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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-5-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one —— C25H26N6O2
(5S)-5-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
—— [(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-[(2S)-oxan-2-yl]methanone —— C25H27N5O2
[(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-[(2S)-oxan-2-yl]methanone
—— [(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-(3-fluorophenyl)methanone —— C26H22FN5O
[(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-(3-fluorophenyl)methanone
—— 1-[2-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2-oxoethyl]pyrrolidin-2-one —— C25H26N6O2
1-[2-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2-oxoethyl]pyrrolidin-2-one
—— [(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-cyclobutylmethanone —— C25H27N5O
[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-cyclobutylmethanone
—— [(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-pyridin-4-ylmethanone —— C26H24N6O
[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-pyridin-4-ylmethanone
—— [(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-cyclopentylmethanone —— C26H29N5O
[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-cyclopentylmethanone
—— 1-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-2-[(1S)-cyclopent-2-en-1-yl]ethanone —— C27H29N5O
1-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-2-[(1S)-cyclopent-2-en-1-yl]ethanone
—— 4-[(2S)-2-(benzylamino)-2-phenylethyl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C24H22N4O
4-[(2S)-2-(benzylamino)-2-phenylethyl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— [(2R)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-pyridin-2-ylmethanone —— C26H24N6O
[(2R)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-pyridin-2-ylmethanone
—— 1-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2-[(1R)-cyclopent-2-en-1-yl]ethanone —— C26H27N5O
1-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2-[(1R)-cyclopent-2-en-1-yl]ethanone
—— 2-[4-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)piperazin-1-yl]acetamide —— C25H29N7O
2-[4-(7-benzyl-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)piperazin-1-yl]acetamide
—— [(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-[(2S)-oxan-2-yl]methanone —— C26H29N5O2
[(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-[(2S)-oxan-2-yl]methanone
—— 7-[[1-(2-Chlorophenyl)pyrrol-2-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H20ClN5O
7-[[1-(2-Chlorophenyl)pyrrol-2-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-(2-fluorophenyl)-N-[(1R)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]acetamide —— C25H21FN4O2
2-(2-fluorophenyl)-N-[(1R)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]acetamide
—— 4-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C22H22N4O2
4-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— N-[(1R)-2-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]cyclohexanecarboxamide —— C24H26N4O2
N-[(1R)-2-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]cyclohexanecarboxamide
—— N-[(1R)-1-(4-fluorophenyl)-2-(6-oxo-2-pyridin-4-yl-1H-pyrimidin-4-yl)ethyl]-2-phenylacetamide —— C25H21FN4O2
N-[(1R)-1-(4-fluorophenyl)-2-(6-oxo-2-pyridin-4-yl-1H-pyrimidin-4-yl)ethyl]-2-phenylacetamide
—— N-[(1S)-2-(2-cyclobutyl-6-oxo-1H-pyrimidin-4-yl)-1-phenylethyl]-2-pyrazol-1-ylacetamide —— C21H23N5O2
N-[(1S)-2-(2-cyclobutyl-6-oxo-1H-pyrimidin-4-yl)-1-phenylethyl]-2-pyrazol-1-ylacetamide
—— N-[(1S)-2-(2-cyclopropyl-6-oxo-1H-pyrimidin-4-yl)-1-phenylethyl]-2-pyridin-2-ylacetamide —— C22H22N4O2
N-[(1S)-2-(2-cyclopropyl-6-oxo-1H-pyrimidin-4-yl)-1-phenylethyl]-2-pyridin-2-ylacetamide
—— 2-[(2R)-1-(2-fluorobenzoyl)pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C20H17FN4O2
2-[(2R)-1-(2-fluorobenzoyl)pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— 4-[4-(2-fluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carbonyl]-1H-pyridin-2-one —— C24H19FN6O2
4-[4-(2-fluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carbonyl]-1H-pyridin-2-one
—— 2-[1-[(2-Fluorophenyl)methylsulfonyl]azetidin-3-yl]-6-thiophen-2-ylpyridazin-3-one —— C18H16FN3O3S2
2-[1-[(2-Fluorophenyl)methylsulfonyl]azetidin-3-yl]-6-thiophen-2-ylpyridazin-3-one
—— (6R)-4-N-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine —— C19H18ClN5
(6R)-4-N-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine
—— 4-pyridin-3-yl-2-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H21N5O
4-pyridin-3-yl-2-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 2-[(3R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-6-thiophen-2-yl-1H-pyrimidin-4-one —— C19H23N3O2S
2-[(3R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-6-thiophen-2-yl-1H-pyrimidin-4-one
—— 2-Pyridin-3-yl-7-(quinolin-6-ylmethyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H19N5O
2-Pyridin-3-yl-7-(quinolin-6-ylmethyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-Pyridin-4-yl-7-(quinolin-6-ylmethyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H19N5O
2-Pyridin-4-yl-7-(quinolin-6-ylmethyl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (3S)-1,1-dioxo-N-[2-(4-pyrazin-2-yl-5-thiophen-2-ylpyrazol-1-yl)ethyl]thiolane-3-carboxamide —— C18H19N5O3S2
(3S)-1,1-dioxo-N-[2-(4-pyrazin-2-yl-5-thiophen-2-ylpyrazol-1-yl)ethyl]thiolane-3-carboxamide
—— 2-[[4-hydroxy-1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]methyl]-6-thiophen-2-ylpyridazin-3-one —— C19H25N3O3S
2-[[4-hydroxy-1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]methyl]-6-thiophen-2-ylpyridazin-3-one
—— N-(2-morpholin-4-ylethyl)-4-(1,3-thiazol-2-yl)-5-thiophen-2-ylpyrimidin-2-amine —— C17H19N5OS2
N-(2-morpholin-4-ylethyl)-4-(1,3-thiazol-2-yl)-5-thiophen-2-ylpyrimidin-2-amine
—— 7-[(6-Fluoroquinolin-2-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H18FN5O
7-[(6-Fluoroquinolin-2-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 4-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-6-one —— C19H20N4OS
4-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-6-one
—— (2S)-N-[2-(4-pyrazin-2-yl-5-thiophen-2-ylpyrazol-1-yl)ethyl]spiro[2.3]hexane-2-carboxamide —— C20H21N5OS
(2S)-N-[2-(4-pyrazin-2-yl-5-thiophen-2-ylpyrazol-1-yl)ethyl]spiro[2.3]hexane-2-carboxamide
—— (2-amino-1,3-thiazol-4-yl)-[4-(4-fluoroanilino)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone —— C22H18FN7OS
(2-amino-1,3-thiazol-4-yl)-[4-(4-fluoroanilino)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]methanone
—— [4-(4-fluoroanilino)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-(2-fluorophenyl)methanone —— C25H19F2N5O
[4-(4-fluoroanilino)-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-(2-fluorophenyl)methanone
—— 2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-6-thiophen-2-yl-1H-pyrimidin-4-one —— C17H19N5OS
2-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-6-thiophen-2-yl-1H-pyrimidin-4-one
—— 6-(Furan-2-yl)-2-[(4-hydroxypiperidin-4-yl)methyl]pyridazin-3-one —— C14H17N3O3
6-(Furan-2-yl)-2-[(4-hydroxypiperidin-4-yl)methyl]pyridazin-3-one
—— 6-[(2S)-1-cyclopentylpiperidin-2-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C19H24N4O
6-[(2S)-1-cyclopentylpiperidin-2-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 3-[(2S)-oxolan-2-yl]-N-[2-(4-pyrazin-2-yl-5-thiophen-2-ylpyrazol-1-yl)ethyl]propanamide —— C20H23N5O2S
3-[(2S)-oxolan-2-yl]-N-[2-(4-pyrazin-2-yl-5-thiophen-2-ylpyrazol-1-yl)ethyl]propanamide
—— (6S)-4-N-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine —— C19H18ClN5
(6S)-4-N-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine
—— 4-pyridin-3-yl-2-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H21N5O
4-pyridin-3-yl-2-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 2-pyridin-3-yl-4-[(2S)-1-(pyridin-3-ylmethyl)piperidin-2-yl]-1H-pyrimidin-6-one —— C20H21N5O
2-pyridin-3-yl-4-[(2S)-1-(pyridin-3-ylmethyl)piperidin-2-yl]-1H-pyrimidin-6-one
—— 1-[(3S)-3-(2,5-dipyridin-4-ylpyrimidin-4-yl)piperidin-1-yl]-2-thiophen-2-ylethanone —— C25H23N5OS
1-[(3S)-3-(2,5-dipyridin-4-ylpyrimidin-4-yl)piperidin-1-yl]-2-thiophen-2-ylethanone
—— 5-cyclopropyl-N-[[4-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)phenyl]methyl]-1,2-oxazole-3-carboxamide —— C19H16N6O2
5-cyclopropyl-N-[[4-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)phenyl]methyl]-1,2-oxazole-3-carboxamide
—— 4-[4-(4-fluorophenoxy)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carbonyl]-1H-pyridin-2-one —— C24H18FN5O3
4-[4-(4-fluorophenoxy)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carbonyl]-1H-pyridin-2-one
—— 4-pyridin-4-yl-2-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H21N5O
4-pyridin-4-yl-2-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 4-pyridin-3-yl-2-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H21N5O
4-pyridin-3-yl-2-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 7-[[4-(2-Oxo-2-pyrrolidin-1-ylethoxy)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H27N5O3
7-[[4-(2-Oxo-2-pyrrolidin-1-ylethoxy)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 4-[(3R)-1-[(4-fluorophenyl)methyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C20H19FN4O
4-[(3R)-1-[(4-fluorophenyl)methyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one