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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[4-[2-(dimethylamino)-5-pyridin-2-ylpyrimidin-4-yl]phenyl]methyl]-4,5-dimethylthiophene-3-carboxamide —— C25H25N5OS
N-[[4-[2-(dimethylamino)-5-pyridin-2-ylpyrimidin-4-yl]phenyl]methyl]-4,5-dimethylthiophene-3-carboxamide
—— 2,4-dimethyl-N-[[4-(2-methyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-1,3-thiazole-5-carboxamide —— C23H21N5OS
2,4-dimethyl-N-[[4-(2-methyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-1,3-thiazole-5-carboxamide
—— N-[(3,5-dimethoxyphenyl)methyl]-4-pyridin-3-yl-5-thiophen-3-ylpyrimidin-2-amine —— C22H20N4O2S
N-[(3,5-dimethoxyphenyl)methyl]-4-pyridin-3-yl-5-thiophen-3-ylpyrimidin-2-amine
—— N-[[4-[2-(dimethylamino)-5-pyridin-2-ylpyrimidin-4-yl]phenyl]methyl]-2-(3-fluorophenyl)acetamide —— C26H24FN5O
N-[[4-[2-(dimethylamino)-5-pyridin-2-ylpyrimidin-4-yl]phenyl]methyl]-2-(3-fluorophenyl)acetamide
—— N-methyl-4-pyridin-3-yl-N-(2-pyridin-2-ylethyl)-5-thiophen-3-ylpyrimidin-2-amine —— C21H19N5S
N-methyl-4-pyridin-3-yl-N-(2-pyridin-2-ylethyl)-5-thiophen-3-ylpyrimidin-2-amine
—— 4-(4-fluorophenyl)-N-[(4-fluorophenyl)methyl]-5-(1H-imidazol-2-yl)pyrimidin-2-amine —— C20H15F2N5
4-(4-fluorophenyl)-N-[(4-fluorophenyl)methyl]-5-(1H-imidazol-2-yl)pyrimidin-2-amine
—— N',N'-diethyl-N-(5-pyridin-2-yl-4-thiophen-2-ylpyrimidin-2-yl)propane-1,3-diamine —— C20H25N5S
N',N'-diethyl-N-(5-pyridin-2-yl-4-thiophen-2-ylpyrimidin-2-yl)propane-1,3-diamine
—— 4-(4-chlorophenyl)-N-(3-ethoxypropyl)-5-(1H-imidazol-2-yl)pyrimidin-2-amine —— C18H20ClN5O
4-(4-chlorophenyl)-N-(3-ethoxypropyl)-5-(1H-imidazol-2-yl)pyrimidin-2-amine
—— (3S)-1-ethyl-N-[[4-(2-methyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-5-oxopyrrolidine-3-carboxamide —— C24H25N5O2
(3S)-1-ethyl-N-[[4-(2-methyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-5-oxopyrrolidine-3-carboxamide
—— (2S,6R)-2,6-dimethyl-4-(4-pyridin-3-yl-5-thiophen-3-ylpyrimidin-2-yl)morpholine —— C19H20N4OS
(2S,6R)-2,6-dimethyl-4-(4-pyridin-3-yl-5-thiophen-3-ylpyrimidin-2-yl)morpholine
—— 7-[[4-(Diethylamino)-2-methoxyphenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H29N5O2
7-[[4-(Diethylamino)-2-methoxyphenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 4-(4-chlorophenyl)-5-(1-methylimidazol-2-yl)-N-(pyridin-4-ylmethyl)pyrimidin-2-amine —— C20H17ClN6
4-(4-chlorophenyl)-5-(1-methylimidazol-2-yl)-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
—— 5-(2,6-dimethoxypyrimidin-4-yl)-N-(pyridin-4-ylmethyl)-4-thiophen-2-ylpyrimidin-2-amine —— C20H18N6O2S
5-(2,6-dimethoxypyrimidin-4-yl)-N-(pyridin-4-ylmethyl)-4-thiophen-2-ylpyrimidin-2-amine
—— N-[[4-[2-(dimethylamino)-5-pyridin-4-ylpyrimidin-4-yl]phenyl]methyl]-3-methoxypropanamide —— C22H25N5O2
N-[[4-[2-(dimethylamino)-5-pyridin-4-ylpyrimidin-4-yl]phenyl]methyl]-3-methoxypropanamide
—— N-[[4-[2-(dimethylamino)-5-pyridin-4-ylpyrimidin-4-yl]phenyl]methyl]-2-[(2S)-oxan-2-yl]acetamide —— C25H29N5O2
N-[[4-[2-(dimethylamino)-5-pyridin-4-ylpyrimidin-4-yl]phenyl]methyl]-2-[(2S)-oxan-2-yl]acetamide
—— (1S,6R)-N-[[4-[2-(dimethylamino)-5-pyridin-4-ylpyrimidin-4-yl]phenyl]methyl]bicyclo[4.1.0]heptane-7-carboxamide —— C26H29N5O
(1S,6R)-N-[[4-[2-(dimethylamino)-5-pyridin-4-ylpyrimidin-4-yl]phenyl]methyl]bicyclo[4.1.0]heptane-7-carboxamide
—— (6Z)-6-{[5-(4-chlorophenyl)furan-2-yl]methylidene}-2-(2-cyclohexylethyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23ClN4O2S
(6Z)-6-{[5-(4-chlorophenyl)furan-2-yl]methylidene}-2-(2-cyclohexylethyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (1R,2S)-N-[[4-(2-cyclopropyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-2-methylcyclopropane-1-carboxamide —— C24H24N4O
(1R,2S)-N-[[4-(2-cyclopropyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-2-methylcyclopropane-1-carboxamide
—— N-cyclopropyl-4-(4-fluorophenyl)-5-(1H-imidazol-2-yl)pyrimidin-2-amine —— C16H14FN5
N-cyclopropyl-4-(4-fluorophenyl)-5-(1H-imidazol-2-yl)pyrimidin-2-amine
—— 4-(2-methylfuran-3-yl)-5-pyrazin-2-yl-N-(3-pyridin-2-ylpropyl)pyrimidin-2-amine —— C21H20N6O
4-(2-methylfuran-3-yl)-5-pyrazin-2-yl-N-(3-pyridin-2-ylpropyl)pyrimidin-2-amine
—— 4-(furan-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine —— C18H15N5O2
4-(furan-3-yl)-5-(3-methyl-1,2-oxazol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
—— 5-(2,6-dimethoxypyrimidin-4-yl)-N-(3-imidazol-1-ylpropyl)-4-thiophen-2-ylpyrimidin-2-amine —— C20H21N7O2S
5-(2,6-dimethoxypyrimidin-4-yl)-N-(3-imidazol-1-ylpropyl)-4-thiophen-2-ylpyrimidin-2-amine
—— N-[4-(4-chlorophenyl)-5-(1H-imidazol-2-yl)pyrimidin-2-yl]-N',N'-dimethylpropane-1,3-diamine —— C18H21ClN6
N-[4-(4-chlorophenyl)-5-(1H-imidazol-2-yl)pyrimidin-2-yl]-N',N'-dimethylpropane-1,3-diamine
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-4-(2-methylfuran-3-yl)-5-pyridin-4-ylpyrimidin-2-amine —— C21H25N5O
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-4-(2-methylfuran-3-yl)-5-pyridin-4-ylpyrimidin-2-amine
—— 5-(1H-imidazol-2-yl)-4-(4-methoxyphenyl)-N-methyl-N-(2-pyridin-2-ylethyl)pyrimidin-2-amine —— C22H22N6O
5-(1H-imidazol-2-yl)-4-(4-methoxyphenyl)-N-methyl-N-(2-pyridin-2-ylethyl)pyrimidin-2-amine
—— (1S,2R)-N-[[4-(2-cyclopropyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-2-methylcyclopropane-1-carboxamide —— C24H24N4O
(1S,2R)-N-[[4-(2-cyclopropyl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]-2-methylcyclopropane-1-carboxamide
—— N-[(5R)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]furan-2-carboxamide —— C20H20N4O2
N-[(5R)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]furan-2-carboxamide
—— 4-(4-chlorophenyl)-5-(1H-imidazol-2-yl)-N,N-dimethylpyrimidin-2-amine —— C15H14ClN5
4-(4-chlorophenyl)-5-(1H-imidazol-2-yl)-N,N-dimethylpyrimidin-2-amine
—— N-(3-ethenoxypropyl)-5-(1H-imidazol-2-yl)-4-(4-methoxyphenyl)pyrimidin-2-amine —— C19H21N5O2
N-(3-ethenoxypropyl)-5-(1H-imidazol-2-yl)-4-(4-methoxyphenyl)pyrimidin-2-amine
—— (2S,6S)-4-[4-(4-chlorophenyl)-5-(1H-imidazol-2-yl)pyrimidin-2-yl]-2,6-dimethylmorpholine —— C19H20ClN5O
(2S,6S)-4-[4-(4-chlorophenyl)-5-(1H-imidazol-2-yl)pyrimidin-2-yl]-2,6-dimethylmorpholine
—— (3S)-1-tert-butyl-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-oxopyrrolidine-3-carboxamide —— C24H31N5O2
(3S)-1-tert-butyl-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-oxopyrrolidine-3-carboxamide
—— (2R,6R)-4-[5-(1H-imidazol-2-yl)-4-(4-methoxyphenyl)pyrimidin-2-yl]-2,6-dimethylmorpholine —— C20H23N5O2
(2R,6R)-4-[5-(1H-imidazol-2-yl)-4-(4-methoxyphenyl)pyrimidin-2-yl]-2,6-dimethylmorpholine
—— 5-(1H-imidazol-2-yl)-4-(4-methoxyphenyl)-N-(2-pyridin-4-ylethyl)pyrimidin-2-amine —— C21H20N6O
5-(1H-imidazol-2-yl)-4-(4-methoxyphenyl)-N-(2-pyridin-4-ylethyl)pyrimidin-2-amine
—— (3R)-1-tert-butyl-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-oxopyrrolidine-3-carboxamide —— C24H31N5O2
(3R)-1-tert-butyl-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-oxopyrrolidine-3-carboxamide
—— N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]cyclopropanecarboxamide —— C19H22N4O
N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]cyclopropanecarboxamide
—— (3R)-N-[[4-[2-(dimethylamino)-5-pyridin-4-ylpyrimidin-4-yl]phenyl]methyl]-2,2-dimethyl-5-oxooxolane-3-carboxamide —— C25H27N5O3
(3R)-N-[[4-[2-(dimethylamino)-5-pyridin-4-ylpyrimidin-4-yl]phenyl]methyl]-2,2-dimethyl-5-oxooxolane-3-carboxamide
—— (3R)-1-cyclohexyl-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-oxopyrrolidine-3-carboxamide —— C26H33N5O2
(3R)-1-cyclohexyl-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-oxopyrrolidine-3-carboxamide
—— N-[(5S)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]furan-2-carboxamide —— C20H20N4O2
N-[(5S)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]furan-2-carboxamide
—— 5-(2,6-dimethoxypyrimidin-4-yl)-4-(furan-2-yl)-N-[(1S)-1-thiophen-2-ylethyl]pyrimidin-2-amine —— C20H19N5O3S
5-(2,6-dimethoxypyrimidin-4-yl)-4-(furan-2-yl)-N-[(1S)-1-thiophen-2-ylethyl]pyrimidin-2-amine
—— N-[(5S)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]-1,3-thiazole-4-carboxamide —— C19H19N5OS
N-[(5S)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]-1,3-thiazole-4-carboxamide
—— (2S)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]oxolane-2-carboxamide —— C20H24N4O2
(2S)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]oxolane-2-carboxamide
—— 5-[(3,3-Dimethylpiperidin-1-yl)methyl]-3-(4-pyrimidin-4-ylphenyl)-1,2,4-oxadiazole —— C20H23N5O
5-[(3,3-Dimethylpiperidin-1-yl)methyl]-3-(4-pyrimidin-4-ylphenyl)-1,2,4-oxadiazole
—— 2-methoxy-N-[[4-(2-propan-2-yl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]acetamide —— C22H24N4O2
2-methoxy-N-[[4-(2-propan-2-yl-5-pyridin-2-ylpyrimidin-4-yl)phenyl]methyl]acetamide
—— N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-[(2S)-oxan-2-yl]acetamide —— C22H28N4O2
N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2-[(2S)-oxan-2-yl]acetamide
—— N-[(5S)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]-3,3-dimethylbutanamide —— C21H28N4O
N-[(5S)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]-3,3-dimethylbutanamide
—— N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]oxane-4-carboxamide —— C21H26N4O2
N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]oxane-4-carboxamide
—— (3S)-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2,2-dimethyl-5-oxooxolane-3-carboxamide —— C22H26N4O3
(3S)-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-2,2-dimethyl-5-oxooxolane-3-carboxamide
—— (3S)-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-1,1-dioxothiolane-3-carboxamide —— C20H24N4O3S
(3S)-N-[(5R)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-1,1-dioxothiolane-3-carboxamide
—— N-[(5S)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]pyridine-4-carboxamide —— C21H21N5O
N-[(5S)-7,7-dimethyl-2-pyridin-3-yl-6,8-dihydro-5H-quinazolin-5-yl]pyridine-4-carboxamide
—— (3S)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-oxo-1-prop-2-enylpyrrolidine-3-carboxamide —— C23H27N5O2
(3S)-N-[(5S)-7,7-dimethyl-2-pyridin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-5-oxo-1-prop-2-enylpyrrolidine-3-carboxamide