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—— (6S)-N-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H14N6O2
(6S)-N-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-(2-phenylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H16N6
(6S)-N-(2-phenylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-Chloro-7-methyl-4-[(4-nitrophenoxy)methyl]chromen-2-one —— C17H12ClNO5
6-Chloro-7-methyl-4-[(4-nitrophenoxy)methyl]chromen-2-one
—— (6R)-N-[[1-(3-fluorophenyl)pyrazol-3-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H17FN6
(6R)-N-[[1-(3-fluorophenyl)pyrazol-3-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H20N6O
(6S)-N-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H20N6O
(6R)-N-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[[1-(3-fluorophenyl)pyrazol-3-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H17FN6
(6S)-N-[[1-(3-fluorophenyl)pyrazol-3-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]amino]pyridine-3-carbonitrile —— C17H16N4O
6-[[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]amino]pyridine-3-carbonitrile
—— [6-(dimethylamino)pyridazin-3-yl]-[(3S)-3-(2-ethylimidazol-1-yl)piperidin-1-yl]methanone —— C17H24N6O
[6-(dimethylamino)pyridazin-3-yl]-[(3S)-3-(2-ethylimidazol-1-yl)piperidin-1-yl]methanone
—— 6-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidine-1-carbonyl]-4H-1,4-benzothiazin-3-one —— C17H18N4O2S
6-[(2R)-2-(1-methylpyrazol-4-yl)pyrrolidine-1-carbonyl]-4H-1,4-benzothiazin-3-one
—— 6-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidine-1-carbonyl]-4H-1,4-benzothiazin-3-one —— C17H18N4O2S
6-[(2S)-2-(1-methylpyrazol-4-yl)pyrrolidine-1-carbonyl]-4H-1,4-benzothiazin-3-one
—— 6-[methyl-[(3R)-1-pyridazin-3-ylpiperidin-3-yl]amino]pyridine-3-carbonitrile —— C16H18N6
6-[methyl-[(3R)-1-pyridazin-3-ylpiperidin-3-yl]amino]pyridine-3-carbonitrile
—— (6S)-2-benzoyl-6-pyridin-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H21N3O2
(6S)-2-benzoyl-6-pyridin-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-[methyl-[(3S)-1-pyridazin-3-ylpiperidin-3-yl]amino]pyridine-3-carbonitrile —— C16H18N6
6-[methyl-[(3S)-1-pyridazin-3-ylpiperidin-3-yl]amino]pyridine-3-carbonitrile
—— (6R)-2-benzoyl-6-pyridin-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H21N3O2
(6R)-2-benzoyl-6-pyridin-2-yl-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-[(2S)-2-(2-chlorophenyl)morpholine-4-carbonyl]-2-methylpyridine-3-carbonitrile —— C18H16ClN3O2
6-[(2S)-2-(2-chlorophenyl)morpholine-4-carbonyl]-2-methylpyridine-3-carbonitrile
—— 6-[(2R)-2-(2-chlorophenyl)morpholine-4-carbonyl]-2-methylpyridine-3-carbonitrile —— C18H16ClN3O2
6-[(2R)-2-(2-chlorophenyl)morpholine-4-carbonyl]-2-methylpyridine-3-carbonitrile
—— 6-[(2S)-2-[(4-methylphenyl)methyl]pyrrolidine-1-carbonyl]-2-propylpyridazin-3-one —— C20H25N3O2
6-[(2S)-2-[(4-methylphenyl)methyl]pyrrolidine-1-carbonyl]-2-propylpyridazin-3-one
—— (6R)-6-[(3-phenylpropylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H23N5O
(6R)-6-[(3-phenylpropylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-N-[(1-benzylimidazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H20N6
(6R)-N-[(1-benzylimidazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-chloro-2-[[(3S)-2-oxoazepan-3-yl]amino]quinoline-4-carbonitrile —— C16H15ClN4O
6-chloro-2-[[(3S)-2-oxoazepan-3-yl]amino]quinoline-4-carbonitrile
—— (6R)-6-(4-methoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C23H24N2O3
(6R)-6-(4-methoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-[(3-phenylpropylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H23N5O
(6S)-6-[(3-phenylpropylamino)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-N-[(1-benzylimidazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H20N6
(6S)-N-[(1-benzylimidazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-5-butanoyl-6-(4-nitrophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C23H23N3O4
(6S)-5-butanoyl-6-(4-nitrophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(2R)-2-[(4-methylphenyl)methyl]pyrrolidine-1-carbonyl]-2-propylpyridazin-3-one —— C20H25N3O2
6-[(2R)-2-[(4-methylphenyl)methyl]pyrrolidine-1-carbonyl]-2-propylpyridazin-3-one
—— (6R)-6-(6-nitro-1,3-benzodioxol-5-yl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C20H17N3O5
(6R)-6-(6-nitro-1,3-benzodioxol-5-yl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(4-methoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C23H24N2O3
(6S)-6-(4-methoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[4-[(2S)-1-acetylazepan-2-yl]piperidin-1-yl]pyridine-3-carbonitrile —— C19H26N4O
6-[4-[(2S)-1-acetylazepan-2-yl]piperidin-1-yl]pyridine-3-carbonitrile
—— (6R)-5-acetyl-6-(4-methylsulfanylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C22H22N2O2S
(6R)-5-acetyl-6-(4-methylsulfanylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-6-(2-methoxyphenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C25H28N2O3
(6R)-6-(2-methoxyphenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-5-benzoyl-6-(4-fluorophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C26H21FN2O2
(6S)-5-benzoyl-6-(4-fluorophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6,7-dimethoxy-2-[(1S)-1-pyridin-4-ylethyl]-3,4-dihydro-1H-isoquinoline —— C18H22N2O2
6,7-dimethoxy-2-[(1S)-1-pyridin-4-ylethyl]-3,4-dihydro-1H-isoquinoline
—— (6R)-6-(3,4-dichlorophenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C22H20Cl2N2O2
(6R)-6-(3,4-dichlorophenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-6-(3,4-dimethoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C24H26N2O4
(6R)-6-(3,4-dimethoxyphenyl)-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-5-benzoyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C24H20N2O3
(6S)-5-benzoyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(2-methoxyphenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C25H28N2O3
(6S)-6-(2-methoxyphenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-6-(3-nitrophenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C24H25N3O4
(6R)-6-(3-nitrophenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-5-benzoyl-6-(4-fluorophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C26H21FN2O2
(6R)-5-benzoyl-6-(4-fluorophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(4-chlorophenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C24H25ClN2O2
(6S)-6-(4-chlorophenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(3-nitrophenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C24H25N3O4
(6S)-6-(3-nitrophenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6,7-dimethoxy-2-[(1R)-1-pyridin-4-ylethyl]-3,4-dihydro-1H-isoquinoline —— C18H22N2O2
6,7-dimethoxy-2-[(1R)-1-pyridin-4-ylethyl]-3,4-dihydro-1H-isoquinoline
—— (6R)-5-acetyl-6-(2,6-dichlorophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C21H18Cl2N2O2
(6R)-5-acetyl-6-(2,6-dichlorophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-N-(imidazo[1,2-a]pyridin-2-ylmethyl)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H18N6
(6R)-N-(imidazo[1,2-a]pyridin-2-ylmethyl)-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-[(7-chloro-1,3-benzodioxol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C14H15ClN4O2
(6R)-N-[(7-chloro-1,3-benzodioxol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-3-methylsulfanyl-6-(5-phenyl-1H-pyrazol-4-yl)-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C20H16N6OS
(6R)-3-methylsulfanyl-6-(5-phenyl-1H-pyrazol-4-yl)-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— (6S)-3-methylsulfanyl-6-(5-phenyl-1H-pyrazol-4-yl)-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C20H16N6OS
(6S)-3-methylsulfanyl-6-(5-phenyl-1H-pyrazol-4-yl)-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— (6S)-N-[(7-chloro-1,3-benzodioxol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C14H15ClN4O2
(6S)-N-[(7-chloro-1,3-benzodioxol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-5-benzoyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C24H20N2O3
(6R)-5-benzoyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(3-ethoxy-4-methoxyphenyl)-3-methylsulfanyl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C20H20N4O3S
(6S)-6-(3-ethoxy-4-methoxyphenyl)-3-methylsulfanyl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine