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—— 7-methyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H23N5O3
7-methyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-fluoro-N-[(2R)-1-hydroxypropan-2-yl]-2-methylquinoline-4-carboxamide —— C14H15FN2O2
7-fluoro-N-[(2R)-1-hydroxypropan-2-yl]-2-methylquinoline-4-carboxamide
—— 7-fluoro-N-[(2S)-2-hydroxypropyl]-2-methylquinoline-4-carboxamide —— C14H15FN2O2
7-fluoro-N-[(2S)-2-hydroxypropyl]-2-methylquinoline-4-carboxamide
—— 7-chloro-N-[(E)-(2,4-dimethoxyphenyl)methylideneamino]quinolin-4-amine —— C18H16ClN3O2
7-chloro-N-[(E)-(2,4-dimethoxyphenyl)methylideneamino]quinolin-4-amine
—— 7-[[(2R)-2-(3,4-dihydro-1H-isoquinolin-2-yl)-3-methylbutyl]amino]-6-nitro-1H-quinazolin-4-one —— C22H25N5O3
7-[[(2R)-2-(3,4-dihydro-1H-isoquinolin-2-yl)-3-methylbutyl]amino]-6-nitro-1H-quinazolin-4-one
—— 7-[[(2S)-2-(3,4-dihydro-1H-isoquinolin-2-yl)-3-methylbutyl]amino]-6-nitro-1H-quinazolin-4-one —— C22H25N5O3
7-[[(2S)-2-(3,4-dihydro-1H-isoquinolin-2-yl)-3-methylbutyl]amino]-6-nitro-1H-quinazolin-4-one
—— 7-cyclopropyl-N-[(2R)-1-hydroxypropan-2-yl]-2,4-dioxo-1-propylpyrido[2,3-d]pyrimidine-5-carboxamide —— C17H22N4O4
7-cyclopropyl-N-[(2R)-1-hydroxypropan-2-yl]-2,4-dioxo-1-propylpyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-N-[(2S)-1-hydroxypropan-2-yl]-2,4-dioxo-1-propylpyrido[2,3-d]pyrimidine-5-carboxamide —— C17H22N4O4
7-cyclopropyl-N-[(2S)-1-hydroxypropan-2-yl]-2,4-dioxo-1-propylpyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-1-ethyl-N-[(2S)-1-hydroxypropan-2-yl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C16H20N4O4
7-cyclopropyl-1-ethyl-N-[(2S)-1-hydroxypropan-2-yl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-[[(2S)-2-(1,3-thiazol-2-yl)morpholin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C14H14N4O2S2
7-[[(2S)-2-(1,3-thiazol-2-yl)morpholin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-methyl-2-[[(2S)-2-(1,3-thiazol-2-yl)morpholin-4-yl]methyl]pyrido[1,2-a]pyrimidin-4-one —— C17H18N4O2S
7-methyl-2-[[(2S)-2-(1,3-thiazol-2-yl)morpholin-4-yl]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-[[(2R)-2-(1,3-thiazol-2-yl)morpholin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C14H14N4O2S2
7-[[(2R)-2-(1,3-thiazol-2-yl)morpholin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-methyl-2-[[(2R)-2-(1,3-thiazol-2-yl)morpholin-4-yl]methyl]pyrido[1,2-a]pyrimidin-4-one —— C17H18N4O2S
7-methyl-2-[[(2R)-2-(1,3-thiazol-2-yl)morpholin-4-yl]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-fluoro-N-[(2S)-1-hydroxypropan-2-yl]-2-methylquinoline-3-carboxamide —— C14H15FN2O2
7-fluoro-N-[(2S)-1-hydroxypropan-2-yl]-2-methylquinoline-3-carboxamide
—— 7-fluoro-N-[(2R)-1-hydroxypropan-2-yl]-2-methylquinoline-3-carboxamide —— C14H15FN2O2
7-fluoro-N-[(2R)-1-hydroxypropan-2-yl]-2-methylquinoline-3-carboxamide
—— 7-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C15H25N3O
7-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C15H17N7
7-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C15H17N7
7-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C15H25N3O
7-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(2R)-4-phenylbutan-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C16H21N3
7-[(2R)-4-phenylbutan-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(1S)-1-(3-fluorophenyl)ethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C14H16FN3
7-[(1S)-1-(3-fluorophenyl)ethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C15H25N3O
7-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C15H25N3O
7-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(1R)-1-(3-fluorophenyl)ethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C14H16FN3
7-[(1R)-1-(3-fluorophenyl)ethyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(2S)-4-phenylbutan-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C16H21N3
7-[(2S)-4-phenylbutan-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-methyl-2-[[(3S)-3-[(pyridin-2-ylamino)methyl]pyrrolidin-1-yl]methyl]pyrido[1,2-a]pyrimidin-4-one —— C20H23N5O
7-methyl-2-[[(3S)-3-[(pyridin-2-ylamino)methyl]pyrrolidin-1-yl]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-methyl-2-[[(3R)-3-[(pyridin-2-ylamino)methyl]pyrrolidin-1-yl]methyl]pyrido[1,2-a]pyrimidin-4-one —— C20H23N5O
7-methyl-2-[[(3R)-3-[(pyridin-2-ylamino)methyl]pyrrolidin-1-yl]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-chloro-N-[(6R)-3-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide —— C16H17ClN4O3
7-chloro-N-[(6R)-3-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide
—— 7-chloro-N-[(6S)-3-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide —— C16H17ClN4O3
7-chloro-N-[(6S)-3-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide
—— 7-fluoro-3-methyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide —— C18H18FN3O2
7-fluoro-3-methyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide
—— 7-chloro-N-[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide —— C15H15ClN4O3
7-chloro-N-[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide
—— 7-fluoro-3-methyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide —— C18H18FN3O2
7-fluoro-3-methyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide
—— 7-chloro-N-[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide —— C15H15ClN4O3
7-chloro-N-[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide
—— 7-fluoro-2-methyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]quinoline-4-carboxamide —— C19H19FN4O
7-fluoro-2-methyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]quinoline-4-carboxamide
—— 7-fluoro-2-methyl-N-[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]quinoline-3-carboxamide —— C18H18FN5O
7-fluoro-2-methyl-N-[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]quinoline-3-carboxamide
—— 7-fluoro-2-methyl-N-[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]quinoline-3-carboxamide —— C18H18FN5O
7-fluoro-2-methyl-N-[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]quinoline-3-carboxamide
—— 7-fluoro-2-methyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]quinoline-4-carboxamide —— C19H19FN4O
7-fluoro-2-methyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]quinoline-4-carboxamide
—— 7-chloro-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide —— C16H16ClN3O3
7-chloro-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide
—— 7-chloro-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide —— C16H16ClN3O3
7-chloro-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide
—— 7-fluoro-2-methyl-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]quinoline-4-carboxamide —— C18H17FN4O
7-fluoro-2-methyl-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]quinoline-4-carboxamide
—— 7-chloro-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide —— C15H14ClN3O3
7-chloro-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide
—— 7-chloro-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide —— C15H14ClN3O3
7-chloro-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1,3-benzodioxole-5-carboxamide
—— 7-chloro-3-methyl-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide —— C17H16ClN3O2
7-chloro-3-methyl-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide
—— 7-fluoro-3-methyl-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide —— C17H16FN3O2
7-fluoro-3-methyl-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide
—— 7-fluoro-3-methyl-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide —— C17H16FN3O2
7-fluoro-3-methyl-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1-benzofuran-2-carboxamide
—— (7R)-2-[(2Z)-2-butan-2-ylidenehydrazinyl]-7-tert-butyl-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H30N4OS
(7R)-2-[(2Z)-2-butan-2-ylidenehydrazinyl]-7-tert-butyl-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-fluoro-N-[(2R)-2-hydroxypropyl]-2-methylquinoline-3-carboxamide —— C14H15FN2O2
7-fluoro-N-[(2R)-2-hydroxypropyl]-2-methylquinoline-3-carboxamide
—— 7-fluoro-N-[(2S)-2-hydroxypropyl]-2-methylquinoline-3-carboxamide —— C14H15FN2O2
7-fluoro-N-[(2S)-2-hydroxypropyl]-2-methylquinoline-3-carboxamide
—— 7-cyclopropyl-N-[(2S)-2-hydroxypropyl]-2,4-dioxo-1-propylpyrido[2,3-d]pyrimidine-5-carboxamide —— C17H22N4O4
7-cyclopropyl-N-[(2S)-2-hydroxypropyl]-2,4-dioxo-1-propylpyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-N-[(2R)-2-hydroxypropyl]-2,4-dioxo-1-propylpyrido[2,3-d]pyrimidine-5-carboxamide —— C17H22N4O4
7-cyclopropyl-N-[(2R)-2-hydroxypropyl]-2,4-dioxo-1-propylpyrido[2,3-d]pyrimidine-5-carboxamide