-4-yl-1H-pyrimidin-6-one —— C19H18N6O3
2-[(3S)-1-(2-methoxypyrimidine-5-carbonyl)pyrrolidin-3-yl]-4-pyridin-4-yl-1H-pyrimidin-6-one
—— 2-(2-methoxyphenoxy)-N-[(1S)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide —— C23H23N5O4
2-(2-methoxyphenoxy)-N-[(1S)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]acetamide
—— 7-[(2-methoxyphenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C21H22N4O2
7-[(2-methoxyphenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 2-(4,6-dimethyl-2-oxopyrimidin-1-yl)-N-[(2R)-2-(4-methylpiperidin-1-yl)-2-phenylethyl]acetamide —— C22H30N4O2
2-(4,6-dimethyl-2-oxopyrimidin-1-yl)-N-[(2R)-2-(4-methylpiperidin-1-yl)-2-phenylethyl]acetamide
—— [(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-(5-methylthiophen-3-yl)methanone —— C25H23N5OS
[(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-(5-methylthiophen-3-yl)methanone
—— [(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-(5-methylthiophen-3-yl)methanone —— C21H23N5OS
[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-(5-methylthiophen-3-yl)methanone
—— 6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one —— C19H21N5O2S
6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one
—— 2-(4,6-dimethyl-2-oxopyrimidin-1-yl)-N-[(1R)-1-pyridin-2-yl-2-thiophen-3-ylethyl]acetamide —— C19H20N4O2S
2-(4,6-dimethyl-2-oxopyrimidin-1-yl)-N-[(1R)-1-pyridin-2-yl-2-thiophen-3-ylethyl]acetamide
—— 2-(4,6-dimethyl-2-oxopyrimidin-1-yl)-N-[(1S)-1-pyridin-2-yl-2-thiophen-3-ylethyl]acetamide —— C19H20N4O2S
2-(4,6-dimethyl-2-oxopyrimidin-1-yl)-N-[(1S)-1-pyridin-2-yl-2-thiophen-3-ylethyl]acetamide
—— 2-(4-methoxy-3-methylphenyl)-N-[[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]methyl]acetamide —— C21H23N5O2
2-(4-methoxy-3-methylphenyl)-N-[[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]methyl]acetamide
—— N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-3-phenylpropanamide —— C23H23N5O2
N-[(1R)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-3-phenylpropanamide
—— 7-[(2-Methyl-4-morpholin-4-ylphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27N5O2
7-[(2-Methyl-4-morpholin-4-ylphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 6-fluoro-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-2-carboxamide —— C22H20FN5O2S
6-fluoro-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-2-carboxamide
—— 4-[(3R)-1-[2-(2-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C22H22N4O3
4-[(3R)-1-[2-(2-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 4-[(3R)-1-[(2S)-2-(3,5-dimethylphenoxy)propanoyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C24H26N4O3
4-[(3R)-1-[(2S)-2-(3,5-dimethylphenoxy)propanoyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 4-[(3S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C23H26N4O2
4-[(3S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 4-[(3S)-1-[2-(2-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C22H22N4O3
4-[(3S)-1-[2-(2-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 4-[(3S)-1-[2-(2-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C22H22N4O3
4-[(3S)-1-[2-(2-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— 7-[(2,5-Dimethyl-1-pyridin-3-ylpyrrol-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[(2,5-Dimethyl-1-pyridin-3-ylpyrrol-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-[(3S)-1-[(2,3-dimethoxyphenyl)methyl]pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C22H24N4O3
2-[(3S)-1-[(2,3-dimethoxyphenyl)methyl]pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one