Gougerotin

• 分子结构分类: 有机化合物 - 有机酸及其衍生物 - 肽模拟物
• 英文名称: Gougerotin
• 英文别名: 6-(4-amino-2-oxopyrimidin-1-yl)-4,5-dihydroxy-3-[[3-hydroxy-2-[[2-(methylamino)acetyl]amino]propanoyl]amino]oxane-2-carboxamide
• 化学式: C₁₆H₂₅N₇O₈
• 分子量: 443.41
• InChiKey: AMNAZJFEONUVTD-UHFFFAOYSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  -5.4
• 重原子数：
  31
• 可旋转键数：
  8
• 环数：
  2.0
• sp3杂化的碳原子比例：
  0.56
• 拓扑面积：
  242
• 氢给体数：
  8
• 氢受体数：
  9

文献信息

• Process for producing gougerotin employing Streptomyces microflavus strains
  申请人：Bayer CropScience LP

  公开号：EP2765200A1

  公开（公告）日：2014-08-13

  The invention relates to a fermentation broth obtained by cultivating a gougerotin producing Streptomyces strain, wherein the fermentation broth contains at least about 1 g/L gougerotin. The invention also relates to a method of producing a fermentation broth of a gougerotin producing Streptomyces strain, wherein the fermentation broth contains at least about 1 g/L gougerotin, the method comprising cultivating the Streptomyces strain in a culture medium containing a digestible carbon source and a digestible nitrogen source under aerobic conditions, wherein the culture medium contains an amino acid at a concentration effective to achieve a gougerotin concentration of at least 1 g/L.

  本发明涉及一种通过培养产生钩吻菌素的链霉菌株获得的发酵液，其中发酵液含有至少约1 g/L钩吻菌素。 本发明还涉及一种生产产生钩藤素的链霉菌株的发酵液的方法，其中发酵液含有至少约1克/升钩藤素，该方法包括在好氧条件下，在含有可消化碳源和可消化氮源的培养基中培养链霉菌株，其中培养基含有一种氨基酸，其浓度能有效地使钩藤素浓度达到至少1克/升。
• [EN] PHENANTHRENE-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF AS PLANT VIRUCIDES<br/>[FR] COMPOSÉS HÉTÉROCYCLIQUES CONTENANT UN PHÉNANTHRÈNE, LEUR PROCÉDÉ DE PRÉPARATION ET LEUR APPLICATION COMME COMPOSÉS VIRUCIDES POUR LES PLANTES
  申请人：UNIV NANKAI

  公开号：WO2015027772A1

  公开（公告）日：2015-03-05

  公开了通式（I）所示的含菲杂环类化合物及其制备和在农药上的应用。该化合物的合成方法简单，易于工业化生产。所述含菲杂环类化合物可用作抗植物病毒剂来抑制烟草花叶病毒、辣椒病毒、水稻病毒、番茄病毒、甘薯病毒、马铃薯病毒和瓜类病毒及玉米矮花叶病毒等，尤其是抑制烟草花叶病毒。通式（I）中R1、R2、R3、X1-X7、m和n定义如说明书。
• STREPTOMYCES MICROFLAVUS STRAINS AND METHODS OF THEIR USE TO CONTROL PLANT DISEASES AND PESTS
  申请人：Bayer CropScience LP

  公开号：US20150299754A1

  公开（公告）日：2015-10-22

  The present invention relates to novel strains of Streptomyces microflavus and methods of their use for controlling diseases or pests of a plant. The invention also relates to a fermentation broth obtained by cultivating a gougerotin producing Streptomyces strain, wherein the fermentation broth contains at least about 2 g/L gougerotin. The invention also relates to a method of producing a fermentation broth of a gougerotin producing Streptomyces strain, wherein the fermentation broth contains at least about 2 g/L gougerotin, the method comprising cultivating the Streptomyces strain in a culture medium containing a digestible carbon source and a digestible nitrogen source under aerobic conditions.
• COMPOSITIONS COMPRISING GOUGEROTIN AND AN INSECTICIDE
  申请人：BAYER CROPSCIENCE LP

  公开号：US20150366199A1

  公开（公告）日：2015-12-24

  The present invention relates to a composition comprising isolated gougerotin and at least one insecticide in a synergistically effective amount, with the proviso that the insecticide is not gougerotin. Furthermore, the present invention relates to the use of this composition as well as a method for reducing overall damage of plants and plant parts.
• COMPOSITIONS COMPRISING GOUGEROTIN AND A FUNGICIDE
  申请人：BAYER CROPSCIENCE LP

  公开号：US20150359220A1

  公开（公告）日：2015-12-17

  The present invention relates to a composition comprising isolated gougerotin and at least one fungicide (I) in a synergistically effective amount, with the proviso that fungicide (I) is not gougerotin. Furthermore, the present invention relates to the use of this composition as well as a method for reducing overall damage of plants and plant parts.