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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— Methyl 4-chloro-8,12-dioxa-1,3,5-triazatricyclo[8.4.0.02,7]tetradeca-2,4,6-triene-6-carboxylate —— C11H12ClN3O4
Methyl 4-chloro-8,12-dioxa-1,3,5-triazatricyclo[8.4.0.02,7]tetradeca-2,4,6-triene-6-carboxylate
—— (5Z)-5-[[[(2R)-butan-2-yl]amino]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C12H17N3O2S
(5Z)-5-[[[(2R)-butan-2-yl]amino]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 3-Ethoxy-4-[[2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]cyclobut-3-ene-1,2-dione —— C23H17FN6O4
3-Ethoxy-4-[[2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]cyclobut-3-ene-1,2-dione
—— N-tert-butyl-5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-amine —— C21H20F2N6O
N-tert-butyl-5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-amine
—— [3-[[5-Fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]oxetan-3-yl]methanol —— C21H18F2N6O3
[3-[[5-Fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]oxetan-3-yl]methanol
—— N-[(Z)-benzylideneamino]-4,6-diphenylpyrimidine-2-carboxamide —— C24H18N4O
N-[(Z)-benzylideneamino]-4,6-diphenylpyrimidine-2-carboxamide
—— 5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-N-(1,1,1-trifluoro-4-methylsulfonylbutan-2-yl)pyrimidin-4-amine —— C22H19F5N6O3S
5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-N-(1,1,1-trifluoro-4-methylsulfonylbutan-2-yl)pyrimidin-4-amine
—— N-[4,4,4-trifluoro-3-[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]butyl]methanesulfonamide —— C22H20F5N7O3S
N-[4,4,4-trifluoro-3-[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]butyl]methanesulfonamide
—— 2-[[[5-Amino-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]methyl]-1,1,1,3,3,3-hexafluoropropan-2-ol —— C21H16F7N7O2
2-[[[5-Amino-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]methyl]-1,1,1,3,3,3-hexafluoropropan-2-ol
—— 3,3,3-Trifluoro-2-[[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]methyl]propane-1,2-diol —— C21H17F5N6O3
3,3,3-Trifluoro-2-[[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]methyl]propane-1,2-diol
—— (5R)-3-[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]-5-(hydroxymethyl)-1,3-oxazolidin-2-one —— C21H16F2N6O4
(5R)-3-[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]-5-(hydroxymethyl)-1,3-oxazolidin-2-one
—— 5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-N-(oxolan-3-yl)pyrimidin-4-amine —— C21H18F2N6O2
5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-N-(oxolan-3-yl)pyrimidin-4-amine
—— 1,1,1-trifluoro-N-[2-[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]ethyl]methanesulfonamide —— C20H16F5N7O3S
1,1,1-trifluoro-N-[2-[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]ethyl]methanesulfonamide
—— 2-[[[2-[1-[(2,3-Difluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-5-fluoropyrimidin-4-yl]amino]methyl]-1,1,1,3,3,3-hexafluoropropan-2-ol —— C21H13F9N6O2
2-[[[2-[1-[(2,3-Difluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-5-fluoropyrimidin-4-yl]amino]methyl]-1,1,1,3,3,3-hexafluoropropan-2-ol
—— 5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-N-[1-(trifluoromethylsulfonyl)azetidin-3-yl]pyrimidin-4-amine —— C21H16F5N7O3S
5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-N-[1-(trifluoromethylsulfonyl)azetidin-3-yl]pyrimidin-4-amine
—— 5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-N-[[1-(1H-imidazol-2-yl)cyclopropyl]methyl]pyrimidin-4-amine —— C24H20F2N8O
5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]-N-[[1-(1H-imidazol-2-yl)cyclopropyl]methyl]pyrimidin-4-amine
—— 2-[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]-N-methylethanesulfonamide —— C20H19F2N7O3S
2-[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]-N-methylethanesulfonamide
—— N-[(2S)-2,3-dihydroxypropyl]-2-[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]ethanesulfonamide —— C22H23F2N7O5S
N-[(2S)-2,3-dihydroxypropyl]-2-[[5-fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]amino]ethanesulfonamide
—— 1-[5-Fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]-3-methyl-3-methylsulfonylpyrrolidin-2-one —— C23H20F2N6O4S
1-[5-Fluoro-2-[1-[(2-fluorophenyl)methyl]-5-(1,2-oxazol-3-yl)pyrazol-3-yl]pyrimidin-4-yl]-3-methyl-3-methylsulfonylpyrrolidin-2-one
—— 5-fluoro-2-(5-(isoxazol-3-yl)-1-(3,3,3-trifluoropropyl)-1H-pyrazol-3-yl)pyrimidin-4-ol —— C13H9F4N5O2
5-fluoro-2-(5-(isoxazol-3-yl)-1-(3,3,3-trifluoropropyl)-1H-pyrazol-3-yl)pyrimidin-4-ol
—— (6-Methyl-3-pyrimidin-2-ylpyridin-2-yl)-[2-[[5-(trifluoromethyl)pyridin-2-yl]amino]-7-azabicyclo[2.2.1]heptan-7-yl]methanone —— C23H21F3N6O
(6-Methyl-3-pyrimidin-2-ylpyridin-2-yl)-[2-[[5-(trifluoromethyl)pyridin-2-yl]amino]-7-azabicyclo[2.2.1]heptan-7-yl]methanone
—— (5E,6E)-3-(1,1-difluoroprop-2-enyl)-6-ethylidene-5-prop-2-enylidenepyrazin-2-one —— C12H12F2N2O
(5E,6E)-3-(1,1-difluoroprop-2-enyl)-6-ethylidene-5-prop-2-enylidenepyrazin-2-one
—— [2-[(4,6-Dimethylpyrimidin-2-yl)amino]-7-azabicyclo[2.2.1]heptan-7-yl]-(6-methyl-3-pyrimidin-2-ylpyridin-2-yl)methanone —— C23H25N7O
[2-[(4,6-Dimethylpyrimidin-2-yl)amino]-7-azabicyclo[2.2.1]heptan-7-yl]-(6-methyl-3-pyrimidin-2-ylpyridin-2-yl)methanone
—— Tert-butyl 4-carbonochloridoyl-10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-11-carboxylate —— C20H23ClN4O4
Tert-butyl 4-carbonochloridoyl-10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-11-carboxylate
—— propan-2-yl N-[4-[2-[2-chloro-5-(pyrrolidine-1-carbonylamino)phenyl]imidazo[1,2-a]pyrimidin-6-yl]phenyl]carbamate —— C27H27ClN6O3
propan-2-yl N-[4-[2-[2-chloro-5-(pyrrolidine-1-carbonylamino)phenyl]imidazo[1,2-a]pyrimidin-6-yl]phenyl]carbamate
—— 2,3-Dimethylpyrazino[2,3-d]pyridazine —— C8H8N4
2,3-Dimethylpyrazino[2,3-d]pyridazine
—— 3-Prop-1-ynylpyridazine —— C7H6N2
3-Prop-1-ynylpyridazine
—— 7-Methyl-[1,3]dioxolo[4,5-d]pyrimidine —— C6H6N2O2
7-Methyl-[1,3]dioxolo[4,5-d]pyrimidine
—— N-[6-[(5R,6S)-3-amino-5-methyl-2-oxa-4-azabicyclo[4.1.0]hept-3-en-5-yl]-5-fluoropyridin-2-yl]-5-methoxypyrazine-2-carboxamide —— C17H17FN6O3
N-[6-[(5R,6S)-3-amino-5-methyl-2-oxa-4-azabicyclo[4.1.0]hept-3-en-5-yl]-5-fluoropyridin-2-yl]-5-methoxypyrazine-2-carboxamide
—— 2-Amino-1-methyl-5,6,7,8-tetrahydropyrazolo[1,2-a]pyridazin-3-one —— C8H13N3O
2-Amino-1-methyl-5,6,7,8-tetrahydropyrazolo[1,2-a]pyridazin-3-one
—— 7-Propan-2-yl-[1,3]dioxolo[4,5-d]pyrimidine —— C8H10N2O2
7-Propan-2-yl-[1,3]dioxolo[4,5-d]pyrimidine
—— 1-[2-(C-methyl-N-phenylcarbonimidoyl)pyrimidin-4-yl]-N-phenylethanimine —— C20H18N4
1-[2-(C-methyl-N-phenylcarbonimidoyl)pyrimidin-4-yl]-N-phenylethanimine
—— (5Z)-1-cyclopropyl-5-[(cyclopropylamino)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C11H13N3O2S
(5Z)-1-cyclopropyl-5-[(cyclopropylamino)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— Methyl 6-amino-5-methoxy-2-phenylpyrimidine-4-carboxylate —— C13H13N3O3
Methyl 6-amino-5-methoxy-2-phenylpyrimidine-4-carboxylate
—— 6-Amino-5-methoxy-2-phenylpyrimidine-4-carboxylic acid —— C12H11N3O3
6-Amino-5-methoxy-2-phenylpyrimidine-4-carboxylic acid
—— Methyl 6-amino-5-chloro-2-(4-chloro-3-fluoro-2-methylphenyl)pyrimidine-4-carboxylate —— C13H10Cl2FN3O2
Methyl 6-amino-5-chloro-2-(4-chloro-3-fluoro-2-methylphenyl)pyrimidine-4-carboxylate
—— 6-Amino-2-(4-ethynylphenyl)-5-methoxypyrimidine-4-carboxylic acid —— C14H11N3O3
6-Amino-2-(4-ethynylphenyl)-5-methoxypyrimidine-4-carboxylic acid
—— Methyl 6-amino-2-(2,5-difluoro-4-methylphenyl)-5-methoxypyrimidine-4-carboxylate —— C14H13F2N3O3
Methyl 6-amino-2-(2,5-difluoro-4-methylphenyl)-5-methoxypyrimidine-4-carboxylate
—— Methyl 6-amino-2-(4-bromophenyl)-5-methoxypyrimidine-4-carboxylate —— C13H12BrN3O3
Methyl 6-amino-2-(4-bromophenyl)-5-methoxypyrimidine-4-carboxylate
—— 6-Amino-2-(2,5-difluoro-4-methylphenyl)-5-methoxypyrimidine-4-carboxylic acid —— C13H11F2N3O3
6-Amino-2-(2,5-difluoro-4-methylphenyl)-5-methoxypyrimidine-4-carboxylic acid
—— 6-Amino-2-[4-(difluoromethyl)-2,5-difluorophenyl]-5-methoxypyrimidine-4-carboxylic acid —— C13H9F4N3O3
6-Amino-2-[4-(difluoromethyl)-2,5-difluorophenyl]-5-methoxypyrimidine-4-carboxylic acid
—— Methyl 6-amino-2-(4-ethynyl-2-fluorophenyl)-5-methoxypyrimidine-4-carboxylate —— C15H12FN3O3
Methyl 6-amino-2-(4-ethynyl-2-fluorophenyl)-5-methoxypyrimidine-4-carboxylate
—— Methyl 6-amino-2-(4-ethynylphenyl)-5-methoxypyrimidine-4-carboxylate —— C15H13N3O3
Methyl 6-amino-2-(4-ethynylphenyl)-5-methoxypyrimidine-4-carboxylate
—— Methyl 6-amino-2-(4-cyanophenyl)-5-methoxypyrimidine-4-carboxylate —— C14H12N4O3
Methyl 6-amino-2-(4-cyanophenyl)-5-methoxypyrimidine-4-carboxylate
—— Tert-butyl 6-[4-amino-3-[4-(2-benzyl-1-methyl-6-oxopyrimidin-5-yl)-2-fluorophenyl]pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.3]heptane-2-carboxylate —— C34H35FN8O3
Tert-butyl 6-[4-amino-3-[4-(2-benzyl-1-methyl-6-oxopyrimidin-5-yl)-2-fluorophenyl]pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.3]heptane-2-carboxylate
—— 6-Amino-2-(4-ethynyl-2-fluorophenyl)-5-methoxypyrimidine-4-carboxylic acid —— C14H10FN3O3
6-Amino-2-(4-ethynyl-2-fluorophenyl)-5-methoxypyrimidine-4-carboxylic acid
—— Methyl 6-amino-2-(3-fluoro-4-methylphenyl)-5-methoxypyrimidine-4-carboxylate —— C14H14FN3O3
Methyl 6-amino-2-(3-fluoro-4-methylphenyl)-5-methoxypyrimidine-4-carboxylate
—— (5Z)-1-cyclopropyl-5-[(furan-2-ylmethylamino)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C13H13N3O3S
(5Z)-1-cyclopropyl-5-[(furan-2-ylmethylamino)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 4-amino-1-[(2R)-3-hydroxy-2-[[2-octadecoxyethoxy(phenylmethoxy)phosphoryl]methoxy]propyl]pyrimidin-2-one —— C35H60N3O7P
4-amino-1-[(2R)-3-hydroxy-2-[[2-octadecoxyethoxy(phenylmethoxy)phosphoryl]methoxy]propyl]pyrimidin-2-one
—— 4-Amino-1-[3-hydroxy-2-[[2-octadecoxyethoxy(phenylmethoxy)phosphoryl]methoxy]propyl]pyrimidin-2-one —— C35H60N3O7P
4-Amino-1-[3-hydroxy-2-[[2-octadecoxyethoxy(phenylmethoxy)phosphoryl]methoxy]propyl]pyrimidin-2-one