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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]pyridine-4-carboxamide —— C22H19N5O2
N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]pyridine-4-carboxamide
—— (1S,3S)-3-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]cyclohexane-1-carboxamide —— C26H32N4O3
(1S,3S)-3-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]cyclohexane-1-carboxamide
—— N-[[4-[2-(dimethylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-3-[(2S)-oxolan-2-yl]propanamide —— C24H29N5O3
N-[[4-[2-(dimethylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-3-[(2S)-oxolan-2-yl]propanamide
—— N-[(1S)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-4,5-dimethylthiophene-2-carboxamide —— C21H21N5O2S
N-[(1S)-1-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]-4,5-dimethylthiophene-2-carboxamide
—— 3,5-dimethyl-4-[(2S)-2-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]pyrrolidin-1-yl]sulfonyl-1,2-oxazole —— C18H21N5O4S
3,5-dimethyl-4-[(2S)-2-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]pyrrolidin-1-yl]sulfonyl-1,2-oxazole
—— 2-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]propanamide —— C19H20N4O2
2-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]propanamide
—— 2-(2-methoxyphenyl)-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]acetamide —— C25H24N4O3
2-(2-methoxyphenyl)-N-[[4-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]acetamide
—— 2-methyl-N-[(5R)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazolin-5-yl]propanamide —— C17H20N4O
2-methyl-N-[(5R)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazolin-5-yl]propanamide
—— (3S)-N-methyl-N-[[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]methyl]-1,1-dioxothiolane-3-sulfonamide —— C17H24N4O5S2
(3S)-N-methyl-N-[[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]methyl]-1,1-dioxothiolane-3-sulfonamide
—— (3R)-N-[[2-(cyclopropylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]methyl]-N-methyloxolane-3-carboxamide —— C18H23N5O3
(3R)-N-[[2-(cyclopropylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]methyl]-N-methyloxolane-3-carboxamide
—— [(2S)-2-(5-methyl-1,2-oxazol-3-yl)azepan-1-yl]-pyrazin-2-ylmethanone —— C15H18N4O2
[(2S)-2-(5-methyl-1,2-oxazol-3-yl)azepan-1-yl]-pyrazin-2-ylmethanone
—— 4-(5-methyl-1,2-oxazol-3-yl)-2-pyridin-2-yl-1H-pyrimidin-6-one —— C13H10N4O2
4-(5-methyl-1,2-oxazol-3-yl)-2-pyridin-2-yl-1H-pyrimidin-6-one
—— [2-(dimethylamino)pyrimidin-5-yl]-[(3S)-3-(4-methyl-6-thiophen-2-ylpyrimidin-2-yl)piperidin-1-yl]methanone —— C21H24N6OS
[2-(dimethylamino)pyrimidin-5-yl]-[(3S)-3-(4-methyl-6-thiophen-2-ylpyrimidin-2-yl)piperidin-1-yl]methanone
—— (1R,3R)-3-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]cyclohexane-1-carboxamide —— C26H32N4O3
(1R,3R)-3-methoxy-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]cyclohexane-1-carboxamide
—— 1-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-2-methylpropan-1-one —— C24H27N5O
1-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-2-methylpropan-1-one
—— (2S)-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]oxolane-2-carboxamide —— C23H26N4O3
(2S)-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-propan-2-ylpyrimidin-4-yl]phenyl]methyl]oxolane-2-carboxamide
—— N-[[2-(cyclopropylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]methyl]-N-methyl-3-[(2R)-oxolan-2-yl]propanamide —— C20H27N5O3
N-[[2-(cyclopropylamino)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]methyl]-N-methyl-3-[(2R)-oxolan-2-yl]propanamide
—— (2-methoxypyrimidin-5-yl)-[(3R)-3-(4-methyl-6-thiophen-2-ylpyrimidin-2-yl)piperidin-1-yl]methanone —— C20H21N5O2S
(2-methoxypyrimidin-5-yl)-[(3R)-3-(4-methyl-6-thiophen-2-ylpyrimidin-2-yl)piperidin-1-yl]methanone
—— 1-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2-methylpropan-1-one —— C23H25N5O
1-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2-methylpropan-1-one
—— 2-[1-(2-methylpropanoyl)piperidin-4-yl]-4-[(3S)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C23H30N6O3
2-[1-(2-methylpropanoyl)piperidin-4-yl]-4-[(3S)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(3S)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C23H29N7O
(5-tert-butyl-1H-pyrazol-3-yl)-[(3S)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methanone
—— [(5aS,8aR)-2-tert-butyl-4,5,5a,6,8,8a-hexahydropyrrolo[3,4-g]indazol-7-yl]-pyrazin-2-ylmethanone —— C18H23N5O
[(5aS,8aR)-2-tert-butyl-4,5,5a,6,8,8a-hexahydropyrrolo[3,4-g]indazol-7-yl]-pyrazin-2-ylmethanone
—— (2-Tert-butylpyrimidin-5-yl)-[4-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C25H31N7O
(2-Tert-butylpyrimidin-5-yl)-[4-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methanone
—— tert-butyl N-[(1R)-2-(4-oxo-2-pyridin-3-yl-1H-pyrimidin-6-yl)-1-phenylethyl]carbamate —— C22H24N4O3
tert-butyl N-[(1R)-2-(4-oxo-2-pyridin-3-yl-1H-pyrimidin-6-yl)-1-phenylethyl]carbamate
—— 2-[1-(2-methylpropanoyl)piperidin-4-yl]-4-[(3R)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C23H30N6O3
2-[1-(2-methylpropanoyl)piperidin-4-yl]-4-[(3R)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C23H29N7O
(5-tert-butyl-1H-pyrazol-3-yl)-[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methanone
—— 1-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2-methylpropan-1-one —— C23H25N5O
1-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2-methylpropan-1-one
—— 5-tert-butyl-2-methyl-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]pyrazole-3-carboxamide —— C22H28N6O2S
5-tert-butyl-2-methyl-N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]pyrazole-3-carboxamide
—— tert-butyl N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]carbamate —— C18H24N4O3S
tert-butyl N-[(1R)-3-methylsulfanyl-1-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)propyl]carbamate
—— 1-[4-(3-fluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-3,3-dimethylbutan-1-one —— C24H26FN5O
1-[4-(3-fluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-3,3-dimethylbutan-1-one
—— 5-tert-butyl-2-methyl-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]pyrazole-3-carboxamide —— C22H28N6O2S
5-tert-butyl-2-methyl-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]pyrazole-3-carboxamide
—— (2R)-2-(4-fluorophenoxy)-N-[[4-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)phenyl]methyl]propanamide —— C21H18FN5O2
(2R)-2-(4-fluorophenoxy)-N-[[4-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)phenyl]methyl]propanamide
—— 1-[4-(3,5-difluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2,2-dimethylpropan-1-one —— C23H23F2N5O
1-[4-(3,5-difluoroanilino)-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl]-2,2-dimethylpropan-1-one
—— 2,2-dimethyl-1-[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]propan-1-one —— C20H27N5O
2,2-dimethyl-1-[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]propan-1-one
—— 3,3-dimethyl-1-[(3S)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]butan-1-one —— C21H29N5O
3,3-dimethyl-1-[(3S)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]butan-1-one
—— 1-[(2R)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one —— C24H27N5O
1-[(2R)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one
—— 1-[(1S,9R)-3-(cyclopropylamino)-5-pyridin-4-yl-4,6,12-triazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-trien-12-yl]-3,3-dimethylbutan-1-one —— C23H29N5O
1-[(1S,9R)-3-(cyclopropylamino)-5-pyridin-4-yl-4,6,12-triazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-trien-12-yl]-3,3-dimethylbutan-1-one
—— (5-Tert-butyl-2-methylpyrazol-3-yl)-[4-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C25H33N7O
(5-Tert-butyl-2-methylpyrazol-3-yl)-[4-[6-(dimethylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]methanone
—— 1-(4-anilino-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)-2,2-dimethylpropan-1-one —— C23H25N5O
1-(4-anilino-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-6-yl)-2,2-dimethylpropan-1-one
—— 2,2-dimethyl-1-[(2S)-2-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)morpholin-4-yl]propan-1-one —— C15H19N5O3
2,2-dimethyl-1-[(2S)-2-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)morpholin-4-yl]propan-1-one
—— 4-[(3R)-1-[(2S)-2-(2-fluorophenoxy)propanoyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one —— C22H21FN4O3
4-[(3R)-1-[(2S)-2-(2-fluorophenoxy)propanoyl]pyrrolidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-6-one
—— N-[3-[6-[(3R)-piperidin-3-yl]-2-pyridin-4-ylpyrimidin-4-yl]oxyphenyl]acetamide —— C22H23N5O2
N-[3-[6-[(3R)-piperidin-3-yl]-2-pyridin-4-ylpyrimidin-4-yl]oxyphenyl]acetamide
—— 1-[(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one —— C24H27N5O
1-[(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one
—— N-[(1S)-2-(2-cyclobutyl-4-oxo-1H-pyrimidin-6-yl)-1-phenylethyl]acetamide —— C18H21N3O2
N-[(1S)-2-(2-cyclobutyl-4-oxo-1H-pyrimidin-6-yl)-1-phenylethyl]acetamide
—— N-[4-[(4-oxo-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-7-yl)methyl]phenyl]acetamide —— C22H23N5O2
N-[4-[(4-oxo-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-7-yl)methyl]phenyl]acetamide
—— 4-[(3S)-1-[(2S)-2-(2-fluorophenoxy)propanoyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C22H21FN4O3
4-[(3S)-1-[(2S)-2-(2-fluorophenoxy)propanoyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 4-[(3S)-1-[(2R)-2-(2-fluorophenoxy)propanoyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C22H21FN4O3
4-[(3S)-1-[(2R)-2-(2-fluorophenoxy)propanoyl]pyrrolidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 1-[4-[6-(Methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]ethanone —— C17H21N5O
1-[4-[6-(Methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]ethanone
—— 6-chloro-N-[(Z)-(3-fluorophenyl)methylideneamino]-4-phenylquinazolin-2-amine —— C21H14ClFN4
6-chloro-N-[(Z)-(3-fluorophenyl)methylideneamino]-4-phenylquinazolin-2-amine
—— Methyl 4-hydroxy-6-(methylsulfanyl)-2-(2-phenylvinyl)-5-pyrimidinecarboxylate —— C15H14N2O3S
Methyl 4-hydroxy-6-(methylsulfanyl)-2-(2-phenylvinyl)-5-pyrimidinecarboxylate