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—— (7R)-7-(4-bromophenyl)-3-N-(4-fluorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C27H21BrFN5O2
(7R)-7-(4-bromophenyl)-3-N-(4-fluorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-7-(4-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7R)-7-(4-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-2-benzylsulfanyl-7-(4-bromophenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26BrN5OS
(7S)-2-benzylsulfanyl-7-(4-bromophenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrClN5OS
(7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H19BrN4O3
(7S)-7-(4-bromophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22BrN5OS
(7R)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-(1,3-benzodioxol-5-yl)-7-(4-bromophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C17H12BrN5O2
(7R)-5-(1,3-benzodioxol-5-yl)-7-(4-bromophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7S)-7-(4-bromophenyl)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H28BrN5O2
(7S)-7-(4-bromophenyl)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(4-bromophenyl)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H26BrN5O2
(7S)-7-(4-bromophenyl)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrFN5OS
(7S)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7S)-7-(4-bromophenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrClN5OS
(7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7S)-7-(4-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(4-bromophenyl)-6-N-(2,4-dimethylphenyl)-3-N-(4-fluorophenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H25BrFN5O2
(7R)-7-(4-bromophenyl)-6-N-(2,4-dimethylphenyl)-3-N-(4-fluorophenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-5-(1,3-benzodioxol-5-yl)-7-(4-bromophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C17H12BrN5O2
(7S)-5-(1,3-benzodioxol-5-yl)-7-(4-bromophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21BrClN5OS
(7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C20H15BrN4O3
(7R)-7-(4-bromophenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H23BrClN5O2
(7S)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(4-bromophenyl)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrFN5OS
(7S)-7-(4-bromophenyl)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24BrN5OS
(7R)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrFN5OS
(7R)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21BrClN5OS
(7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H24BrN5O2
(7S)-7-(4-bromophenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrFN5OS
(7R)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H23BrClN5O2
(7R)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22BrN5OS
(7S)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrFN5OS
(7R)-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26BrN5OS
(7R)-2-benzylsulfanyl-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24BrN5OS
(7S)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrClN5OS
(7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28BrN5OS
(7R)-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrFN5OS
(7R)-7-(4-bromophenyl)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-N-(4-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H20BrCl2N5OS
(7S)-7-(4-bromophenyl)-N-(4-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-(4-bromophenyl)-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C16H13BrN4S
(7S)-5-(4-bromophenyl)-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrClN5OS
(7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24BrN5OS
(7S)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21BrFN5OS
(7S)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromo-2-fluorophenyl)-5-(4-bromophenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine —— C16H10Br2FN5
(7S)-7-(5-bromo-2-fluorophenyl)-5-(4-bromophenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrClN5OS
(7R)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-2-[(3-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrClN5OS
(7S)-7-(4-bromophenyl)-2-[(3-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrClN5OS
(7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(5-bromo-2-fluorophenyl)-5-(4-bromophenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine —— C16H10Br2FN5
(7R)-7-(5-bromo-2-fluorophenyl)-5-(4-bromophenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7R)-7-(4-bromophenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H24BrN5O2
(7R)-7-(4-bromophenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrClN5OS
(7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrClN5OS
(7S)-7-(4-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21BrFN5OS
(7R)-7-(4-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-(4-bromophenyl)-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C16H13BrN4S
(7R)-5-(4-bromophenyl)-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-5-(4-bromophenyl)-7-(2-fluorophenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine —— C16H11BrFN5
(7R)-5-(4-bromophenyl)-7-(2-fluorophenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7S)-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28BrN5OS
(7S)-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-bromo-4-fluorophenyl)-5-(4-bromophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C17H11Br2FN4
(7S)-7-(3-bromo-4-fluorophenyl)-5-(4-bromophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine