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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R,S)-3-mercaptomethyl-2,3-dihydro-5H-thiazolo[2,3-b]chinazolin-5-on 363178-89-6 C11H10N2OS2
(R,S)-3-mercaptomethyl-2,3-dihydro-5H-thiazolo[2,3-b]chinazolin-5-on
—— 4-(2-pyridyl)-5-(4-pyridyl)-2-pyrimidinylamine 371230-39-6 C14H11N5
4-(2-pyridyl)-5-(4-pyridyl)-2-pyrimidinylamine
—— 2-(5-bromo-3-pyridyl)methyl-1,4,5,6-tetrahydropyrimidine 371122-04-2 C10H12BrN3
2-(5-bromo-3-pyridyl)methyl-1,4,5,6-tetrahydropyrimidine
—— (E)-N-(3-methylbenzyl)cinnamamidine 381689-93-6 C17H18N2
(E)-N-(3-methylbenzyl)cinnamamidine
—— (1S,5R)-6-(5-bromo-3-pyridinyl)-3,6-diazabicyclo[3.2.0]heptane 370881-53-1 C10H12BrN3
(1S,5R)-6-(5-bromo-3-pyridinyl)-3,6-diazabicyclo[3.2.0]heptane
—— 5,8-dimethyl-6,7-dioxo-5,8,14-triazatetracyclo[10.3.1.02,11.04,9]hexadeca-2(11),3,9-triene 357424-08-9 C15H17N3O2
5,8-dimethyl-6,7-dioxo-5,8,14-triazatetracyclo[10.3.1.02,11.04,9]hexadeca-2(11),3,9-triene
—— 1-(2-aminopropyl)-3,7,8,9-tetrahydro-pyrano[3,2-e]indol-8-ol 362603-47-2 C14H18N2O2
1-(2-aminopropyl)-3,7,8,9-tetrahydro-pyrano[3,2-e]indol-8-ol
—— 2-thio-3'-deoxy-uridine 37097-53-3 C9H12N2O4S
2-thio-3'-deoxy-uridine
—— 4-bromo-3-Pyridinesulfonamide 361544-09-4 C5H5BrN2O2S
4-bromo-3-Pyridinesulfonamide
—— furan-3-ylmethyl-(3-[1H-1,2,3-triazol-4-yl]phenyl)amine 369363-86-0 C13H12N4O
furan-3-ylmethyl-(3-[1H-1,2,3-triazol-4-yl]phenyl)amine
—— 2-(1-cyclohexen-1-ylethynyl)-5-nitro-1,3-thiazole 329202-27-9 C11H10N2O2S
2-(1-cyclohexen-1-ylethynyl)-5-nitro-1,3-thiazole
—— ((3R,5S)-1-Hydroxymethyl-3,5-dimethyl-cyclohexyl)-acetic acid, sodium salt 344574-37-4 C11H19O3*Na
((3R,5S)-1-Hydroxymethyl-3,5-dimethyl-cyclohexyl)-acetic acid, sodium salt
—— 4-[2-(2-naphthyl)ethynyl]pyridine 364064-85-7 C17H11N
4-[2-(2-naphthyl)ethynyl]pyridine
—— 3-(5-Ethyl-3-pyridyl)-3,7-diazabicyclo[3.3.0]octane 345317-13-7 C13H19N3
3-(5-Ethyl-3-pyridyl)-3,7-diazabicyclo[3.3.0]octane
—— 3-(3-Pyridyl)-3,7-diazabicyclo[3.3.2]decane 345317-27-3 C13H19N3
3-(3-Pyridyl)-3,7-diazabicyclo[3.3.2]decane
—— 2-(3-thienyl)methyl-1,4,5, 6-tetrahydropyrimidine 371122-30-4 C9H12N2S
2-(3-thienyl)methyl-1,4,5, 6-tetrahydropyrimidine
—— 1,2-propylene glycol monopivalate 37086-87-6 C8H16O3
1,2-propylene glycol monopivalate
—— 2-(5-methyl-3-pyridyl)methyl-1,4,5,6-tetrahydropyrimidine 371123-03-4 C11H15N3
2-(5-methyl-3-pyridyl)methyl-1,4,5,6-tetrahydropyrimidine
—— (8aS)-7-[5-(4-fluorophenyl)-4-pyridin-4-yl-1H-pyrrol-3-yl]-1,2,3,5,6,8a-hexahydroindolizine 321344-57-4 C23H22FN3
(8aS)-7-[5-(4-fluorophenyl)-4-pyridin-4-yl-1H-pyrrol-3-yl]-1,2,3,5,6,8a-hexahydroindolizine
—— 2-{4-[2-methyl-2-(nitrosothio)propyl]piperazinyl}ethyl 2-{2-[(2,6-dichlorophenyl)amino]phenyl}acetate citrate 364055-65-2 C6H8O7*C24H30Cl2N4O3S
2-{4-[2-methyl-2-(nitrosothio)propyl]piperazinyl}ethyl 2-{2-[(2,6-dichlorophenyl)amino]phenyl}acetate citrate
—— Ethyl (E)-3-[5,6-bis-([1,1'-biphenyl]-4-ylmethoxy)-3-(4-chlorophenoxy)-benzo[b]thiophen-2-yl]-propenoate 334720-03-5 C45H35ClO5S
Ethyl (E)-3-[5,6-bis-([1,1'-biphenyl]-4-ylmethoxy)-3-(4-chlorophenoxy)-benzo[b]thiophen-2-yl]-propenoate
—— 4-[({4-[(4-chlorophenyl)amino]furo[2,3-d]pyridazin-7-yl}oxy)methyl]-N-methyl-2-pyridinecarboxamide 4-chlorobenzenesulfonate 332013-25-9 C6H5ClO3S*C20H16ClN5O3
4-[({4-[(4-chlorophenyl)amino]furo[2,3-d]pyridazin-7-yl}oxy)methyl]-N-methyl-2-pyridinecarboxamide 4-chlorobenzenesulfonate
—— 5-[[1-(3-amino-1,2-benzisoxazol-5-yl)-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl]-8-[2-(aminosulfonyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzoxazepine 321435-83-0 C27H21F3N6O5S
5-[[1-(3-amino-1,2-benzisoxazol-5-yl)-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl]-8-[2-(aminosulfonyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzoxazepine
—— 2-(1,1-dimethylethoxycarbonylamino)-8-{3-[4-(5-chloro-2-methoxyphenyl)-1-piperazinyl]-propylcarbamoyl}-3-methyl-4-oxo-4H-1-benzopyran 335086-88-9 C30H37ClN4O6
2-(1,1-dimethylethoxycarbonylamino)-8-{3-[4-(5-chloro-2-methoxyphenyl)-1-piperazinyl]-propylcarbamoyl}-3-methyl-4-oxo-4H-1-benzopyran
—— 2-[(2,4-dichloro-6-methylphenyl)amino]-5-ethylbenzeneacetic acid 346670-74-4 C17H17Cl2NO2
2-[(2,4-dichloro-6-methylphenyl)amino]-5-ethylbenzeneacetic acid
—— 4-{2-[3,4-Bis(difluoromethoxy)phenyl]-2-[6-(4-fluorophenylmethanesulfonyl)3-pyridyl]ethyl}pyridine-N-oxide 308281-64-3 C27H21F5N2O5S
4-{2-[3,4-Bis(difluoromethoxy)phenyl]-2-[6-(4-fluorophenylmethanesulfonyl)3-pyridyl]ethyl}pyridine-N-oxide
—— (2S,3R)-3-(2,4-Difluoro-benzylsulfanyl)-2-(4'-methoxy-biphenyl-4-sulfonylamino)-3-phenyl-propionic acid 334991-42-3 C29H25F2NO5S2
(2S,3R)-3-(2,4-Difluoro-benzylsulfanyl)-2-(4'-methoxy-biphenyl-4-sulfonylamino)-3-phenyl-propionic acid
—— (2S,3R)-2-(4'-Bromo-biphenyl-4-sulfonylamino)-3-phenyl-3-(pyrimidin-2-ylsulfanyl)-propionic acid 334991-28-5 C25H20BrN3O4S2
(2S,3R)-2-(4'-Bromo-biphenyl-4-sulfonylamino)-3-phenyl-3-(pyrimidin-2-ylsulfanyl)-propionic acid
—— 1-[2-(4-{4-[3-(3-Amino-pyrrolidin-1-yl)-propyl]-piperidin-1-yl}-phenylamino)-pteridin-7-yl]-3-tert-butyl-urea 330550-91-9 C29H42N10O
1-[2-(4-{4-[3-(3-Amino-pyrrolidin-1-yl)-propyl]-piperidin-1-yl}-phenylamino)-pteridin-7-yl]-3-tert-butyl-urea
—— 3-(2-(R)-cyclopropylmethyl-3-(S)-hydroxyl-1-oxoheptyl)amino-1-cyclopropylmethyl-5-(4-trifluoromethylphenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one 330840-50-1 C31H36F3N3O3
3-(2-(R)-cyclopropylmethyl-3-(S)-hydroxyl-1-oxoheptyl)amino-1-cyclopropylmethyl-5-(4-trifluoromethylphenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one
—— 1-tert-Butyl-3-(2-{4-[4-(3-piperazin-1-yl-propyl)-piperidin-1-yl]-phenylamino}-pteridin-7-yl)-urea 330550-90-8 C29H42N10O
1-tert-Butyl-3-(2-{4-[4-(3-piperazin-1-yl-propyl)-piperidin-1-yl]-phenylamino}-pteridin-7-yl)-urea
—— 2-[5-chloro-2-({3-[(4,4-diphenyl-1-piperidinyl)methyl]-1H-pyrazol-1-yl}methyl)phenoxy]-N,N-dimethylacetamide 321403-94-5 C32H35ClN4O2
2-[5-chloro-2-({3-[(4,4-diphenyl-1-piperidinyl)methyl]-1H-pyrazol-1-yl}methyl)phenoxy]-N,N-dimethylacetamide
—— 3-(2 (R)-Cyclopentylmethyl-3(S)-hydroxyl-1-oxo-5-phenylpentyl)amino-1-methyl-5-(4-fluoro-phenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one 330839-29-7 C33H36FN3O3
3-(2 (R)-Cyclopentylmethyl-3(S)-hydroxyl-1-oxo-5-phenylpentyl)amino-1-methyl-5-(4-fluoro-phenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one
—— 2-[(S)-1-(3-Trifluoromethylphenyl)ethylamino]-4-[5-(pyridin-4-yl)benzimidazol-1-yl]-6-[2-methylphenyl]pyrimidine 317829-64-4 C32H25F3N6
2-[(S)-1-(3-Trifluoromethylphenyl)ethylamino]-4-[5-(pyridin-4-yl)benzimidazol-1-yl]-6-[2-methylphenyl]pyrimidine
—— 1-[[1-[3-(aminoiminomethyl)phenyl]-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl]-2,3-dihydro-5-[2-(methylsulfonyl)phenyl]-1H-indole 321435-84-1 C27H22F3N5O3S
1-[[1-[3-(aminoiminomethyl)phenyl]-3-(trifluoromethyl)-1H-pyrazol-5-yl]carbonyl]-2,3-dihydro-5-[2-(methylsulfonyl)phenyl]-1H-indole
—— (2S,3R)-2-(4'-methoxy-biphenyl-4-sulfonylamino)-3-phenyl-3-(pyridin-2-ylmethylsulfanyl)-propionic acid 334991-45-6 C28H26N2O5S2
(2S,3R)-2-(4'-methoxy-biphenyl-4-sulfonylamino)-3-phenyl-3-(pyridin-2-ylmethylsulfanyl)-propionic acid
—— (2S,3R)-2-(4'-Methoxy-biphenyl-4-sulfonylamino)-3-(5-methyl-oxazol-2-ylmethylsulfanyl)-3-phenyl-propionic acid 334991-46-7 C27H26N2O6S2
(2S,3R)-2-(4'-Methoxy-biphenyl-4-sulfonylamino)-3-(5-methyl-oxazol-2-ylmethylsulfanyl)-3-phenyl-propionic acid
—— 2-[(3S)-3-({[4-(4-Chlorophenyl)phenyl]sulfonyl}amino)-2-oxopiperidyl]-N-[2-(amidinoaminooxy)ethyl]acetamide 330668-15-0 C22H27ClN6O5S
2-[(3S)-3-({[4-(4-Chlorophenyl)phenyl]sulfonyl}amino)-2-oxopiperidyl]-N-[2-(amidinoaminooxy)ethyl]acetamide
—— 6-[7-(3-benzyl-ureido)-2,5-dioxo-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-3-phenyl-hexanoic acid 320385-77-1 C29H30N4O5
6-[7-(3-benzyl-ureido)-2,5-dioxo-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-3-phenyl-hexanoic acid
—— 2'-(3-trifluoromethylphenylsulfonylaminomethyl)biphenyl-2-carboxylic acid benzylamide 332378-56-0 C28H23F3N2O3S
2'-(3-trifluoromethylphenylsulfonylaminomethyl)biphenyl-2-carboxylic acid benzylamide
—— 1-Ethyl-3-methyl-N-[3-[[3-[(1E)-2-(2-pyridinyl)ethenyl]-1H-indazol-6-yl]carbonyl]phenyl]-1H-pyrazole-5-carboxamide 319460-86-1 C28H24N6O2
1-Ethyl-3-methyl-N-[3-[[3-[(1E)-2-(2-pyridinyl)ethenyl]-1H-indazol-6-yl]carbonyl]phenyl]-1H-pyrazole-5-carboxamide
—— 4-[Bis(4-chlorophenyl)methoxymethyl]-1-(2,2-diphenylethyl)piperidine 300554-51-2 C33H33Cl2NO
4-[Bis(4-chlorophenyl)methoxymethyl]-1-(2,2-diphenylethyl)piperidine
—— 3-(2-(R)-iso-butyl-3-(S)-hydroxyl-1-oxoheptyl)amino-1-methyl-5-(4-trifluoromethylphenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one 330840-05-6 C28H34F3N3O3
3-(2-(R)-iso-butyl-3-(S)-hydroxyl-1-oxoheptyl)amino-1-methyl-5-(4-trifluoromethylphenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one
—— 8-Cyclopentyl-2-{4-[4-(3-piperazin-1-yl-propyl)-piperidin-1-yl]-phenylamino}-8H-pteridin-7-one 330550-59-9 C29H40N8O
8-Cyclopentyl-2-{4-[4-(3-piperazin-1-yl-propyl)-piperidin-1-yl]-phenylamino}-8H-pteridin-7-one
—— 3-(4-methylpiperazin-1-yl)carbonyl-4-(naphthalen-1-yl)-1-{1-[2-(thiophen-2-yl)ethyl]-1H-imidazol-5-yl}methyl-1H-pyrrole 303778-46-3 C30H31N5OS
3-(4-methylpiperazin-1-yl)carbonyl-4-(naphthalen-1-yl)-1-{1-[2-(thiophen-2-yl)ethyl]-1H-imidazol-5-yl}methyl-1H-pyrrole
—— 5H-[1,4]oxathiepino[6,5-b]pyridine-8-carboxylic acid, 9-(2-chloro-6-fluorophenyl)-2,3,6,9-tetrahydro-7-methyl-, 2-[(cyclopropylcarbonyl)oxy]ethyl ester, 1,1-dioxide 319909-04-1 C22H23ClFNO7S
5H-[1,4]oxathiepino[6,5-b]pyridine-8-carboxylic acid, 9-(2-chloro-6-fluorophenyl)-2,3,6,9-tetrahydro-7-methyl-, 2-[(cyclopropylcarbonyl)oxy]ethyl ester, 1,1-dioxide
—— 2-(oxalyl-amino)-5-(1,1,3-trioxo-5-phenyl-1,3-dihydro-isothiazol-2-ylmethyl)-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid 330193-31-2 C20H16N2O9S2
2-(oxalyl-amino)-5-(1,1,3-trioxo-5-phenyl-1,3-dihydro-isothiazol-2-ylmethyl)-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid
—— 3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[(4-acetylaminophenoxy)methyl]propanoic acid 321584-98-9 C24H22ClNO6S
3-[(4'-chloro[1,1'-biphenyl]-4-yl)sulfonyl]-2-[(4-acetylaminophenoxy)methyl]propanoic acid
—— 4-[2-(7-{2-[4-(tert-butoxy)phenoxy]ethyl}-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl)ethoxy]isophthalonitrile 335620-67-2 C28H34N4O4
4-[2-(7-{2-[4-(tert-butoxy)phenoxy]ethyl}-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl)ethoxy]isophthalonitrile
—— 4-(3-{7-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl]-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl}-2-hydroxypropoxy)benzonitrile 335619-40-4 C26H29N3O6
4-(3-{7-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl]-9-oxa-3,7-diazabicyclo[3.3.1]non-3-yl}-2-hydroxypropoxy)benzonitrile