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—— 6-amino-5-[2-[[(1R)-1-(2,5-difluorophenyl)ethyl]-methylamino]acetyl]-1-(2-methylpropyl)pyrimidine-2,4-dione —— C19H24F2N4O3
6-amino-5-[2-[[(1R)-1-(2,5-difluorophenyl)ethyl]-methylamino]acetyl]-1-(2-methylpropyl)pyrimidine-2,4-dione
—— 6-methoxy-3-[[(2S)-2-(pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl]-1H-quinolin-2-one —— C20H24N4O3
6-methoxy-3-[[(2S)-2-(pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl]-1H-quinolin-2-one
—— 6-(diethylaminomethyl)-N-[(1R)-1-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C16H22N8O2
6-(diethylaminomethyl)-N-[(1R)-1-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-ethoxy-3-[[methyl-[(1S)-1-pyrimidin-4-ylethyl]amino]methyl]-1H-quinolin-2-one —— C19H22N4O2
6-ethoxy-3-[[methyl-[(1S)-1-pyrimidin-4-ylethyl]amino]methyl]-1H-quinolin-2-one
—— 6-[[(2S)-oxan-2-yl]methylamino]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide —— C20H26N4O2
6-[[(2S)-oxan-2-yl]methylamino]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide
—— (6R)-6-(3-hydroxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C16H17N3O2
(6R)-6-(3-hydroxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— 6-ethoxy-3-[[methyl-[(1R)-1-pyrimidin-4-ylethyl]amino]methyl]-1H-quinolin-2-one —— C19H22N4O2
6-ethoxy-3-[[methyl-[(1R)-1-pyrimidin-4-ylethyl]amino]methyl]-1H-quinolin-2-one
—— (6S)-6-(4-fluorophenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C16H16FN3O
(6S)-6-(4-fluorophenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— 6-(diethylaminomethyl)-N-[(1S)-1-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C16H22N8O2
6-(diethylaminomethyl)-N-[(1S)-1-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6,8-dimethyl-3-[5-phenyl-3-[(3S)-pyrrolidin-3-yl]imidazol-4-yl]-1H-quinolin-2-one —— C24H24N4O
6,8-dimethyl-3-[5-phenyl-3-[(3S)-pyrrolidin-3-yl]imidazol-4-yl]-1H-quinolin-2-one
—— 6,8-dimethyl-3-[5-phenyl-3-[(3R)-pyrrolidin-3-yl]imidazol-4-yl]-1H-quinolin-2-one —— C24H24N4O
6,8-dimethyl-3-[5-phenyl-3-[(3R)-pyrrolidin-3-yl]imidazol-4-yl]-1H-quinolin-2-one
—— 6-[[(2R)-oxan-2-yl]methylamino]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide —— C20H26N4O2
6-[[(2R)-oxan-2-yl]methylamino]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide
—— (6R)-6-(4-fluorophenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C16H16FN3O
(6R)-6-(4-fluorophenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— 6-(1-methylimidazol-2-yl)-N-[(1S)-1-phenylethyl]pyridazin-3-amine —— C16H17N5
6-(1-methylimidazol-2-yl)-N-[(1S)-1-phenylethyl]pyridazin-3-amine
—— (6S)-4-[[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane —— C20H27N3O3
(6S)-4-[[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane
—— (6R)-4-[[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane —— C20H27N3O3
(6R)-4-[[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl]-1,11-dioxa-4,8-diazaspiro[5.6]dodecane
—— (6S)-6-(3-hydroxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C16H17N3O2
(6S)-6-(3-hydroxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— 6-[5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1,2-dihydropyrazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C18H21N5O2
6-[5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1,2-dihydropyrazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— [6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2S)-2-pyridin-3-ylpiperidin-1-yl]methanone —— C22H28N6O
[6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2S)-2-pyridin-3-ylpiperidin-1-yl]methanone
—— [6-[(2R)-2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]pyridin-3-yl]-morpholin-4-ylmethanone —— C19H21N3O3
[6-[(2R)-2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]pyridin-3-yl]-morpholin-4-ylmethanone
—— 6-Chloro-7-methyl-4-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]chromen-2-one —— C16H16ClN3O2S
6-Chloro-7-methyl-4-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]chromen-2-one
—— [6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2R)-2-pyridin-3-ylpiperidin-1-yl]methanone —— C22H28N6O
[6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2R)-2-pyridin-3-ylpiperidin-1-yl]methanone
—— (6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 2-(2,4-dimethylphenyl)sulfanylacetate —— C21H19ClO4S
(6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 2-(2,4-dimethylphenyl)sulfanylacetate
—— (6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 2-(3,4-dimethylphenyl)sulfanylacetate —— C21H19ClO4S
(6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 2-(3,4-dimethylphenyl)sulfanylacetate
—— [6-[(2S)-2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]pyridin-3-yl]-morpholin-4-ylmethanone —— C19H21N3O3
[6-[(2S)-2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]pyridin-3-yl]-morpholin-4-ylmethanone
—— 6-(1-methylimidazol-2-yl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyridazin-3-amine —— C13H16N8
6-(1-methylimidazol-2-yl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyridazin-3-amine
—— 6-[(2S)-2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-N,N-dimethylpyrazine-2-carboxamide —— C16H17FN4O2
6-[(2S)-2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-N,N-dimethylpyrazine-2-carboxamide
—— 6-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carboxylic acid —— C16H19N3O4
6-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carboxylic acid
—— 6-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carboxylic acid —— C16H19N3O4
6-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carboxylic acid
—— 6-methyl-N-[2-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]ethyl]pyridine-2-carboxamide —— C20H26N4O
6-methyl-N-[2-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]ethyl]pyridine-2-carboxamide
—— 6-amino-N-[[(3R)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]methyl]pyridine-3-carboxamide —— C18H24N4OS
6-amino-N-[[(3R)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]methyl]pyridine-3-carboxamide
—— [6-[(2S)-2-methylpyrrolidin-1-yl]pyridin-3-yl]-[4-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone —— C21H29N5O
[6-[(2S)-2-methylpyrrolidin-1-yl]pyridin-3-yl]-[4-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone
—— [6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(3R)-3,4-dimethylpiperazin-1-yl]methanone —— C18H28N6O
[6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(3R)-3,4-dimethylpiperazin-1-yl]methanone
—— 6-amino-N-[[(3S)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]methyl]pyridine-3-carboxamide —— C18H24N4OS
6-amino-N-[[(3S)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl]methyl]pyridine-3-carboxamide
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carboxylate —— C19H19ClO4S
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-2-carboxylate
—— 6-methyl-N-[2-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]ethyl]pyridine-2-carboxamide —— C20H26N4O
6-methyl-N-[2-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]ethyl]pyridine-2-carboxamide
—— 6-(1-methylimidazol-2-yl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyridazin-3-amine —— C13H16N8
6-(1-methylimidazol-2-yl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyridazin-3-amine
—— [6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(3S)-3,4-dimethylpiperazin-1-yl]methanone —— C18H28N6O
[6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(3S)-3,4-dimethylpiperazin-1-yl]methanone
—— [6-[(2R)-2-methylpyrrolidin-1-yl]pyridin-3-yl]-[4-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone —— C21H29N5O
[6-[(2R)-2-methylpyrrolidin-1-yl]pyridin-3-yl]-[4-(2-pyrazol-1-ylethyl)piperidin-1-yl]methanone
—— 6-[3-[(1R)-1-methoxyethyl]phenyl]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide —— C23H25N3O2
6-[3-[(1R)-1-methoxyethyl]phenyl]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide
—— 6-[3-[(1S)-1-methoxyethyl]phenyl]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide —— C23H25N3O2
6-[3-[(1S)-1-methoxyethyl]phenyl]-N-(3-pyridin-2-ylpropyl)pyridine-3-carboxamide
—— (6S)-6-[(E)-1-phenylprop-1-en-2-yl]-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C19H21N3O
(6S)-6-[(E)-1-phenylprop-1-en-2-yl]-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— 6-(aminomethyl)-N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]pyrimidin-4-amine —— C12H18N6
6-(aminomethyl)-N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]pyrimidin-4-amine
—— [6-[[(2S)-2-hydroxypropyl]amino]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone —— C18H28N4O3
[6-[[(2S)-2-hydroxypropyl]amino]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone
—— 6-(3-methoxyphenyl)-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C20H24N4O2S
6-(3-methoxyphenyl)-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— 6-(aminomethyl)-N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]pyrimidin-4-amine —— C12H18N6
6-(aminomethyl)-N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]pyrimidin-4-amine
—— 6-(3-methoxyphenyl)-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C20H24N4O2S
6-(3-methoxyphenyl)-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— 6-(diethylaminomethyl)-N-[(2S)-1-hydroxypropan-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H23N5O2
6-(diethylaminomethyl)-N-[(2S)-1-hydroxypropan-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-6-[(E)-1-phenylprop-1-en-2-yl]-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C19H21N3O
(6R)-6-[(E)-1-phenylprop-1-en-2-yl]-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— 6-(diethylaminomethyl)-N-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H25N5O2
6-(diethylaminomethyl)-N-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide