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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1,5-anhydro-3-O-benzyl-2,4-dideoxy-4-[(imidazo[1,2-a]pyrimidin-2-ylcarbonyl)amino]-D-erythro-pentitol —— C19H20N4O3
1,5-anhydro-3-O-benzyl-2,4-dideoxy-4-[(imidazo[1,2-a]pyrimidin-2-ylcarbonyl)amino]-D-erythro-pentitol
—— 1-[5-(Pyrazin-2-ylacetyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]ethane-1,2-diol —— C14H17N5O3
1-[5-(Pyrazin-2-ylacetyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]ethane-1,2-diol
—— N-(cis-3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}cyclobutyl)-3-(4,6-dimethyl-2-oxopyrimidin-1(2H)-yl)propanamide —— C19H29N7O2
N-(cis-3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}cyclobutyl)-3-(4,6-dimethyl-2-oxopyrimidin-1(2H)-yl)propanamide
—— 1,5-anhydro-2-{[(2-cyclopropylpyrimidin-5-yl)carbonyl]amino}-2,4-dideoxy-3-O-(pyridin-2-ylmethyl)-D-threo-pentitol —— C19H22N4O3
1,5-anhydro-2-{[(2-cyclopropylpyrimidin-5-yl)carbonyl]amino}-2,4-dideoxy-3-O-(pyridin-2-ylmethyl)-D-threo-pentitol
—— 2-cyclopropyl-6-(trans-3-{[4-methyl-6-(methylamino)pyrimidin-2-yl]amino}cyclobutyl)pyrimidin-4(3H)-one —— C17H22N6O
2-cyclopropyl-6-(trans-3-{[4-methyl-6-(methylamino)pyrimidin-2-yl]amino}cyclobutyl)pyrimidin-4(3H)-one
—— 1,5-anhydro-3-O-(cyclopropylmethyl)-4-{[(2-cyclopropyl-6-oxo-1,6-dihydropyrimidin-5-yl)carbonyl]amino}-2,4-dideoxy-D-erythro-pentitol —— C17H23N3O4
1,5-anhydro-3-O-(cyclopropylmethyl)-4-{[(2-cyclopropyl-6-oxo-1,6-dihydropyrimidin-5-yl)carbonyl]amino}-2,4-dideoxy-D-erythro-pentitol
—— 6-(cis-3-aminocyclobutyl)-N~4~-[3-(cyclopentyloxy)propyl]pyrimidine-2,4-diamine —— C16H27N5O
6-(cis-3-aminocyclobutyl)-N~4~-[3-(cyclopentyloxy)propyl]pyrimidine-2,4-diamine
—— 2-(4,6-dimethyl-2-oxopyrimidin-1(2H)-yl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}acetamide —— C17H23N5O2
2-(4,6-dimethyl-2-oxopyrimidin-1(2H)-yl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}acetamide
—— N-methyl-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzisoxazol-3-ylmethyl)propanamide —— C16H22N4O3
N-methyl-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzisoxazol-3-ylmethyl)propanamide
—— N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide —— C14H18ClN5O2
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
—— (5Z)-5-[[4-(azepan-1-yl)phenyl]methylidene]-1-butan-2-yl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C21H27N3O2S
(5Z)-5-[[4-(azepan-1-yl)phenyl]methylidene]-1-butan-2-yl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 1,5-anhydro-2,3-dideoxy-3-{[(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)carbonyl]amino}-4-O-(1,3-thiazol-4-ylmethyl)-D-threo-pentitol —— C16H20N4O5S
1,5-anhydro-2,3-dideoxy-3-{[(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)carbonyl]amino}-4-O-(1,3-thiazol-4-ylmethyl)-D-threo-pentitol
—— 2-[(2Z)-2-butan-2-ylidenehydrazinyl]-5-butyl-4-methyl-1H-pyrimidin-6-one —— C13H22N4O
2-[(2Z)-2-butan-2-ylidenehydrazinyl]-5-butyl-4-methyl-1H-pyrimidin-6-one
—— 4-{[6-(aminocarbonyl)pyrazin-2-yl]amino}-1,5-anhydro-2,4-dideoxy-3-O-(1,3-thiazol-4-ylmethyl)-D-erythro-pentitol —— C14H17N5O3S
4-{[6-(aminocarbonyl)pyrazin-2-yl]amino}-1,5-anhydro-2,4-dideoxy-3-O-(1,3-thiazol-4-ylmethyl)-D-erythro-pentitol
—— N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3,5-dimethylisoxazole-4-carboxamide —— C12H15N5O3
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3,5-dimethylisoxazole-4-carboxamide
—— N-[(2-methylpyridin-4-yl)methyl]-2-(methylthio)pyrimidine-5-carboxamide —— C13H14N4OS
N-[(2-methylpyridin-4-yl)methyl]-2-(methylthio)pyrimidine-5-carboxamide
—— N-(2-pyrazin-2-ylethyl)-2-(2,2,3,3-tetrafluoropropoxy)acetamide —— C11H13F4N3O2
N-(2-pyrazin-2-ylethyl)-2-(2,2,3,3-tetrafluoropropoxy)acetamide
—— 2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]acetamide —— C15H22N6O2
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]acetamide
—— 1,5-anhydro-2-O-benzyl-3,4-dideoxy-3-{[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)carbonyl]amino}-D-threo-pentitol —— C17H19N3O5
1,5-anhydro-2-O-benzyl-3,4-dideoxy-3-{[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)carbonyl]amino}-D-threo-pentitol
—— 6-{[2-(hydroxymethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]carbonyl}-1,3-dimethylpyrimidine-2,4(1H,3H)-dione —— C15H19N5O4
6-{[2-(hydroxymethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]carbonyl}-1,3-dimethylpyrimidine-2,4(1H,3H)-dione
—— 6-(3-aminocyclobutyl)-N~4~-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine —— C13H20N8
6-(3-aminocyclobutyl)-N~4~-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine
—— 1-{3-[2-[cyclopropyl(hydroxy)methyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]-3-oxopropyl}-4,6-dimethylpyrimidin-2(1H)-one —— C19H25N5O3
1-{3-[2-[cyclopropyl(hydroxy)methyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]-3-oxopropyl}-4,6-dimethylpyrimidin-2(1H)-one
—— N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide —— C15H20N6O2
N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
—— 1,5-anhydro-2-O-benzyl-3-{[(5-chloro-2-methylpyrimidin-4-yl)carbonyl]amino}-3,4-dideoxy-D-threo-pentitol —— C18H20ClN3O3
1,5-anhydro-2-O-benzyl-3-{[(5-chloro-2-methylpyrimidin-4-yl)carbonyl]amino}-3,4-dideoxy-D-threo-pentitol
—— 6-(3-aminocyclobutyl)-N~4~-[2-(2-methylphenyl)ethyl]pyrimidine-2,4-diamine —— C17H23N5
6-(3-aminocyclobutyl)-N~4~-[2-(2-methylphenyl)ethyl]pyrimidine-2,4-diamine
—— 6-(trans-3-aminocyclobutyl)-2-methyl-N-[1-(2-thienylmethyl)piperidin-4-yl]pyrimidin-4-amine —— C19H27N5S
6-(trans-3-aminocyclobutyl)-2-methyl-N-[1-(2-thienylmethyl)piperidin-4-yl]pyrimidin-4-amine
—— N-(cis-3-{6-[(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethyl)amino]-2-methylpyrimidin-4-yl}cyclobutyl)acetamide —— C19H24N6O
N-(cis-3-{6-[(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethyl)amino]-2-methylpyrimidin-4-yl}cyclobutyl)acetamide
—— 6-(trans-3-aminocyclobutyl)-N-{3-[(2-chlorobenzyl)thio]propyl}pyrimidin-4-amine —— C18H23ClN4S
6-(trans-3-aminocyclobutyl)-N-{3-[(2-chlorobenzyl)thio]propyl}pyrimidin-4-amine
—— 3-(2-{[2-Amino-6-(3-aminocyclobutyl)pyrimidin-4-YL]amino}ethyl)-1,3-oxazinan-2-one —— C14H22N6O2
3-(2-{[2-Amino-6-(3-aminocyclobutyl)pyrimidin-4-YL]amino}ethyl)-1,3-oxazinan-2-one
—— 6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-(2-pyrazin-2-ylethyl)pyrimidin-4-amine —— C16H22N6O
6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-(2-pyrazin-2-ylethyl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidine-2,4-diamine —— C13H18N6S
6-(3-aminocyclobutyl)-N~4~-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidine-2,4-diamine
—— 1,5-anhydro-4-{[(2-cyclopropylpyrimidin-5-yl)carbonyl]amino}-2,4-dideoxy-3-O-(3-fluorophenyl)-D-erythro-pentitol —— C19H20FN3O3
1,5-anhydro-4-{[(2-cyclopropylpyrimidin-5-yl)carbonyl]amino}-2,4-dideoxy-3-O-(3-fluorophenyl)-D-erythro-pentitol
—— 5-[(E)-pent-3-en-2-yl]-5-prop-2-enyl-1,3-diazinane-2,4,6-trione —— C12H16N2O3
5-[(E)-pent-3-en-2-yl]-5-prop-2-enyl-1,3-diazinane-2,4,6-trione
—— ethyl 6-[[(E)-but-2-enoyl]oxymethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H18N2O5S
ethyl 6-[[(E)-but-2-enoyl]oxymethyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1,5-anhydro-2,4-dideoxy-3-O-[2-(dimethylamino)-2-oxoethyl]-4-[(2-ethyl-6-methylpyrimidin-4-yl)amino]-D-erythro-pentitol —— C16H26N4O3
1,5-anhydro-2,4-dideoxy-3-O-[2-(dimethylamino)-2-oxoethyl]-4-[(2-ethyl-6-methylpyrimidin-4-yl)amino]-D-erythro-pentitol
—— 6-(3-aminocyclobutyl)-4-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]pyrimidine-2,4-diamine —— C16H25N7
6-(3-aminocyclobutyl)-4-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]pyrimidine-2,4-diamine
—— N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-(methylthio)pyrimidine-5-carboxamide —— C9H11N7OS
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-(methylthio)pyrimidine-5-carboxamide
—— 6-isobutyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-oxo-1,2-dihydropyrimidine-4-carboxamide —— C13H17N5O2S
6-isobutyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-oxo-1,2-dihydropyrimidine-4-carboxamide
—— 1,5-anhydro-2-{[(2-cyclopropyl-6-oxo-1,6-dihydropyrimidin-5-yl)carbonyl]amino}-2,4-dideoxy-3-O-pyridin-2-yl-D-threo-pentitol —— C18H20N4O4
1,5-anhydro-2-{[(2-cyclopropyl-6-oxo-1,6-dihydropyrimidin-5-yl)carbonyl]amino}-2,4-dideoxy-3-O-pyridin-2-yl-D-threo-pentitol
—— 1,5-anhydro-2,3-dideoxy-3-[(2-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]-4-O-(1,3-thiazol-4-ylmethyl)-D-threo-pentitol —— C17H22N4O2S
1,5-anhydro-2,3-dideoxy-3-[(2-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]-4-O-(1,3-thiazol-4-ylmethyl)-D-threo-pentitol
—— 6-(3-aminocyclobutyl)-N-[(3-pyridin-3-ylisoxazol-5-yl)methyl]pyrimidin-4-amine —— C17H18N6O
6-(3-aminocyclobutyl)-N-[(3-pyridin-3-ylisoxazol-5-yl)methyl]pyrimidin-4-amine
—— 5-hydroxy-N-{[3-(2-methoxyphenyl)isoxazol-5-yl]methyl}pyrazine-2-carboxamide —— C16H14N4O4
5-hydroxy-N-{[3-(2-methoxyphenyl)isoxazol-5-yl]methyl}pyrazine-2-carboxamide
—— N-(1-{[2-(methylthio)pyrimidin-5-yl]carbonyl}piperidin-4-yl)methanesulfonamide —— C12H18N4O3S2
N-(1-{[2-(methylthio)pyrimidin-5-yl]carbonyl}piperidin-4-yl)methanesulfonamide
—— 1,5-anhydro-2,4-dideoxy-2-[(3,6-dimethylisoxazolo[5,4-d]pyrimidin-4-yl)amino]-3-O-(pyridin-2-ylmethyl)-D-threo-pentitol —— C18H21N5O3
1,5-anhydro-2,4-dideoxy-2-[(3,6-dimethylisoxazolo[5,4-d]pyrimidin-4-yl)amino]-3-O-(pyridin-2-ylmethyl)-D-threo-pentitol
—— N-{cis-3-[2-amino-6-(methylamino)pyrimidin-4-yl]cyclobutyl}-3,5-dimethylisoxazole-4-sulfonamide —— C14H20N6O3S
N-{cis-3-[2-amino-6-(methylamino)pyrimidin-4-yl]cyclobutyl}-3,5-dimethylisoxazole-4-sulfonamide
—— N-{trans-3-[4-ethyl-5-(hydroxymethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide —— C16H18N6O3S
N-{trans-3-[4-ethyl-5-(hydroxymethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
—— 2-methyl-5-{[3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]carbonyl}pyrimidin-4(3H)-one —— C18H18N6O3
2-methyl-5-{[3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]carbonyl}pyrimidin-4(3H)-one
—— 1,5-anhydro-3-{[(2-cyclopropyl-6-oxo-1,6-dihydropyrimidin-5-yl)carbonyl]amino}-2,3-dideoxy-D-threo-pentitol —— C13H17N3O4
1,5-anhydro-3-{[(2-cyclopropyl-6-oxo-1,6-dihydropyrimidin-5-yl)carbonyl]amino}-2,3-dideoxy-D-threo-pentitol
—— 6-(cis-3-aminocyclobutyl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]pyrimidin-4-amine —— C13H18N6
6-(cis-3-aminocyclobutyl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]pyrimidin-4-amine
—— N-(2-pyrazin-2-ylethyl)-2-(tetrahydro-2H-pyran-2-ylmethoxy)acetamide —— C14H21N3O3
N-(2-pyrazin-2-ylethyl)-2-(tetrahydro-2H-pyran-2-ylmethoxy)acetamide