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—— 6-[2-[[(1R,8S)-8,11,11-trimethyl-3,4,6-triazatricyclo[6.2.1.02,7]undeca-2(7),3,5-trien-5-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one —— C21H22N4O3S
6-[2-[[(1R,8S)-8,11,11-trimethyl-3,4,6-triazatricyclo[6.2.1.02,7]undeca-2(7),3,5-trien-5-yl]sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one
—— 6-[[(5R)-5-hydroxy-3-phenyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]-sulfanylmethylidene]cyclohexa-2,4-dien-1-one —— C17H13F3N2O2S
6-[[(5R)-5-hydroxy-3-phenyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]-sulfanylmethylidene]cyclohexa-2,4-dien-1-one
—— (6R)-2-methyl-N-[1-(4-methylphenyl)tetrazol-5-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H18N8
(6R)-2-methyl-N-[1-(4-methylphenyl)tetrazol-5-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-6-[[[(S)-cyclopropyl(phenyl)methyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H23N5O
(6S)-6-[[[(S)-cyclopropyl(phenyl)methyl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-chloro-N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]quinoline-8-carboxamide —— C18H23ClN4O
6-chloro-N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]quinoline-8-carboxamide
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-chlorobenzoate —— C19H15ClO4
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-chlorobenzoate
—— 6-chloro-N-[(2R)-2-(4-methylpiperazin-1-yl)propyl]quinoline-8-carboxamide —— C18H23ClN4O
6-chloro-N-[(2R)-2-(4-methylpiperazin-1-yl)propyl]quinoline-8-carboxamide
—— (6-methoxypyridin-3-yl)-[(3S)-3-(4-propan-2-yl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone —— C17H23N5O2
(6-methoxypyridin-3-yl)-[(3S)-3-(4-propan-2-yl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone
—— 6-amino-1,3-dimethyl-5-[2-[(2S)-2-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]acetyl]pyrimidine-2,4-dione —— C17H20N4O4
6-amino-1,3-dimethyl-5-[2-[(2S)-2-methyl-2,3-dihydro-1,4-benzoxazin-4-yl]acetyl]pyrimidine-2,4-dione
—— (6-methoxypyridin-3-yl)-[(3R)-3-(4-propan-2-yl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone —— C17H23N5O2
(6-methoxypyridin-3-yl)-[(3R)-3-(4-propan-2-yl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-bromobenzoate —— C16H12BrClO4
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 2-bromobenzoate
—— 6-[(2,4-Dichlorophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H15Cl2N5O
6-[(2,4-Dichlorophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[5-[(E)-2-(4-fluorophenyl)ethenyl]-2-phenyl-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C22H16FN3O
6-[5-[(E)-2-(4-fluorophenyl)ethenyl]-2-phenyl-1H-1,2,4-triazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— (6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-bromobenzoate —— C19H15BrO4
(6,7-Dimethyl-2-oxochromen-4-yl)methyl 2-bromobenzoate
—— 6-[4-[(2S)-2-hydroxy-2-phenylethyl]piperazine-1-carbonyl]-2-methylpyridazin-3-one —— C18H22N4O3
6-[4-[(2S)-2-hydroxy-2-phenylethyl]piperazine-1-carbonyl]-2-methylpyridazin-3-one
—— 6-[2-(4-Chlorophenyl)-2-oxoethyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C20H16ClN5O2
6-[2-(4-Chlorophenyl)-2-oxoethyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(3-Chlorophenyl)methyl]-3-(3,4-dimethoxyphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H16ClN5O3
6-[(3-Chlorophenyl)methyl]-3-(3,4-dimethoxyphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(3-chloro-4-methylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H21ClN6O2
6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(3-chloro-4-methylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-Benzyl-3-(3-chloro-4-methylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C18H14ClN5O
6-Benzyl-3-(3-chloro-4-methylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-Benzyl-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H17N5O
6-Benzyl-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-Benzyl-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H17N5O
6-Benzyl-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-(4-Chlorophenyl)-2-oxoethyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C20H16ClN5O2
6-[2-(4-Chlorophenyl)-2-oxoethyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C20H24N6O3
6-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C20H24N6O3
6-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— (6S)-3-methyl-6-(2-methylpropyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one —— C15H18N4O
(6S)-3-methyl-6-(2-methylpropyl)-6,7-dihydro-[1,2,4]triazino[2,3-c]quinazolin-2-one
—— 6-[(2-Chlorophenyl)methyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one —— C17H10ClF2N5O
6-[(2-Chlorophenyl)methyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(2-Chlorophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H16ClN5O
6-[(2-Chlorophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[4-[(2R)-2-hydroxy-2-phenylethyl]piperazine-1-carbonyl]-2-methylpyridazin-3-one —— C18H22N4O3
6-[4-[(2R)-2-hydroxy-2-phenylethyl]piperazine-1-carbonyl]-2-methylpyridazin-3-one
—— 6-(2-Oxopropyl)-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one —— C14H10F3N5O3
6-(2-Oxopropyl)-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one
—— 6-[(2-Methylphenyl)methyl]-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one —— C19H14F3N5O2
6-[(2-Methylphenyl)methyl]-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one
—— 6-(2-Piperidin-1-ylethyl)-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one —— C18H19F3N6O2
6-(2-Piperidin-1-ylethyl)-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C20H24N6O3
6-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(2-Chloro-6-fluorophenyl)methyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H15ClFN5O
6-[(2-Chloro-6-fluorophenyl)methyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H22N6O2
6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[4-[[(2R)-1-methylpiperidin-2-yl]methyl]piperazin-1-yl]pyridine-3-carbonitrile —— C17H25N5
6-[4-[[(2R)-1-methylpiperidin-2-yl]methyl]piperazin-1-yl]pyridine-3-carbonitrile
—— 6-(2-Pyrrolidin-1-ylethyl)-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one —— C17H17F3N6O2
6-(2-Pyrrolidin-1-ylethyl)-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one
—— 6-[(2,4-Dichlorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C18H13Cl2N5O
6-[(2,4-Dichlorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(4-Bromophenyl)methyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H16BrN5O
6-[(4-Bromophenyl)methyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C20H24N6O3
6-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one —— C18H18F2N6O2
6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(3-Chlorophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H16ClN5O
6-[(3-Chlorophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(3-Fluorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C18H14FN5O
6-[(3-Fluorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C20H24N6O2
6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(3,4-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(4-Chlorophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H16ClN5O
6-[(4-Chlorophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-Benzyl-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one —— C17H11F2N5O
6-Benzyl-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(2-Chloro-6-fluorophenyl)methyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one —— C17H9ClF3N5O
6-[(2-Chloro-6-fluorophenyl)methyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(4-Fluorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C18H14FN5O
6-[(4-Fluorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(3,4-Dichlorophenyl)methyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one —— C17H9Cl2F2N5O
6-[(3,4-Dichlorophenyl)methyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(2-Chlorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C18H14ClN5O
6-[(2-Chlorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(4-Bromophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H16BrN5O
6-[(4-Bromophenyl)methyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one