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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N,N-dimethyl-6-[(1S)-1-[(6-methylpyridin-2-yl)methylamino]-2-phenylethyl]-2-pyridin-3-ylpyrimidin-4-amine —— C26H28N6
N,N-dimethyl-6-[(1S)-1-[(6-methylpyridin-2-yl)methylamino]-2-phenylethyl]-2-pyridin-3-ylpyrimidin-4-amine
—— 4-methyl-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-2-carboxamide —— C23H23N5O2S
4-methyl-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-2-carboxamide
—— 4-[(3R)-1-[2-(2,6-dimethylphenoxy)acetyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C23H24N4O3
4-[(3R)-1-[2-(2,6-dimethylphenoxy)acetyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 7-[(6-methylpyridin-2-yl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H21N5O
7-[(6-methylpyridin-2-yl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-(2-methylphenyl)acetamide —— C24H22N4O2
N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-(2-methylphenyl)acetamide
—— 4-[(2R)-1-[(6-methylpyridin-2-yl)methyl]piperidin-2-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C21H23N5O
4-[(2R)-1-[(6-methylpyridin-2-yl)methyl]piperidin-2-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— 2-[(2S)-1-[2-(2-methylphenyl)acetyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C22H22N4O2
2-[(2S)-1-[2-(2-methylphenyl)acetyl]pyrrolidin-2-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— (2,6-dimethoxypyrimidin-4-yl)-[3-(2,6-dimethylanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methanone —— C21H23N5O4
(2,6-dimethoxypyrimidin-4-yl)-[3-(2,6-dimethylanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methanone
—— N-[(1S)-2-[2-cyclopropyl-6-(dimethylamino)pyrimidin-4-yl]-1-(3-methylphenyl)ethyl]-2,4-dimethylpyrimidine-5-carboxamide —— C25H30N6O
N-[(1S)-2-[2-cyclopropyl-6-(dimethylamino)pyrimidin-4-yl]-1-(3-methylphenyl)ethyl]-2,4-dimethylpyrimidine-5-carboxamide
—— N-[(1S)-2-[2-cyclopropyl-6-(methylamino)pyrimidin-4-yl]-1-(3-methylphenyl)ethyl]-2,4-dimethylpyrimidine-5-carboxamide —— C24H28N6O
N-[(1S)-2-[2-cyclopropyl-6-(methylamino)pyrimidin-4-yl]-1-(3-methylphenyl)ethyl]-2,4-dimethylpyrimidine-5-carboxamide
—— (3S)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-1-(2,3-dimethylphenyl)-5-oxopyrrolidine-3-carboxamide —— C25H28N6O2
(3S)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-1-(2,3-dimethylphenyl)-5-oxopyrrolidine-3-carboxamide
—— N-[(1S)-2-[2-cyclopropyl-6-(methylamino)pyrimidin-4-yl]-1-(3-methylphenyl)ethyl]-2-pyridin-3-ylacetamide —— C24H27N5O
N-[(1S)-2-[2-cyclopropyl-6-(methylamino)pyrimidin-4-yl]-1-(3-methylphenyl)ethyl]-2-pyridin-3-ylacetamide
—— 1,5-dimethyl-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]indole-2-carboxamide —— C24H25N5O2S
1,5-dimethyl-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]indole-2-carboxamide
—— (3R)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-1-(2,3-dimethylphenyl)-5-oxopyrrolidine-3-carboxamide —— C25H28N6O2
(3R)-N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-1-(2,3-dimethylphenyl)-5-oxopyrrolidine-3-carboxamide
—— 4-[3-(2,6-dimethylanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-6-(2-methylpropyl)-1H-pyrimidin-2-one —— C23H27N5O3
4-[3-(2,6-dimethylanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-6-(2-methylpropyl)-1H-pyrimidin-2-one
—— 2-[5-Amino-3-(5-methylfuran-2-yl)-6-oxopyridazin-1-yl]acetamide —— C11H12N4O3
2-[5-Amino-3-(5-methylfuran-2-yl)-6-oxopyridazin-1-yl]acetamide
—— 5-methyl-N-[(1S)-2-methyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1-benzofuran-2-carboxamide —— C23H22N4O3
5-methyl-N-[(1S)-2-methyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1-benzofuran-2-carboxamide
—— N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-2-(6-methyl-1-benzofuran-3-yl)acetamide —— C23H23N5O2
N-[[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]-2-(6-methyl-1-benzofuran-3-yl)acetamide
—— N,N-Dimethyl-2-[1-[2-pyrimidyl]ethylidene]hydrazidocarbothioamide —— C9H13N5S
N,N-Dimethyl-2-[1-[2-pyrimidyl]ethylidene]hydrazidocarbothioamide
—— (2R)-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]propanamide —— C21H24N4O4S
(2R)-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]propanamide
—— 3,5-dimethyl-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]-1-benzofuran-2-carboxamide —— C24H24N4O3S
3,5-dimethyl-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]-1-benzofuran-2-carboxamide
—— N-[(1S)-2-[2-cyclopropyl-6-(methylamino)pyrimidin-4-yl]-1-(3-methylphenyl)ethyl]cyclopropanecarboxamide —— C21H26N4O
N-[(1S)-2-[2-cyclopropyl-6-(methylamino)pyrimidin-4-yl]-1-(3-methylphenyl)ethyl]cyclopropanecarboxamide
—— (2S)-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]propanamide —— C21H24N4O4S
(2S)-2-[4-(3-methyl-1,2-oxazol-5-yl)-3-(5-methylthiophen-2-yl)-6-oxopyridazin-1-yl]-N-[[(2S)-oxolan-2-yl]methyl]propanamide
—— 5-(6-methylpyridin-3-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H14N4O
5-(6-methylpyridin-3-yl)-3-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-N-[(1R)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]thiophene-2-carboxamide —— C23H20N4O2S
5-methyl-N-[(1R)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]thiophene-2-carboxamide
—— 1-[(3S)-3-[2-(dimethylamino)-6-(4-methylphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethanone —— C26H30N4O2
1-[(3S)-3-[2-(dimethylamino)-6-(4-methylphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethanone
—— (2S)-2-(3,4-dimethylphenoxy)-N-[[4-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)phenyl]methyl]propanamide —— C23H23N5O2
(2S)-2-(3,4-dimethylphenoxy)-N-[[4-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)phenyl]methyl]propanamide
—— 5-(2-methoxypyridin-3-yl)-2-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H16N4O2
5-(2-methoxypyridin-3-yl)-2-(4-methylphenyl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 2-(4-methylphenyl)-N-[(1R)-2-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]acetamide —— C26H24N4O2
2-(4-methylphenyl)-N-[(1R)-2-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)-1-phenylethyl]acetamide
—— [(4S)-5-ethoxycarbonyl-4-(furan-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl]methyl 2-(4-methoxyphenyl)-1,3-thiazole-4-carboxylate —— C23H21N3O7S
[(4S)-5-ethoxycarbonyl-4-(furan-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl]methyl 2-(4-methoxyphenyl)-1,3-thiazole-4-carboxylate
—— 2-(2-methoxy-5-methylphenyl)-1-[(3S)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]ethanone —— C25H29N5O2
2-(2-methoxy-5-methylphenyl)-1-[(3S)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]ethanone
—— 2-[(3R)-1-(6-methyl-2-oxo-1H-pyridine-3-carbonyl)pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C20H19N5O3
2-[(3R)-1-(6-methyl-2-oxo-1H-pyridine-3-carbonyl)pyrrolidin-3-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— 1-[(3S)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-2-(2-methoxy-5-methylphenyl)ethanone —— C26H31N5O2
1-[(3S)-3-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]-2-(2-methoxy-5-methylphenyl)ethanone
—— 6-[1-(2-fluoro-5-methylphenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C22H24FN5O2S
6-[1-(2-fluoro-5-methylphenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(2-methoxy-4-methylphenoxy)acetamide —— C23H22FN5O3
N-[(1S)-1-[7-(2-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-2-(2-methoxy-4-methylphenoxy)acetamide
—— 2-(dimethylamino)-N,N-dimethyl-4-[4-[[(6-methyl-2-oxo-1H-pyridine-3-carbonyl)amino]methyl]phenyl]pyrimidine-5-carboxamide —— C23H26N6O3
2-(dimethylamino)-N,N-dimethyl-4-[4-[[(6-methyl-2-oxo-1H-pyridine-3-carbonyl)amino]methyl]phenyl]pyrimidine-5-carboxamide
—— [(4R)-5-ethoxycarbonyl-4-(furan-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl]methyl 2-(4-methoxyphenyl)-1,3-thiazole-4-carboxylate —— C23H21N3O7S
[(4R)-5-ethoxycarbonyl-4-(furan-2-yl)-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl]methyl 2-(4-methoxyphenyl)-1,3-thiazole-4-carboxylate
—— N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-[(2S)-oxolan-2-yl]acetamide —— C21H22N4O3
N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-[(2S)-oxolan-2-yl]acetamide
—— 2-(4-fluorophenyl)-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]acetamide —— C24H21FN4O2
2-(4-fluorophenyl)-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]acetamide
—— 3-(2-methoxyphenyl)-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]propanamide —— C25H24N4O3
3-(2-methoxyphenyl)-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]propanamide
—— (2S)-N-[[2-(cyclopropylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]methyl]-N-methyloxolane-2-carboxamide —— C18H23N5O3
(2S)-N-[[2-(cyclopropylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]methyl]-N-methyloxolane-2-carboxamide
—— (2S,6S)-2,6-dimethyl-4-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]morpholine —— C23H28N6O3
(2S,6S)-2,6-dimethyl-4-[5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)pyrimidin-2-yl]morpholine
—— (1R,2R)-2-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]cyclopropane-1-carboxamide —— C20H20N4O2
(1R,2R)-2-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]cyclopropane-1-carboxamide
—— 5-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]thiophene-2-carboxamide —— C21H18N4O3S
5-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]thiophene-2-carboxamide
—— 5-(2-methoxypyridin-3-yl)-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C13H12N4O2
5-(2-methoxypyridin-3-yl)-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-(3-propan-2-yloxypropyl)pyrimidin-2-amine —— C23H30N6O3
5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-(3-propan-2-yloxypropyl)pyrimidin-2-amine
—— 2-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]acetamide —— C18H18N4O3
2-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]acetamide
—— (1S,3R)-3-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]cyclohexane-1-carboxamide —— C26H32N4O3
(1S,3R)-3-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]cyclohexane-1-carboxamide
—— (3S)-N-[[2-(cyclopropylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]methyl]-N-methyloxolane-3-carboxamide —— C18H23N5O3
(3S)-N-[[2-(cyclopropylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]methyl]-N-methyloxolane-3-carboxamide
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-(thiophen-2-ylmethyl)pyrimidin-2-amine —— C22H22N6O2S
5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-(thiophen-2-ylmethyl)pyrimidin-2-amine