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—— (6-ethoxy-1H-indol-2-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone —— C19H22N4O2
(6-ethoxy-1H-indol-2-yl)-[(3R)-3-imidazol-1-ylpiperidin-1-yl]methanone
—— 6-methyl-2-[[[(3R)-1-pyridazin-3-ylpiperidin-3-yl]amino]methyl]pyridin-3-ol —— C16H21N5O
6-methyl-2-[[[(3R)-1-pyridazin-3-ylpiperidin-3-yl]amino]methyl]pyridin-3-ol
—— (6S)-N-(2-naphthalen-2-yloxyethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H20N4O
(6S)-N-(2-naphthalen-2-yloxyethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[2-[(2S)-2-[(2R)-1-ethylpyrrolidin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]-methylamino]pyridine-3-carbonitrile —— C19H27N5O
6-[[2-[(2S)-2-[(2R)-1-ethylpyrrolidin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]-methylamino]pyridine-3-carbonitrile
—— (6S)-2-ethyl-N-[(2-pyridin-2-yl-1,3-thiazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H20N6S
(6S)-2-ethyl-N-[(2-pyridin-2-yl-1,3-thiazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-4-(1-tert-butyl-3,5-dimethylpyrazol-4-yl)sulfonyl-2,2,6-trimethylmorpholine —— C16H29N3O3S
(6S)-4-(1-tert-butyl-3,5-dimethylpyrazol-4-yl)sulfonyl-2,2,6-trimethylmorpholine
—— (6R)-2-ethyl-N-[(2-pyridin-2-yl-1,3-thiazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H20N6S
(6R)-2-ethyl-N-[(2-pyridin-2-yl-1,3-thiazol-4-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-4-(1-tert-butyl-3,5-dimethylpyrazol-4-yl)sulfonyl-2,2,6-trimethylmorpholine —— C16H29N3O3S
(6R)-4-(1-tert-butyl-3,5-dimethylpyrazol-4-yl)sulfonyl-2,2,6-trimethylmorpholine
—— 6-ethoxy-N-[(2R)-1-ethylsulfonylpropan-2-yl]-1H-indole-2-carboxamide —— C16H22N2O4S
6-ethoxy-N-[(2R)-1-ethylsulfonylpropan-2-yl]-1H-indole-2-carboxamide
—— 6-((2-(1,3-dioxolan-2-yl)ethyl)thio)-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one —— C10H12N4O3S
6-((2-(1,3-dioxolan-2-yl)ethyl)thio)-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one
—— 6-[(2S)-butan-2-yl]sulfanyl-1,5-dihydropyrazolo[3,4-d]pyrimidin-4-one —— C9H12N4OS
6-[(2S)-butan-2-yl]sulfanyl-1,5-dihydropyrazolo[3,4-d]pyrimidin-4-one
—— 6-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-4H-1,4-benzothiazin-3-one —— C17H18N4O2S
6-[(2R)-2-(pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-4H-1,4-benzothiazin-3-one
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 3-hydroxybenzoate —— C19H16O5
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 3-hydroxybenzoate
—— 6-methyl-2-[[[(3S)-1-pyridazin-3-ylpiperidin-3-yl]amino]methyl]pyridin-3-ol —— C16H21N5O
6-methyl-2-[[[(3S)-1-pyridazin-3-ylpiperidin-3-yl]amino]methyl]pyridin-3-ol
—— 6-ethoxy-N-[(2S)-1-ethylsulfonylpropan-2-yl]-1H-indole-2-carboxamide —— C16H22N2O4S
6-ethoxy-N-[(2S)-1-ethylsulfonylpropan-2-yl]-1H-indole-2-carboxamide
—— 6-bromo-3-(4-phenylpiperazin-1-yl)-4H-thiochromen-4-one —— C19H17BrN2OS
6-bromo-3-(4-phenylpiperazin-1-yl)-4H-thiochromen-4-one
—— 6-bromo-3-[(2R)-2-methyl-2,3-dihydroindol-1-yl]thiochromen-4-one —— C18H14BrNOS
6-bromo-3-[(2R)-2-methyl-2,3-dihydroindol-1-yl]thiochromen-4-one
—— (6R)-6-[[[(2S)-2-methoxy-2-phenylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H23N5O2
(6R)-6-[[[(2S)-2-methoxy-2-phenylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-Bromo-3-morpholin-4-ylthiochromen-4-one —— C13H12BrNO2S
6-Bromo-3-morpholin-4-ylthiochromen-4-one
—— 6-Bromo-3-(1,2,3,4-tetrahydroisoquinolin-2-YL)-4H-thiochromen-4-one —— C18H14BrNOS
6-Bromo-3-(1,2,3,4-tetrahydroisoquinolin-2-YL)-4H-thiochromen-4-one
—— 6-bromo-3-[(2S)-2-ethylpiperidin-1-yl]thiochromen-4-one —— C16H18BrNOS
6-bromo-3-[(2S)-2-ethylpiperidin-1-yl]thiochromen-4-one
—— (6S)-6-[[[(1R)-1-(3-ethoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O2
(6S)-6-[[[(1R)-1-(3-ethoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-bromo-3-[(2R)-2-ethylpiperidin-1-yl]thiochromen-4-one —— C16H18BrNOS
6-bromo-3-[(2R)-2-ethylpiperidin-1-yl]thiochromen-4-one
—— [6-[(3-Fluorophenyl)methyl]furo[2,3-b]pyrrol-5-yl]-pyrrolidin-1-ylmethanone —— C18H17FN2O2
[6-[(3-Fluorophenyl)methyl]furo[2,3-b]pyrrol-5-yl]-pyrrolidin-1-ylmethanone
—— (6S)-N-[(5-phenyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H17N5O
(6S)-N-[(5-phenyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-bromo-3-[(3S,5S)-3,5-dimethylpiperidin-1-yl]thiochromen-4-one —— C16H18BrNOS
6-bromo-3-[(3S,5S)-3,5-dimethylpiperidin-1-yl]thiochromen-4-one
—— 6-bromo-3-(4-ethylpiperazin-1-yl)-4H-thiochromen-4-one —— C15H17BrN2OS
6-bromo-3-(4-ethylpiperazin-1-yl)-4H-thiochromen-4-one
—— 6-bromo-3-[(3R,5R)-3,5-dimethylpiperidin-1-yl]thiochromen-4-one —— C16H18BrNOS
6-bromo-3-[(3R,5R)-3,5-dimethylpiperidin-1-yl]thiochromen-4-one
—— 6-[[(1R)-1-[5-fluoro-2-(4-hydroxypiperidin-1-yl)phenyl]ethyl]amino]pyridine-3-carbonitrile —— C19H21FN4O
6-[[(1R)-1-[5-fluoro-2-(4-hydroxypiperidin-1-yl)phenyl]ethyl]amino]pyridine-3-carbonitrile
—— 6-methyl-N-[[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C13H17N7S
6-methyl-N-[[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— 6-Bromo-3-pyrrolidin-1-ylthiochromen-4-one —— C13H12BrNOS
6-Bromo-3-pyrrolidin-1-ylthiochromen-4-one
—— (6R)-6-[[[(1R)-1-(3-ethoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O2
(6R)-6-[[[(1R)-1-(3-ethoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(2R)-2-methoxy-2-phenylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H23N5O2
(6R)-6-[[[(2R)-2-methoxy-2-phenylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[(2R)-2-methoxy-2-phenylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H23N5O2
(6S)-6-[[[(2R)-2-methoxy-2-phenylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-chloro-3-ethyl-2-[(1R)-1-[(3R)-3-methylpiperazine-1,4-diium-1-yl]ethyl]quinazolin-4-one —— C17H25ClN4O+2
6-chloro-3-ethyl-2-[(1R)-1-[(3R)-3-methylpiperazine-1,4-diium-1-yl]ethyl]quinazolin-4-one
—— 6-[(2-methylphenyl)methyl]-N-propylthieno[2,3-b]pyrrole-5-carboxamide —— C18H20N2OS
6-[(2-methylphenyl)methyl]-N-propylthieno[2,3-b]pyrrole-5-carboxamide
—— (6R)-6-[[[(1S)-1-(3-ethoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O2
(6R)-6-[[[(1S)-1-(3-ethoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[3-(cyclopropanecarbonylamino)phenyl]-N,N,8-trimethyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C21H26N4O2S
(6S)-6-[3-(cyclopropanecarbonylamino)phenyl]-N,N,8-trimethyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— (6S)-6-[[[(1S)-1-(3-ethoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O2
(6S)-6-[[[(1S)-1-(3-ethoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-Bromo-3-[di(propan-2-yl)amino]thiochromen-4-one —— C15H18BrNOS
6-Bromo-3-[di(propan-2-yl)amino]thiochromen-4-one
—— (6S)-2-ethyl-N-[(5-phenyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H21N5O
(6S)-2-ethyl-N-[(5-phenyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-2-ethyl-N-[(5-phenyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H21N5O
(6R)-2-ethyl-N-[(5-phenyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-2-ethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H21N5O
(6R)-2-ethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-methyl-N-[[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C13H17N7S
6-methyl-N-[[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— (6S)-2-ethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H21N5O
(6S)-2-ethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-[3-(4-fluorophenyl)sulfonylpropyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H19FN4O2S
(6R)-N-[3-(4-fluorophenyl)sulfonylpropyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[(1S)-1-[5-fluoro-2-(4-hydroxypiperidin-1-yl)phenyl]ethyl]amino]pyridine-3-carbonitrile —— C19H21FN4O
6-[[(1S)-1-[5-fluoro-2-(4-hydroxypiperidin-1-yl)phenyl]ethyl]amino]pyridine-3-carbonitrile
—— (6S)-N-[3-(4-fluorophenyl)sulfonylpropyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H19FN4O2S
(6S)-N-[3-(4-fluorophenyl)sulfonylpropyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-[(4-methyl-2-phenyl-1,3-thiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H19N5S
(6R)-N-[(4-methyl-2-phenyl-1,3-thiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[(4-methyl-2-phenyl-1,3-thiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H19N5S
(6S)-N-[(4-methyl-2-phenyl-1,3-thiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine