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—— 6-(2-chlorophenyl)-N-[(3S)-2-oxopiperidin-3-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C17H15ClN4O2S
6-(2-chlorophenyl)-N-[(3S)-2-oxopiperidin-3-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— 6-chloro-2-[2-[(3S)-3-(4-ethyl-1-methyl-5-oxo-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C16H21ClN6O3
6-chloro-2-[2-[(3S)-3-(4-ethyl-1-methyl-5-oxo-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— 6-(1-methylimidazol-2-yl)-N-[(2S)-2-pyridin-3-yloxypropyl]pyridazin-3-amine —— C16H18N6O
6-(1-methylimidazol-2-yl)-N-[(2S)-2-pyridin-3-yloxypropyl]pyridazin-3-amine
—— [6-[[(3R)-oxolan-3-yl]methylamino]pyridin-3-yl]-[4-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C20H27N5O2
[6-[[(3R)-oxolan-3-yl]methylamino]pyridin-3-yl]-[4-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— 6-(2-chlorophenyl)-N-[(3R)-2-oxopiperidin-3-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C17H15ClN4O2S
6-(2-chlorophenyl)-N-[(3R)-2-oxopiperidin-3-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— 6-(3,4-dimethylphenyl)-3-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C18H16N4S
6-(3,4-dimethylphenyl)-3-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— 6-(diethylaminomethyl)-N-[(3R)-1-methyl-6-oxopiperidin-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H26N6O2
6-(diethylaminomethyl)-N-[(3R)-1-methyl-6-oxopiperidin-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [6-[[(3S)-oxolan-3-yl]methylamino]pyridin-3-yl]-[4-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C20H27N5O2
[6-[[(3S)-oxolan-3-yl]methylamino]pyridin-3-yl]-[4-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— [6-[[(1S)-1-cyclopropylethyl]amino]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone —— C20H30N4O2
[6-[[(1S)-1-cyclopropylethyl]amino]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone
—— 6-chloro-2-[2-[(3R)-3-(4-ethyl-1-methyl-5-oxo-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C16H21ClN6O3
6-chloro-2-[2-[(3R)-3-(4-ethyl-1-methyl-5-oxo-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— 6-(2-aminoethyl)-2-methyl-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]pyrimidin-4-amine —— C14H25N5
6-(2-aminoethyl)-2-methyl-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]pyrimidin-4-amine
—— 6-(4-methyl-3-oxopiperazin-1-yl)-N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide —— C20H31N5O2
6-(4-methyl-3-oxopiperazin-1-yl)-N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide
—— 6-(4-methyl-3-oxopiperazin-1-yl)-N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide —— C20H31N5O2
6-(4-methyl-3-oxopiperazin-1-yl)-N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]pyridine-3-carboxamide
—— [6-[[(1R)-1-cyclopropylethyl]amino]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone —— C20H30N4O2
[6-[[(1R)-1-cyclopropylethyl]amino]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone
—— 6-(aminomethyl)-N-[(2S)-1-thiophen-3-ylpropan-2-yl]pyrimidin-4-amine —— C12H16N4S
6-(aminomethyl)-N-[(2S)-1-thiophen-3-ylpropan-2-yl]pyrimidin-4-amine
—— 6-(aminomethyl)-N-[(2R)-1-thiophen-3-ylpropan-2-yl]pyrimidin-4-amine —— C12H16N4S
6-(aminomethyl)-N-[(2R)-1-thiophen-3-ylpropan-2-yl]pyrimidin-4-amine
—— 6-[(2S)-2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]pyridine-3-carboxamide —— C15H14ClN3O2
6-[(2S)-2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]pyridine-3-carboxamide
—— 6-chloro-N-[(1R,2R)-2-(3-fluorophenyl)cyclopropyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C17H14ClFN2O4S
6-chloro-N-[(1R,2R)-2-(3-fluorophenyl)cyclopropyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— 6-chloro-N-[(1S,2R)-2-(3-fluorophenyl)cyclopropyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C17H14ClFN2O4S
6-chloro-N-[(1S,2R)-2-(3-fluorophenyl)cyclopropyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— (6R)-6-(3,5-dimethoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C18H21N3O3
(6R)-6-(3,5-dimethoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— 6-chloro-N-[(1S,2S)-2-(3-fluorophenyl)cyclopropyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C17H14ClFN2O4S
6-chloro-N-[(1S,2S)-2-(3-fluorophenyl)cyclopropyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— 6-Methyl-2-{4-[3-(trifluoromethyl)benzoyl]piperazin-1-yl}-1,3-benzothiazole —— C20H18F3N3OS
6-Methyl-2-{4-[3-(trifluoromethyl)benzoyl]piperazin-1-yl}-1,3-benzothiazole
—— 6-[[(5R)-2,9-diazaspiro[4.5]decan-2-yl]sulfonyl]-4H-1,4-benzoxazin-3-one —— C16H21N3O4S
6-[[(5R)-2,9-diazaspiro[4.5]decan-2-yl]sulfonyl]-4H-1,4-benzoxazin-3-one
—— [6-[(2S)-2-methylpyrrolidin-1-yl]pyridin-3-yl]-(4-pyrimidin-2-yl-1,4-diazepan-1-yl)methanone —— C20H26N6O
[6-[(2S)-2-methylpyrrolidin-1-yl]pyridin-3-yl]-(4-pyrimidin-2-yl-1,4-diazepan-1-yl)methanone
—— (6S)-6-(3,5-dimethoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C18H21N3O3
(6S)-6-(3,5-dimethoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— [6-[(2R)-2-methylpyrrolidin-1-yl]pyridin-3-yl]-(4-pyrimidin-2-yl-1,4-diazepan-1-yl)methanone —— C20H26N6O
[6-[(2R)-2-methylpyrrolidin-1-yl]pyridin-3-yl]-(4-pyrimidin-2-yl-1,4-diazepan-1-yl)methanone
—— 6-[[(5S)-2,9-diazaspiro[4.5]decan-2-yl]sulfonyl]-4H-1,4-benzoxazin-3-one —— C16H21N3O4S
6-[[(5S)-2,9-diazaspiro[4.5]decan-2-yl]sulfonyl]-4H-1,4-benzoxazin-3-one
—— (6S)-6-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one —— C15H17N3OS2
(6S)-6-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one
—— [6-[(2R)-2-ethylmorpholin-4-yl]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone —— C21H32N4O3
[6-[(2R)-2-ethylmorpholin-4-yl]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone
—— [6-[(2S)-2-ethylmorpholin-4-yl]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone —— C21H32N4O3
[6-[(2S)-2-ethylmorpholin-4-yl]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone
—— 6-(2-methoxyphenyl)-N-[[(3S)-oxolan-3-yl]methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C18H19N3O3S
6-(2-methoxyphenyl)-N-[[(3S)-oxolan-3-yl]methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— 6-oxo-N-[4-[(2S)-oxolan-2-yl]butyl]-4,5-dihydro-1H-pyridazine-3-carboxamide —— C13H21N3O3
6-oxo-N-[4-[(2S)-oxolan-2-yl]butyl]-4,5-dihydro-1H-pyridazine-3-carboxamide
—— 6-(2-methoxyphenyl)-N-[[(3R)-oxolan-3-yl]methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C18H19N3O3S
6-(2-methoxyphenyl)-N-[[(3R)-oxolan-3-yl]methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— (6R)-6-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one —— C15H17N3OS2
(6R)-6-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one
—— (6R)-6-(1-methyltetrazol-5-yl)sulfanyl-6,7,8,9-tetrahydrobenzo[7]annulen-5-one —— C13H14N4OS
(6R)-6-(1-methyltetrazol-5-yl)sulfanyl-6,7,8,9-tetrahydrobenzo[7]annulen-5-one
—— 6-Fluoro-2-[4-(3-methoxybenzoyl)piperazin-1-yl]-1,3-benzothiazole —— C19H18FN3O2S
6-Fluoro-2-[4-(3-methoxybenzoyl)piperazin-1-yl]-1,3-benzothiazole
—— (6S)-6-[[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one —— C16H19N3O2S
(6S)-6-[[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one
—— 6-oxo-N-[4-[(2R)-oxolan-2-yl]butyl]-4,5-dihydro-1H-pyridazine-3-carboxamide —— C13H21N3O3
6-oxo-N-[4-[(2R)-oxolan-2-yl]butyl]-4,5-dihydro-1H-pyridazine-3-carboxamide
—— (6S)-6-(1-methyltetrazol-5-yl)sulfanyl-6,7,8,9-tetrahydrobenzo[7]annulen-5-one —— C13H14N4OS
(6S)-6-(1-methyltetrazol-5-yl)sulfanyl-6,7,8,9-tetrahydrobenzo[7]annulen-5-one
—— (6S)-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one —— C14H15N3OS
(6S)-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one
—— (6R)-2-methyl-2,8-diazaspiro[5.5]undecan-3-one —— C10H18N2O
(6R)-2-methyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-methyl-2,8-diazaspiro[5.5]undecan-3-one —— C10H18N2O
(6S)-2-methyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one —— C16H19N3O2S
(6R)-6-[[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one
—— (6R)-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one —— C14H15N3OS
(6R)-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]-6,7,8,9-tetrahydrobenzo[7]annulen-5-one
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 5-chloro-2-methoxybenzoate —— C20H17ClO5
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 5-chloro-2-methoxybenzoate
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4,5-dimethoxy-2-nitrobenzoate —— C18H16ClNO8
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4,5-dimethoxy-2-nitrobenzoate
—— 6-[4-[(S)-(4-chlorophenyl)-hydroxymethyl]piperidin-1-yl]pyridine-3-carbonitrile —— C18H18ClN3O
6-[4-[(S)-(4-chlorophenyl)-hydroxymethyl]piperidin-1-yl]pyridine-3-carbonitrile
—— 6-[4-[(R)-(4-chlorophenyl)-hydroxymethyl]piperidin-1-yl]pyridine-3-carbonitrile —— C18H18ClN3O
6-[4-[(R)-(4-chlorophenyl)-hydroxymethyl]piperidin-1-yl]pyridine-3-carbonitrile
—— 6-[[(2R)-2-hydroxy-2-naphthalen-2-ylethyl]amino]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C18H17N5O2
6-[[(2R)-2-hydroxy-2-naphthalen-2-ylethyl]amino]-1-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6,7-Dimethyl-4-[(2-oxochromen-7-yl)oxymethyl]chromen-2-one —— C21H16O5
6,7-Dimethyl-4-[(2-oxochromen-7-yl)oxymethyl]chromen-2-one