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—— (7,8-dimethyl-2-oxochromen-4-yl)methyl (2S)-2-[(4-methoxyphenyl)sulfonylamino]-3-methylbutanoate —— C24H27NO7S
(7,8-dimethyl-2-oxochromen-4-yl)methyl (2S)-2-[(4-methoxyphenyl)sulfonylamino]-3-methylbutanoate
—— (7-ethyl-2-oxochromen-4-yl)methyl (2R)-2-[(2-chloro-4-nitrobenzoyl)amino]-3-methylbutanoate —— C24H23ClN2O7
(7-ethyl-2-oxochromen-4-yl)methyl (2R)-2-[(2-chloro-4-nitrobenzoyl)amino]-3-methylbutanoate
—— [7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl (2R)-2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate —— C24H26N2O8
[7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl (2R)-2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate
—— [7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl (2S)-2-[(3aR,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate —— C24H26N2O8
[7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl (2S)-2-[(3aR,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate
—— (7-ethyl-2-oxochromen-4-yl)methyl (2R)-2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate —— C23H25NO6
(7-ethyl-2-oxochromen-4-yl)methyl (2R)-2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate
—— (7-methoxy-2-oxochromen-4-yl)methyl (2R)-2-[(4-methoxyphenyl)sulfonylamino]propanoate —— C21H21NO8S
(7-methoxy-2-oxochromen-4-yl)methyl (2R)-2-[(4-methoxyphenyl)sulfonylamino]propanoate
—— [7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 4-[[(2R)-oxolan-2-yl]methoxy]benzoate —— C25H25NO8
[7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 4-[[(2R)-oxolan-2-yl]methoxy]benzoate
—— (7-acetamido-2-oxochromen-4-yl)methyl (2S,3R)-2-(1,3-dioxoisoindol-2-yl)-3-methylpentanoate —— C26H24N2O7
(7-acetamido-2-oxochromen-4-yl)methyl (2S,3R)-2-(1,3-dioxoisoindol-2-yl)-3-methylpentanoate
—— [7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 4-[[(2S)-oxolan-2-yl]methoxy]benzoate —— C25H25NO8
[7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 4-[[(2S)-oxolan-2-yl]methoxy]benzoate
—— (7-acetamido-2-oxochromen-4-yl)methyl (2R,3R)-2-(1,3-dioxoisoindol-2-yl)-3-methylpentanoate —— C26H24N2O7
(7-acetamido-2-oxochromen-4-yl)methyl (2R,3R)-2-(1,3-dioxoisoindol-2-yl)-3-methylpentanoate
—— (7-acetamido-2-oxochromen-4-yl)methyl (2S,3S)-2-(1,3-dioxoisoindol-2-yl)-3-methylpentanoate —— C26H24N2O7
(7-acetamido-2-oxochromen-4-yl)methyl (2S,3S)-2-(1,3-dioxoisoindol-2-yl)-3-methylpentanoate
—— [7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]acetate —— C23H24N2O8
[7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 2-[(3aS,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]acetate
—— [7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]acetate —— C23H24N2O8
[7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 2-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]acetate
—— (7-Chloro-1,3-benzodioxol-5-yl)-[4-(pyridin-4-ylmethyl)piperazin-1-yl]methanone —— C18H18ClN3O3
(7-Chloro-1,3-benzodioxol-5-yl)-[4-(pyridin-4-ylmethyl)piperazin-1-yl]methanone
—— (7-methoxy-2-oxochromen-4-yl)methyl (2S,3R)-2-[(4-chlorobenzoyl)amino]-3-methylpentanoate —— C24H24ClNO6
(7-methoxy-2-oxochromen-4-yl)methyl (2S,3R)-2-[(4-chlorobenzoyl)amino]-3-methylpentanoate
—— (7-methoxy-2-oxochromen-4-yl)methyl (2R,3R)-2-[(4-chlorobenzoyl)amino]-3-methylpentanoate —— C24H24ClNO6
(7-methoxy-2-oxochromen-4-yl)methyl (2R,3R)-2-[(4-chlorobenzoyl)amino]-3-methylpentanoate
—— (7-ethyl-2-oxochromen-4-yl)methyl 4-methoxy-3-[(2R)-2-methylpiperidin-1-yl]sulfonylbenzoate —— C26H29NO7S
(7-ethyl-2-oxochromen-4-yl)methyl 4-methoxy-3-[(2R)-2-methylpiperidin-1-yl]sulfonylbenzoate
—— (7-ethyl-2-oxochromen-4-yl)methyl 4-methoxy-3-[(2S)-2-methylpiperidin-1-yl]sulfonylbenzoate —— C26H29NO7S
(7-ethyl-2-oxochromen-4-yl)methyl 4-methoxy-3-[(2S)-2-methylpiperidin-1-yl]sulfonylbenzoate
—— (7-methoxy-2-oxochromen-4-yl)methyl (2R)-2-(1,3-dioxoisoindol-2-yl)-3-phenylpropanoate —— C28H21NO7
(7-methoxy-2-oxochromen-4-yl)methyl (2R)-2-(1,3-dioxoisoindol-2-yl)-3-phenylpropanoate
—— (7-acetamido-2-oxochromen-4-yl)methyl 2-[(5S,7S)-3-bromo-1-adamantyl]acetate —— C24H26BrNO5
(7-acetamido-2-oxochromen-4-yl)methyl 2-[(5S,7S)-3-bromo-1-adamantyl]acetate
—— (7-acetamido-2-oxochromen-4-yl)methyl 2-[(5R,7R)-3-bromo-1-adamantyl]acetate —— C24H26BrNO5
(7-acetamido-2-oxochromen-4-yl)methyl 2-[(5R,7R)-3-bromo-1-adamantyl]acetate
—— 7-[[methyl-[[4-(trifluoromethyl)phenyl]methyl]amino]methyl]-8H-[1,3]thiazolo[3,2-a]pyrimidin-4-ium-5-one —— C16H15F3N3OS+
7-[[methyl-[[4-(trifluoromethyl)phenyl]methyl]amino]methyl]-8H-[1,3]thiazolo[3,2-a]pyrimidin-4-ium-5-one
—— (7-acetamido-2-oxochromen-4-yl)methyl 2-[(5S,7R)-3-bromo-1-adamantyl]acetate —— C24H26BrNO5
(7-acetamido-2-oxochromen-4-yl)methyl 2-[(5S,7R)-3-bromo-1-adamantyl]acetate
—— (7,8-dimethyl-2-oxochromen-4-yl)methyl (2R)-2-(furan-2-carbonylamino)-3-phenylpropanoate —— C26H23NO6
(7,8-dimethyl-2-oxochromen-4-yl)methyl (2R)-2-(furan-2-carbonylamino)-3-phenylpropanoate
—— [7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl (2R)-2-benzamido-3-methylbutanoate —— C25H26N2O7
[7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl (2R)-2-benzamido-3-methylbutanoate
—— (7E)-1,3-dimethyl-7-[(5-nitrofuran-2-yl)methylidene]purino[8,9-b][1,3]thiazole-2,4,8-trione —— C14H9N5O6S
(7E)-1,3-dimethyl-7-[(5-nitrofuran-2-yl)methylidene]purino[8,9-b][1,3]thiazole-2,4,8-trione
—— (7S)-7-(4-bromophenyl)-5-(4-ethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C19H17BrN4O
(7S)-7-(4-bromophenyl)-5-(4-ethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-2-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H24N2O3S2
(7R)-2-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-(4-bromophenyl)-5-(4-ethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C19H17BrN4O
(7R)-7-(4-bromophenyl)-5-(4-ethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7S)-2-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H24N2O3S2
(7S)-2-[(1S)-1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-chloro-2-[(2S)-1-[(2R)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]sulfanyl-3-(3-methoxypropyl)quinazolin-4-one —— C22H30ClN3O3S
7-chloro-2-[(2S)-1-[(2R)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]sulfanyl-3-(3-methoxypropyl)quinazolin-4-one
—— (7R)-2-[(1R)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24N4O3S2
(7R)-2-[(1R)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24N4O3S2
(7S)-2-[(1R)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-chloro-2-[(2R)-1-[(2R)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]sulfanyl-3-(3-methoxypropyl)quinazolin-4-one —— C22H30ClN3O3S
7-chloro-2-[(2R)-1-[(2R)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]sulfanyl-3-(3-methoxypropyl)quinazolin-4-one
—— (7S)-2-[(1S)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24N4O3S2
(7S)-2-[(1S)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24N4O3S2
(7R)-2-[(1S)-1-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-chloro-2-[(2R)-1-[(2S)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]sulfanyl-3-(3-methoxypropyl)quinazolin-4-one —— C22H30ClN3O3S
7-chloro-2-[(2R)-1-[(2S)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]sulfanyl-3-(3-methoxypropyl)quinazolin-4-one
—— 7-chloro-2-[(2S)-1-[(2S)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]sulfanyl-3-(3-methoxypropyl)quinazolin-4-one —— C22H30ClN3O3S
7-chloro-2-[(2S)-1-[(2S)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]sulfanyl-3-(3-methoxypropyl)quinazolin-4-one
—— 7-fluoro-3-methyl-N-[[2-(pyrrolidin-1-ylmethyl)phenyl]methyl]-1-benzofuran-2-carboxamide —— C22H23FN2O2
7-fluoro-3-methyl-N-[[2-(pyrrolidin-1-ylmethyl)phenyl]methyl]-1-benzofuran-2-carboxamide
—— 7-[(2-methoxyacetyl)amino]-1-methyl-2-phenyl-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide —— C28H30N4O3
7-[(2-methoxyacetyl)amino]-1-methyl-2-phenyl-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide
—— 7-[(2-methoxyacetyl)amino]-1-methyl-2-phenyl-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide —— C28H30N4O3
7-[(2-methoxyacetyl)amino]-1-methyl-2-phenyl-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide
—— 7-[(2-methoxyacetyl)amino]-1-methyl-2-phenyl-N-[[(1R,2S,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide —— C28H30N4O3
7-[(2-methoxyacetyl)amino]-1-methyl-2-phenyl-N-[[(1R,2S,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide
—— (7-Chloro-1,3-benzodioxol-5-yl)-(4-pyrimidin-2-ylpiperazin-1-yl)methanone —— C16H15ClN4O3
(7-Chloro-1,3-benzodioxol-5-yl)-(4-pyrimidin-2-ylpiperazin-1-yl)methanone
—— 7-(cyclobutanecarbonylamino)-1-methyl-2-pyridin-4-yl-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide —— C29H31N5O2
7-(cyclobutanecarbonylamino)-1-methyl-2-pyridin-4-yl-N-[[(1R,2R,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide
—— (7Z)-7-[2-(4-cyclohexylphenyl)-2-oxoethylidene]-1,3,5,8-tetrahydroimidazo[4,5-g]quinoxaline-2,6-dione —— C23H22N4O3
(7Z)-7-[2-(4-cyclohexylphenyl)-2-oxoethylidene]-1,3,5,8-tetrahydroimidazo[4,5-g]quinoxaline-2,6-dione
—— 7-(cyclobutanecarbonylamino)-1-methyl-2-pyridin-4-yl-N-[[(1R,2S,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide —— C29H31N5O2
7-(cyclobutanecarbonylamino)-1-methyl-2-pyridin-4-yl-N-[[(1R,2S,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide
—— 7-(cyclobutanecarbonylamino)-1-methyl-2-pyridin-4-yl-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide —— C29H31N5O2
7-(cyclobutanecarbonylamino)-1-methyl-2-pyridin-4-yl-N-[[(1R,2R,4S)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide
—— 7-(cyclobutanecarbonylamino)-1-methyl-2-pyridin-4-yl-N-[[(1R,2S,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide —— C29H31N5O2
7-(cyclobutanecarbonylamino)-1-methyl-2-pyridin-4-yl-N-[[(1R,2S,4R)-spiro[bicyclo[2.2.1]hept-5-ene-7,1'-cyclopropane]-2-yl]methyl]benzimidazole-5-carboxamide
—— 7-[[5-(Cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C13H13N5OS3
7-[[5-(Cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (7-methyl-2-oxochromen-4-yl)methyl (2R)-2-[(4-bromophenyl)sulfonylamino]-3-hydroxypropanoate —— C20H18BrNO7S
(7-methyl-2-oxochromen-4-yl)methyl (2R)-2-[(4-bromophenyl)sulfonylamino]-3-hydroxypropanoate