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—— 3-(5-cyclopentyl-2-(R)-cyclopropylmethyl-3-(S)-hydroxyl-1-oxopentyl)amino-1-methyl-5-(4-trifluoromethylphenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one 330840-21-6 C31H36F3N3O3
3-(5-cyclopentyl-2-(R)-cyclopropylmethyl-3-(S)-hydroxyl-1-oxopentyl)amino-1-methyl-5-(4-trifluoromethylphenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one
—— N-[5-Bromo-2-[3-chloro-4-(3-chloro-2-methylbenzoyl)-phenylamino]phenyl]-succinamic acid 321371-64-6 C24H19BrCl2N2O4
N-[5-Bromo-2-[3-chloro-4-(3-chloro-2-methylbenzoyl)-phenylamino]phenyl]-succinamic acid
—— N-[3-(2,6-dichloro-phenyl)-5isopropyl-2-methyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)ethane-1,2-diamine 332179-03-0 C27H32Cl2N8
N-[3-(2,6-dichloro-phenyl)-5isopropyl-2-methyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-pyrimidin-2-yl-piperidin-4-yl)ethane-1,2-diamine
—— 3-Z-[1-(4-(N-dimethylaminocarbonylmethyl-N-methylsulphonyl-amino)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone 334949-35-8 C28H28N4O6S
3-Z-[1-(4-(N-dimethylaminocarbonylmethyl-N-methylsulphonyl-amino)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone
—— [1-(3-amino-1,2-benzisoxazol-5-yl)-3-(trifluoromethyl)-1H-pyrazol-5-yl][6-[2-[(dimethylamino)methyl]phenyl]-3-benzofuranyl]methanone 321435-94-3 C29H22F3N5O3
[1-(3-amino-1,2-benzisoxazol-5-yl)-3-(trifluoromethyl)-1H-pyrazol-5-yl][6-[2-[(dimethylamino)methyl]phenyl]-3-benzofuranyl]methanone
—— 3-[[[1-[[(1S,4R)-4-[(4,5-dihydro-1H-imidazol-2-yl)amino]-2-cyclopenten-1-yl]carbonyl]-4-piperidinyl]carbonyl]amino]-N-[(phenylmethoxy)carbonyl]-L-alanine 332185-26-9 C26H34N6O6
3-[[[1-[[(1S,4R)-4-[(4,5-dihydro-1H-imidazol-2-yl)amino]-2-cyclopenten-1-yl]carbonyl]-4-piperidinyl]carbonyl]amino]-N-[(phenylmethoxy)carbonyl]-L-alanine
—— (2R)-2-([4-[1-(4-octylphenyl)-5-methyl-1H-pyrrol-2-yl]phenyl]oxy)-3-phenylpropanoic acid 376639-78-0 C34H39NO3
(2R)-2-([4-[1-(4-octylphenyl)-5-methyl-1H-pyrrol-2-yl]phenyl]oxy)-3-phenylpropanoic acid
—— 1-[3-(aminomethyl)phenyl]-N-[4-(2,3-dihydro-1,1-dioxido-1,2-benzisothiazol-7-yl)phenyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide 300710-16-1 C25H20F3N5O3S
1-[3-(aminomethyl)phenyl]-N-[4-(2,3-dihydro-1,1-dioxido-1,2-benzisothiazol-7-yl)phenyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
—— (S)-3-{4-[(6,7-Dimethoxy-4-quinazolinyl)amino]phenyl}-2-[(2-N,N-diethylamino-3,4-dioxocyclobut-1-enyl)amino]propanoic acid 312292-72-1 C27H29N5O6
(S)-3-{4-[(6,7-Dimethoxy-4-quinazolinyl)amino]phenyl}-2-[(2-N,N-diethylamino-3,4-dioxocyclobut-1-enyl)amino]propanoic acid
—— (2S,3R)-2-(4'-methoxy-biphenyl-4-sulfonylamino)-3-(1-methyl-1H-imidazol-2-ylsulfanyl)-3-phenyl-propionic acid 334991-31-0 C26H25N3O5S2
(2S,3R)-2-(4'-methoxy-biphenyl-4-sulfonylamino)-3-(1-methyl-1H-imidazol-2-ylsulfanyl)-3-phenyl-propionic acid
—— 4-(5,6-dichloro-1H-indol-2-yl)-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)-3-ethoxybenzamide 318262-49-6 C27H33Cl2N3O2
4-(5,6-dichloro-1H-indol-2-yl)-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)-3-ethoxybenzamide
—— 4-[4-(3-chloro-4-ethoxybenzylamino)-[1]benzothieno[2,3-d]pyrimidin-2-yl]phenylacetic acid 329928-11-2 C27H22ClN3O3S
4-[4-(3-chloro-4-ethoxybenzylamino)-[1]benzothieno[2,3-d]pyrimidin-2-yl]phenylacetic acid
—— (S)-3-[4-([2,6-Naphthyridin-1-yl]oxy)phenyl]-2-[(2-N,N-dipropylamino-3,4-dioxocyclobut-1-enyl)amino]propanoic acid 312292-44-7 C27H28N4O5
(S)-3-[4-([2,6-Naphthyridin-1-yl]oxy)phenyl]-2-[(2-N,N-dipropylamino-3,4-dioxocyclobut-1-enyl)amino]propanoic acid
—— (S)-1-Phenyl-N-{4-[2-(azetidin-3-yl-methyl)-3-methyl-5-(3-trifluoromethyl-phenyl)-3H-imidazol-4-yl]-pyridin-2-yl}-ethylamine 319469-66-4 C28H28F3N5
(S)-1-Phenyl-N-{4-[2-(azetidin-3-yl-methyl)-3-methyl-5-(3-trifluoromethyl-phenyl)-3H-imidazol-4-yl]-pyridin-2-yl}-ethylamine
—— N-{(R)-1-(Cyanomethyl-carbamoyl)-2-[2-(1,1-difluoro-methoxy)-phenylmethane-sulfonyl]-ethyl}-3,4-difluro-benzamide 330475-09-7 C20H17F4N3O5S
N-{(R)-1-(Cyanomethyl-carbamoyl)-2-[2-(1,1-difluoro-methoxy)-phenylmethane-sulfonyl]-ethyl}-3,4-difluro-benzamide
—— 3-[(4-hydroxycarbamoyltetrahydropyran-4-yl)-(4-phenoxybenzenesulfonyl)amino]-propionic acid ethyl ester 332049-53-3 C23H28N2O8S
3-[(4-hydroxycarbamoyltetrahydropyran-4-yl)-(4-phenoxybenzenesulfonyl)amino]-propionic acid ethyl ester
—— tert-butyl 2-[7-(2-{4-[(methylsulfonyl)amino]phenoxy}ethyl)-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl]ethylcarbamate 335620-92-3 C22H36N4O6S
tert-butyl 2-[7-(2-{4-[(methylsulfonyl)amino]phenoxy}ethyl)-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl]ethylcarbamate
—— 1-(5-(2-(2,4-Dimethoxycinnamoylamino)ethyl)-2-methoxyphenylsulfonyl)-3-ethylurea 308336-13-2 C23H29N3O7S
1-(5-(2-(2,4-Dimethoxycinnamoylamino)ethyl)-2-methoxyphenylsulfonyl)-3-ethylurea
—— (2R,3R)-3-hydroxy-2-(4'-methoxy-biphenyl-4-sulfonylamino)-6-phenoxy-hexanoic acid 334991-75-2 C25H27NO7S
(2R,3R)-3-hydroxy-2-(4'-methoxy-biphenyl-4-sulfonylamino)-6-phenoxy-hexanoic acid
—— 3-(3-bromobenzyl)-1-(3,5-dichlorophenyl)-4-hydroxy-3-methyl-1,3-dihydroindol-2-one 321981-76-4 C22H16BrCl2NO2
3-(3-bromobenzyl)-1-(3,5-dichlorophenyl)-4-hydroxy-3-methyl-1,3-dihydroindol-2-one
—— 4-(1-Ethyl-5-trifluoromethanesulfonyl-1-benzoimidazol-2-yl)-N-(2-pyrrolidin-1-yl-ethyl)-benzamide 329317-66-0 C23H25F3N4O3S
4-(1-Ethyl-5-trifluoromethanesulfonyl-1-benzoimidazol-2-yl)-N-(2-pyrrolidin-1-yl-ethyl)-benzamide
—— 5-(4-acetylamino-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid 330191-57-6 C21H17N3O9S
5-(4-acetylamino-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid
—— 4-Bromo-2'-[3-chloro-4-(2-methylbenzoyl)-phenylamino]butananilide 321371-39-5 C24H22BrClN2O2
4-Bromo-2'-[3-chloro-4-(2-methylbenzoyl)-phenylamino]butananilide
—— 7-[4-(3,4-ethylenedioxybenzylamino)benzothieno[2,3-d]pyrimidin-2-yl]heptanoic acid 329927-90-4 C26H27N3O4S
7-[4-(3,4-ethylenedioxybenzylamino)benzothieno[2,3-d]pyrimidin-2-yl]heptanoic acid
—— 3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[[(4-hydroxy-6-methyl-2-pyrimidinyl)sulfanyl]methyl]propanoic acid 321585-00-6 C21H19ClN2O5S2
3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[[(4-hydroxy-6-methyl-2-pyrimidinyl)sulfanyl]methyl]propanoic acid
—— 3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[[(5-amino-1,3,4-thiadiazol-2-yl)-sulfanyl]-methyl]propanoic acid 321584-84-3 C18H16ClN3O4S3
3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[[(5-amino-1,3,4-thiadiazol-2-yl)-sulfanyl]-methyl]propanoic acid
—— 1-(2,6-dichlorophenyl)-3-[7-(3-morpholinopropoxy)quinazolin-4-yl]urea 320363-14-2 C22H23Cl2N5O3
1-(2,6-dichlorophenyl)-3-[7-(3-morpholinopropoxy)quinazolin-4-yl]urea
—— 3-[[4-[(4-chlorobenzoyl)amino]phenyl]sulfonyl]-2-(phenoxymethyl)propanoic acid 321585-06-2 C23H20ClNO6S
3-[[4-[(4-chlorobenzoyl)amino]phenyl]sulfonyl]-2-(phenoxymethyl)propanoic acid
—— 3-[[4-[(4-cyanobenzoyl)amino]phenyl]sulfonyl]-2-(phenoxymethyl)propanoic acid 321585-08-4 C24H20N2O6S
3-[[4-[(4-cyanobenzoyl)amino]phenyl]sulfonyl]-2-(phenoxymethyl)propanoic acid
—— 2-(oxalyl-amino)-7-(1,1,3-trioxo-1,3-dihydro-1H-benzo[d]isothiazol-2-ylmethyl)-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid 330191-58-7 C18H14N2O9S2
2-(oxalyl-amino)-7-(1,1,3-trioxo-1,3-dihydro-1H-benzo[d]isothiazol-2-ylmethyl)-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid
—— 7-(5-methoxy-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,7-dihydro-5h-thieno[2,3-c]pyran-3-carboxylic acid 330191-26-9 C20H16N2O9S
7-(5-methoxy-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,7-dihydro-5h-thieno[2,3-c]pyran-3-carboxylic acid
—— 3-(2-(R)-cyclopropylmethyl-3-(S)-hydroxyl-1-oxoheptyl)amino-5-(2-fluorophenyl)-1-methyl-2,3-dihydro-1H-1,4-benzodiazepin-2-one 330839-84-4 C27H32FN3O3
3-(2-(R)-cyclopropylmethyl-3-(S)-hydroxyl-1-oxoheptyl)amino-5-(2-fluorophenyl)-1-methyl-2,3-dihydro-1H-1,4-benzodiazepin-2-one
—— N-[3-(2,6-dichloro-phenyl)-2,5-dimethyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-ethyl-piperidin-3-yl)-ethane-1,2-diamine 332178-82-2 C23H30Cl2N6
N-[3-(2,6-dichloro-phenyl)-2,5-dimethyl-pyrazolo[1,5-a]pyrimidin-7-yl]-N'-(1-ethyl-piperidin-3-yl)-ethane-1,2-diamine
—— N-methyl-4-{[(4-{[4-(4-morpholinyl)phenyl]amino}furo[2,3-d]pyridazin-7-yl)oxy]methyl}-2-pyridinecarboxamide 332012-68-7 C24H24N6O4
N-methyl-4-{[(4-{[4-(4-morpholinyl)phenyl]amino}furo[2,3-d]pyridazin-7-yl)oxy]methyl}-2-pyridinecarboxamide
—— 4-[4-(3-Chloro-5-methoxyphenoxy)anilino]-6,7-dimethoxyquinoline-3-carbonitrile 306997-92-2 C25H20ClN3O4
4-[4-(3-Chloro-5-methoxyphenoxy)anilino]-6,7-dimethoxyquinoline-3-carbonitrile
—— [2-(2,4-dichlorophenyl)ethyl](2-phenyl-7-pyridin-4-yl[1,2,4]triazolo[1,5-a]pyridin-5-yl)amine 329972-14-7 C25H19Cl2N5
[2-(2,4-dichlorophenyl)ethyl](2-phenyl-7-pyridin-4-yl[1,2,4]triazolo[1,5-a]pyridin-5-yl)amine
—— 1-{[2-(4-chlorobenzyl)-1-methyl-1H-imidazol-5-yl]methyl}-4,4-diphenylpiperidine 321405-25-8 C29H30ClN3
1-{[2-(4-chlorobenzyl)-1-methyl-1H-imidazol-5-yl]methyl}-4,4-diphenylpiperidine
—— (R)-N-[2-chloro-3-morpholino-4-(isopropylsulphonyl)phenyl]-2-hydroxy-2-methyl-3,3,3-trifluoropropanamide 329926-37-6 C17H22ClF3N2O5S
(R)-N-[2-chloro-3-morpholino-4-(isopropylsulphonyl)phenyl]-2-hydroxy-2-methyl-3,3,3-trifluoropropanamide
—— 2-(tert-butylamino)-1-[4-hydroxy-3[4-oxo-(4-nitroxybutyloxy)butyryloxy]methylphenyl]ethanol 301669-68-1 C21H32N2O9
2-(tert-butylamino)-1-[4-hydroxy-3[4-oxo-(4-nitroxybutyloxy)butyryloxy]methylphenyl]ethanol
—— N-(5-Bromo-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-bromo-4-ethoxybenzamide 318528-37-9 C18H18Br2N2O2
N-(5-Bromo-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-bromo-4-ethoxybenzamide
—— Ethyl 5-Amino-2-(4-chlorobenzylthio)-4-phenyl-thieno[2,3-d]pyrimidine-6-carboxylate 301846-14-0 C22H18ClN3O2S2
Ethyl 5-Amino-2-(4-chlorobenzylthio)-4-phenyl-thieno[2,3-d]pyrimidine-6-carboxylate
—— 2-(4-Fluorophenyl)-1-(2-cyclopropylamino-4-pyrimidinyl)-5-(4-methyl-1-piperazinyl)imidazo[4,5-b]pyridine 337902-53-1 C24H25FN8
2-(4-Fluorophenyl)-1-(2-cyclopropylamino-4-pyrimidinyl)-5-(4-methyl-1-piperazinyl)imidazo[4,5-b]pyridine
—— N-hydroxy-2-[2-[5-(4-nitrophenyl)furan-2-yl]-4-oxo-1,3-thiazolidin-3-yl]-3-phenylpropanamide 302826-92-2 C22H19N3O6S
N-hydroxy-2-[2-[5-(4-nitrophenyl)furan-2-yl]-4-oxo-1,3-thiazolidin-3-yl]-3-phenylpropanamide
—— 3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[(2-methyl-2H-1,2,3-triazol-4-yl)sulfanylmethyl]propanoic acid 321584-86-5 C19H18ClN3O4S2
3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[(2-methyl-2H-1,2,3-triazol-4-yl)sulfanylmethyl]propanoic acid
—— N-(1,3-benzothiazol-6-yl)-N-(4-{[4-(1-piperidinyl)phenyl]amino}-1-phthalazinyl)amine 332013-17-9 C26H24N6S
N-(1,3-benzothiazol-6-yl)-N-(4-{[4-(1-piperidinyl)phenyl]amino}-1-phthalazinyl)amine
—— 3-Z-[1-(4-(1-methyl-imidazol-2-yl)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone 334949-31-4 C27H22N4O3
3-Z-[1-(4-(1-methyl-imidazol-2-yl)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone
—— 5-(S)-(7-Methoxy-1-oxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid 330191-97-4 C20H19N3O7S
5-(S)-(7-Methoxy-1-oxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid
—— 4-[2-(2,3-difluorobenzoylamino)phenoxy]phthalic acid dimethyl ester 332369-76-3 C23H17F2NO6
4-[2-(2,3-difluorobenzoylamino)phenoxy]phthalic acid dimethyl ester
—— 3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[[(1-methyl-1H-imidazol-2-yl)sulfanyl]methyl]propanoic acid 321584-88-7 C20H19ClN2O4S2
3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[[(1-methyl-1H-imidazol-2-yl)sulfanyl]methyl]propanoic acid
—— 2-[3-Chloro-4-(3-chloro-pyrrolidin-1-yl)-phenylamino]-8-cyclopentyl-8H-pteridin-7-one 330550-66-8 C21H22Cl2N6O
2-[3-Chloro-4-(3-chloro-pyrrolidin-1-yl)-phenylamino]-8-cyclopentyl-8H-pteridin-7-one