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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-N-[2-chloro-3-(1-oxothiomorpholino)-4-(ethyl-sulphonyl)phenyl]-2-hydroxy-2-methyl-3,3,3-trifluoropropanamide 329925-69-1 C16H20ClF3N2O5S2
(R)-N-[2-chloro-3-(1-oxothiomorpholino)-4-(ethyl-sulphonyl)phenyl]-2-hydroxy-2-methyl-3,3,3-trifluoropropanamide
—— 2-(Oxalyl-amino)-5-(S)-((4-phenoxy-benzylamino)methyl)-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid 330191-99-6 C24H23N3O6S
2-(Oxalyl-amino)-5-(S)-((4-phenoxy-benzylamino)methyl)-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid
—— N-methyl-4-{[(4-{[4-(trifluoromethoxy)phenyl]amino}thieno[2,3-d]pyridazin-7-yl)oxy]methyl}-2-pyridinecarboxamide 332012-91-6 C21H16F3N5O3S
N-methyl-4-{[(4-{[4-(trifluoromethoxy)phenyl]amino}thieno[2,3-d]pyridazin-7-yl)oxy]methyl}-2-pyridinecarboxamide
—— 1-(5-benzyl-2-isopropoxy-3-[1,2,4]triazol-1-ylmethylphenyl)-3-(4-methyl-pyridin-2-yl)propane-1,3-dione 317333-08-7 C28H28N4O3
1-(5-benzyl-2-isopropoxy-3-[1,2,4]triazol-1-ylmethylphenyl)-3-(4-methyl-pyridin-2-yl)propane-1,3-dione
—— 1-(2,6-difluorophenyl)-3-[6-methoxy-7-(3-morpholinopropoxy)quinazolin-4-yl]urea 320363-44-8 C23H25F2N5O4
1-(2,6-difluorophenyl)-3-[6-methoxy-7-(3-morpholinopropoxy)quinazolin-4-yl]urea
—— (S)-3-[4-(2,6-Naphthyridin-1-ylamino)phenyl]-2-[2-(N-ethyl-N-iso-propylamino)-3,4-dioxocyclobut-1-enylamino]propanoic acid 312292-36-7 C26H27N5O4
(S)-3-[4-(2,6-Naphthyridin-1-ylamino)phenyl]-2-[2-(N-ethyl-N-iso-propylamino)-3,4-dioxocyclobut-1-enylamino]propanoic acid
—— 3-(3-aminomethyl-cyclohexylmethyl)-2-([2,2']bithiophenyl-5-yl)-6-methoxy-3H-quinazolin-4-one 332121-24-1 C25H27N3O2S2
3-(3-aminomethyl-cyclohexylmethyl)-2-([2,2']bithiophenyl-5-yl)-6-methoxy-3H-quinazolin-4-one
—— 1-(5-(2-(2,4-Dimethylcinnamoylamino)ethyl)-2-methoxyphenylsulfonyl)-3-methylthiourea 308336-14-3 C22H27N3O4S2
1-(5-(2-(2,4-Dimethylcinnamoylamino)ethyl)-2-methoxyphenylsulfonyl)-3-methylthiourea
—— tert-butyl 2-({7-[2-(4-cyanophenoxy)ethyl]-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl}methyl)-1-pyrrolidinecarboxylate 335620-88-7 C25H36N4O4
tert-butyl 2-({7-[2-(4-cyanophenoxy)ethyl]-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl}methyl)-1-pyrrolidinecarboxylate
—— Ethyl 2'-[3-chloro-4-(2-methylbenzoyl)-phenylamino]succinanilate 321371-40-8 C26H25ClN2O4
Ethyl 2'-[3-chloro-4-(2-methylbenzoyl)-phenylamino]succinanilate
—— 4-[4-(1-Amino-1-methylethyl)phenyl]-5-chloro-N-[4-(2-(piperidin-1-yl)ethyl)phenyl]pyrimidine-2-amine 335592-56-8 C26H32ClN5
4-[4-(1-Amino-1-methylethyl)phenyl]-5-chloro-N-[4-(2-(piperidin-1-yl)ethyl)phenyl]pyrimidine-2-amine
—— N-methyl-4-{[(4-{[4-(trifluoromethoxy)phenyl]amino}-furo[2,3-d]pyridazin-7-yl)oxy]methyl}-2-pyridinecarboxamide 332012-65-4 C21H16F3N5O4
N-methyl-4-{[(4-{[4-(trifluoromethoxy)phenyl]amino}-furo[2,3-d]pyridazin-7-yl)oxy]methyl}-2-pyridinecarboxamide
—— 2-Bromo-4H-thieno[3,2-b]pyrrole-5-carboxylic acid [(1S)-benzyl-2-(3-hydroxy-azetidin-1-yl)-2-oxo-ethyl]-amide 332098-67-6 C19H18BrN3O3S
2-Bromo-4H-thieno[3,2-b]pyrrole-5-carboxylic acid [(1S)-benzyl-2-(3-hydroxy-azetidin-1-yl)-2-oxo-ethyl]-amide
—— 3-(Octahydro-7-indolizinyl)-2,5-dichlorobenzenesulfonyl-5-azaindole 325975-39-1 C21H21Cl2N3O2S
3-(Octahydro-7-indolizinyl)-2,5-dichlorobenzenesulfonyl-5-azaindole
—— 3-{2-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazolo[1,5-a]pyrimidin-7-ylamino]-ethylamino}-propane-1,2-diol 332178-53-7 C20H25Cl2N5O3
3-{2-[3-(2,6-dichloro-4-methoxy-phenyl)-2,5-dimethyl-pyrazolo[1,5-a]pyrimidin-7-ylamino]-ethylamino}-propane-1,2-diol
—— 3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[(2-pyridinylsulfanyl)methyl]propanoic acid 321584-78-5 C21H18ClNO4S2
3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[(2-pyridinylsulfanyl)methyl]propanoic acid
—— N-[2-(Benzo[b]thiophen-5-yl-methanesulfonyl)-1-(3,4-dichlorophenyl)-ethyl]-N-hydroxy-formamide 376386-98-0 C18H15Cl2NO4S2
N-[2-(Benzo[b]thiophen-5-yl-methanesulfonyl)-1-(3,4-dichlorophenyl)-ethyl]-N-hydroxy-formamide
—— 2-[(S)-1-(3-Nitrophenyl)ethylamino]-4-[5-(pyridazin-3-yl)benzimidazol-1-yl]pyrimidine 317829-46-2 C23H18N8O2
2-[(S)-1-(3-Nitrophenyl)ethylamino]-4-[5-(pyridazin-3-yl)benzimidazol-1-yl]pyrimidine
—— 25-(N-ethyl-N-methylamino)-3-hydroxy-24-homo-19-nor-cholest-1,3,5(10),16-tetraene 305812-21-9 C30H47NO
25-(N-ethyl-N-methylamino)-3-hydroxy-24-homo-19-nor-cholest-1,3,5(10),16-tetraene
—— 1-[2-[3-chloro-4-(2-methylbenzoyl)-phenylamino]phenyl]-3-iso-propylurea 321438-14-6 C24H24ClN3O2
1-[2-[3-chloro-4-(2-methylbenzoyl)-phenylamino]phenyl]-3-iso-propylurea
—— (2R)-1-[(N-benzyl-N-methyl)amino]-3-[3-(thieno[2,3-d]isoxazol-3-yl)phenoxy]-2-propanol hydrochloride 330650-04-9 C22H22N2O3S*ClH
(2R)-1-[(N-benzyl-N-methyl)amino]-3-[3-(thieno[2,3-d]isoxazol-3-yl)phenoxy]-2-propanol hydrochloride
—— 4-({3-[7-(phenylsulfonyl)-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl]propyl}amino)benzonitrile 335620-94-5 C22H26N4O3S
4-({3-[7-(phenylsulfonyl)-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl]propyl}amino)benzonitrile
—— N-(3-acetylphenyl)-N'-[1-[[(3S)-3-[(4-fluorophenyl)methyl]piperidinyl]methyl]cyclopropyl]-urea 383430-04-4 C25H30FN3O2
N-(3-acetylphenyl)-N'-[1-[[(3S)-3-[(4-fluorophenyl)methyl]piperidinyl]methyl]cyclopropyl]-urea
—— [2-(2-chlorophenyl)ethyl](2-phenyl-7-pyridin-4-yl[1,2,4]triazolo[1,5-a]pyridin-5-yl)amine 329972-13-6 C25H20ClN5
[2-(2-chlorophenyl)ethyl](2-phenyl-7-pyridin-4-yl[1,2,4]triazolo[1,5-a]pyridin-5-yl)amine
—— 6-(3Chlorophenyl)-4-cyclopropyl-1-(4-methoxybenzyl)-1H-quinazolin-2-one 304857-62-3 C25H21ClN2O2
6-(3Chlorophenyl)-4-cyclopropyl-1-(4-methoxybenzyl)-1H-quinazolin-2-one
—— N-(5-Trifluoromethyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-4-methoxy-3-trifluoromethylbenzamide 318528-40-4 C19H16F6N2O2
N-(5-Trifluoromethyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-4-methoxy-3-trifluoromethylbenzamide
—— (2R,3R)-5-tert-butoxycarbonylamino-3-hydroxy-2-(4-methoxy-benzenesulfonylamino)-pentanoic acid 334991-82-1 C17H26N2O8S
(2R,3R)-5-tert-butoxycarbonylamino-3-hydroxy-2-(4-methoxy-benzenesulfonylamino)-pentanoic acid
—— N-(5-Bromo-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-chloro-4-ethoxybenzamide 318528-36-8 C18H18BrClN2O2
N-(5-Bromo-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-chloro-4-ethoxybenzamide
—— 2-{[4-(3-chloropropoxy)-benzenesulfonyl]-pyridin-3-ylmethyl-amino}-N-hydroxy-acetamide 325785-01-1 C17H20ClN3O5S
2-{[4-(3-chloropropoxy)-benzenesulfonyl]-pyridin-3-ylmethyl-amino}-N-hydroxy-acetamide
—— 3-(2 (R)-Isobutyl-3(S)-hydroxyl-1-oxo-butyl)amino-1-methyl-5-phenyl-2,3-dihydro-1H-1,4-benzodiazepin-2-one 330839-73-1 C24H29N3O3
3-(2 (R)-Isobutyl-3(S)-hydroxyl-1-oxo-butyl)amino-1-methyl-5-phenyl-2,3-dihydro-1H-1,4-benzodiazepin-2-one
—— methyl 4-((4-((5 S)-5-((acetylamino)methyl)-2-oxo-1,3-oxazolidin-3-yl)-2-fluorophenyl)ethynyl)benzoate 355004-55-6 C22H19FN2O5
methyl 4-((4-((5 S)-5-((acetylamino)methyl)-2-oxo-1,3-oxazolidin-3-yl)-2-fluorophenyl)ethynyl)benzoate
—— (R)-1-(4-benzo[b]thiophen-3-yl-phenoxy)-3-(4-fluoro-benzylamino)-propan-2-ol 330669-78-8 C24H22FNO2S
(R)-1-(4-benzo[b]thiophen-3-yl-phenoxy)-3-(4-fluoro-benzylamino)-propan-2-ol
—— 3-chloro-6,7-dimethoxy-N-(4-phenoxyphenyl)quinolin-4-amine 304904-43-6 C23H19ClN2O3
3-chloro-6,7-dimethoxy-N-(4-phenoxyphenyl)quinolin-4-amine
—— 8-(4-Fluoro-2-methyl-phenyl)-4-(3-imidazol-1-yl-phenyl)-1,3-dihydro-benzo[b][1,4]diazepin-2-one 335258-30-5 C25H19FN4O
8-(4-Fluoro-2-methyl-phenyl)-4-(3-imidazol-1-yl-phenyl)-1,3-dihydro-benzo[b][1,4]diazepin-2-one
—— dimethyl-[3-(8-oxa-1-thia-dibenzo[e,h]azulene-2-ylmethoxy)-propyl]-amine hydrochloride 374799-32-3 C22H23NO2S*ClH
dimethyl-[3-(8-oxa-1-thia-dibenzo[e,h]azulene-2-ylmethoxy)-propyl]-amine hydrochloride
—— 1-[5-(3,4-Dichlorophenyl)-4-pyridin-4-yl-1H-imidazol-2-yl]-1-piperidin-1-yl-methanone 359888-77-0 C20H18Cl2N4O
1-[5-(3,4-Dichlorophenyl)-4-pyridin-4-yl-1H-imidazol-2-yl]-1-piperidin-1-yl-methanone
—— ethyl (3S,4aR,6S,8aR)-6-[[(2S)-2-ethoxycarbonyl-4,4-difluoropyrrolidin-1-yl]methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylate 317844-31-8 C20H32F2N2O4
ethyl (3S,4aR,6S,8aR)-6-[[(2S)-2-ethoxycarbonyl-4,4-difluoropyrrolidin-1-yl]methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylate
—— N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3,4-dichlorobenzyl)-4-piperidinamine 328082-02-6 C18H23Cl3N4
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3,4-dichlorobenzyl)-4-piperidinamine
—— N-[5-(2-chlorophenyl)-3-methyl-2,10-dihydropyrazolo[3,4-b][1,4]benzodiazepin-7-yl]methanesulfonamide 303196-54-5 C18H16ClN5O2S
N-[5-(2-chlorophenyl)-3-methyl-2,10-dihydropyrazolo[3,4-b][1,4]benzodiazepin-7-yl]methanesulfonamide
—— 4-[{[4-(3,5-ditert-butyl-4-hydroxyphenyl)-1,3-thiazol-2-yl]methyl}(methyl)amino]butanenitrile 335242-81-4 C23H33N3OS
4-[{[4-(3,5-ditert-butyl-4-hydroxyphenyl)-1,3-thiazol-2-yl]methyl}(methyl)amino]butanenitrile
—— 2-(4-{[2-(4-pyridyl)-2,8-diazaspiro[4.5]dec-8-yl]carbonyl}phenoxy)acetic acid 336190-85-3 C22H25N3O4
2-(4-{[2-(4-pyridyl)-2,8-diazaspiro[4.5]dec-8-yl]carbonyl}phenoxy)acetic acid
—— 3-[5-(2-hydroxy-4-isopropoxybenzoyl)-2-isobutoxyphenyl] propanoic acid 374893-06-8 C23H28O6
3-[5-(2-hydroxy-4-isopropoxybenzoyl)-2-isobutoxyphenyl] propanoic acid
—— 3-anilino-5-(2-(4-chlorophenyl)-thiazol-4-ylmethylthio)-1,2,4-triazole 334538-64-6 C18H14ClN5S2
3-anilino-5-(2-(4-chlorophenyl)-thiazol-4-ylmethylthio)-1,2,4-triazole
—— 4-Chloro-N-[3-(3,4-dichloro-phenoxy)-propyl]-benzenesulfonamide 333799-61-4 C15H14Cl3NO3S
4-Chloro-N-[3-(3,4-dichloro-phenoxy)-propyl]-benzenesulfonamide
—— 3(S)-(2-Methyl-pyrimidin-5-yl)-5-hydroxy-9-(5,6,7,8-tetrahydro-[1,8]-naphthyridin-2-yl)-nonanoic acid 312261-80-6 C22H30N4O3
3(S)-(2-Methyl-pyrimidin-5-yl)-5-hydroxy-9-(5,6,7,8-tetrahydro-[1,8]-naphthyridin-2-yl)-nonanoic acid
—— 1-benzyl-4-[(5,6-dimethoxy-2-amino-1-indanon)-2-yl]methylpiperidine 329010-77-7 C24H30N2O3
1-benzyl-4-[(5,6-dimethoxy-2-amino-1-indanon)-2-yl]methylpiperidine
—— 2-(p-(2,4-dioxothiazolidin-5-ylmethyl)phenoxy)ethel-5-methoxyindole 311312-29-5 C21H20N2O4S
2-(p-(2,4-dioxothiazolidin-5-ylmethyl)phenoxy)ethel-5-methoxyindole
—— 7-(N-cyclopropyl-carbamoyl)-5-(4-amino-3-methyl-phenyl)-8-methyl-7H-1,3-dioxolo[4,5-h][2,3]benzodiazepine 319907-75-0 C22H22N4O3
7-(N-cyclopropyl-carbamoyl)-5-(4-amino-3-methyl-phenyl)-8-methyl-7H-1,3-dioxolo[4,5-h][2,3]benzodiazepine
—— 3-(2-chlorophenyl)-7-(4-oxo-cyclohexylamino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one 335652-22-7 C19H20ClN5O2
3-(2-chlorophenyl)-7-(4-oxo-cyclohexylamino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one
—— 1-(6,7,8,9-tetrahydro-5H-10-oxabenzo[a]azulene-2-sulfonylamino)cyclopentane carboxylic acid hydroxyamide 326499-89-2 C19H24N2O5S
1-(6,7,8,9-tetrahydro-5H-10-oxabenzo[a]azulene-2-sulfonylamino)cyclopentane carboxylic acid hydroxyamide