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—— (7S)-7-(3-bromophenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7S)-7-(3-bromophenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(3-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H20BrFN6OS
(7S)-7-(3-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-bromophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H19BrN4O3
(7S)-7-(3-bromophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(3-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28BrN5OS
(7R)-7-(3-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C22H19BrN4O3
(7R)-7-(3-bromophenyl)-3-[(3,4-dimethylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7R)-7-(3-bromophenyl)-N-(4-chlorophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H20BrCl2N5OS
(7R)-7-(3-bromophenyl)-N-(4-chlorophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21BrClN5OS
(7S)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(3-bromophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22BrN5OS
(7R)-2-benzylsulfanyl-7-(3-bromophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-bromophenyl)-N-(4-chlorophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H20BrCl2N5OS
(7S)-7-(3-bromophenyl)-N-(4-chlorophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-(3-bromophenyl)-7-(2-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C16H11BrFN5
(7R)-5-(3-bromophenyl)-7-(2-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7S)-7-(5-bromo-2-fluorophenyl)-5-(3-bromophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C17H11Br2FN4
(7S)-7-(5-bromo-2-fluorophenyl)-5-(3-bromophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21BrClN5OS
(7R)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H20BrFN6OS
(7R)-7-(3-bromophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrClN5OS
(7R)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrClN5OS
(7R)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-(3-bromophenyl)-7-(2-chloro-6-fluorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C17H11BrClFN4
(7R)-5-(3-bromophenyl)-7-(2-chloro-6-fluorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-7-(5-bromo-2-fluorophenyl)-5-(3-bromophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C17H11Br2FN4
(7R)-7-(5-bromo-2-fluorophenyl)-5-(3-bromophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7S)-7-(3-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28BrN5OS
(7S)-7-(3-bromophenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromophenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C21H17BrN4O3
(7R)-7-(3-bromophenyl)-3-[(2-methylphenyl)carbamoyl]-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(3-bromophenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid —— C20H15BrN4O3
(7S)-7-(3-bromophenyl)-3-(phenylcarbamoyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-7-(3-bromophenyl)-2-[(3-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrClN5OS
(7S)-7-(3-bromophenyl)-2-[(3-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H25BrClN5OS
(7S)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-(3-bromophenyl)-7-(2-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C16H11BrFN5
(7S)-5-(3-bromophenyl)-7-(2-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7S)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrClN5OS
(7S)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-(3-bromophenyl)-7-(2-chloro-6-fluorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C17H11BrClFN4
(7S)-5-(3-bromophenyl)-7-(2-chloro-6-fluorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7S)-2-benzylsulfanyl-7-(3-bromophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22BrN5OS
(7S)-2-benzylsulfanyl-7-(3-bromophenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromo-2-fluorophenyl)-5-(3-bromophenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine —— C16H10Br2FN5
(7S)-7-(5-bromo-2-fluorophenyl)-5-(3-bromophenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7S)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrClN5OS
(7S)-7-(3-bromophenyl)-2-[(2-chlorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-Methyl-2,2-di(propan-2-yl)-1,2-benzoxasiline —— C15H22OSi
7-Methyl-2,2-di(propan-2-yl)-1,2-benzoxasiline
—— 7-deacetylgedunin —— C26H32O6
7-deacetylgedunin
—— 7-Desacetoxy-7-oxo-14(15)-desoxygedunin —— C26H30O5
7-Desacetoxy-7-oxo-14(15)-desoxygedunin
—— (7S)-5-(5-bromothiophen-2-yl)-7-(2-chloro-6-fluorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C15H9BrClFN4S
(7S)-5-(5-bromothiophen-2-yl)-7-(2-chloro-6-fluorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7S)-7-(5-bromofuran-2-yl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H21BrFN5O2S
(7S)-7-(5-bromofuran-2-yl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23BrFN5O2S
(7S)-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-(5-bromothiophen-2-yl)-7-(2-chloro-6-fluorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C15H9BrClFN4S
(7R)-5-(5-bromothiophen-2-yl)-7-(2-chloro-6-fluorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-7-(5-bromothiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxylic acid —— C10H7BrN4O2S
(7R)-7-(5-bromothiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxylic acid
—— (7S)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H22BrN5O2S
(7S)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromofuran-2-yl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23BrClN5O2S
(7S)-7-(5-bromofuran-2-yl)-2-[(2-chlorophenyl)methylsulfanyl]-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H24BrN5O2S
(7R)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-(5-bromothiophen-2-yl)-7-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C16H13BrN4S
(7S)-5-(5-bromothiophen-2-yl)-7-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7S)-5-(5-bromothiophen-2-yl)-7-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C15H12BrN5S
(7S)-5-(5-bromothiophen-2-yl)-7-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7R)-5-(5-bromothiophen-2-yl)-7-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C16H13BrN4S
(7R)-5-(5-bromothiophen-2-yl)-7-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-5-(5-bromothiophen-2-yl)-7-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C15H12BrN5S
(7R)-5-(5-bromothiophen-2-yl)-7-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7R)-7-(5-bromofuran-2-yl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H21BrFN5O2S
(7R)-7-(5-bromofuran-2-yl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(5-bromofuran-2-yl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H21BrFN5O2S
(7R)-7-(5-bromofuran-2-yl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H22BrN5O2S
(7S)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-(2-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-chloro-2,8-dimethyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one —— C22H29ClN2O
7-chloro-2,8-dimethyl-3-[[(1S,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methyl]-1H-quinolin-4-one
—— (7R)-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23BrFN5O2S
(7R)-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H20BrN5O2S
(7S)-2-benzylsulfanyl-7-(5-bromofuran-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromothiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxylic acid —— C10H7BrN4O2S
(7S)-7-(5-bromothiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxylic acid