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—— (6R,9R)-6-(2-chloro-6-fluorophenyl)-9-phenyl-5,6,6a,8,9,10-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H20ClFN2O
(6R,9R)-6-(2-chloro-6-fluorophenyl)-9-phenyl-5,6,6a,8,9,10-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R,6aR,9R)-9-(4-methoxyphenyl)-3-methyl-6-thiophen-2-yl-5,6,6a,8,9,10-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H24N2O2S
(6R,6aR,9R)-9-(4-methoxyphenyl)-3-methyl-6-thiophen-2-yl-5,6,6a,8,9,10-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-chloro-4-N-[[(3R)-1-(2-morpholin-4-ylethyl)pyrrolidin-3-yl]methyl]pyrimidine-2,4-diamine —— C15H25ClN6O
6-chloro-4-N-[[(3R)-1-(2-morpholin-4-ylethyl)pyrrolidin-3-yl]methyl]pyrimidine-2,4-diamine
—— (6R)-2-(4-methoxyphenyl)imino-N-(2-methyl-4-nitrophenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C19H18N4O5S
(6R)-2-(4-methoxyphenyl)imino-N-(2-methyl-4-nitrophenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S)-2-(azepan-1-yl)-6-ethyl-5-phenyl-6H-1,3,4-thiadiazine —— C17H23N3S
(6S)-2-(azepan-1-yl)-6-ethyl-5-phenyl-6H-1,3,4-thiadiazine
—— 6-chloro-4-N-[[(3S)-1-(2-morpholin-4-ylethyl)pyrrolidin-3-yl]methyl]pyrimidine-2,4-diamine —— C15H25ClN6O
6-chloro-4-N-[[(3S)-1-(2-morpholin-4-ylethyl)pyrrolidin-3-yl]methyl]pyrimidine-2,4-diamine
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C17H15ClN4O4
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate
—— 6-[[[(6R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C15H22N6O2
6-[[[(6R)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 5-nitrothiophene-2-carboxylate —— C14H10ClNO6S
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 5-nitrothiophene-2-carboxylate
—— 6-chloro-3-oxo-N-[(R)-(4-propan-2-ylphenyl)-thiophen-2-ylmethyl]-4H-1,4-benzoxazine-7-sulfonamide —— C22H21ClN2O4S2
6-chloro-3-oxo-N-[(R)-(4-propan-2-ylphenyl)-thiophen-2-ylmethyl]-4H-1,4-benzoxazine-7-sulfonamide
—— 6-chloro-3-oxo-N-[(S)-(4-propan-2-ylphenyl)-thiophen-2-ylmethyl]-4H-1,4-benzoxazine-7-sulfonamide —— C22H21ClN2O4S2
6-chloro-3-oxo-N-[(S)-(4-propan-2-ylphenyl)-thiophen-2-ylmethyl]-4H-1,4-benzoxazine-7-sulfonamide
—— 6-[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]pyridine-3-carbonitrile —— C13H14N6
6-[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]pyridine-3-carbonitrile
—— 6-[[[(6S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C15H22N6O2
6-[[[(6S)-2-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— (6S)-2-ethyl-N-[[3-(furan-3-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H18N6O2
(6S)-2-ethyl-N-[[3-(furan-3-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-2-ethyl-N-[[3-(furan-3-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H18N6O2
(6R)-2-ethyl-N-[[3-(furan-3-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[(2S)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]pyridine-3-carbonitrile —— C13H14N6
6-[(2S)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]pyridine-3-carbonitrile
—— 6-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole —— C13H16N6S
6-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]imidazo[2,1-b][1,3]thiazole
—— 6-tert-butyl-2-[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole —— C15H21N7S
6-tert-butyl-2-[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole
—— 6-chloro-8-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]quinoline —— C17H18ClN5
6-chloro-8-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]quinoline
—— 6-tert-butyl-2-[(2S)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole —— C15H21N7S
6-tert-butyl-2-[(2S)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole
—— 6-chloro-8-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]quinoline —— C17H18ClN5
6-chloro-8-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)pyrrolidin-1-yl]methyl]quinoline
—— 6-chloro-4-N-methyl-4-N-[(7R)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]pyrimidine-2,4-diamine —— C13H16ClN5S
6-chloro-4-N-methyl-4-N-[(7R)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]pyrimidine-2,4-diamine
—— (6S)-N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H18N6O
(6S)-N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-[[3-[(4-fluorophenoxy)methyl]-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H17FN6O2
(6R)-N-[[3-[(4-fluorophenoxy)methyl]-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[[3-[(4-fluorophenoxy)methyl]-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H17FN6O2
(6S)-N-[[3-[(4-fluorophenoxy)methyl]-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-6-[[[(1S)-2-methyl-1-thiophen-2-ylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C16H23N5OS
(6R)-6-[[[(1S)-2-methyl-1-thiophen-2-ylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-N-[[5-(3-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H18N6O
(6S)-N-[[5-(3-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-chloro-4-N-methyl-4-N-[(7S)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]pyrimidine-2,4-diamine —— C13H16ClN5S
6-chloro-4-N-methyl-4-N-[(7S)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-yl]pyrimidine-2,4-diamine
—— (6S)-6-[[[(1R)-2-methyl-1-thiophen-2-ylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C16H23N5OS
(6S)-6-[[[(1R)-2-methyl-1-thiophen-2-ylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-N-(2-benzhydryloxyethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C21H24N4O
(6S)-N-(2-benzhydryloxyethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-[(4-piperidin-1-ylphenyl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H25N5
(6R)-N-[(4-piperidin-1-ylphenyl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-(cyclopropylamino)-N-[(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl]pyridine-3-carboxamide —— C17H24N4O2
6-(cyclopropylamino)-N-[(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl]pyridine-3-carboxamide
—— (6R)-N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H18N6O
(6R)-N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-6-[[[(1S)-2-methyl-1-thiophen-2-ylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C16H23N5OS
(6S)-6-[[[(1S)-2-methyl-1-thiophen-2-ylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-N-[(4-piperidin-1-ylphenyl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H25N5
(6S)-N-[(4-piperidin-1-ylphenyl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-6-[[[(1R)-2-methyl-1-thiophen-2-ylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C16H23N5OS
(6R)-6-[[[(1R)-2-methyl-1-thiophen-2-ylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(1S)-2-methyl-1-phenylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O
(6R)-6-[[[(1S)-2-methyl-1-phenylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(1R)-2-methyl-1-phenylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O
(6R)-6-[[[(1R)-2-methyl-1-phenylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[(1R)-2-methyl-1-phenylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O
(6S)-6-[[[(1R)-2-methyl-1-phenylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(1R)-1-phenylbutyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O
(6R)-6-[[[(1R)-1-phenylbutyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[(1S)-2-methyl-1-phenylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O
(6S)-6-[[[(1S)-2-methyl-1-phenylpropyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-Amino-5-[2-(2,5-dimethylphenyl)sulfanylacetyl]-1-propylpyrimidine-2,4-dione —— C17H21N3O3S
6-Amino-5-[2-(2,5-dimethylphenyl)sulfanylacetyl]-1-propylpyrimidine-2,4-dione
—— (6R)-6-[[[(1S)-1-phenylbutyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O
(6R)-6-[[[(1S)-1-phenylbutyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-chloro-3-piperidin-1-ium-4-yl-1H-benzimidazol-2-one —— C12H15ClN3O+
6-chloro-3-piperidin-1-ium-4-yl-1H-benzimidazol-2-one
—— (6S)-5-oxo-7,8-dihydro-6H-thieno[2,3-b]indolizine-6-carbonitrile —— C11H8N2OS
(6S)-5-oxo-7,8-dihydro-6H-thieno[2,3-b]indolizine-6-carbonitrile
—— (6R)-6-(4-chlorophenyl)-9,9-dimethyl-5-(2-methylpropanoyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H27ClN2O2
(6R)-6-(4-chlorophenyl)-9,9-dimethyl-5-(2-methylpropanoyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-5-oxo-7,8-dihydro-6H-thieno[2,3-b]indolizine-6-carbonitrile —— C11H8N2OS
(6R)-5-oxo-7,8-dihydro-6H-thieno[2,3-b]indolizine-6-carbonitrile
—— 6-Chloro-4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanylmethyl)-7-methylchromen-2-one —— C19H15ClO4S
6-Chloro-4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanylmethyl)-7-methylchromen-2-one
—— (6S)-6-[[[(1S)-1-phenylbutyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O
(6S)-6-[[[(1S)-1-phenylbutyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-methyl-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-5-phenylthieno[2,3-d]pyrimidin-4-one —— C21H23N3O2S
6-methyl-3-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-5-phenylthieno[2,3-d]pyrimidin-4-one