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—— [7-dibenzothiophen-2-yl-9-[[(3R)-oxolan-3-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-thiazol-5-yl)methanone —— C30H26N2O4S2
[7-dibenzothiophen-2-yl-9-[[(3R)-oxolan-3-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-thiazol-5-yl)methanone
—— (7S)-7-(4-methoxyphenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O4
(7S)-7-(4-methoxyphenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(4-fluorophenyl)-3-[(4-fluorophenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C20H14F2N4O3
(7R)-7-(4-fluorophenyl)-3-[(4-fluorophenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-fluorophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H19FN4O3
(7R)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-fluorophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-3-[(4-fluorophenyl)carbamoyl]-7-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17FN4O4
(7S)-3-[(4-fluorophenyl)carbamoyl]-7-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(3-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7R)-7-(3-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-chlorophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H19ClN4O3
(7S)-7-(4-chlorophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-3-[(3,4-dimethylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O3
(7R)-3-[(3,4-dimethylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-3-[(4-ethoxyphenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H22N4O4
(7R)-3-[(4-ethoxyphenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-3-[(3-methylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H18N4O3
(7S)-3-[(3-methylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-methoxyphenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O4
(7S)-7-(4-methoxyphenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-3-[(3,4-dimethylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O3
(7S)-3-[(3,4-dimethylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(2-ethoxyphenyl)-3-N-(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H28FN5O4
(7R)-7-(2-ethoxyphenyl)-3-N-(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-3-[(4-fluorophenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H17FN4O3
(7R)-3-[(4-fluorophenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-3-[(3-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H20N4O3
(7R)-3-[(3-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-7-(4-methylsulfanylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26ClN5O2S2
(7S)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-7-(4-methylsulfanylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-3-[(3,4-dimethylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C24H22N4O3
(7S)-3-[(3,4-dimethylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-(3,4,5-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C30H29ClN4O4
(7R)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-(3,4,5-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-5-(4-bromophenyl)-N-(4-chlorophenyl)-7-(2-fluorophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H17BrClFN4O
(7R)-5-(4-bromophenyl)-N-(4-chlorophenyl)-7-(2-fluorophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-7-(3,4-dimethoxyphenyl)-2-[(3-fluorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28FN5O4S
(7R)-7-(3,4-dimethoxyphenyl)-2-[(3-fluorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-chlorophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H19ClN4O3
(7R)-7-(4-chlorophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— 7-[2-(3,4-dimethoxyphenyl)ethyl]-6-imino-2-oxo-N-[(1R)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C30H29N5O4
7-[2-(3,4-dimethoxyphenyl)ethyl]-6-imino-2-oxo-N-[(1R)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (7R)-2-[(3-fluorophenyl)methylsulfanyl]-N-(4-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H30FN5O5S
(7R)-2-[(3-fluorophenyl)methylsulfanyl]-N-(4-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-3-[(4-methylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H18N4O3
(7S)-3-[(4-methylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(5-bromo-2-fluorophenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H27BrFN5O2S
(7R)-7-(5-bromo-2-fluorophenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3-[(3-methylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H18N4O3
(7R)-3-[(3-methylphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-5-(4-bromophenyl)-N-(4-chlorophenyl)-7-(2-fluorophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H17BrClFN4O
(7S)-5-(4-bromophenyl)-N-(4-chlorophenyl)-7-(2-fluorophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-3-[(4-fluorophenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C20H15FN4O3
(7R)-3-[(4-fluorophenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-7-(4-methylsulfanylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26ClN5O2S2
(7R)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-7-(4-methylsulfanylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-octyl-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide —— C24H30N2O3
(7R)-N-octyl-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide
—— (7R)-7-(4-fluorophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17FN4O3
(7R)-7-(4-fluorophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— 7-[2-(3,4-dimethoxyphenyl)ethyl]-6-imino-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C30H29N5O4
7-[2-(3,4-dimethoxyphenyl)ethyl]-6-imino-2-oxo-N-[(1S)-1-phenylethyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (7S)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-(3-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H23BrClN5O2
(7S)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-(3-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(3,4-dimethoxyphenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O3S
(7S)-7-(3,4-dimethoxyphenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-acetamidophenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H30N6O2S
(7S)-7-(4-acetamidophenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-methoxyphenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O4
(7R)-7-(4-methoxyphenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-2-[(4-chlorophenyl)methylsulfanyl]-7-(3,4-dimethoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28ClN5O4S
(7R)-2-[(4-chlorophenyl)methylsulfanyl]-7-(3,4-dimethoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2-chlorophenyl)-2-[(3-fluorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClFN5O2S
(7R)-7-(2-chlorophenyl)-2-[(3-fluorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-methylphenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O3
(7R)-7-(4-methylphenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-N-octyl-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide —— C24H30N2O3
(7S)-N-octyl-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide
—— (7R)-7-(3,4-dimethoxyphenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O3S
(7R)-7-(3,4-dimethoxyphenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-[(2,4-dimethylphenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-7-(4-propan-2-ylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C32H35N5O2S
(7S)-2-[(2,4-dimethylphenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-7-(4-propan-2-ylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-hydroxy-3,5-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O5S
(7S)-2-benzylsulfanyl-7-(4-hydroxy-3,5-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-3-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-7-(3,4-dimethoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione —— C26H21BrN2O4S
(7S)-3-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-7-(3,4-dimethoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-7-(2-chlorophenyl)-2-[(3-fluorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClFN5O2S
(7S)-7-(2-chlorophenyl)-2-[(3-fluorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H30ClN5O5S
(7R)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-N-(2-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O5S
(7R)-2-benzylsulfanyl-N-(2-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-acetamidophenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H30N6O2S
(7R)-7-(4-acetamidophenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-N-(2-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O5S
(7S)-2-benzylsulfanyl-N-(2-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2-ethoxyphenyl)-3-N-(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H28FN5O4
(7S)-7-(2-ethoxyphenyl)-3-N-(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide