trans-3-(2,2-dichloro-vinyl)-2,2-dimethyl-cyclopropane-1R-carboxylic acidα-(S)-cyano-3-phenoxy-4-fluoro-benzyl ester

• 分子结构分类: 有机化合物 - 脂质和类脂质分子 - 脂肪酰基
• 英文名称: trans-3-(2,2-dichloro-vinyl)-2,2-dimethyl-cyclopropane-1R-carboxylic acidα-(S)-cyano-3-phenoxy-4-fluoro-benzyl ester
• 英文别名: (R)-α-cyano-4-fluoro-3-phenoxybenzyl (1R,cis)-3-(2,2-dichlorovinyl)-2,2-dimethylcyclopropane carboxylate；[cyano-(4-fluoro-3-phenoxyphenyl)methyl] (1R,3R)-3-(2,2-dichloroethenyl)-2,2-dimethylcyclopropane-1-carboxylate
• 化学式: C₂₂H₁₈Cl₂FNO₃
• 分子量: 434.294
• InChiKey: QQODLKZGRKWIFG-JSFUQZLZSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  6.2
• 重原子数：
  29
• 可旋转键数：
  7
• 环数：
  3.0
• sp3杂化的碳原子比例：
  0.27
• 拓扑面积：
  59.3
• 氢给体数：
  0
• 氢受体数：
  5

文献信息

• ALPHA-CYANO-4-FLUORO-3-PHENOXYBENZYL META-HALO PYRETHRATE, A PROCESS FOR PREPARING THE SAME AND THE USES THEREOF
  申请人：Zou Xinzhuo

  公开号：US20100286265A1

  公开（公告）日：2010-11-11

  The present invention relates to a compound of formula (I), stereoisomers thereof or the mixture of these stereoisomers, wherein: X represents a halogen atom, i.e. F, Cl, Br. The present invention also relates to a process for preparing the compound, and to a use of the compound in the preparation of an insecticide for controlling or killing vectors in the public hygiene and disease control, and to a use of the compound in the preparation of an insecticide for controlling or killing insects, nematodes, and mites in agriculture or horticulture.

  本发明涉及公式(I)的化合物及其立体异构体或这些立体异构体的混合物，其中：X代表卤素原子，即F，Cl，Br。本发明还涉及制备该化合物的方法，以及在公共卫生和疾病控制中控制或杀灭媒介生物的杀虫剂的制备中使用该化合物的用途，以及在农业或园艺中控制或杀灭昆虫，线虫和螨类的杀虫剂的制备中使用该化合物的用途。
• DEUTERATED BENZYLBENZENE DERIVATIVES AND METHODS OF USE
  申请人：Seed Brian

  公开号：US20100063141A1

  公开（公告）日：2010-03-11

  Provided are compounds having an inhibitory effect on sodium-dependent glucose cotransporter SGLT. The invention also provides pharmaceutical compositions, methods of preparing the compounds, synthetic intermediates, and methods of using the compounds, independently or in combination with other therapeutic agents, for treating diseases and conditions that are affected by SGLT inhibition.

  提供了对钠依赖性葡萄糖共转运体SGLT具有抑制作用的化合物。本发明还提供了制备这些化合物的药物组合物、制备方法、合成中间体以及使用这些化合物的方法，独立或与其他治疗剂联合治疗受SGLT抑制影响的疾病和病况。
• Pesticidal methods and compositions
  申请人：SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V.

  公开号：EP0647401A1

  公开（公告）日：1995-04-12

  A pesticidal composition which includes a substituted 1,2,4-triazole compound and a pyrethroid insecticide is disclosed. The pesticidal composition is particularly effective against aphid pests.

  本发明公开了一种杀虫组合物，其中包括一种取代的 1,2,4-三唑化合物和一种拟除虫菊酯杀虫剂。该杀虫组合物对蚜虫特别有效。
• Synergistic compositions with diafenthiuron
  申请人：CIBA-GEIGY AG

  公开号：EP0736252A2

  公开（公告）日：1996-10-09

  There are described a pesticidal composition which comprises a pesticidally-synergistically active combination, in various proportions, of the active ingredient of the formula in free form or in the form of an agrochemically acceptable salt, and one or more pesticidally active compound(s) (I) to (LXIX) as described in claim 1, a method of controlling pests, a process for the preparation of the composition, its use, and plant propagation material treated therewith, and the use of the compound of the formula (A) for the preparation of the composition.

  描述了一种杀虫组合物，该组合物包括不同比例的杀虫增效活性组合物，其活性成分的式为 以游离形式或以农用化学品可接受的盐的形式、 和权利要求1所述的一种或多种农药活性化合物(I)至(LXIX)、 3.一种防治害虫的方法、一种制备组合物的工艺、其用途和用其处理的植物繁殖材料，以及使用式(A)化合物制备组合物。
• Method for the enhancement of the residual activity of pesticide formulations
  申请人：American Cyanamid Company

  公开号：EP0981957A1

  公开（公告）日：2000-03-01

  The present invention relates to the preparation of novel solid pesticide formulations which, after application, provide a dry, coherent deposit of the pesticidal agent on the target, resulting in increased residual activity and greater efficacy when applied to various agricultural products, especially food crops. This enhanced residual activity results from formulation of the pesticidal agent with 10-75% by weight of a polyvinylpyrrolidone polymer or copolymer and application of the formulation to the target.

  本发明涉及新型固体农药制剂的制备，施用该制剂后，杀虫剂会在目标物上形成干燥、连贯的沉积物，从而在施用到各种农产品，特别是粮食作物上时，可提高残留活性和药效。将杀虫剂与 10-75% （按重量计）的聚乙烯吡咯烷酮聚合物或共聚物配制成制剂并施用到目标物上，可提高残留活性。