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—— (6R)-6-[[[(2S)-1-(4-methylphenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O2
(6R)-6-[[[(2S)-1-(4-methylphenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(2R)-1-(4-methylphenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O2
(6R)-6-[[[(2R)-1-(4-methylphenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-[(2R)-4-hydroxy-5-oxo-2-phenyl-3-[(E)-3-phenylprop-2-enoyl]-2H-pyrrol-1-yl]hexanoic acid —— C25H25NO5
6-[(2R)-4-hydroxy-5-oxo-2-phenyl-3-[(E)-3-phenylprop-2-enoyl]-2H-pyrrol-1-yl]hexanoic acid
—— (6R)-N-(3-naphthalen-1-yloxypropyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C19H22N4O
(6R)-N-(3-naphthalen-1-yloxypropyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[(2S)-2-(4-hydroxyphenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]hexanoate —— C23H22NO6-
6-[(2S)-2-(4-hydroxyphenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]hexanoate
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4-fluorobenzoate —— C16H12ClFO4
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4-fluorobenzoate
—— 6-[[(2R)-4-ethylmorpholin-2-yl]methylamino]pyridine-3-carbonitrile —— C13H18N4O
6-[[(2R)-4-ethylmorpholin-2-yl]methylamino]pyridine-3-carbonitrile
—— (6S)-2-methyl-N-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H17N5
(6S)-2-methyl-N-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[(2S)-4-ethylmorpholin-2-yl]methylamino]pyridine-3-carbonitrile —— C13H18N4O
6-[[(2S)-4-ethylmorpholin-2-yl]methylamino]pyridine-3-carbonitrile
—— 6-[(3S)-4-(2-methoxyethyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile —— C14H20N4O
6-[(3S)-4-(2-methoxyethyl)-3-methylpiperazin-1-yl]pyridine-3-carbonitrile
—— (6S)-N-(3-naphthalen-1-yloxypropyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C19H22N4O
(6S)-N-(3-naphthalen-1-yloxypropyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-6-[[(1-phenylcyclopentyl)methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H27N5O
(6S)-6-[[(1-phenylcyclopentyl)methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-methyl-N-[[(6R)-3-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C15H21N7S
6-methyl-N-[[(6R)-3-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— (6R)-6-[(2-phenoxyethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C16H21N5O2
(6R)-6-[(2-phenoxyethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[(2-phenoxyethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C16H21N5O2
(6S)-6-[(2-phenoxyethylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[(1S)-1-naphthalen-1-ylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H23N5O
(6S)-6-[[[(1S)-1-naphthalen-1-ylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[(1-phenylcyclopentyl)methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H27N5O
(6R)-6-[[(1-phenylcyclopentyl)methylamino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[(1R)-1-naphthalen-1-ylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H23N5O
(6S)-6-[[[(1R)-1-naphthalen-1-ylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(1R)-1-naphthalen-1-ylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H23N5O
(6R)-6-[[[(1R)-1-naphthalen-1-ylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-2-methyl-N-[(3-methylthiophen-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H18N4S
(6R)-2-methyl-N-[(3-methylthiophen-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-2-methyl-N-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H17N5
(6R)-2-methyl-N-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-2-methyl-N-[(3-methylthiophen-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H18N4S
(6S)-2-methyl-N-[(3-methylthiophen-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-6-[[[(1R)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6R)-6-[[[(1R)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(1S)-1-naphthalen-1-ylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H23N5O
(6R)-6-[[[(1S)-1-naphthalen-1-ylethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[[[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6R)-6-[[[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6S)-6-[[[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-tert-butyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C15H21N7S
6-tert-butyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— (6S)-6-[[[(1R)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6S)-6-[[[(1R)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-[(2R)-4-hydroxy-5-oxo-2-phenyl-3-[(E)-3-phenylprop-2-enoyl]-2H-pyrrol-1-yl]hexanoate —— C25H24NO5-
6-[(2R)-4-hydroxy-5-oxo-2-phenyl-3-[(E)-3-phenylprop-2-enoyl]-2H-pyrrol-1-yl]hexanoate
—— 6-[(2S)-4-hydroxy-5-oxo-2-phenyl-3-[(E)-3-phenylprop-2-enoyl]-2H-pyrrol-1-yl]hexanoic acid —— C25H25NO5
6-[(2S)-4-hydroxy-5-oxo-2-phenyl-3-[(E)-3-phenylprop-2-enoyl]-2H-pyrrol-1-yl]hexanoic acid
—— 6-[(2S)-2-(4-hydroxyphenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]hexanoic acid —— C23H23NO6
6-[(2S)-2-(4-hydroxyphenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]hexanoic acid
—— 6-[(2R)-2-(4-hydroxyphenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]hexanoate —— C23H22NO6-
6-[(2R)-2-(4-hydroxyphenyl)-3-[hydroxy(phenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]hexanoate
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 4-fluorobenzoate —— C19H15FO4
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 4-fluorobenzoate
—— (6-Chloro-7-hydroxy-3,4-dimethyl-2-oxochromen-8-yl)methyl-diethylazanium —— C16H21ClNO3+
(6-Chloro-7-hydroxy-3,4-dimethyl-2-oxochromen-8-yl)methyl-diethylazanium
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl pyridine-4-carboxylate —— C15H12ClNO4
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl pyridine-4-carboxylate
—— (6-Chloro-7-methyl-2-oxochromen-4-yl)methyl pyridine-4-carboxylate —— C17H12ClNO4
(6-Chloro-7-methyl-2-oxochromen-4-yl)methyl pyridine-4-carboxylate
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 4-hydroxybenzoate —— C19H16O5
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 4-hydroxybenzoate
—— 6-[[(5S)-5-hydroxy-3-phenyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]-sulfanylmethylidene]cyclohexa-2,4-dien-1-one —— C17H13F3N2O2S
6-[[(5S)-5-hydroxy-3-phenyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]-sulfanylmethylidene]cyclohexa-2,4-dien-1-one
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl pyridine-2-carboxylate —— C18H15NO4
(6,7-Dimethyl-2-oxochromen-4-yl)methyl pyridine-2-carboxylate
—— (6S)-2-methyl-N-[1-(4-methylphenyl)tetrazol-5-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H18N8
(6S)-2-methyl-N-[1-(4-methylphenyl)tetrazol-5-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[2-[[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]ethoxy]-3,4-dihydro-1H-quinolin-2-one —— C18H23N5O2
6-[2-[[(6R)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]ethoxy]-3,4-dihydro-1H-quinolin-2-one
—— 6-[2-[[(1S,8R)-8,11,11-trimethyl-3,4,6-triazatricyclo[6.2.1.02,7]undeca-2(7),3,5-trien-5-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one —— C21H22N4O3S
6-[2-[[(1S,8R)-8,11,11-trimethyl-3,4,6-triazatricyclo[6.2.1.02,7]undeca-2(7),3,5-trien-5-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one
—— (6R)-N,N-bis[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C24H22N8O2
(6R)-N,N-bis[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-6-[[[(S)-cyclopropyl(phenyl)methyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H23N5O
(6R)-6-[[[(S)-cyclopropyl(phenyl)methyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-N-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H16ClN5O
(6S)-N-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[2-[[(6S)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]ethoxy]-3,4-dihydro-1H-quinolin-2-one —— C18H23N5O2
6-[2-[[(6S)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-yl]amino]ethoxy]-3,4-dihydro-1H-quinolin-2-one
—— (6S)-6-[[[(R)-cyclopropyl(phenyl)methyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H23N5O
(6S)-6-[[[(R)-cyclopropyl(phenyl)methyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-N-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H16ClN5O
(6R)-N-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[5-[(E)-2-(5-methylfuran-2-yl)ethenyl]-2-phenyl-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C21H17N3O2
6-[5-[(E)-2-(5-methylfuran-2-yl)ethenyl]-2-phenyl-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— (6S)-N,N-bis[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C24H22N8O2
(6S)-N,N-bis[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine