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—— 6-methyl-1-[3-oxo-3-[3-[(2S)-oxolan-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propyl]pyridin-2-one —— C19H25N5O3
6-methyl-1-[3-oxo-3-[3-[(2S)-oxolan-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propyl]pyridin-2-one
—— [6-[[(1R)-1-(1H-imidazol-2-yl)ethyl]amino]pyridin-3-yl]-(4-pyridin-3-yloxypiperidin-1-yl)methanone —— C21H24N6O2
[6-[[(1R)-1-(1H-imidazol-2-yl)ethyl]amino]pyridin-3-yl]-(4-pyridin-3-yloxypiperidin-1-yl)methanone
—— 6-[(3S)-3-(aminomethyl)piperidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide —— C22H30N4O2
6-[(3S)-3-(aminomethyl)piperidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
—— 6-[(3R)-3-(aminomethyl)piperidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide —— C22H30N4O2
6-[(3R)-3-(aminomethyl)piperidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
—— 6-(4-Fluorophenyl)sulfonyl-2-[(3-methylphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H20FN3O3S
6-(4-Fluorophenyl)sulfonyl-2-[(3-methylphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(4-fluorophenyl)-N-methyl-N-[(1R)-1-pyridin-3-ylpropyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C21H19FN4OS
6-(4-fluorophenyl)-N-methyl-N-[(1R)-1-pyridin-3-ylpropyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— 6-[[(3S)-oxolan-3-yl]methylamino]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide —— C19H24N4O2
6-[[(3S)-oxolan-3-yl]methylamino]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide
—— 6-[(2R)-2-chloropropanoyl]-2-[(2-methoxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H20ClN3O3
6-[(2R)-2-chloropropanoyl]-2-[(2-methoxyphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3R)-3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-2-carbonitrile —— C21H21N5
6-[(3R)-3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-2-carbonitrile
—— 6-[(3S)-3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-2-carbonitrile —— C21H21N5
6-[(3S)-3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-2-carbonitrile
—— 6-[(3S)-3-ethylpiperazin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide —— C22H30N4O2
6-[(3S)-3-ethylpiperazin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
—— 6-[[(3S)-3-methylpiperazin-1-yl]methyl]-3-phenylpyrazolo[1,5-a]pyrimidine —— C18H21N5
6-[[(3S)-3-methylpiperazin-1-yl]methyl]-3-phenylpyrazolo[1,5-a]pyrimidine
—— 6-[[(3R)-3-methylpiperazin-1-yl]methyl]-3-phenylpyrazolo[1,5-a]pyrimidine —— C18H21N5
6-[[(3R)-3-methylpiperazin-1-yl]methyl]-3-phenylpyrazolo[1,5-a]pyrimidine
—— [6-(2,3-dihydro-1-benzofuran-7-yl)pyridin-3-yl]-[(3R)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methanone —— C23H29N3O2
[6-(2,3-dihydro-1-benzofuran-7-yl)pyridin-3-yl]-[(3R)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methanone
—— 6-ethoxy-3-[[methyl-[[(2R)-1-methylpyrrolidin-2-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C19H27N3O2
6-ethoxy-3-[[methyl-[[(2R)-1-methylpyrrolidin-2-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 6-chloro-2-methyl-N-[2-[(3S)-1-methylpiperidin-3-yl]ethyl]imidazo[1,2-a]pyridine-3-carboxamide —— C17H23ClN4O
6-chloro-2-methyl-N-[2-[(3S)-1-methylpiperidin-3-yl]ethyl]imidazo[1,2-a]pyridine-3-carboxamide
—— 6-chloro-2-methyl-N-[2-[(3R)-1-methylpiperidin-3-yl]ethyl]imidazo[1,2-a]pyridine-3-carboxamide —— C17H23ClN4O
6-chloro-2-methyl-N-[2-[(3R)-1-methylpiperidin-3-yl]ethyl]imidazo[1,2-a]pyridine-3-carboxamide
—— 6-chloro-N-[(E)-1-(4-nitrophenyl)ethylideneamino]-4-phenylquinolin-2-amine —— C23H17ClN4O2
6-chloro-N-[(E)-1-(4-nitrophenyl)ethylideneamino]-4-phenylquinolin-2-amine
—— 6-[(3R)-3-ethylpiperazin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide —— C22H30N4O2
6-[(3R)-3-ethylpiperazin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
—— 6-ethoxy-3-[[methyl-[[(2S)-1-methylpyrrolidin-2-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C19H27N3O2
6-ethoxy-3-[[methyl-[[(2S)-1-methylpyrrolidin-2-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— (6R)-2-[(3-ethoxybenzoyl)amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H22N2O3S
(6R)-2-[(3-ethoxybenzoyl)amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6S)-2-[(3-ethoxybenzoyl)amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H22N2O3S
(6S)-2-[(3-ethoxybenzoyl)amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— [6-(2,3-dihydro-1-benzofuran-7-yl)pyridin-3-yl]-[(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methanone —— C23H29N3O2
[6-(2,3-dihydro-1-benzofuran-7-yl)pyridin-3-yl]-[(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methanone
—— [6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(3R)-3-(methoxymethyl)pyrrolidin-1-yl]methanone —— C18H27N5O2
[6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(3R)-3-(methoxymethyl)pyrrolidin-1-yl]methanone
—— 6-methyl-N-[(E)-[(1S,6S)-6-methyl-4-(4-methylpent-3-enyl)cyclohex-3-en-1-yl]methylideneamino]-5H-[1,2,4]triazino[5,6-b]indol-3-amine —— C24H30N6
6-methyl-N-[(E)-[(1S,6S)-6-methyl-4-(4-methylpent-3-enyl)cyclohex-3-en-1-yl]methylideneamino]-5H-[1,2,4]triazino[5,6-b]indol-3-amine
—— 6-methyl-N-[(E)-[(1R,6S)-6-methyl-4-(4-methylpent-3-enyl)cyclohex-3-en-1-yl]methylideneamino]-5H-[1,2,4]triazino[5,6-b]indol-3-amine —— C24H30N6
6-methyl-N-[(E)-[(1R,6S)-6-methyl-4-(4-methylpent-3-enyl)cyclohex-3-en-1-yl]methylideneamino]-5H-[1,2,4]triazino[5,6-b]indol-3-amine
—— [6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(3S)-3-(methoxymethyl)pyrrolidin-1-yl]methanone —— C18H27N5O2
[6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(3S)-3-(methoxymethyl)pyrrolidin-1-yl]methanone
—— 6-[(2S)-2-methylpyrrolidin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide —— C18H24N4O2
6-[(2S)-2-methylpyrrolidin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
—— 6-[(2R)-2-methylpyrrolidin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide —— C18H24N4O2
6-[(2R)-2-methylpyrrolidin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
—— 6-[(3S)-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl]-7H-purine —— C19H18FN7
6-[(3S)-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl]-7H-purine
—— 6-methyl-5-[(2Z)-2-[(2-phenylmethoxynaphthalen-1-yl)methylidene]hydrazinyl]-2H-1,2,4-triazin-3-one —— C22H19N5O2
6-methyl-5-[(2Z)-2-[(2-phenylmethoxynaphthalen-1-yl)methylidene]hydrazinyl]-2H-1,2,4-triazin-3-one
—— (6R)-N-[(E)-(2-fluorophenyl)methylideneamino]-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-amine —— C15H16FN3S
(6R)-N-[(E)-(2-fluorophenyl)methylideneamino]-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-amine
—— (6S)-2-[[(2R)-2-(2,4-difluorophenoxy)propanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H20F2N2O3S
(6S)-2-[[(2R)-2-(2,4-difluorophenoxy)propanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-methyl-5-[(2Z)-2-[[4-[(4-methylphenyl)methoxy]phenyl]methylidene]hydrazinyl]-2H-1,2,4-triazin-3-one —— C19H19N5O2
6-methyl-5-[(2Z)-2-[[4-[(4-methylphenyl)methoxy]phenyl]methylidene]hydrazinyl]-2H-1,2,4-triazin-3-one
—— (6R)-N-[(4-ethylphenyl)methylideneamino]-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-amine —— C17H21N3S
(6R)-N-[(4-ethylphenyl)methylideneamino]-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-amine
—— 6-ethoxy-3-[[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-quinolin-2-one —— C21H23N3O2
6-ethoxy-3-[[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-quinolin-2-one
—— 6-(diethylaminomethyl)-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22N6OS
6-(diethylaminomethyl)-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-[[(2S)-2-methylpiperazin-1-yl]methyl]-3-phenylpyrazolo[1,5-a]pyrimidine —— C18H21N5
6-[[(2S)-2-methylpiperazin-1-yl]methyl]-3-phenylpyrazolo[1,5-a]pyrimidine
—— 6-ethoxy-3-[[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-quinolin-2-one —— C21H23N3O2
6-ethoxy-3-[[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-quinolin-2-one
—— 6-fluoro-N-[(1S)-1-(4-methylpyridin-2-yl)propyl]-2-oxo-1H-quinoline-4-carboxamide —— C19H18FN3O2
6-fluoro-N-[(1S)-1-(4-methylpyridin-2-yl)propyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-[(3S)-3-methoxypiperidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide —— C21H31N5O2
6-[(3S)-3-methoxypiperidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide
—— 6-[(3R)-3-methoxypiperidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide —— C21H31N5O2
6-[(3R)-3-methoxypiperidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide
—— 6-[[(2R)-2,3-dihydroxypropyl]-methylamino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide —— C16H23N5O4
6-[[(2R)-2,3-dihydroxypropyl]-methylamino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide
—— 6-oxo-N-[[(3S)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]-1H-pyridine-2-carboxamide —— C20H23N3O2
6-oxo-N-[[(3S)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]-1H-pyridine-2-carboxamide
—— (6S)-2-[[(2S)-2-(2,4-difluorophenoxy)propanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H20F2N2O3S
(6S)-2-[[(2S)-2-(2,4-difluorophenoxy)propanoyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— [6-(2,6-dimethoxy-4-methylphenyl)pyridin-3-yl]-[(3R)-3-(methoxymethyl)piperidin-1-yl]methanone —— C22H28N2O4
[6-(2,6-dimethoxy-4-methylphenyl)pyridin-3-yl]-[(3R)-3-(methoxymethyl)piperidin-1-yl]methanone
—— 6-oxo-N-[[(3R)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]-1H-pyridine-2-carboxamide —— C20H23N3O2
6-oxo-N-[[(3R)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]-1H-pyridine-2-carboxamide
—— 6-[[(2S)-2,3-dihydroxypropyl]-methylamino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide —— C16H23N5O4
6-[[(2S)-2,3-dihydroxypropyl]-methylamino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide
—— 6-(4-fluorophenyl)-N-methyl-N-[[(2R)-oxolan-2-yl]methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C18H18FN3O2S
6-(4-fluorophenyl)-N-methyl-N-[[(2R)-oxolan-2-yl]methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— [6-(2,6-dimethoxy-4-methylphenyl)pyridin-3-yl]-[(3S)-3-(methoxymethyl)piperidin-1-yl]methanone —— C22H28N2O4
[6-(2,6-dimethoxy-4-methylphenyl)pyridin-3-yl]-[(3S)-3-(methoxymethyl)piperidin-1-yl]methanone