Palladium-catalyzed arylation of methyl 2-(acetoxymethyl)acrylate with aryl iodides afforded the primary acetates of Morita–Baylis–Hillman adducts in good yields with high stereoselectivity under mild conditions (50 °C).
2-(乙酰氧基甲基)
丙烯酸甲酯与芳基
碘化物的
钯催化芳基化反应可在温和的条件下(50°C)以良好的产率和高的立体选择性提供森田-贝利斯-希尔曼加合物的初级
乙酸酯。