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—— 7-methoxy-3-({(E)-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methylidene}amino)-3,5-dihydro-4H-pyrimido[5,4-b]indol-4-one —— C24H25N5O3
7-methoxy-3-({(E)-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methylidene}amino)-3,5-dihydro-4H-pyrimido[5,4-b]indol-4-one
—— (7R)-3-[(4-ethoxyphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O4
(7R)-3-[(4-ethoxyphenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-methylphenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H18N4O3
(7S)-7-(4-methylphenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— [7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2R)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-fluorophenyl)methanone —— C27H23ClF4N2O4
[7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2R)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-fluorophenyl)methanone
—— (7S)-7-(4-methylphenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O3
(7S)-7-(4-methylphenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(2,5-dimethoxyphenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C24H24N4O5
(7S)-7-(2,5-dimethoxyphenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(2-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7R)-7-(2-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-3-[(4-fluorophenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C20H15FN4O3
(7S)-3-[(4-fluorophenyl)carbamoyl]-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(4-methylphenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H18N4O3
(7R)-7-(4-methylphenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(2,5-dimethoxyphenyl)-3-[(4-fluorophenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H19FN4O5
(7R)-7-(2,5-dimethoxyphenyl)-3-[(4-fluorophenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— [7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2S)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-fluorophenyl)methanone —— C27H23ClF4N2O4
[7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2S)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-fluorophenyl)methanone
—— (7S)-3-[(2-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H20N4O3
(7S)-3-[(2-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— [7-dibenzothiophen-2-yl-9-[[(3S)-oxolan-3-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyridin-2-ylmethanone —— C32H28N2O4S
[7-dibenzothiophen-2-yl-9-[[(3S)-oxolan-3-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyridin-2-ylmethanone
—— (7R)-3-[(2-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H20N4O3
(7R)-3-[(2-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— [7-dibenzothiophen-2-yl-9-[[(3R)-oxolan-3-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyridin-2-ylmethanone —— C32H28N2O4S
[7-dibenzothiophen-2-yl-9-[[(3R)-oxolan-3-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyridin-2-ylmethanone
—— (7R)-7-(4-methoxyphenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O4
(7R)-7-(4-methoxyphenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H22N4O3
(7R)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-3-[(4-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H20N4O3
(7R)-3-[(4-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(3,4-dimethoxyphenyl)-2-[(3-fluorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28FN5O4S
(7S)-7-(3,4-dimethoxyphenyl)-2-[(3-fluorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-methylphenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O3
(7R)-7-(4-methylphenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H22N4O3
(7S)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— [7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2S)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-cyclohexylmethanone —— C27H30ClF3N2O4
[7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2S)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-cyclohexylmethanone
—— (7R)-7-(4-methoxyphenyl)-3-[(4-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O4
(7R)-7-(4-methoxyphenyl)-3-[(4-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-fluorophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17FN4O3
(7S)-7-(4-fluorophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(3-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7S)-7-(3-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-methylphenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O3
(7S)-7-(4-methylphenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-methoxyphenyl)-3-[(4-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O4
(7S)-7-(4-methoxyphenyl)-3-[(4-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H22N4O4
(7S)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-N-(4-ethoxyphenyl)-5-(4-ethylphenyl)-7-(2,4,5-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C32H34N4O5
(7S)-N-(4-ethoxyphenyl)-5-(4-ethylphenyl)-7-(2,4,5-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-7-(2,4-dichlorophenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25Cl2N5OS
(7R)-7-(2,4-dichlorophenyl)-2-[(2,4-dimethylphenyl)methylsulfanyl]-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H22N4O4
(7R)-3-[(3,4-dimethylphenyl)carbamoyl]-7-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(2-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7S)-7-(2-bromophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-chlorophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17ClN4O3
(7S)-7-(4-chlorophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-3-[(4-fluorophenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H17FN4O3
(7S)-3-[(4-fluorophenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— [7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2R)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-methylthiophen-2-yl)methanone —— C26H24ClF3N2O4S
[7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2R)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-methylthiophen-2-yl)methanone
—— [7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2R)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-cyclohexylmethanone —— C27H30ClF3N2O4
[7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2R)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-cyclohexylmethanone
—— (7S)-3-[(4-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H20N4O3
(7S)-3-[(4-methylphenyl)carbamoyl]-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-3-[(4-fluorophenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17FN4O3
(7R)-3-[(4-fluorophenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-N-(4-ethoxyphenyl)-5-(4-ethylphenyl)-7-(2,4,5-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C32H34N4O5
(7R)-N-(4-ethoxyphenyl)-5-(4-ethylphenyl)-7-(2,4,5-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-(3,4,5-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C30H29ClN4O4
(7S)-5-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-(3,4,5-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-2-[(3-fluorophenyl)methylsulfanyl]-N-(4-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H30FN5O5S
(7S)-2-[(3-fluorophenyl)methylsulfanyl]-N-(4-methoxyphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— [7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2S)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-methylthiophen-2-yl)methanone —— C26H24ClF3N2O4S
[7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2S)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(3-methylthiophen-2-yl)methanone
—— (7S)-3-(phenylcarbamoyl)-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H18N4O3
(7S)-3-(phenylcarbamoyl)-7-[(E)-2-phenylethenyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-2-[(4-chlorophenyl)methylsulfanyl]-7-(3,4-dimethoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28ClN5O4S
(7S)-2-[(4-chlorophenyl)methylsulfanyl]-7-(3,4-dimethoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-hydroxy-3,5-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O5S
(7R)-2-benzylsulfanyl-7-(4-hydroxy-3,5-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-3-[(4-ethoxyphenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C23H22N4O4
(7S)-3-[(4-ethoxyphenyl)carbamoyl]-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(4-methylphenyl)-3-[(4-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H20N4O3
(7S)-7-(4-methylphenyl)-3-[(4-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-3-[(4-fluorophenyl)carbamoyl]-7-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17FN4O4
(7R)-3-[(4-fluorophenyl)carbamoyl]-7-(4-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— [7-dibenzothiophen-2-yl-9-[[(3S)-oxolan-3-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-thiazol-5-yl)methanone —— C30H26N2O4S2
[7-dibenzothiophen-2-yl-9-[[(3S)-oxolan-3-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-thiazol-5-yl)methanone
—— (7R)-7-(4-chlorophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17ClN4O3
(7R)-7-(4-chlorophenyl)-3-[(3-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid