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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl 1-[(2R)-2-[[(3R)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carbonyl]amino]-3-(4-chlorophenyl)propanoyl]-4-cyclohexylpiperidine-4-carboxylate 312639-65-9 C33H48ClN3O4
ethyl 1-[(2R)-2-[[(3R)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carbonyl]amino]-3-(4-chlorophenyl)propanoyl]-4-cyclohexylpiperidine-4-carboxylate
—— 1-[[1-[3-(Aminomethyl)phenyl]-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl]-5-[2-(aminosulfonyl)phenyl]-2,3-dihydro-1H-indole 321435-61-4 C26H22F3N5O3S
1-[[1-[3-(Aminomethyl)phenyl]-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl]-5-[2-(aminosulfonyl)phenyl]-2,3-dihydro-1H-indole
—— (3S)-3-{3-[2-methyl-(1S)-1-(2-naphthalenecarbonylamino)-propyl]-4,5-dihydro-isoxazole-5-carbonylamino}-4-keto-5-phenoxy-pentanoic acid 331778-78-0 C30H31N3O7
(3S)-3-{3-[2-methyl-(1S)-1-(2-naphthalenecarbonylamino)-propyl]-4,5-dihydro-isoxazole-5-carbonylamino}-4-keto-5-phenoxy-pentanoic acid
—— ethyl 2-{2-methyl-4-[({4-methyl-2-[3,5-bis(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy}acetate 317318-81-3 C24H21F6NO3S2
ethyl 2-{2-methyl-4-[({4-methyl-2-[3,5-bis(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy}acetate
—— 1-tert-Butyl-3-(2-{4-[4-(3-morpholin-4-yl-propyl)-piperidin-1-yl]-phenylamino}-pteridin-7-yl)-urea 330550-89-5 C29H41N9O2
1-tert-Butyl-3-(2-{4-[4-(3-morpholin-4-yl-propyl)-piperidin-1-yl]-phenylamino}-pteridin-7-yl)-urea
—— 4-(4-fluor-phenyl)-2-piperazin-1-yl-pyrimidine-5-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide 311340-28-0 C25H22F7N5O
4-(4-fluor-phenyl)-2-piperazin-1-yl-pyrimidine-5-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide
—— 5-(4-benzyloxy-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid 330191-42-9 C26H20N2O9S
5-(4-benzyloxy-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid
—— 4-[4-[7-(butylsulfonyl)-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl]-1-(3,4-dimethoxyphenoxy)butyl]benzonitrile 335619-26-6 C29H39N3O6S
4-[4-[7-(butylsulfonyl)-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl]-1-(3,4-dimethoxyphenoxy)butyl]benzonitrile
—— 5-Bromo-N-(4-Bromophenyl)-2-(4-methoxyphenylsulfonamido)benzamide 320715-37-5 C20H16Br2N2O4S
5-Bromo-N-(4-Bromophenyl)-2-(4-methoxyphenylsulfonamido)benzamide
—— 1-acetyl-4-(4-{2-[3-methoxy-4-(3-o-tolyl-ureido)-phenyl]-acetylamino}-phenyl)-pyrrolidine-3-carboxylic acid 306305-23-7 C30H32N4O6
1-acetyl-4-(4-{2-[3-methoxy-4-(3-o-tolyl-ureido)-phenyl]-acetylamino}-phenyl)-pyrrolidine-3-carboxylic acid
—— 1-[1-(3-benzyloxypropyl)-1H-imidazol-5-yl]methyl-3-(morpholin-4-yl) carbonyl-4-(naphthalen-1-yl)-1H-pyrrole 303778-37-2 C33H34N4O3
1-[1-(3-benzyloxypropyl)-1H-imidazol-5-yl]methyl-3-(morpholin-4-yl) carbonyl-4-(naphthalen-1-yl)-1H-pyrrole
—— (2S)-N-[(3S)-5-methyl-2-oxo-1-(2,3,4,5-tetrahydro-1,4-benzothiazepin-4-yl)-3-hexyl]-2-benzyloxycarbonylamino-4-methylpentanamide 352356-18-4 C30H41N3O4S
(2S)-N-[(3S)-5-methyl-2-oxo-1-(2,3,4,5-tetrahydro-1,4-benzothiazepin-4-yl)-3-hexyl]-2-benzyloxycarbonylamino-4-methylpentanamide
—— 2'-(4-trifluoromethylbenzyloxycarbonylaminomethyl)biphenyl-2-carboxylic acid phenethylamide 332378-34-4 C31H27F3N2O3
2'-(4-trifluoromethylbenzyloxycarbonylaminomethyl)biphenyl-2-carboxylic acid phenethylamide
—— 1-[3-benzyl-5-(4-methyl-5-thioxo-3-trifluoromethyl-4,5-dihydro-[1,24]-triazol-1-ylmethyl)phenyl]-3-(4-methylpyridin-2-yl)propane-1,3-dione 317333-56-5 C27H23F3N4O2S
1-[3-benzyl-5-(4-methyl-5-thioxo-3-trifluoromethyl-4,5-dihydro-[1,24]-triazol-1-ylmethyl)phenyl]-3-(4-methylpyridin-2-yl)propane-1,3-dione
—— 5-(4-benzyloxy-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid 330192-04-6 C26H21N3O8S
5-(4-benzyloxy-1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl)-2-(oxalyl-amino)-4,5,6,7-tetrahydro-thieno[2,3-c]pyridine-3-carboxylic acid
—— 5-Bromo-N-(4-bromophenyl)-2-(2-fluorophenylsulfonamido)benzamide 314018-68-3 C19H13Br2FN2O3S
5-Bromo-N-(4-bromophenyl)-2-(2-fluorophenylsulfonamido)benzamide
—— 4-[4,5-dichloro-2-(3-nitrobenzoylamino)phenoxy]phthalic acid dimethyl ester 332370-23-7 C23H16Cl2N2O8
4-[4,5-dichloro-2-(3-nitrobenzoylamino)phenoxy]phthalic acid dimethyl ester
—— 6-(3,5-Dimethoxyphenyl)-8-ethyl-2-[[4-[2-(diethylamino)ethoxy]-phenyl]amino]-8H-pteridin-7-one 330550-49-7 C28H34N6O4
6-(3,5-Dimethoxyphenyl)-8-ethyl-2-[[4-[2-(diethylamino)ethoxy]-phenyl]amino]-8H-pteridin-7-one
—— 1-[2-(2-(2-chlorophenyl)ethylamino)pyrimidin-4-yl]-2-(3-trifluoromethylphenyl)-1H-imidazole4-carboxylic acid ethyl ester 306297-74-5 C25H21ClF3N5O2
1-[2-(2-(2-chlorophenyl)ethylamino)pyrimidin-4-yl]-2-(3-trifluoromethylphenyl)-1H-imidazole4-carboxylic acid ethyl ester
—— 5H-[1,4]oxathiepino[6,5-b]pyridine-8-carboxylic acid, 2,3,6,9-tetrahydro-7-methyl-9-(3-nitrophenyl), 2-[methyl(phenylmethyl)amino]ethyl ester, 1,1-dioxide 319908-90-2 C26H29N3O7S
5H-[1,4]oxathiepino[6,5-b]pyridine-8-carboxylic acid, 2,3,6,9-tetrahydro-7-methyl-9-(3-nitrophenyl), 2-[methyl(phenylmethyl)amino]ethyl ester, 1,1-dioxide
—— tris(2-(1,1-dimethylpropyl)phenyl)phosphite 31570-01-1 C33H45O3P
tris(2-(1,1-dimethylpropyl)phenyl)phosphite
—— 4-[(N-{[4-({[(2-methylphenyl)amino]carbonyl}amino)phenyl]acetyl}-L-leucyl)amino]benzoic acid 370596-25-1 C29H32N4O5
4-[(N-{[4-({[(2-methylphenyl)amino]carbonyl}amino)phenyl]acetyl}-L-leucyl)amino]benzoic acid
—— 1-(3-carbamimidoylphenyl)-N-[2-chloro-4-(2-sulfamoylphenyl)phenyl]piperidine-2-carboxamide 308108-26-1 C25H26ClN5O3S
1-(3-carbamimidoylphenyl)-N-[2-chloro-4-(2-sulfamoylphenyl)phenyl]piperidine-2-carboxamide
—— (2S)-3-[4-(2-{4-[(tert-Butoxycarbonyl)amino]phenyl}ethoxy)phenyl]-2-ethoxypropyl methanesulfonate 343880-35-3 C25H35NO7S
(2S)-3-[4-(2-{4-[(tert-Butoxycarbonyl)amino]phenyl}ethoxy)phenyl]-2-ethoxypropyl methanesulfonate
—— 25-benzamido-3-hydroxy-24-homo-19-nor-cholest-1,3,5(10),16-tetraene 305812-25-3 C34H45NO2
25-benzamido-3-hydroxy-24-homo-19-nor-cholest-1,3,5(10),16-tetraene
—— 3-Z-[1-(4-(N-((2-dimethylamino-ethyl)-carbonyl)-N-methyl-amino)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone 334949-36-9 C29H30N4O4
3-Z-[1-(4-(N-((2-dimethylamino-ethyl)-carbonyl)-N-methyl-amino)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone
—— 1-[[1-[3-(aminomethyl)phenyl]-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl]-2,3-dihydro-5-(1-pyrrolidinylcarbonyl)-1H-indole 321435-77-2 C25H24F3N5O2
1-[[1-[3-(aminomethyl)phenyl]-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl]-2,3-dihydro-5-(1-pyrrolidinylcarbonyl)-1H-indole
—— 2-(4-fluoro-2-methyl-phenyl)-3-methyl-piperazine-1-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide 334476-73-2 C23H24F7N3O
2-(4-fluoro-2-methyl-phenyl)-3-methyl-piperazine-1-carboxylic acid (3,5-bis-trifluoromethyl-benzyl)-methyl-amide
—— 2-((3S)-2-Oxo-3-{[(4-pyrimidin-5-ylphenyl)sulfonyl]amino}piperidyl)-N-[2-(amidinoaminooxy)ethyl]acetamide 330668-17-2 C20H26N8O5S
2-((3S)-2-Oxo-3-{[(4-pyrimidin-5-ylphenyl)sulfonyl]amino}piperidyl)-N-[2-(amidinoaminooxy)ethyl]acetamide
—— (2R,3R)-5-tert-butoxycarbonylamino-3-hydroxy-2-(4'-methoxy-biphenyl-4-sulfonylamino)-pentanoic acid 334991-80-9 C23H30N2O8S
(2R,3R)-5-tert-butoxycarbonylamino-3-hydroxy-2-(4'-methoxy-biphenyl-4-sulfonylamino)-pentanoic acid
—— (2R,3S)-3-hydroxy-2-(4'-methoxy-biphenyl-4-sulfonylamino)-4-(1-methyl-1H-imidazol-2-ylsulfanyl)-butyric acid 334991-66-1 C21H23N3O6S2
(2R,3S)-3-hydroxy-2-(4'-methoxy-biphenyl-4-sulfonylamino)-4-(1-methyl-1H-imidazol-2-ylsulfanyl)-butyric acid
—— 1-(4-Acetoaminophenyl)-4-(4-fluorophenyl)-2-(3-phenylpropyl)-3-(4-pyridyl)pyrrole 308280-12-8 C32H28FN3O
1-(4-Acetoaminophenyl)-4-(4-fluorophenyl)-2-(3-phenylpropyl)-3-(4-pyridyl)pyrrole
—— 3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[(1H-benzimidazol-2-ylsulfanyl)methyl]propanoic acid 321585-12-0 C23H19ClN2O4S2
3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[(1H-benzimidazol-2-ylsulfanyl)methyl]propanoic acid
—— 2-[[3-(aminooxoacetyl)-2-ethyl-1-(phenylmethyl)-1H-indol-4-yl]oxy]-N-(methyl)-N-(phenyloxy)acetamide 331441-05-5 C28H27N3O5
2-[[3-(aminooxoacetyl)-2-ethyl-1-(phenylmethyl)-1H-indol-4-yl]oxy]-N-(methyl)-N-(phenyloxy)acetamide
—— (R)-2-{(Benzo[b]thiophen-5-ylmethanesulfonyl)[2-(2-methoxyethoxy)-ethyl]amino}-N-hydroxy-2-phenylacetamide 355851-01-3 C22H26N2O6S2
(R)-2-{(Benzo[b]thiophen-5-ylmethanesulfonyl)[2-(2-methoxyethoxy)-ethyl]amino}-N-hydroxy-2-phenylacetamide
—— 3-[[4-(4-chlorophenoxy)benzenesulfonyl]-(1-hydroxycarbamoylcyclopentyl)amino]-propionic acid 332049-59-9 C21H23ClN2O7S
3-[[4-(4-chlorophenoxy)benzenesulfonyl]-(1-hydroxycarbamoylcyclopentyl)amino]-propionic acid
—— (S)-3-[4-([2,6-Naphthyridin-1-yl]amino)phenyl]-2-[(2-N,N-dipropylamino-3,4-dioxocyclobut-1-enyl)amino]propanoic acid 312292-29-8 C27H29N5O4
(S)-3-[4-([2,6-Naphthyridin-1-yl]amino)phenyl]-2-[(2-N,N-dipropylamino-3,4-dioxocyclobut-1-enyl)amino]propanoic acid
—— 2-[5-[2-(benzylamino)-2-oxoethyl]-2-(4-methoxyphenyl)-4-oxo-1,3-thiazolidin-3-yl]-N-hydroxy-4-methylpentanamide 302829-86-3 C25H31N3O5S
2-[5-[2-(benzylamino)-2-oxoethyl]-2-(4-methoxyphenyl)-4-oxo-1,3-thiazolidin-3-yl]-N-hydroxy-4-methylpentanamide
—— 4-[4-(3,4-ethylenedioxybenzylamino)benzothieno[2,3-d]pyrimidin-2-yl]cyclohexanecarboxylic acid 329927-92-6 C26H25N3O4S
4-[4-(3,4-ethylenedioxybenzylamino)benzothieno[2,3-d]pyrimidin-2-yl]cyclohexanecarboxylic acid
—— 1-{[1-(4-chloro-2-methoxybenzyl)-1H-pyrazol-3-yl]methyl}-4,4-diphenylpiperidine 321405-16-7 C29H30ClN3O
1-{[1-(4-chloro-2-methoxybenzyl)-1H-pyrazol-3-yl]methyl}-4,4-diphenylpiperidine
—— (2R,3S)-4-(3,3-dimethyl-butoxy)-3-hydroxy-2-(4'-methoxy-biphenyl-4-sulfonylamino)-butyric acid 334991-76-3 C23H31NO7S
(2R,3S)-4-(3,3-dimethyl-butoxy)-3-hydroxy-2-(4'-methoxy-biphenyl-4-sulfonylamino)-butyric acid
—— N-hydroxy 2-[(4-{4-[3-(2-hydroxyethoxy)-1H-pyrazol-1-yl]-3-methylphenyl}piperidin-1-yl)sulphonyl]-2-methylpropanamide 312930-93-1 C21H30N4O6S
N-hydroxy 2-[(4-{4-[3-(2-hydroxyethoxy)-1H-pyrazol-1-yl]-3-methylphenyl}piperidin-1-yl)sulphonyl]-2-methylpropanamide
—— 3-(2-(R)-iso-butyl-3-(S)-hydroxyl-1-oxoheptyl)amino-5-(4-fluorophenyl)-1-methyl-2,3-dihydro-1H-1,4-benzodiazepin-2-one 330840-18-1 C27H34FN3O3
3-(2-(R)-iso-butyl-3-(S)-hydroxyl-1-oxoheptyl)amino-5-(4-fluorophenyl)-1-methyl-2,3-dihydro-1H-1,4-benzodiazepin-2-one
—— {4-[4-(8-Cyclopentyl-5-methyl-7-oxo-5,6,7,8-tetrahydro-pteridin-2-ylamino)-phenyl]-piperazin-1-yl}-acetic acid 330550-85-1 C24H31N7O3
{4-[4-(8-Cyclopentyl-5-methyl-7-oxo-5,6,7,8-tetrahydro-pteridin-2-ylamino)-phenyl]-piperazin-1-yl}-acetic acid
—— 2-[(S)-1-(3-Trifluoromethylphenyl)ethylamino]-4-[5-(pyridazin-3-yl)benzimidazol-1-yl]pyrimidine 317829-47-3 C24H18F3N7
2-[(S)-1-(3-Trifluoromethylphenyl)ethylamino]-4-[5-(pyridazin-3-yl)benzimidazol-1-yl]pyrimidine
—— 5-[7-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-4-benzothiophenyl-methyl]-2,4-thiazolidinedione 385395-39-1 C24H20N2O4S2
5-[7-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-4-benzothiophenyl-methyl]-2,4-thiazolidinedione
—— 5-((benzyloxy)(1-methyl-1H-imidazol-5-yl)methyl)-2'-isopropyl(1,1'-biphenyl)-2-carbonitrile hydrochloride 371761-30-7 C28H27N3O*ClH
5-((benzyloxy)(1-methyl-1H-imidazol-5-yl)methyl)-2'-isopropyl(1,1'-biphenyl)-2-carbonitrile hydrochloride
—— 3-[2-[(phenylmethyl)amino]4-pyridinyl]-2-[3-(trifluoromethyl)phenyl]-imidazo[1,2-a]pyrimidin-7-amine 340042-04-8 C25H19F3N6
3-[2-[(phenylmethyl)amino]4-pyridinyl]-2-[3-(trifluoromethyl)phenyl]-imidazo[1,2-a]pyrimidin-7-amine
—— {(R)-1-(Cyanomethyl-carbamoyl)-2-[2-(1,1-difluoro-methoxy)-phenylmethane-sulfonyl]-ethyl}-carbamic acid isobutyl ester 330475-07-5 C18H23F2N3O6S
{(R)-1-(Cyanomethyl-carbamoyl)-2-[2-(1,1-difluoro-methoxy)-phenylmethane-sulfonyl]-ethyl}-carbamic acid isobutyl ester
—— 2-[3-chloro-4-({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methoxy)phenyl]acetic acid 317318-40-4 C20H15ClF3NO3S
2-[3-chloro-4-({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methoxy)phenyl]acetic acid