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—— (6R)-6-[(3-methylpyridin-1-ium-2-yl)amino]-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one —— C12H12F3N4OS+
(6R)-6-[(3-methylpyridin-1-ium-2-yl)amino]-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one
—— 6-amino-N-[[(3R)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]pyridine-3-carboxamide —— C20H24N4O
6-amino-N-[[(3R)-1-[(E)-3-phenylprop-2-enyl]pyrrolidin-3-yl]methyl]pyridine-3-carboxamide
—— (6S)-6-[(3-methylpyridin-2-yl)amino]-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one —— C12H11F3N4OS
(6S)-6-[(3-methylpyridin-2-yl)amino]-6-(trifluoromethyl)-2,3-dihydroimidazo[2,1-b][1,3]thiazol-5-one
—— 6-(2-cyanophenyl)-N-[2-[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]ethyl]pyridine-3-carboxamide —— C23H19N3O3
6-(2-cyanophenyl)-N-[2-[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]ethyl]pyridine-3-carboxamide
—— 6-(2-cyanophenyl)-N-[2-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]ethyl]pyridine-3-carboxamide —— C23H19N3O3
6-(2-cyanophenyl)-N-[2-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]ethyl]pyridine-3-carboxamide
—— 6-[4-(2,4-dimethoxyphenyl)-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C19H18N2O3
6-[4-(2,4-dimethoxyphenyl)-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— [6-[[(2S)-2,3-dihydroxypropyl]amino]pyridin-3-yl]-(4-pyrimidin-2-yl-1,4-diazepan-1-yl)methanone —— C18H24N6O3
[6-[[(2S)-2,3-dihydroxypropyl]amino]pyridin-3-yl]-(4-pyrimidin-2-yl-1,4-diazepan-1-yl)methanone
—— [(6R,8R,8aR)-5,7,7-tricyano-2-ethyl-8-thiophen-2-yl-2,6,8,8a-tetrahydro-1H-isoquinolin-2-ium-6-yl]azanium —— C18H19N5S+2
[(6R,8R,8aR)-5,7,7-tricyano-2-ethyl-8-thiophen-2-yl-2,6,8,8a-tetrahydro-1H-isoquinolin-2-ium-6-yl]azanium
—— (6S)-6-(4-propan-2-ylphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C19H23N3O
(6S)-6-(4-propan-2-ylphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— [6-[2-[(3R)-3-(4-fluorophenyl)oxolan-3-yl]imidazol-1-yl]-1H-benzimidazol-2-yl]methanol —— C21H19FN4O2
[6-[2-[(3R)-3-(4-fluorophenyl)oxolan-3-yl]imidazol-1-yl]-1H-benzimidazol-2-yl]methanol
—— [6-[2-[(3S)-3-(4-fluorophenyl)oxolan-3-yl]imidazol-1-yl]-1H-benzimidazol-2-yl]methanol —— C21H19FN4O2
[6-[2-[(3S)-3-(4-fluorophenyl)oxolan-3-yl]imidazol-1-yl]-1H-benzimidazol-2-yl]methanol
—— 6-oxo-N-[(2S)-4-pyrazol-1-ylbutan-2-yl]-1H-pyrazine-3-carboxamide —— C12H15N5O2
6-oxo-N-[(2S)-4-pyrazol-1-ylbutan-2-yl]-1H-pyrazine-3-carboxamide
—— 6-[(2R)-3-(azepan-1-yl)-2-hydroxypropyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carbonitrile —— C18H22N4O3
6-[(2R)-3-(azepan-1-yl)-2-hydroxypropyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carbonitrile
—— (6R)-6-tert-butyl-N-[(E)-(5-methylthiophen-2-yl)methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H24N2OS2
(6R)-6-tert-butyl-N-[(E)-(5-methylthiophen-2-yl)methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(2R)-2-methylpyrrolidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide —— C20H29N5O
6-[(2R)-2-methylpyrrolidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide
—— 6-(2-methylphenyl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C18H18N6OS
6-(2-methylphenyl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— [6-(1-methylpyrazol-4-yl)pyridin-3-yl]-[(4S)-4-phenylazepan-1-yl]methanone —— C22H24N4O
[6-(1-methylpyrazol-4-yl)pyridin-3-yl]-[(4S)-4-phenylazepan-1-yl]methanone
—— (6R)-6-(4-propan-2-ylphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C19H23N3O
(6R)-6-(4-propan-2-ylphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— 6-(aminomethyl)-N-[(2S)-2-morpholin-4-yl-2-pyridin-2-ylethyl]pyrimidin-4-amine —— C16H22N6O
6-(aminomethyl)-N-[(2S)-2-morpholin-4-yl-2-pyridin-2-ylethyl]pyrimidin-4-amine
—— (6R)-6-[5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenylimidazol-1-yl]-2-methylheptan-2-ol —— C22H30N4O
(6R)-6-[5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenylimidazol-1-yl]-2-methylheptan-2-ol
—— [6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2S)-2-propylpyrrolidin-1-yl]methanone —— C19H29N5O
[6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2S)-2-propylpyrrolidin-1-yl]methanone
—— 6-oxo-N-[(2R)-4-pyrazol-1-ylbutan-2-yl]-1H-pyrazine-3-carboxamide —— C12H15N5O2
6-oxo-N-[(2R)-4-pyrazol-1-ylbutan-2-yl]-1H-pyrazine-3-carboxamide
—— 6-[(2S)-2-methylpyrrolidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide —— C20H29N5O
6-[(2S)-2-methylpyrrolidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide
—— 6-chloro-N,N-dimethyl-3-[[(3S)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine-2-carboxamide —— C21H30ClN5O2
6-chloro-N,N-dimethyl-3-[[(3S)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine-2-carboxamide
—— 6-[(2S)-3-(azepan-1-yl)-2-hydroxypropyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carbonitrile —— C18H22N4O3
6-[(2S)-3-(azepan-1-yl)-2-hydroxypropyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carbonitrile
—— 6-chloro-N,N-dimethyl-3-[[(3R)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine-2-carboxamide —— C21H30ClN5O2
6-chloro-N,N-dimethyl-3-[[(3R)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine-2-carboxamide
—— 6-(diethylaminomethyl)-N-[[(2S)-1,4-dioxan-2-yl]methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H25N5O3
6-(diethylaminomethyl)-N-[[(2S)-1,4-dioxan-2-yl]methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2R)-2-propylpyrrolidin-1-yl]methanone —— C19H29N5O
[6-(diethylaminomethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2R)-2-propylpyrrolidin-1-yl]methanone
—— (6S)-6-[5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenylimidazol-1-yl]-2-methylheptan-2-ol —— C22H30N4O
(6S)-6-[5-(3,5-dimethyl-1H-pyrazol-4-yl)-4-phenylimidazol-1-yl]-2-methylheptan-2-ol
—— 6-(diethylaminomethyl)-N-[[(2R)-1,4-dioxan-2-yl]methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H25N5O3
6-(diethylaminomethyl)-N-[[(2R)-1,4-dioxan-2-yl]methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-(2-methylphenyl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C18H18N6OS
6-(2-methylphenyl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— 6-[[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]amino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide —— C19H25N7O2
6-[[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]amino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide
—— 6-[[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]amino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide —— C19H25N7O2
6-[[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]amino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide
—— 6-(4-chlorophenyl)-N-[2-[(3S)-oxolan-3-yl]ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C18H18ClN3O2S
6-(4-chlorophenyl)-N-[2-[(3S)-oxolan-3-yl]ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— (6R)-6-(1,3-benzodioxol-5-yl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one —— C17H17N3O3
(6R)-6-(1,3-benzodioxol-5-yl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
—— 6-[[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]amino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide —— C17H22N8O2
6-[[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]amino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide
—— 6-amino-N-cyclopentyl-7-(2-hydroxyethyl)-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide —— C19H22N5O3+
6-amino-N-cyclopentyl-7-(2-hydroxyethyl)-2-oxo-1,9-diaza-7-azoniatricyclo[8.4.0.03,8]tetradeca-3,5,7,9,11,13-hexaene-5-carboxamide
—— 6-[[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]amino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide —— C17H22N8O2
6-[[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]amino]-N-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]pyridine-3-carboxamide
—— (6S)-N-(1-adamantylmethyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C21H29NOS
(6S)-N-(1-adamantylmethyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(4S,7R)-4-methyl-7-propan-2-yl-1,2,4,5,6,7-hexahydroindazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C17H22N2O
6-[(4S,7R)-4-methyl-7-propan-2-yl-1,2,4,5,6,7-hexahydroindazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— 6-methyl-2-[(4-methylpiperazine-1,4-diium-1-yl)methyl]-5-phenyl-3H-thieno[2,3-d]pyrimidin-4-one —— C19H24N4OS+2
6-methyl-2-[(4-methylpiperazine-1,4-diium-1-yl)methyl]-5-phenyl-3H-thieno[2,3-d]pyrimidin-4-one
—— [6-(1-methylpyrazol-4-yl)pyridin-3-yl]-[(4R)-4-phenylazepan-1-yl]methanone —— C22H24N4O
[6-(1-methylpyrazol-4-yl)pyridin-3-yl]-[(4R)-4-phenylazepan-1-yl]methanone
—— 6-(diethylaminomethyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H21N9O
6-(diethylaminomethyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 6-[(3R)-3-(hydroxymethyl)pyrrolidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide —— C20H29N5O2
6-[(3R)-3-(hydroxymethyl)pyrrolidin-1-yl]-N-[3-(2-propan-2-ylimidazol-1-yl)propyl]pyridine-3-carboxamide
—— 6-[(4S,7S)-4-methyl-7-propan-2-yl-1,2,4,5,6,7-hexahydroindazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C17H22N2O
6-[(4S,7S)-4-methyl-7-propan-2-yl-1,2,4,5,6,7-hexahydroindazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— [6-[(3R)-3,4-dimethylpiperazin-1-yl]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone —— C21H33N5O2
[6-[(3R)-3,4-dimethylpiperazin-1-yl]pyridin-3-yl]-(4-morpholin-4-ylpiperidin-1-yl)methanone
—— 6-[[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-3-phenylpyrazolo[1,5-a]pyrimidine —— C22H24N6
6-[[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-3-phenylpyrazolo[1,5-a]pyrimidine
—— 6-(4-chlorophenyl)-N-[2-[(3R)-oxolan-3-yl]ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide —— C18H18ClN3O2S
6-(4-chlorophenyl)-N-[2-[(3R)-oxolan-3-yl]ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
—— 6-[2-[(2S)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carbonitrile —— C17H20N4O3
6-[2-[(2S)-2-(hydroxymethyl)piperidin-1-yl]ethyl]-2,5-dioxo-1H-1,6-naphthyridine-3-carbonitrile
—— 6-[(4R,7R)-4-methyl-7-propan-2-yl-1,2,4,5,6,7-hexahydroindazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C17H22N2O
6-[(4R,7R)-4-methyl-7-propan-2-yl-1,2,4,5,6,7-hexahydroindazol-3-ylidene]cyclohexa-2,4-dien-1-one