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—— (7S)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H24BrN5O2S
(7S)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(5-bromofuran-2-yl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23BrClN5O2S
(7R)-7-(5-bromofuran-2-yl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromofuran-2-yl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H19BrFN5O2S
(7S)-7-(5-bromofuran-2-yl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromo-3-hydroxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrClN5O2S
(7S)-7-(4-bromo-3-hydroxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H22BrN5O2S
(7R)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H22BrN5O2S
(7R)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromo-3-hydroxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21BrClN5O2S
(7S)-7-(4-bromo-3-hydroxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H20BrN5O2S
(7R)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[2-(3,4-dimethoxyphenyl)ethyl]-6-imino-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C27H29N5O5
7-[2-(3,4-dimethoxyphenyl)ethyl]-6-imino-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— (7R)-7-(4-bromo-3-hydroxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21BrClN5O2S
(7R)-7-(4-bromo-3-hydroxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromo-3-hydroxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrClN5O2S
(7R)-7-(4-bromo-3-hydroxyphenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-(4-bromophenyl)-N-[(2R)-2-(furan-2-yl)-2-morpholin-4-ylethyl]-5-phenylpyrrolo[2,3-d]pyrimidin-4-amine —— C28H26BrN5O2
7-(4-bromophenyl)-N-[(2R)-2-(furan-2-yl)-2-morpholin-4-ylethyl]-5-phenylpyrrolo[2,3-d]pyrimidin-4-amine
—— (7R,11R,23S,27R)-9,25-dioxaoctacyclo[15.15.0.03,15.05,13.07,11.019,31.021,29.023,27]dotriaconta-1(17),3(15),5(13),19(31),21(29)-pentaene-8,10,24,26-tetrone —— C30H28O6
(7R,11R,23S,27R)-9,25-dioxaoctacyclo[15.15.0.03,15.05,13.07,11.019,31.021,29.023,27]dotriaconta-1(17),3(15),5(13),19(31),21(29)-pentaene-8,10,24,26-tetrone
—— (7R,11R,23R,27R)-9,25-dioxaoctacyclo[15.15.0.03,15.05,13.07,11.019,31.021,29.023,27]dotriaconta-1(17),3(15),5(13),19(31),21(29)-pentaene-8,10,24,26-tetrone —— C30H28O6
(7R,11R,23R,27R)-9,25-dioxaoctacyclo[15.15.0.03,15.05,13.07,11.019,31.021,29.023,27]dotriaconta-1(17),3(15),5(13),19(31),21(29)-pentaene-8,10,24,26-tetrone
—— (7S)-N-(4-bromophenyl)-7-thiophen-2-yl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C25H22BrN3OS2
(7S)-N-(4-bromophenyl)-7-thiophen-2-yl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-9-(4-bromophenyl)-1,7-dimethyl-3-(naphthalen-1-ylmethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C27H24BrN5O2
(7R)-9-(4-bromophenyl)-1,7-dimethyl-3-(naphthalen-1-ylmethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-9-(4-bromophenyl)-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H20BrCl2N5O2
(7R)-9-(4-bromophenyl)-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-9-(4-bromophenyl)-1,7-dimethyl-3-(naphthalen-1-ylmethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C27H24BrN5O2
(7S)-9-(4-bromophenyl)-1,7-dimethyl-3-(naphthalen-1-ylmethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— 7-methoxy-4-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]-5H-pyrimido[5,4-b]indole —— C21H26N4O
7-methoxy-4-[(1R,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]-5H-pyrimido[5,4-b]indole
—— (7S)-9-(4-bromophenyl)-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H20BrCl2N5O2
(7S)-9-(4-bromophenyl)-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26BrN5O2
(7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H19BrN4O3
(7R)-7-(4-bromophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— 7-methoxy-4-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]-5H-pyrimido[5,4-b]indole —— C21H26N4O
7-methoxy-4-[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]-5H-pyrimido[5,4-b]indole
—— (7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23BrN6O2
(7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26BrN5O2
(7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-3-N-(4-fluorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C27H21BrFN5O2
(7S)-7-(4-bromophenyl)-3-N-(4-fluorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25BrN6O2
(7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25BrN6O2
(7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25BrN6O2
(7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24BrN5O2
(7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25BrN6O2
(7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26BrN5O2
(7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23BrN6O2
(7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26BrN5O2
(7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24BrN5O2
(7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24BrN5O2
(7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23BrN6O2
(7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23BrN6O2
(7R)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C27H21BrClN5O2
(7R)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C27H21BrClN5O2
(7S)-7-(4-bromophenyl)-6-N-(4-chlorophenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(4-bromophenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C20H15BrN4O3
(7S)-7-(4-bromophenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24BrN5O2
(7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-N-(4-chlorophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H20BrCl2N5OS
(7R)-7-(4-bromophenyl)-N-(4-chlorophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-N-(4-chlorophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H20BrCl2N5OS
(7S)-7-(4-bromophenyl)-N-(4-chlorophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24BrN5OS
(7R)-2-benzylsulfanyl-7-(4-bromophenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrFN5OS
(7S)-7-(4-bromophenyl)-N-(2,4-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7R)-7-(4-bromophenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-bromophenyl)-5-methyl-3-N-(3-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H24BrN5O2
(7S)-7-(4-bromophenyl)-5-methyl-3-N-(3-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-7-(4-bromophenyl)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H26BrN5O2
(7R)-7-(4-bromophenyl)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-7-(4-bromophenyl)-3-[(2-chlorophenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C20H14BrClN4O3
(7R)-7-(4-bromophenyl)-3-[(2-chlorophenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid