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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[(3R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C23H26N4O2
4-[(3R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— 2-[(3R)-1-[(2,3-dimethoxyphenyl)methyl]pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C22H24N4O3
2-[(3R)-1-[(2,3-dimethoxyphenyl)methyl]pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— 5,6-dimethyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C23H21N5O3
5,6-dimethyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— 2-[(3S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C23H26N4O2
2-[(3S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— 7-[(2,6-dimethoxyphenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C22H24N4O3
7-[(2,6-dimethoxyphenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 4,6-dimethyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C23H21N5O3
4,6-dimethyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— 4-methyl-2-[2-oxo-2-[(3R)-3-(2-pyridin-3-ylpyrimidin-4-yl)piperidin-1-yl]ethyl]phthalazin-1-one —— C25H24N6O2
4-methyl-2-[2-oxo-2-[(3R)-3-(2-pyridin-3-ylpyrimidin-4-yl)piperidin-1-yl]ethyl]phthalazin-1-one
—— (7-fluoro-3-methyl-1-benzofuran-2-yl)-[(3R)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C25H24FN5O2
(7-fluoro-3-methyl-1-benzofuran-2-yl)-[(3R)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]methanone
—— 4-methyl-2-[2-oxo-2-[(3S)-3-(2-pyridin-3-ylpyrimidin-4-yl)piperidin-1-yl]ethyl]phthalazin-1-one —— C25H24N6O2
4-methyl-2-[2-oxo-2-[(3S)-3-(2-pyridin-3-ylpyrimidin-4-yl)piperidin-1-yl]ethyl]phthalazin-1-one
—— 7-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H23N5O2
7-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-[(2S)-1-[(3-methoxyphenyl)methyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C21H22N4O2
2-[(2S)-1-[(3-methoxyphenyl)methyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— (2-tert-butylpyrimidin-5-yl)-[(2R)-2-[5-(4-methyl-1,3-thiazol-5-yl)-1,3,4-oxadiazol-2-yl]piperidin-1-yl]methanone —— C20H24N6O2S
(2-tert-butylpyrimidin-5-yl)-[(2R)-2-[5-(4-methyl-1,3-thiazol-5-yl)-1,3,4-oxadiazol-2-yl]piperidin-1-yl]methanone
—— 2-[1-[3-(3-Methoxyphenyl)propanoyl]azetidin-3-yl]-6-phenylpyridazin-3-one —— C23H23N3O3
2-[1-[3-(3-Methoxyphenyl)propanoyl]azetidin-3-yl]-6-phenylpyridazin-3-one
—— 5-(4-fluorophenyl)-4-(4-methyl-1,3-thiazol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine —— C20H16FN5S
5-(4-fluorophenyl)-4-(4-methyl-1,3-thiazol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
—— 6-methoxy-N-[(1S)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]pyridine-3-carboxamide —— C24H21N5O3
6-methoxy-N-[(1S)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]pyridine-3-carboxamide
—— 5-(4-fluorophenyl)-N-(2-methoxyethyl)-4-(4-methyl-1,3-thiazol-5-yl)pyrimidin-2-amine —— C17H17FN4OS
5-(4-fluorophenyl)-N-(2-methoxyethyl)-4-(4-methyl-1,3-thiazol-5-yl)pyrimidin-2-amine
—— N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-4-methyl-1,3-thiazole-5-carboxamide —— C20H21N5OS
N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-4-methyl-1,3-thiazole-5-carboxamide
—— 2-[(3S)-1-(5-chloro-2-methoxybenzoyl)pyrrolidin-3-yl]-4-(2-methoxypyridin-3-yl)-1H-pyrimidin-6-one —— C22H21ClN4O4
2-[(3S)-1-(5-chloro-2-methoxybenzoyl)pyrrolidin-3-yl]-4-(2-methoxypyridin-3-yl)-1H-pyrimidin-6-one
—— 4-methyl-N-[[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenyl]methyl]-1,3-thiazole-5-carboxamide —— C18H13F3N6OS
4-methyl-N-[[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenyl]methyl]-1,3-thiazole-5-carboxamide
—— 2-[(2R)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C18H18N6O3
2-[(2R)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— 4-[5-(2-aminoethyl)-4-methyl-1,3-thiazol-2-yl]-5-(2-fluorophenyl)-N-[(1R)-1-phenylethyl]pyrimidin-2-amine —— C24H24FN5S
4-[5-(2-aminoethyl)-4-methyl-1,3-thiazol-2-yl]-5-(2-fluorophenyl)-N-[(1R)-1-phenylethyl]pyrimidin-2-amine
—— 4-[(3S)-1-[2-(3,4-dimethoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C23H24N4O4
4-[(3S)-1-[2-(3,4-dimethoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— 5-(4-fluorophenyl)-4-(4-methyl-1,3-thiazol-5-yl)-N-(3-propan-2-yloxypropyl)pyrimidin-2-amine —— C20H23FN4OS
5-(4-fluorophenyl)-4-(4-methyl-1,3-thiazol-5-yl)-N-(3-propan-2-yloxypropyl)pyrimidin-2-amine
—— 4-pyridin-3-yl-2-[(2S)-1-[3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrimidin-6-one —— C22H26N6O2
4-pyridin-3-yl-2-[(2S)-1-[3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrimidin-6-one
—— [4-(3-fluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-(4-methyl-1,2,5-oxadiazol-3-yl)methanone —— C22H18FN7O2
[4-(3-fluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-(4-methyl-1,2,5-oxadiazol-3-yl)methanone
—— 5-[4-[(2,3-Difluorophenyl)methyl]piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-3-ylpyrimidine —— C21H21F2N5O2S
5-[4-[(2,3-Difluorophenyl)methyl]piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-3-ylpyrimidine
—— 6-[(3R)-1-[(1-ethenyl-5-methylpyrazol-4-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one —— C20H23N5OS
6-[(3R)-1-[(1-ethenyl-5-methylpyrazol-4-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one
—— 5-[4-[(3,4-Difluorophenyl)methyl]piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-4-ylpyrimidine —— C21H21F2N5O2S
5-[4-[(3,4-Difluorophenyl)methyl]piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-4-ylpyrimidine
—— 5-[4-[(2-Fluorophenyl)methyl]piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-3-ylpyrimidine —— C21H22FN5O2S
5-[4-[(2-Fluorophenyl)methyl]piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-3-ylpyrimidine
—— 4-pyridin-3-yl-2-[(2S)-1-[2-(3,4,5-trimethylpyrazol-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrimidin-6-one —— C21H24N6O2
4-pyridin-3-yl-2-[(2S)-1-[2-(3,4,5-trimethylpyrazol-1-yl)acetyl]pyrrolidin-2-yl]-1H-pyrimidin-6-one
—— N-[[4-[2-(dimethylamino)-5-(3,4-dimethyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]cyclohexanecarboxamide —— C25H31N5O2
N-[[4-[2-(dimethylamino)-5-(3,4-dimethyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]cyclohexanecarboxamide
—— 3-methyl-5-pyridin-3-yl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C16H12N4OS
3-methyl-5-pyridin-3-yl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— [4-(4,5-Dimethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-pyrazin-2-ylmethanone —— C20H26N6O2
[4-(4,5-Dimethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-pyrazin-2-ylmethanone
—— 2-(4-methoxyphenyl)-N-[[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenyl]methyl]acetamide —— C22H18F3N5O2
2-(4-methoxyphenyl)-N-[[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenyl]methyl]acetamide
—— 5-[4-(3,6-dihydro-2H-pyran-5-ylmethyl)piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-2-ylpyrimidine —— C20H25N5O3S
5-[4-(3,6-dihydro-2H-pyran-5-ylmethyl)piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-2-ylpyrimidine
—— 6-[(6-Methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]-2-pyridin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H18N6OS
6-[(6-Methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]-2-pyridin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 2-[(2R)-1-[3-(4-methoxyphenyl)propanoyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C23H24N4O3
2-[(2R)-1-[3-(4-methoxyphenyl)propanoyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— 6-[(6-Methoxy-1,3-benzodioxol-5-yl)methyl]-2-pyridin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H20N4O4
6-[(6-Methoxy-1,3-benzodioxol-5-yl)methyl]-2-pyridin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 2-[(3S)-1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-4-thiophen-2-yl-1H-pyrimidin-6-one —— C19H19N5O2S
2-[(3S)-1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-4-thiophen-2-yl-1H-pyrimidin-6-one
—— 5-[4-[(3-Methoxyphenyl)methyl]piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-4-ylpyrimidine —— C22H25N5O3S
5-[4-[(3-Methoxyphenyl)methyl]piperazin-1-yl]sulfonyl-4-methyl-2-pyridin-4-ylpyrimidine
—— 4-[(3S)-1-[2-(4-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C22H22N4O3
4-[(3S)-1-[2-(4-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— 2-[(3R)-1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-4-thiophen-2-yl-1H-pyrimidin-6-one —— C19H19N5O2S
2-[(3R)-1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-4-thiophen-2-yl-1H-pyrimidin-6-one
—— N-[[4-[5-(dimethylcarbamoyl)-2-methylpyrimidin-4-yl]phenyl]methyl]-2,4-dimethylpyrimidine-5-carboxamide —— C22H24N6O2
N-[[4-[5-(dimethylcarbamoyl)-2-methylpyrimidin-4-yl]phenyl]methyl]-2,4-dimethylpyrimidine-5-carboxamide
—— [4-(4-fluorophenoxy)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-(4-methylpyrimidin-5-yl)methanone —— C24H19FN6O2
[4-(4-fluorophenoxy)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-(4-methylpyrimidin-5-yl)methanone
—— 2-[(3R)-1-[(2,4-dimethoxyphenyl)methyl]pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C22H24N4O3
2-[(3R)-1-[(2,4-dimethoxyphenyl)methyl]pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— 4-[(3R)-1-[(2-fluoro-5-methoxyphenyl)methyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C21H21FN4O2
4-[(3R)-1-[(2-fluoro-5-methoxyphenyl)methyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— 2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-4-(1,3-thiazol-2-yl)-1H-pyrimidin-6-one —— C19H20N6O2S
2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]-4-(1,3-thiazol-2-yl)-1H-pyrimidin-6-one
—— 4-[(3R)-1-[2-(4-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C22H22N4O3
4-[(3R)-1-[2-(4-methoxyphenyl)acetyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— 2-[(3S)-1-(2,5-dimethoxybenzoyl)pyrrolidin-3-yl]-4-(2-methoxypyridin-3-yl)-1H-pyrimidin-6-one —— C23H24N4O5
2-[(3S)-1-(2,5-dimethoxybenzoyl)pyrrolidin-3-yl]-4-(2-methoxypyridin-3-yl)-1H-pyrimidin-6-one
—— 6-[[4-(2-Hydroxyethoxy)-3-methoxyphenyl]methyl]-2-pyridin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H24N4O4
6-[[4-(2-Hydroxyethoxy)-3-methoxyphenyl]methyl]-2-pyridin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one