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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2R)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]butan-2-yl]-2-(4-methoxyphenyl)acetamide —— C23H23F2N3O3
N-[(2R)-1-[3-(3,4-difluorophenyl)-6-oxopyridazin-1-yl]butan-2-yl]-2-(4-methoxyphenyl)acetamide
—— 5-[(E)-3-(5-nitrofuran-2-yl)prop-2-enylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C11H7N3O5S
5-[(E)-3-(5-nitrofuran-2-yl)prop-2-enylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— Ethyl 1-[[3-(4-pyrimidin-4-ylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperidine-4-carboxylate —— C21H23N5O3
Ethyl 1-[[3-(4-pyrimidin-4-ylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperidine-4-carboxylate
—— Ethyl 1-[4-(furan-2-yl)-5-(2-pyrrolidin-1-ylpyrimidin-4-yl)pyrimidin-2-yl]piperidine-4-carboxylate —— C24H28N6O3
Ethyl 1-[4-(furan-2-yl)-5-(2-pyrrolidin-1-ylpyrimidin-4-yl)pyrimidin-2-yl]piperidine-4-carboxylate
—— 4-ethoxy-N-[(5S)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazolin-5-yl]benzamide —— C22H22N4O2
4-ethoxy-N-[(5S)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazolin-5-yl]benzamide
—— N-[(2R)-1-[3-(4-methoxyphenyl)-6-oxopyridazin-1-yl]butan-2-yl]-1,3-benzodioxole-5-carboxamide —— C23H23N3O5
N-[(2R)-1-[3-(4-methoxyphenyl)-6-oxopyridazin-1-yl]butan-2-yl]-1,3-benzodioxole-5-carboxamide
—— Ethyl 1-[[3-[3-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidine-4-carboxylate —— C22H25N5O3
Ethyl 1-[[3-[3-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidine-4-carboxylate
—— (3R)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-1-ethyl-5-oxopyrrolidine-3-carboxamide —— C22H27N5O2
(3R)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
—— N',N'-diethyl-N-[4-(furan-2-yl)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-2-yl]ethane-1,2-diamine —— C18H23N5O2
N',N'-diethyl-N-[4-(furan-2-yl)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-2-yl]ethane-1,2-diamine
—— tert-butyl 4-[(Z)-1-chloro-2-phenylethenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H21ClN2O3
tert-butyl 4-[(Z)-1-chloro-2-phenylethenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (3R)-N-[[4-(2-methyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-1,1-dioxothiolane-3-carboxamide —— C22H22N4O3S
(3R)-N-[[4-(2-methyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-1,1-dioxothiolane-3-carboxamide
—— N-[[4-(2-cyclopropyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]pyridine-3-carboxamide —— C25H21N5O
N-[[4-(2-cyclopropyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]pyridine-3-carboxamide
—— N-[[4-(2-methyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-2-piperidin-1-ylacetamide —— C24H27N5O
N-[[4-(2-methyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-2-piperidin-1-ylacetamide
—— (1S)-N-[[4-(2-cyclopropyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]cyclohex-3-ene-1-carboxamide —— C26H26N4O
(1S)-N-[[4-(2-cyclopropyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]cyclohex-3-ene-1-carboxamide
—— N-[[(2S)-1,4-dioxan-2-yl]methyl]-4,5-bis(furan-2-yl)pyrimidin-2-amine —— C17H17N3O4
N-[[(2S)-1,4-dioxan-2-yl]methyl]-4,5-bis(furan-2-yl)pyrimidin-2-amine
—— N-(3-ethoxypropyl)-4,5-bis(furan-2-yl)pyrimidin-2-amine —— C17H19N3O3
N-(3-ethoxypropyl)-4,5-bis(furan-2-yl)pyrimidin-2-amine
—— 1-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-fluorobenzene-1,4-dicarboxamide —— C23H22FN5O2
1-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-fluorobenzene-1,4-dicarboxamide
—— N-[2-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]pyridine-4-carboxamide —— C20H18N6O2
N-[2-[7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl]ethyl]pyridine-4-carboxamide
—— 4-(2-methylfuran-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)-N-[2-(4-methylpiperidin-1-yl)ethyl]pyrimidin-2-amine —— C21H27N5O2
4-(2-methylfuran-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)-N-[2-(4-methylpiperidin-1-yl)ethyl]pyrimidin-2-amine
—— (2S)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-(2-methylphenoxy)butanamide —— C26H30N4O2
(2S)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-(2-methylphenoxy)butanamide
—— 4-(2-methylfuran-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)-N-(thiophen-2-ylmethyl)pyrimidin-2-amine —— C18H16N4O2S
4-(2-methylfuran-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)-N-(thiophen-2-ylmethyl)pyrimidin-2-amine
—— N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-3-(1,2-oxazol-5-yl)propanamide —— C21H23N5O2
N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-3-(1,2-oxazol-5-yl)propanamide
—— 5-(2,6-dimethoxypyrimidin-4-yl)-N-(2-pyrrolidin-1-ylethyl)-4-thiophen-2-ylpyrimidin-2-amine —— C20H24N6O2S
5-(2,6-dimethoxypyrimidin-4-yl)-N-(2-pyrrolidin-1-ylethyl)-4-thiophen-2-ylpyrimidin-2-amine
—— N-(3-ethoxypropyl)-4-(furan-3-yl)-5-pyrazin-2-ylpyrimidin-2-amine —— C17H19N5O2
N-(3-ethoxypropyl)-4-(furan-3-yl)-5-pyrazin-2-ylpyrimidin-2-amine
—— (2S)-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-(3-methoxyphenoxy)butanamide —— C26H30N4O3
(2S)-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-(3-methoxyphenoxy)butanamide
—— 4-(2-methylfuran-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C18H20N4O3
4-(2-methylfuran-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-4-(2-methylfuran-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-2-amine —— C20H22N6O2
N-[2-(3,5-dimethylpyrazol-1-yl)ethyl]-4-(2-methylfuran-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-2-amine
—— 2-(dimethylamino)-N,N-dimethyl-4-[4-[[[(1S,2R)-2-methylcyclopropanecarbonyl]amino]methyl]phenyl]pyrimidine-5-carboxamide —— C21H27N5O2
2-(dimethylamino)-N,N-dimethyl-4-[4-[[[(1S,2R)-2-methylcyclopropanecarbonyl]amino]methyl]phenyl]pyrimidine-5-carboxamide
—— 5-(2,6-dimethoxypyrimidin-4-yl)-4-(furan-2-yl)-N-(2-pyrrolidin-1-ylethyl)pyrimidin-2-amine —— C20H24N6O3
5-(2,6-dimethoxypyrimidin-4-yl)-4-(furan-2-yl)-N-(2-pyrrolidin-1-ylethyl)pyrimidin-2-amine
—— (1S,2S)-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-methylcyclopropane-1-carboxamide —— C20H24N4O
(1S,2S)-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-methylcyclopropane-1-carboxamide
—— 2-(4-ethoxyphenyl)-N-[(5S)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide —— C23H24N4O2
2-(4-ethoxyphenyl)-N-[(5S)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
—— 4-(2,4-dimethoxypyrimidin-5-yl)-N-[2-(4-fluorophenyl)ethyl]-5-thiophen-3-ylpyrimidin-2-amine —— C22H20FN5O2S
4-(2,4-dimethoxypyrimidin-5-yl)-N-[2-(4-fluorophenyl)ethyl]-5-thiophen-3-ylpyrimidin-2-amine
—— N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-propyl-1,2-oxazole-3-carboxamide —— C22H25N5O2
N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-propyl-1,2-oxazole-3-carboxamide
—— 2-(2-chloro-4-fluorophenyl)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]acetamide —— C23H22ClFN4O
2-(2-chloro-4-fluorophenyl)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]acetamide
—— 2-[(3R)-1-(1,5-dimethylpyrazol-4-yl)sulfonylpiperidin-3-yl]pyrazine —— C14H19N5O2S
2-[(3R)-1-(1,5-dimethylpyrazol-4-yl)sulfonylpiperidin-3-yl]pyrazine
—— N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-3-methyl-1,2-oxazole-5-carboxamide —— C20H21N5O2
N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-3-methyl-1,2-oxazole-5-carboxamide
—— N-(2-pyridin-4-ylethyl)-4-(1,3-thiazol-2-yl)-5-thiophen-2-ylpyrimidin-2-amine —— C18H15N5S2
N-(2-pyridin-4-ylethyl)-4-(1,3-thiazol-2-yl)-5-thiophen-2-ylpyrimidin-2-amine
—— 4,5-dichloro-N-[(5S)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazolin-5-yl]-1,2-thiazole-3-carboxamide —— C17H13Cl2N5OS
4,5-dichloro-N-[(5S)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazolin-5-yl]-1,2-thiazole-3-carboxamide
—— 4,5-bis(furan-2-yl)-N-prop-2-enylpyrimidin-2-amine —— C15H13N3O2
4,5-bis(furan-2-yl)-N-prop-2-enylpyrimidin-2-amine
—— 2-[1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one —— C24H26N4O3
2-[1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl]-4-pyridin-3-yl-1H-pyrimidin-6-one
—— N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-[(3S)-1,1-dioxothiolan-3-yl]acetamide —— C21H26N4O3S
N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-[(3S)-1,1-dioxothiolan-3-yl]acetamide
—— 3,5-Dimethyl-4-(5-pyrazin-2-yl-2-pyridin-3-ylpyrimidin-4-yl)-1,2-oxazole —— C18H14N6O
3,5-Dimethyl-4-(5-pyrazin-2-yl-2-pyridin-3-ylpyrimidin-4-yl)-1,2-oxazole
—— (2R)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-(2-methylphenoxy)butanamide —— C26H30N4O2
(2R)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-(2-methylphenoxy)butanamide
—— 2-[3-(furan-2-yl)-4-(3-methyl-1,2-oxazol-5-yl)-6-oxopyridazin-1-yl]-N-(2-methylpropyl)acetamide —— C18H20N4O4
2-[3-(furan-2-yl)-4-(3-methyl-1,2-oxazol-5-yl)-6-oxopyridazin-1-yl]-N-(2-methylpropyl)acetamide
—— N-[[(2R)-1,4-dioxan-2-yl]methyl]-4,5-bis(furan-2-yl)pyrimidin-2-amine —— C17H17N3O4
N-[[(2R)-1,4-dioxan-2-yl]methyl]-4,5-bis(furan-2-yl)pyrimidin-2-amine
—— N,N,2-trimethyl-4-[4-[[[(1R,2R)-2-methylcyclopropanecarbonyl]amino]methyl]phenyl]pyrimidine-5-carboxamide —— C20H24N4O2
N,N,2-trimethyl-4-[4-[[[(1R,2R)-2-methylcyclopropanecarbonyl]amino]methyl]phenyl]pyrimidine-5-carboxamide
—— N'-[7-[(4-fluorophenyl)methyl]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-N,N,2,2-tetramethylpropane-1,3-diamine —— C26H33FN6
N'-[7-[(4-fluorophenyl)methyl]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-N,N,2,2-tetramethylpropane-1,3-diamine
—— N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-4-methoxy-3-prop-2-enylbenzamide —— C26H28N4O2
N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-4-methoxy-3-prop-2-enylbenzamide
—— [(3S)-3-[2-(dimethylamino)-6-(4-methylphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(2-methoxyphenyl)methanone —— C25H28N4O2
[(3S)-3-[2-(dimethylamino)-6-(4-methylphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(2-methoxyphenyl)methanone
—— 2-[(3R)-3-methylpiperidin-1-yl]-4-(6-methylpyridin-3-yl)-5-pyridin-4-ylpyrimidine —— C21H23N5
2-[(3R)-3-methylpiperidin-1-yl]-4-(6-methylpyridin-3-yl)-5-pyridin-4-ylpyrimidine